Crystallography Open Database

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7150278 CIFC20 H24 O SP 21 21 219.932; 11.5642; 14.7502
90; 90; 90
1694.14Hitchcock, Peter B.; Rowlands, Gareth J.; Seacome, Richard J.
The synthesis and directed ortho-lithiation of 4-tert-butylsulfinyl[2.2]paracyclophane.
Organic & biomolecular chemistry, 2005, 3, 3873-3876
7150279 CIFC20 H24 O SP 21 21 219.9622; 11.5421; 14.9696
90; 90; 90
1721.28Hitchcock, Peter B.; Rowlands, Gareth J.; Seacome, Richard J.
The synthesis and directed ortho-lithiation of 4-tert-butylsulfinyl[2.2]paracyclophane.
Organic & biomolecular chemistry, 2005, 3, 3873-3876
7150291 CIFC23 H25 N O2 SP 21 21 2110.712; 13.782; 14.26
90; 90; 90
2105.24Betson, Mark S.; Clayden, Jonathan; Helliwell, Madeleine; Mitjans, David
Kinetic and thermodynamic stereocontrol in the atroposelective formation of sulfoxides by oxidation of 2-sulfanyl-1-naphthamides.
Organic & biomolecular chemistry, 2005, 3, 3898-3904
7150300 CIFC20 H34 O7P 21 21 219.2857; 10.4352; 21.127
90; 90; 90
2047.17Ley, Steven V.; Dixon, Darren J.; Guy, Richard T.; Rodríguez, Félix; Sheppard, Tom D.
Michael, Michael-aldol and Michael-Michael reactions of enolate equivalents of butane-2,3-diacetal protected glycolic acid derivatives.
Organic & biomolecular chemistry, 2005, 3, 4095-4107
7150303 CIFC17 H28 O6P 21 21 217.9383; 14.4423; 15.4979
90; 90; 90
1776.79Ley, Steven V.; Dixon, Darren J.; Guy, Richard T.; Rodríguez, Félix; Sheppard, Tom D.
Michael, Michael-aldol and Michael-Michael reactions of enolate equivalents of butane-2,3-diacetal protected glycolic acid derivatives.
Organic & biomolecular chemistry, 2005, 3, 4095-4107
7150304 CIFC14 H22 O6P 21 21 218.5902; 10.0809; 16.5589
90; 90; 90
1433.95Ley, Steven V.; Dixon, Darren J.; Guy, Richard T.; Rodríguez, Félix; Sheppard, Tom D.
Michael, Michael-aldol and Michael-Michael reactions of enolate equivalents of butane-2,3-diacetal protected glycolic acid derivatives.
Organic & biomolecular chemistry, 2005, 3, 4095-4107
7150332 CIFC78 H87 Cl6 N3 O9P 21 21 2130.941; 23.839; 10.252
90; 90; 90
7562Toda, Fumio; Yoshizawa, Kazuhiro; Hyoda, Shunji; Toyota, Shinji; Chatziefthimiou, Spyros; Mavridis, Irene M.
Efficient resolution of 2,2'-dihydroxy-1,1'-binaphthyl by inclusion complexation with chiral N-(3-chloro-2-hydroxypropyl)-N,N,N-trimethylammonium chloride.
Organic & biomolecular chemistry, 2004, 2, 449-451
7150344 CIFC23 H36 N2 O5P 21 21 219.005; 16.541; 16.841
90; 90; 90
2508.5Charrier, Jean-Damien; Hadfield, David S.; Hitchcock, Peter B.; Young, Douglas W.
Synthesis of (2S,4S)- and (2S,4R)-5-fluoroleucine and (2S,4S)-[5,5-2H2]-5-fluoroleucine.
Organic & biomolecular chemistry, 2004, 2, 474-482
7150351 CIFC66 H83 N5 O9 Si3P 21 21 2120.698; 28.908; 11.465
90; 90; 90
6859.9Takasawa, Ryoichi; Yoshikawa, Isao; Araki, Koji
Use of an adjustable soft segment as an effective molecular design for crystal engineering of hydrogen-bonded tape motifs.
Organic & biomolecular chemistry, 2004, 2, 1125-1132
7150357 CIFC22 H41 N5 O3 Si2P 21 21 217.5; 8.329; 43.319
90; 90; 90
2706.03Takasawa, Ryoichi; Yoshikawa, Isao; Araki, Koji
Use of an adjustable soft segment as an effective molecular design for crystal engineering of hydrogen-bonded tape motifs.
Organic & biomolecular chemistry, 2004, 2, 1125-1132
7150362 CIFC15 H17 F O3P 21 21 216.8956; 8.0263; 25.0635
90; 90; 90
1387.17Buffet, Marianne F.; Dixon, Darren J.; Ley, Steven V.; Reynolds, Dominic J.; Storer, R. Ian
Anomeric oxygen to carbon rearrangements of alkynyl tributylstannane derivatives of furanyl (gamma)- and pyranyl (delta)-lactols.
Organic & biomolecular chemistry, 2004, 2, 1145-1154
7150384 CIFC38 H53 N5 O6 SP 21 21 2111.234; 16.394; 20.993
90; 90; 90
3866.28Nyangulu, James M.; Nelson, Ken M.; Rose, Patricia A.; Gai, Yuanzhu; Loewen, Mary; Lougheed, Brenda; Quail, J. Wilson; Cutler, Adrian J.; Abrams, Suzanne R.
Synthesis and biological activity of tetralone abscisic acid analogues.
Organic & biomolecular chemistry, 2006, 4, 1400-1412
7150406 CIFC18 H19 N O3 SeP 21 21 214.8305; 13.532; 26.21
90; 90; 90
1713.3Fenner, Tahli; White, Jonathan M.; Schiesser, Carl H.
Preparation of 2,3-dihydroselenolo[2,3-b]pyridines and related compounds by free-radical means.
Organic & biomolecular chemistry, 2006, 4, 466-474
7150416 CIFC12 H24 N2 O3P 21 21 218.73; 9.741; 17.509
90; 90; 90
1488.9Sengupta, Anindita; Roy, Rituparna S.; Sabareesh, Varatharajan; Shamala, Narayanaswamy; Balaram, Padmanabhan
Aggregation modes in sheets formed by protected beta-amino acids and beta-peptides.
Organic & biomolecular chemistry, 2006, 4, 1166-1173
7150418 CIFC18 H34 N2 O5P 21 21 219.3852; 11.899; 19.199
90; 90; 90
2144Sengupta, Anindita; Roy, Rituparna S.; Sabareesh, Varatharajan; Shamala, Narayanaswamy; Balaram, Padmanabhan
Aggregation modes in sheets formed by protected beta-amino acids and beta-peptides.
Organic & biomolecular chemistry, 2006, 4, 1166-1173
7150419 CIFC18 H34 N2 O5P 21 21 215.17; 10.86; 37.3
90; 90; 90
2094Sengupta, Anindita; Roy, Rituparna S.; Sabareesh, Varatharajan; Shamala, Narayanaswamy; Balaram, Padmanabhan
Aggregation modes in sheets formed by protected beta-amino acids and beta-peptides.
Organic & biomolecular chemistry, 2006, 4, 1166-1173
7150424 CIFC22 H28 N4 O SiP 21 21 217.4112; 15.3453; 19.811
90; 90; 90
2253Morrison, Christopher F.; Vaters, Jamie P.; Miller, David O.; Burnell, D. Jean
Facial selectivity in the 4 + 2 reactions of a diene derived from carvone
Organic & Biomolecular Chemistry, 2006, 4, 1160
7150425 CIFC22 H28 N4 O SiP 21 21 2117.488; 17.514; 7.601
90; 90; 90
2328.1Morrison, Christopher F.; Vaters, Jamie P.; Miller, David O.; Burnell, D. Jean
Facial selectivity in the 4 + 2 reactions of a diene derived from carvone
Organic & Biomolecular Chemistry, 2006, 4, 1160
7150432 CIFC23 H25 F N2 O3P 21 21 2112.174; 21.549; 7.6755
90; 90; 90
2013.6Peng, Hairuo; Carrico, Dora; Thai, Van; Blaskovich, Michelle; Bucher, Cynthia; Pusateri, Erin E.; Sebti, Said M.; Hamilton, Andrew D.
Synthesis and evaluation of potent, highly-selective, 3-aryl-piperazinone inhibitors of protein geranylgeranyltransferase-I.
Organic & biomolecular chemistry, 2006, 4, 1768-1784
7150434 CIFC11 H15 N O5P 21 21 216.0153; 12.4888; 15.2629
90; 90; 90
1146.61Li, Hongqing; Schütz, Catherine; Favre, Sylvain; Zhang, Yongmin; Vogel, Pierre; Sinaÿ, Pierre; Blériot, Yves
Nucleophilic opening of epoxyazepanes: expanding the family of polyhydroxyazepane-based glycosidase inhibitors.
Organic & biomolecular chemistry, 2006, 4, 1653-1662
7150436 CIFC22 H29 NP 21 21 219.807; 11.749; 16.027
90; 90; 90
1846.7Petersen, Michael Axman; Nielsen, Iben B.; Kristensen, Michael B.; Kadziola, Anders; Lammich, Lutz; Andersen, Lars H.; Nielsen, Mogens Brøndsted
Novel retinylidene iminium salts for defining opsin shifts: synthesis and intrinsic chromophoric properties.
Organic & biomolecular chemistry, 2006, 4, 1546-1554
7150437 CIFC22 H29 NP 21 21 219.884; 11.711; 16.091
90; 90; 90
1862.6Petersen, Michael Axman; Nielsen, Iben B.; Kristensen, Michael B.; Kadziola, Anders; Lammich, Lutz; Andersen, Lars H.; Nielsen, Mogens Brøndsted
Novel retinylidene iminium salts for defining opsin shifts: synthesis and intrinsic chromophoric properties.
Organic & biomolecular chemistry, 2006, 4, 1546-1554
7150439 CIFC12 H19 N3 O4P 21 21 215.6733; 11.538; 21.3149
90; 90; 90
1395.24Ahmed, Omar; Hitchcock, Peter B.; Young, Douglas W.
Investigation of a route to ibotenic acid analogues via a reduced pyroglutamate template.
Organic & biomolecular chemistry, 2006, 4, 1596-1603
7150451 CIFC32 H28 N8 O7P 21 21 217.688; 13.2934; 31.112
90; 90; 90
3179.64Rosenbohm, Christoph; Christensen, Signe M.; Sørensen, Mads D.; Pedersen, Daniel Sejer; Larsen, Lotte-Emilie; Wengel, Jesper; Koch, Troels
Synthesis of 2'-amino-LNA: a new strategyElectronic supplementary information (ESI) available: further experimental details and the structure of compound S11 (.pdb file). See http://www.rsc.org/suppdata/ob/b2/b208864a/
Organic & Biomolecular Chemistry, 2003, 1, 655
7150455 CIFC10 H16 OP 21 21 215.9714; 20.5466; 22.5632
90; 90; 90
2768.32Amelia García Fraile; David G. Morris; Antonio García Martínez; Santiago de la Moya Cerero; Kenneth W. Muir; Karl S. Ryder; Enrique Teso Vilar
Self-recognition and hydrogen bonding by polycyclic bridgehead monoalcohols
Org. Biomol. Chem., 2003, 1, 700-704
7150461 CIFC22 H23 N O7P 21 21 219.3201; 12.5782; 17.9679
90; 90; 90
2106.38Anat Reizelman; Suzanne C. M. Wigchert; Cinzia del-Bianco; Binne Zwanenburg
Synthesis and bioactivity of labelled germination stimulants for the isolation and identification of the strigolactone receptor
Org. Biomol. Chem., 2003, 1, 950-959
7150476 CIFC32 H39 N O12P 21 21 217.917; 19.736; 21.32
90; 90; 90
3331.2Liao, Jian; Peng, Xiaohua; Zhang, Juhua; Yu, Kaibei; Cui, Xin; Zhu, Jin; Deng, Jingen
Facile resolution of racemic terbutaline and a study of molecular recognition through chiral supramolecules based on enantiodifferentiating self-assemblyElectronic supplementary information (ESI) available: 1) 1H and 13C NMR analyses of (R)-1·4 and (S)-1·4; 2) ORTEP views and stacking structures of crystals 5, 7 and 8; 3) DSC and TG analyses of the more- and less-soluble salts. See http://www.rsc.org/suppdata/ob/b2/b211327a/
Organic & Biomolecular Chemistry, 2003, 1, 1080
7150479 CIFC35 H45 N O13P 21 21 217.81; 21.431; 21.948
90; 90; 90
3673.6Liao, Jian; Peng, Xiaohua; Zhang, Juhua; Yu, Kaibei; Cui, Xin; Zhu, Jin; Deng, Jingen
Facile resolution of racemic terbutaline and a study of molecular recognition through chiral supramolecules based on enantiodifferentiating self-assemblyElectronic supplementary information (ESI) available: 1) 1H and 13C NMR analyses of (R)-1·4 and (S)-1·4; 2) ORTEP views and stacking structures of crystals 5, 7 and 8; 3) DSC and TG analyses of the more- and less-soluble salts. See http://www.rsc.org/suppdata/ob/b2/b211327a/
Organic & Biomolecular Chemistry, 2003, 1, 1080
7150529 CIFC20 H27 N O6 SP 21 21 216.5353; 9.8759; 30.2519
90; 90; 90
1952.52Evans, Amanda C.; Longbottom, Deborah A.; Matsuoka, Masato; Davies, John E.; Turner, Richard; Franckevičius, Vilius; Ley, Steven V.
Highly diastereoselective desymmetrisation of cyclic meso-anhydrides and derivatisation for use in natural product synthesis
Organic & Biomolecular Chemistry, 2009, 7, 747-760
7150530 CIFC14 H22 O3P 21 21 215.797; 12.152; 20.075
90; 90; 90
1414.2Zhang, Xue-jing; Yan, Ming; Huang, Dan
Catalyzed addition of diazoacetoacetates to imines: synthesis of highly functionalized aziridines
Organic & Biomolecular Chemistry, 2009, 7, 187-192
7150564 CIFC26 H24 N2 O2P 21 21 219.0438; 14.174; 19.0124
90; 90; 90
2437.1Libendi, Samuel Shikuku; Demizu, Yosuke; Onomura, Osamu
Direct electrochemical α-cyanation of N-protected cyclic amines
Organic & Biomolecular Chemistry, 2009, 7, 351-356
7150569 CIFC45 H91.249 O43.6245P 21 21 2115.5665; 23.5385; 33.1929
90; 90; 90
12162.3Osaki, Motofumi; Takashima, Yoshinori; Yamaguchi, Hiroyasu; Harada, Akira
Switching of polymerization activity of cinnamoyl-α-cyclodextrin
Organic & Biomolecular Chemistry, 2009, 7, 1646-1651
7150570 CIFC29 H39 N O4P 21 21 2111.5712; 13.9737; 17.038
90; 90; 90
2754.92Davies, Stephen G.; Durbin, Matthew J.; Goddard, Euan C.; Kelly, Peter M.; Kurosawa, Wataru; Lee, James A.; Nicholson, Rebecca L.; Price, Paul D.; Roberts, Paul M.; Russell, Angela J.; Scott, Philip M.; Smith, Andrew D.
Doubly diastereoselective conjugate addition of homochiral lithium amides to homochiral α,β-unsaturated esters containing cis- and trans-dioxolane units
Organic & Biomolecular Chemistry, 2009, 7, 761-776
7150573 CIFC15 H16 O4P 21 21 216.5457; 12.2932; 30.973
90; 90; 90
2492.3Li, Yi; Nawrat, Christopher C.; Pattenden, Gerald; Winne, Johan M.
A concise total synthesis of (±)-anthecularin
Organic & Biomolecular Chemistry, 2009, 7, 639-640
7150577 CIFC15 H21 N O2 SP 21 21 216.237; 12.419; 17.923
90; 90; 90
1388.3Klein, Johannes E. M. N.; Müller-Bunz, Helge; Evans, Paul
Studies concerning the electrophilic amino-alkene cyclisation for the synthesis of bicyclic amines
Organic & Biomolecular Chemistry, 2009, 7, 986-995
7150581 CIFC65 H89 I N2 O8P 21 21 2111.2099; 15.8759; 35.534
90; 90; 90
6323.9Podoprygorina, Ganna; Bolte, Michael; Böhmer, Volker
Tetra-urea calix[4]arenes 1,3-bridged at the narrow rim
Organic & Biomolecular Chemistry, 2009, 7, 1592-1598
7150624 CIFC16 H19 Br O5P 21 21 219.648; 9.9528; 17.941
90; 90; 90
1722.8Yang, Jin; Wang, Ting; Ding, Zhenhua; Shen, Zongxuan; Zhang, Yawen
Highly diastereo- and enantioselective organocatalytic addition of acetone to β-substituted α-ketoesters via dynamic kinetic resolution
Organic & Biomolecular Chemistry, 2009, 7, 2208-2213
7150625 CIFC18 H21 N3 OP 21 21 216.1265; 13.8082; 19.2305
90; 90; 90
1626.82Coeffard, Vincent; Müller-Bunz, Helge; Guiry, Patrick J.
The synthesis of new oxazoline-containing bifunctional catalysts and their application in the addition of diethylzinc to aldehydes
Organic & Biomolecular Chemistry, 2009, 7, 1723-1734
7150626 CIFC18 H21 Cl2 N3 O ZnP 21 21 2110.4417; 11.1428; 17.018
90; 90; 90
1980.04Coeffard, Vincent; Müller-Bunz, Helge; Guiry, Patrick J.
The synthesis of new oxazoline-containing bifunctional catalysts and their application in the addition of diethylzinc to aldehydes
Organic & Biomolecular Chemistry, 2009, 7, 1723-1734
7150655 CIFC23 H23 N3 O3P 21 21 217.9563; 8.4315; 28.798
90; 90; 90
1931.9Walton, Jeffrey G. A.; Patterson, Stephen; Liu, Gu; Haraldsen, Jeralyn D.; Hollick, Jonathan J.; Slawin, Alexandra M. Z.; Ward, Gary E.; Westwood, Nicholas J.
Synthesis and biological evaluation of functionalised tetrahydro-β-carboline analogues as inhibitors of Toxoplasma gondii invasion
Organic & Biomolecular Chemistry, 2009, 7, 3049
7150656 CIFC11 H16 O3P 21 21 217.475; 8.234; 16.061
90; 90; 90
988.5Stevens, Anne T.; Caira, Mino R.; Bull, James R.; Chibale, Kelly
Cycloaddition and one-carbon homologation studies in the synthesis of advanced iridoid precursors
Organic & Biomolecular Chemistry, 2009, 7, 3527-3536
7150662 CIFC29 H32.33 N O2P 21 21 218.9487; 5.1851; 52.29
90; 90; 90
2426.25Davies, Stephen G.; Garner, A. Christopher; Nicholson, Rebecca L.; Osborne, James; Roberts, Paul M.; Savory, Edward D.; Smith, Andrew D.; Thomson, James E.
Doubly diastereoselective [3,3]-sigmatropic aza-Claisen rearrangements
Organic & Biomolecular Chemistry, 2009, 7, 2604-2611
7150701 CIFC12 H21 N O3P 21 21 219.725; 6.479; 20.325
90; 90; 90
1280.6Pandey, Ganesh; Grahacharya, Debasish; Shashidhara, K. S.; Khan, M. Islam; Puranik, Vedavati G.
Synthesis of polyfunctional quinolizidine alkaloids: development towards selective glycosidase inhibitors
Organic & Biomolecular Chemistry, 2009, 7, 3300-3307
7150702 CIFC13 H23 N O4P 21 21 215.3743; 10.2506; 24.3106
90; 90; 90
1339.27Pandey, Ganesh; Grahacharya, Debasish; Shashidhara, K. S.; Khan, M. Islam; Puranik, Vedavati G.
Synthesis of polyfunctional quinolizidine alkaloids: development towards selective glycosidase inhibitors
Organic & Biomolecular Chemistry, 2009, 7, 3300-3307
7150703 CIFC14 H28 N4 O7P 21 21 217.814; 14.5374; 16.0994
90; 90; 90
1828.82Fernández-Tejada, Alberto; Corzana, Francisco; Busto, Jesús H.; Avenoza, Alberto; Peregrina, Jesús M.
Stabilizing unusual conformations in small peptides and glucopeptides using a hydroxylated cyclobutane amino acid
Organic & Biomolecular Chemistry, 2009, 7, 2885-2893
7150705 CIFC25 H25 N5 OP 21 21 215.1252; 17.913; 23.305
90; 90; 90
2139.6Ghiviriga, Ion; El-Gendy, Bahaa El-Dien M.; Steel, Peter J.; Katritzky, Alan R.
Tautomerism of guanidines studied by 15N NMR: 2-hydrazono-3-phenylquinazolin-4(3H)-ones and related compounds
Organic & Biomolecular Chemistry, 2009, 7, 4110-4119
7150712 CIFC17 H15 N O2P 21 21 216.0167; 10.2379; 22.355
90; 90; 90
1377Lu, Ting; Hayashi, Ryuji; Hsung, Richard P.; DeKorver, Kyle A.; Lohse, Andrew G.; Song, Zhenlei; Tang, Yu
Synthesis of amido-spiro[2.2]pentanes via Simmons–Smith cyclopropanation of allenamides
Organic & Biomolecular Chemistry, 2009, 7, 3331-3337
7150715 CIFC14 H15 N O2P 21 21 216.4331; 11.657; 15.86
90; 90; 90
1189.4Lu, Ting; Hayashi, Ryuji; Hsung, Richard P.; DeKorver, Kyle A.; Lohse, Andrew G.; Song, Zhenlei; Tang, Yu
Synthesis of amido-spiro[2.2]pentanes via Simmons–Smith cyclopropanation of allenamides
Organic & Biomolecular Chemistry, 2009, 7, 3331-3337
7150722 CIFC25 H28 N2 O6P 21 21 217.67; 14.837; 20.519
90; 90; 90
2335.06Cheeseman, Matt; Davies, Iwan R.; Axe, Phil; Johnson, Andrew L.; Bull, Steven D.
A temporary stereocentre approach for the asymmetric synthesis of chiral cyclopropane-carboxaldehydes
Organic & Biomolecular Chemistry, 2009, 7, 3537-3548
7150727 CIFC18 H19 N2 O4 PP 21 21 216.0491; 8.3323; 34.349
90; 90; 90
1731.3Hou, Jian-Bo; Zhang, Hui; Guo, Jian-Nan; Liu, Yan; Xu, Peng-Xiang; Zhao, Yu-Fen; Blackburn, G. Michael
Chirality at phosphorus in pentacoordinate spirophosphoranes: stereochemistry by X-ray structure and spectroscopic analysis
Organic & Biomolecular Chemistry, 2009, 7, 3020
7150728 CIFC18 H19 N2 O4 PP 21 21 216.0474; 8.329; 34.27
90; 90; 90
1726.14Hou, Jian-Bo; Zhang, Hui; Guo, Jian-Nan; Liu, Yan; Xu, Peng-Xiang; Zhao, Yu-Fen; Blackburn, G. Michael
Chirality at phosphorus in pentacoordinate spirophosphoranes: stereochemistry by X-ray structure and spectroscopic analysis
Organic & Biomolecular Chemistry, 2009, 7, 3020
7150730 CIFC37 H52 Cl2 N2 O13 SP 21 21 217.4542; 23.187; 23.706
90; 90; 90
4097.4Bragnier, Nicolas; Guillot, Regis; Scherrmann, Marie-Christine
Diastereoselective addition of sugar radicals to camphorsultam glyoxilic oxime ether: a route toward C-glycosylthreonine and allothreonine
Organic & Biomolecular Chemistry, 2009, 7, 3918-3921
7150731 CIFC36 H50 N2 O13 SP 21 21 2112.629; 14.954; 20.739
90; 90; 90
3917Bragnier, Nicolas; Guillot, Regis; Scherrmann, Marie-Christine
Diastereoselective addition of sugar radicals to camphorsultam glyoxilic oxime ether: a route toward C-glycosylthreonine and allothreonine
Organic & Biomolecular Chemistry, 2009, 7, 3918-3921
7150732 CIFC18 H26 O11P 21 21 219.9034; 10.2924; 20.413
90; 90; 90
2080.7Bragnier, Nicolas; Guillot, Regis; Scherrmann, Marie-Christine
Diastereoselective addition of sugar radicals to camphorsultam glyoxilic oxime ether: a route toward C-glycosylthreonine and allothreonine
Organic & Biomolecular Chemistry, 2009, 7, 3918-3921
7150772 CIFC19 H20 O3 SP 21 21 215.6114; 11.6946; 25.505
90; 90; 90
1673.7Stalford, Susanne A.; Kilner, Colin A.; Leach, Andrew G.; Turnbull, W. Bruce
Neighbouring group participation vs. addition to oxacarbenium ions: studies on the synthesis of mycobacterial oligosaccharides
Organic & Biomolecular Chemistry, 2009, 7, 4842-4852
7150789 CIFC23 H21 N O3P 21 21 219.729; 10.168; 18.965
90; 90; 90
1876.1Jennings, W. Brian; McCarthy, Noel J. P.; Kelly, Padraig; Malone, John F.
Topically resolved intramolecular CH-π interactions in phenylalanine derivatives
Organic & Biomolecular Chemistry, 2009, 7, 5156-5162
7150791 CIFC23 H21 N O3P 21 21 219.212; 10.822; 19.309
90; 90; 90
1925Jennings, W. Brian; McCarthy, Noel J. P.; Kelly, Padraig; Malone, John F.
Topically resolved intramolecular CH-π interactions in phenylalanine derivatives
Organic & Biomolecular Chemistry, 2009, 7, 5156-5162
7150792 CIFC16 H11 N3 OP 21 21 215.6393; 11.9631; 38.0483
90; 90; 90
2566.87Tran, Tuan P.; Patel, Nandini; Samas, Brian; Schwarz, Jacob B.
Robust preparation of novel imidazo[5,1-b][1,3,4]oxadiazoles
Organic & Biomolecular Chemistry, 2009, 7, 5063-5066
7150794 CIFC20 H28 N2 O8P 21 21 218.681; 9.784; 24.875
90; 90; 90
2112.8Hartmann, Caroline E.; Gross, Patrick J.; Nieger, Martin; Bräse, Stefan
Towards an asymmetric synthesis of the bacterial peptide deformylase (PDF) inhibitor fumimycin
Organic & Biomolecular Chemistry, 2009, 7, 5059-5062
7150795 CIFC24 H30 N4 O4P 21 21 218.771; 9.743; 26.204
90; 90; 90
2239.3Jiang, Jun; Chen, Xiaohong; Wang, Jun; Hui, Yonghai; Liu, Xiaohua; Lin, Lili; Feng, Xiaoming
Chiral biphenylamide derivative: an efficient organocatalyst for the enantioselective synthesis of α-hydroxy phosphonates
Organic & Biomolecular Chemistry, 2009, 7, 4355-4357
7150803 CIFC23 H22 Co2 N2 O12P 21 21 218.7674; 9.3303; 31.529
90; 90; 90
2579.2Sergeant, Craig D.; Ott, Ingo; Sniady, Adam; Meneni, Srinivasarao; Gust, Ronald; Rheingold, Arnold L.; Dembinski, Roman
Metallo-nucleosides: synthesis and biological evaluation of hexacarbonyl dicobalt 5-alkynyl-2′-deoxyuridines
Organic & Biomolecular Chemistry, 2008, 6, 73-80
7150815 CIFC28 H46 O5 SiP 21 21 218.43; 16.304; 20.801
90; 90; 90
2858.9Burton, Jonathan W.; Anderson, Edward A.; O'Sullivan, Paul T.; Collins, Ian; Davies, John E.; Bond, Andrew D.; Feeder, Neil; Holmes, Andrew B.
The Claisen rearrangement approach to fused bicyclic medium-ring oxacycles
Organic & Biomolecular Chemistry, 2008, 6, 693-702
7150817 CIFC12 H14 O5P 21 21 217.8054; 10.1991; 14.3886
90; 90; 90
1145.45Burton, Jonathan W.; Anderson, Edward A.; O'Sullivan, Paul T.; Collins, Ian; Davies, John E.; Bond, Andrew D.; Feeder, Neil; Holmes, Andrew B.
The Claisen rearrangement approach to fused bicyclic medium-ring oxacycles
Organic & Biomolecular Chemistry, 2008, 6, 693-702
7150818 CIFC26 H44 O5 SiP 21 21 218.04; 16.929; 19.604
90; 90; 90
2668.3Burton, Jonathan W.; Anderson, Edward A.; O'Sullivan, Paul T.; Collins, Ian; Davies, John E.; Bond, Andrew D.; Feeder, Neil; Holmes, Andrew B.
The Claisen rearrangement approach to fused bicyclic medium-ring oxacycles
Organic & Biomolecular Chemistry, 2008, 6, 693-702
7150834 CIFC17 H27 Cu F6 N3 O4P 21 21 218.3666; 15.4945; 16.3029
90; 90; 90
2113.45Stones, Graham; Tripoli, Régis; McDavid, Colin L.; Roux-Duplâtre, Kewin; Kennedy, Alan R.; Sherrington, David C.; Gibson, Colin L.
Investigation of macrocyclisation routes to 1,4,7-triazacyclononanes: efficient syntheses from 1,2-ditosylamides
Organic & Biomolecular Chemistry, 2008, 6, 374-384
7150838 CIFC14 H15.3 N5 O6.15P 21 21 215.9329; 14.5318; 18.898
90; 90; 90
1629.3Anegundi, Ramakrishna I.; Puranik, Vedavati G.; Hotha, Srinivas
Synthesis of 1,2,3-triazole and 1,2,3,4-tetrazole-fused glycosides and nucleosides by an intramolecular 1,3-dipolar cycloaddition reaction
Organic & Biomolecular Chemistry, 2008, 6, 779-786
7150839 CIFC10 H14 N4 O4P 21 21 215.6672; 9.8214; 21.2188
90; 90; 90
1181.03Anegundi, Ramakrishna I.; Puranik, Vedavati G.; Hotha, Srinivas
Synthesis of 1,2,3-triazole and 1,2,3,4-tetrazole-fused glycosides and nucleosides by an intramolecular 1,3-dipolar cycloaddition reaction
Organic & Biomolecular Chemistry, 2008, 6, 779-786
7150840 CIFC11 H15 N3 O4P 21 21 215.495; 10.054; 21.33
90; 90; 90
1178.4Anegundi, Ramakrishna I.; Puranik, Vedavati G.; Hotha, Srinivas
Synthesis of 1,2,3-triazole and 1,2,3,4-tetrazole-fused glycosides and nucleosides by an intramolecular 1,3-dipolar cycloaddition reaction
Organic & Biomolecular Chemistry, 2008, 6, 779-786
7150843 CIFC48 H67 N O5P 21 21 216.3023; 19.07; 35.095
90; 90; 90
4217.9Taniguchi, Kayoko; Aruga, Marie; Yasutake, Mikio; Hirose, Takuji
Solvent control of optical resolution of 2-amino-1-phenylethanol using dehydroabietic acid
Organic & Biomolecular Chemistry, 2008, 6, 458-463
7150849 CIFC17 H28 N6 O2 S3P 21 21 218.4053; 14.8272; 18.2296
90; 90; 90
2271.9Basheer, Ahmad; Rappoport, Zvi
Enols and thioenols of substituted cyanomonothiocarbonylmalonamides: structures, enolization vs. thioenolization, equilibria and conformations
Organic & Biomolecular Chemistry, 2008, 6, 1071-1082
7150858 CIFC55 H66 N6 O9 S2P 21 21 2113.819; 17.9176; 21.6376
90; 90; 90
5357.5Meshcheryakov, Denys; Arnaud-Neu, Françoise; Böhmer, Volker; Bolte, Michael; Hubscher-Bruder, Véronique; Jobin, Emilie; Thondorf, Iris; Werner, Sabine
Cyclic triureas—synthesis, crystal structures and properties
Organic & Biomolecular Chemistry, 2008, 6, 1004-1014
7150873 CIFC22 H25 N3 O4P 21 21 2111.3216; 13.2699; 13.7391
90; 90; 90
2064.11Sakamoto, Masami; Sato, Naoto; Mino, Takashi; Kasashima, Yoshio; Fujita, Tsutomu
Crystallization-induced diastereomer transformation of 2-quinolone-4-carboxamide followed by stereoselective intermolecular photocycloaddition reaction
Organic & Biomolecular Chemistry, 2008, 6, 848-850
7150874 CIFC22 H25 N3 O4P 21 21 218.0817; 14.5195; 17.141
90; 90; 90
2011.4Sakamoto, Masami; Sato, Naoto; Mino, Takashi; Kasashima, Yoshio; Fujita, Tsutomu
Crystallization-induced diastereomer transformation of 2-quinolone-4-carboxamide followed by stereoselective intermolecular photocycloaddition reaction
Organic & Biomolecular Chemistry, 2008, 6, 848-850
7150879 CIFC28 H23 N O3 SP 21 21 216.6262; 16.496; 21.207
90; 90; 90
2318Duguet, Nicolas; Campbell, Craig D.; Slawin, Alexandra M. Z.; Smith, Andrew D.
N-Heterocyclic carbene catalysed β-lactam synthesis
Organic & Biomolecular Chemistry, 2008, 6, 1108-1113
7150886 CIFC26 H40 N4 O6P 21 21 219.3903; 16.0688; 19.4462
90; 90; 90
2934.3Fischer, Lucile; Didierjean, Claude; Jolibois, Franck; Semetey, Vincent; Manuel Lozano, Jose; Briand, Jean-Paul; Marraud, Michel; Poteau, Romuald; Guichard, Gilles
Propensity for local folding induced by the urea fragment in short-chain oligomers
Organic & Biomolecular Chemistry, 2008, 6, 2596-2610
7150887 CIFC17 H27 N3 O3P 21 21 215.241; 17.883; 19.356
90; 90; 90
1814.1Fischer, Lucile; Didierjean, Claude; Jolibois, Franck; Semetey, Vincent; Manuel Lozano, Jose; Briand, Jean-Paul; Marraud, Michel; Poteau, Romuald; Guichard, Gilles
Propensity for local folding induced by the urea fragment in short-chain oligomers
Organic & Biomolecular Chemistry, 2008, 6, 2596-2610
7150895 CIFC51 H84 O3P 21 21 216.429; 13.631; 50.896
90; 90; 90
4460.2Winne, Johan M.; De Clercq, Pierre J.; Milanesio, Marco; Pattison, Philip; Viterbo, Davide
Nonenzymic polycyclisation of analogues of oxidosqualene with a preformed C-ring
Organic & Biomolecular Chemistry, 2008, 6, 1918-1925
7150898 CIFC12 H13 N O5P 21 21 216.566; 7.3847; 24.1727
90; 90; 90
1172.08Alcaide, Benito; Almendros, Pedro; Luna, Amparo; Torres, M. Rosario
Stereoselective NaN3-catalyzed halonitroaldol-type reaction of azetidine-2,3-diones in aqueous media
Organic & Biomolecular Chemistry, 2008, 6, 1635-1640
7150903 CIFC18 H20 Cl N O SiP 21 21 215.99; 15.612; 19.9389
90; 90; 90
1864.6Karatas, Betül; Rendler, Sebastian; Fröhlich, Roland; Oestreich, Martin
Kinetic resolution of donor-functionalised tertiary alcohols by Cu–H-catalysed stereoselective silylation using a strained silicon-stereogenic silane
Organic & Biomolecular Chemistry, 2008, 6, 1435-1440
7150916 CIFC14 H14 N2 O3P 21 21 2111.014; 13.24; 17.939
90; 90; 90
2616Berini, Christophe; Minassian, Frédéric; Pelloux-Léon, Nadia; Denis, Jean-Noël; Vallée, Yannick; Philouze, Christian
Efficient stereoselective nucleophilic addition of pyrroles to chiral nitrones
Organic & Biomolecular Chemistry, 2008, 6, 2574-2586
7150917 CIFC14 H14 N2 O3P 21 21 215.96; 12.835; 16.626
90; 90; 90
1271.8Berini, Christophe; Minassian, Frédéric; Pelloux-Léon, Nadia; Denis, Jean-Noël; Vallée, Yannick; Philouze, Christian
Efficient stereoselective nucleophilic addition of pyrroles to chiral nitrones
Organic & Biomolecular Chemistry, 2008, 6, 2574-2586
7150924 CIFC15 H18 N2 O3P 21 21 217.4315; 8.443; 21.576
90; 90; 90
1353.8Zezula, Josef; Singer, Lisa; Przybył, Anna K.; Hashimoto, Akihiro; Dersch, Christina M.; Rothman, Richard B.; Deschamps, Jeffrey; Lee, Yong Sok; Jacobson, Arthur E.; Rice, Kenner C.
Synthesis and pharmacological effects of the enantiomers of the N-phenethyl analogues of the ortho and para e- and f-oxide-bridged phenylmorphans
Organic & Biomolecular Chemistry, 2008, 6, 2868-2883
7150925 CIFC36.5 H43 F N2 O12.5P 21 21 218.7028; 13.9149; 30.493
90; 90; 90
3692.7Zezula, Josef; Singer, Lisa; Przybył, Anna K.; Hashimoto, Akihiro; Dersch, Christina M.; Rothman, Richard B.; Deschamps, Jeffrey; Lee, Yong Sok; Jacobson, Arthur E.; Rice, Kenner C.
Synthesis and pharmacological effects of the enantiomers of the N-phenethyl analogues of the ortho and para e- and f-oxide-bridged phenylmorphans
Organic & Biomolecular Chemistry, 2008, 6, 2868-2883
7150926 CIFC25 H33 Br N2 O7 SP 21 21 217.719; 13.922; 24.899
90; 90; 90
2675.7Zezula, Josef; Singer, Lisa; Przybył, Anna K.; Hashimoto, Akihiro; Dersch, Christina M.; Rothman, Richard B.; Deschamps, Jeffrey; Lee, Yong Sok; Jacobson, Arthur E.; Rice, Kenner C.
Synthesis and pharmacological effects of the enantiomers of the N-phenethyl analogues of the ortho and para e- and f-oxide-bridged phenylmorphans
Organic & Biomolecular Chemistry, 2008, 6, 2868-2883
7150927 CIFC22 H26 Br N O2P 21 21 217.5366; 11.9922; 21.9804
90; 90; 90
1986.6Zezula, Josef; Singer, Lisa; Przybył, Anna K.; Hashimoto, Akihiro; Dersch, Christina M.; Rothman, Richard B.; Deschamps, Jeffrey; Lee, Yong Sok; Jacobson, Arthur E.; Rice, Kenner C.
Synthesis and pharmacological effects of the enantiomers of the N-phenethyl analogues of the ortho and para e- and f-oxide-bridged phenylmorphans
Organic & Biomolecular Chemistry, 2008, 6, 2868-2883
7150932 CIFC35 H31 N3 O2P 21 21 2112.2155; 14.8014; 15.6657
90; 90; 90
2832.46Klosterman, Jeremy K.; Linden, Anthony; Siegel, Jay S.
Synthesis of aryl-substituted 2-pyridyl-1,10-phenanthrolines; a series of oriented terpyridine analogues
Organic & Biomolecular Chemistry, 2008, 6, 2755-2764
7150958 CIFC13 H20 Cl3 N O2 SiP 21 21 218.03; 10.027; 22.837
90; 90; 90
1838.8Pattenden, Gerald; Rescourio, Gwenaëlla
A new synthetic approach to (+)-lactacystin based on radical cyclisation of enantiopure α-ethynyl substituted serine derivatives to 4-methylenepyrrolidinones
Organic & Biomolecular Chemistry, 2008, 6, 3428-3438
7150976 CIFC14 H19 BrP 21 21 217.76; 10.508; 15.461
90; 90; 90
1260.7Christie, Victoria B.; Barnard, Jonathan H.; Batsanov, Andrei S.; Bridgens, Caroline E.; Cartmell, Emily B.; Collings, Jonathan C.; Maltman, Daniel J.; Redfern, Christopher P. F.; Marder, Todd B.; Przyborski, Stefan; Whiting, Andrew
Synthesis and evaluation of synthetic retinoid derivatives as inducers of stem cell differentiation
Organic & Biomolecular Chemistry, 2008, 6, 3497-3507
7150977 CIFC19 H28 SiP 21 21 216.0434; 13.3512; 22.597
90; 90; 90
1823.3Christie, Victoria B.; Barnard, Jonathan H.; Batsanov, Andrei S.; Bridgens, Caroline E.; Cartmell, Emily B.; Collings, Jonathan C.; Maltman, Daniel J.; Redfern, Christopher P. F.; Marder, Todd B.; Przyborski, Stefan; Whiting, Andrew
Synthesis and evaluation of synthetic retinoid derivatives as inducers of stem cell differentiation
Organic & Biomolecular Chemistry, 2008, 6, 3497-3507
7151007 CIFC24 H24 N2 O4P 21 21 2110.4911; 12.2289; 16.1319
90; 90; 90
2069.64Farran, Daniel; Parrot, Isabelle; Toupet, Loïc; Martinez, Jean; Dewynter, Georges
Transannular rearrangement of activated 2,5-diketopiperazines: a key route to original scaffolds
Organic & Biomolecular Chemistry, 2008, 6, 3989-3996
7151010 CIFC55 H61 F6 N3 O P2 PdP 21 21 2114.3877; 16.3592; 21.4727
90; 90; 90
5054.1Maxwell, Aoife C.; Franc, Celine; Pouchain, Laurent; Müller-Bunz, Helge; Guiry, Patrick J.
Electronically varied quinazolinaps for asymmetric catalysis
Organic & Biomolecular Chemistry, 2008, 6, 3848-3853
7151012 CIFC13 H17 N O3 SP 21 21 219.8353; 17.4256; 31.038
90; 90; 90
5319.5Coote, Susannah C.; O'Brien, Peter; Whitwood, Adrian C.
Stereoselective aziridination of cyclic allylic alcohols using chloramine-T
Organic & Biomolecular Chemistry, 2008, 6, 4299-4314
7151014 CIFC36 H51 N O4P 21 21 219.2925; 12.9908; 28.111
90; 90; 90
3393.48Tayama, Eiji; Orihara, Kiwako; Kimura, Hiroshi
New synthetic routes to optically active α-quaternary α-aryl amino acid derivatives via the diastereoselective Stevens and Sommelet–Hauser rearrangements
Organic & Biomolecular Chemistry, 2008, 6, 3673-3680
7151018 CIFC22 H32 N O8 PP 21 21 218.0227; 8.8488; 31.8469
90; 90; 90
2260.85Liu, Xue-Wei; Le, Thanh Nguyen; Lu, Yunpeng; Xiao, Yongjun; Ma, Jimei; Li, Xingwei
An efficient synthesis of chiral phosphinyl oxide pyrrolidines and their application to asymmetric direct aldol reactions
Organic & Biomolecular Chemistry, 2008, 6, 3997-4003
7151024 CIFC30 H31 N3 O9P 21 21 216.48; 10.5889; 41.9162
90; 90; 90
2876.12Driller, Katrin Marie; Libnow, Stefanie; Hein, Martin; Harms, Manuela; Wende, Kristian; Lalk, Michael; Michalik, Dirk; Reinke, Helmut; Langer, Peter
Synthesis of 6H-indolo[2,3-b]quinoxaline-N-glycosides and their cytotoxic activity against human ceratinocytes (HaCaT)
Organic & Biomolecular Chemistry, 2008, 6, 4218-4223
7151025 CIFC26 H25 N3 O7P 21 21 216.3601; 11.2214; 35.0578
90; 90; 90
2502.05Driller, Katrin Marie; Libnow, Stefanie; Hein, Martin; Harms, Manuela; Wende, Kristian; Lalk, Michael; Michalik, Dirk; Reinke, Helmut; Langer, Peter
Synthesis of 6H-indolo[2,3-b]quinoxaline-N-glycosides and their cytotoxic activity against human ceratinocytes (HaCaT)
Organic & Biomolecular Chemistry, 2008, 6, 4218-4223
7151026 CIFC24 H29 N O6 SP 21 21 215.7683; 9.0468; 43.5087
90; 90; 90
2270.49Paixão, Márcio W.; Nielsen, Martin; Jacobsen, Christian Borch; Jørgensen, Karl Anker
Organocatalytic asymmetric ring-opening of aziridines
Organic & Biomolecular Chemistry, 2008, 6, 3467-3470
7151035 CIFC36 H47 N O8 SP 21 21 216.008; 17.848; 30.989
90; 90; 90
3323Chen, Qiao-Hong; Ganesh, Thota; Brodie, Peggy; Slebodnick, Carla; Jiang, Yi; Banerjee, Abhijit; Bane, Susan; Snyder, James P.; Kingston, David G. I.
Design, synthesis and biological evaluation of bridged epothilone D analogues
Organic & Biomolecular Chemistry, 2008, 6, 4542-4552
7151036 CIFC27 H46 O2P 21 21 2134.899; 9.3865; 7.5
90; 90; 90
2456.8Martin, René; Däbritz, Frank; Entchev, Eugeni V.; Kurzchalia, Teymuras V.; Knölker, Hans-Joachim
Stereoselective synthesis of the hormonally active (25S)-Δ7-dafachronic acid, (25S)-Δ4-dafachronic acid, (25S)-dafachronic acid, and (25S)-cholestenoic acid
Organic & Biomolecular Chemistry, 2008, 6, 4293-4295
7151037 CIFC6 H13 N O4P 21 21 215.9247; 7.2417; 17.4475
90; 90; 90
748.58Donohoe, Timothy J.; Cheeseman, Matthew D.; O'Riordan, Timothy J. C.; Kershaw, Jessica A.
Synthesis of (+)-DGDP and (−)-7-epialexine
Organic & Biomolecular Chemistry, 2008, 6, 3896-3898
7151039 CIFC34 H36P 21 21 219.7582; 14.4454; 17.915
90; 90; 90
2525.3Ter Wiel, Matthijs K. J.; Kwit, Marcin G.; Meetsma, Auke; Feringa, Ben L.
Synthesis, stereochemistry, and photochemical and thermal behaviour of bis-tert-butyl substituted overcrowded alkenes.
Organic & biomolecular chemistry, 2007, 5, 87-96
7151042 CIFC31 H33 N7 O6P 21 21 2111.581; 14.4762; 17.7027
90; 90; 90
2967.84Tan, T. H. Samuel; Worthington, Roberta J.; Pritchard, Robin G.; Morral, Jordi; Micklefield, Jason
Homopolymeric pyrrolidine-amide oligonucleotide mimics: Fmoc-synthesis and DNA/RNA binding properties.
Organic & biomolecular chemistry, 2007, 5, 239-248
7151044 CIFC24 H35 N7 O6P 21 21 217.7564; 13.3948; 25.589
90; 90; 90
2658.6Worthington, Roberta J.; O'Rourke, Adam P; Morral, Jordi; Tan, T. H. Samuel; Micklefield, Jason
Mixed-sequence pyrrolidine-amide oligonucleotide mimics: Boc(Z) synthesis and DNA/RNA binding properties.
Organic & biomolecular chemistry, 2007, 5, 249-259
7151045 CIFC10 H11 Cl OP 21 21 214.9735; 10.531; 17.521
90; 90; 90
917.7Haak, Robert M.; Tarabiono, Chiara; Janssen, Dick B.; Minnaard, Adriaan J.; de Vries, Johannes G.; Feringa, Ben L.
Synthesis of enantiopure chloroalcohols by enzymatic kinetic resolution.
Organic & biomolecular chemistry, 2007, 5, 318-323
7151064 CIFC20 H20 Cl N O2P 21 21 215.148; 15.808; 21.3073
90; 90; 90
1733.98Chen, Wei; Du, Wei; Yue, Lei; Li, Rui; Wu, Yong; Ding, Li-Sheng; Chen, Ying-Chun
Organocatalytic enantioselective indole alkylations of alpha,beta-unsaturated ketones.
Organic & biomolecular chemistry, 2007, 5, 816-821
7151097 CIFC26 H29 N O2P 21 21 218.4065; 9.6892; 26.482
90; 90; 90
2157McGhee, Andrea M.; Kizirian, Jean-Claude; Procter, David J.
Synthesis and evaluation of a new polymer-supported pseudoephedrine auxiliary for asymmetric alkylations on solid phase.
Organic & biomolecular chemistry, 2007, 5, 1021-1024
7151100 CIFC38 H43 N O4P 21 21 2111.264; 16.634; 17.048
90; 90; 90
3194.2Davies, Stephen G.; Roberts, Paul M.; Smith, Andrew D.
Asymmetric three- and [2 + 1]-component conjugate addition reactions for the stereoselective synthesis of polysubstituted piperidinones.
Organic & biomolecular chemistry, 2007, 5, 1405-1415
7151101 CIFC19 H22 N2 O4 SP 21 21 219.416; 13.56; 15.727
90; 90; 90
2008Zhu, Qing; Liu, Mei-Fang; Wang, Bo; Cheng, Ying
An unprecedented tandem 1,3-dipolar cycloaddition-cheletropic elimination: a facial approach to novel push-pull olefins.
Organic & biomolecular chemistry, 2007, 5, 1282-1286
7151103 CIFC27 H21 N3 O2P 21 21 2110.052; 15.052; 42.205
90; 90; 90
6386Bouet, Alexis; Deguest, Geoffrey; Heller, Barbara; Papamicaël, Cyril; Dupas, Georges; Oudeyer, Sylvain; Marsais, Francis; Levacher, Vincent
Preparation of new axially chiral bridged 2,2'-bipyridines and pyridyl monooxazolines (pymox). Evaluation in copper(I)-catalyzed enantioselective cyclopropanation.
Organic & biomolecular chemistry, 2007, 5, 1397-1404
7151106 CIFC26 H33 N6 O6 P SiP 21 21 2110.9131; 13.5228; 20.2901
90; 90; 90
2994.33Andrei, Mioara; Bjørnstad, Vidar; Langli, Geir; Rømming, Christian; Klaveness, Jo; Taskén, Kjetil; Undheim, Kjell
Stereoselective preparation of (RP)-8-hetaryladenosine-3',5'-cyclic phosphorothioic acids.
Organic & biomolecular chemistry, 2007, 5, 2070-2080
7151107 CIFC27 H35 N6 O6 P SiP 21 21 2110.8533; 13.3879; 20.9242
90; 90; 90
3040.3Andrei, Mioara; Bjørnstad, Vidar; Langli, Geir; Rømming, Christian; Klaveness, Jo; Taskén, Kjetil; Undheim, Kjell
Stereoselective preparation of (RP)-8-hetaryladenosine-3',5'-cyclic phosphorothioic acids.
Organic & biomolecular chemistry, 2007, 5, 2070-2080
7151113 CIFC24 H26 N6 O10P 21 21 217.5396; 7.9351; 43.1982
90; 90; 90
2584.44Xia, Yi; Li, Wei; Qu, Fanqi; Fan, Zhijin; Liu, Xiufeng; Berro, Charles; Rauzy, Evelyne; Peng, Ling
Synthesis of bitriazolyl nucleosides and unexpectedly different reactivity of azidotriazole nucleoside isomers in the Huisgen reaction.
Organic & biomolecular chemistry, 2007, 5, 1695-1701
7151123 CIFC31 H43 N3 O7P 21 21 219.415; 33.845; 9.568
90; 90; 90
3048.85Davies, Stephen G.; Garner, A. Christopher; Ouzman, Jaqueline V. A.; Roberts, Paul M.; Smith, Andrew D.; Snow, Emma J.; Thomson, James E.; Tamayo, Juan A.; Vickers, Richard J.
Diastereoselective synthesis of quaternary alpha-amino acids from diketopiperazine templates.
Organic & biomolecular chemistry, 2007, 5, 2138-2147
7151126 CIFC13 H18 O4P 21 21 217.2231; 9.3503; 17.2474
90; 90; 90
1164.86McGowan, Craig A.; Schmieder, Ann-Kathrin; Roberts, Lee; Greaney, Michael F.
Synthesis of the guanacastepene A-B hydrazulene ring system through photochemical ring transposition.
Organic & biomolecular chemistry, 2007, 5, 1522-1524
7151134 CIFC39 H46 O6P 21 21 216.052; 23.756; 23.944
90; 90; 90
3442.46Risseeuw, Martijn D. P.; Mazurek, Jaroslaw; van Langenvelde, Arjan; van der Marel, Gijsbert A.; Overkleeft, Herman S.; Overhand, Mark
Synthesis of alkylated sugar amino acids: conformationally restricted L-Xaa-L-Ser/Thr mimics.
Organic & biomolecular chemistry, 2007, 5, 2311-2314
7151145 CIFC32 H38 N2 O4P 21 21 218.6876; 14.8422; 22.3552
90; 90; 90
2882.55Beddow, James E.; Davies, Stephen G.; Ling, Kenneth B.; Roberts, Paul M.; Russell, Angela J.; Smith, Andrew D.; Thomson, James E.
Asymmetric synthesis of beta2-amino acids: 2-substituted-3-aminopropanoic acids from N-acryloyl SuperQuat derivatives.
Organic & biomolecular chemistry, 2007, 5, 2812-2825
7151146 CIFC29 H40 N2 O4P 21 21 2111.5661; 12.049; 20.5677
90; 90; 90
2866.31Beddow, James E.; Davies, Stephen G.; Ling, Kenneth B.; Roberts, Paul M.; Russell, Angela J.; Smith, Andrew D.; Thomson, James E.
Asymmetric synthesis of beta2-amino acids: 2-substituted-3-aminopropanoic acids from N-acryloyl SuperQuat derivatives.
Organic & biomolecular chemistry, 2007, 5, 2812-2825
7151163 CIFC15 H20 O4 S5P 21 21 219.3614; 10.3321; 20.0889
90; 90; 90
1943.1Brown, R. James; Brooks, Andrew C.; Griffiths, Jon-Paul; Vital, Betrand; Day, Peter; Wallis, John D.
Synthesis of bis(ethylenedithio)tetrathiafulvalene (BEDT-TTF) derivatives functionalised with two, four or eight hydroxyl groups.
Organic & biomolecular chemistry, 2007, 5, 3172-3182
7151165 CIFC12 H12 O4 SP 21 21 217.5636; 10.4554; 15.375
90; 90; 90
1215.9Evans, Lyndsay Ann; Adams, Harry; Barber, Christopher G.; Caggiano, Lorenzo; Jackson, Richard F. W.
Stereoselective synthesis of 2,3-difunctionalised thioesters using nucleophilic epoxidation of 1-arylthio-1-nitroalkenes.
Organic & biomolecular chemistry, 2007, 5, 3156-3163
7151170 CIFC42 H34 Cl2 N2 O6 P2 PtP 21 21 2111.1024; 13.8168; 26.9261
90; 90; 90
4130.5Eberhardt, Luc; Armspach, Dominique; Matt, Dominique; Oswald, Benoît; Toupet, Loic
Efficient asymmetric hydrogenation of olefins with hydrazine-derived diphosphoramidites.
Organic & biomolecular chemistry, 2007, 5, 3340-3346
7151174 CIFC21 H24 N2 OP 21 21 215.3478; 13.519; 23.99
90; 90; 90
1734.4Mikata, Yuji; Aida, Shiho; Inaba, Yoko; Yano, Shigenobu
Consideration of molecular arrangements in regio- and enantioselective reduction of an NAD model compound controlled by carbonyl oxygen orientation.
Organic & biomolecular chemistry, 2007, 5, 3834-3841
7151182 CIFC13 H16 N2 O5 SP 21 21 217.7577; 17.7377; 20.872
90; 90; 90
2872.1Curtis, Kim L.; Evinson, Emma L.; Handa, Sandeep; Singh, Kuldip
Asymmetric synthesis of 3-amino-4-hydroxy-2-(hydroxymethyl)pyrrolidines as potential glycosidase inhibitors.
Organic & biomolecular chemistry, 2007, 5, 3544-3553
7151184 CIFC12 H16 Br N O4 SP 21 21 217.5443; 10.6588; 17.4366
90; 90; 90
1402.1Curtis, Kim L.; Evinson, Emma L.; Handa, Sandeep; Singh, Kuldip
Asymmetric synthesis of 3-amino-4-hydroxy-2-(hydroxymethyl)pyrrolidines as potential glycosidase inhibitors.
Organic & biomolecular chemistry, 2007, 5, 3544-3553
7151186 CIFC13 H15 N2 O5 SP 21 21 215.6923; 15.7807; 33.089
90; 90; 90
2972.3Curtis, Kim L.; Evinson, Emma L.; Handa, Sandeep; Singh, Kuldip
Asymmetric synthesis of 3-amino-4-hydroxy-2-(hydroxymethyl)pyrrolidines as potential glycosidase inhibitors.
Organic & biomolecular chemistry, 2007, 5, 3544-3553
7151192 CIFC34 H35 Br N3 O3 ReP 21 21 217.893; 14.212; 28.551
90; 90; 90
3202.7Yeung, Chi-Tung; Teng, Pang-Fei; Yeung, Ho-Lun; Wong, Wing-Tak; Kwong, Hoi-Lun
Catalytic and asymmetric cyclopropanation of alkenes catalysed by rhenium(I) bipyridine and terpyridine tricarbonyl complexes.
Organic & biomolecular chemistry, 2007, 5, 3859-3864
7151200 CIFC16 H14 F2 O2 SP 21 21 217.8387; 11.645; 15.4763
90; 90; 90
1412.7Wyatt, Paul; Hudson, Andrew; Charmant, Jonathan; Orpen, A. Guy; Phetmung, Hirihattaya
Synthesis and chemistry of enantiomerically pure 10,11-dihydrodibenzo[b,f]thiepines.
Organic & biomolecular chemistry, 2006, 4, 2218-2232
7151204 CIFC12 H15 N O3P 21 21 215.644; 8.477; 25.121
90; 90; 90
1201.89Mitchell, Claire E. T.; Brenner, Stacey E.; García-Fortanet, Jorge; Ley, Steven V.
An efficient, asymmetric organocatalyst-mediated conjugate addition of nitroalkanes to unsaturated cyclic and acyclic ketones.
Organic & biomolecular chemistry, 2006, 4, 2039-2049
7151217 CIFC21 H30 O4 S2P 21 21 218.1371; 9.7341; 26.6319
90; 90; 90
2109.44Zinzalla, Giovanna; Milroy, Lech-Gustav; Ley, Steven V.
Chemical variation of natural product-like scaffolds: design and synthesis of spiroketal derivatives.
Organic & biomolecular chemistry, 2006, 4, 1977-2002
7151218 CIFC21 H30 O4 S2P 21 21 218.1836; 11.8557; 21.3327
90; 90; 90
2069.75Zinzalla, Giovanna; Milroy, Lech-Gustav; Ley, Steven V.
Chemical variation of natural product-like scaffolds: design and synthesis of spiroketal derivatives.
Organic & biomolecular chemistry, 2006, 4, 1977-2002
7151220 CIFC20 H25 N O6P 21 21 215.5259; 10.0212; 34.6
90; 90; 90
1916Markad, Shankar D.; Karanjule, Narayan S.; Sharma, Tarun; Sabharwal, Sushma G.; Puranik, Vedavati G.; Dhavale, Dilip D.
Synthesis of tetrahydroxy perhydroaza-azulenes: tandem Johnson-Claisen rearrangement of D-glucose-derived allylic alcohols.
Organic & biomolecular chemistry, 2006, 4, 2549-2555
7151224 CIFC23 H33 Cl2 N O5 SP 21 21 219.7734; 13.3223; 20.38
90; 90; 90
2653.6Besong, Gilbert; Jarowicki, Krzysztof; Kocienski, Philip J.; Sliwinski, Eric; Boyle, F. Thomas
Synthesis of (S)-(-)-N-acetylcolchinol using intramolecular biaryl oxidative coupling.
Organic & biomolecular chemistry, 2006, 4, 2193-2207
7151228 CIFC40 H40 N4 O4P 21 21 2110.0407; 15.0369; 22.816
90; 90; 90
3444.8Srimurugan, Sankareswaran; Viswanathan, Balasubramanian; Varadarajan, Thirukallam Kanthadai; Varghese, Babu
Synthesis and crystal structure of [2 + 2] calixsalens.
Organic & biomolecular chemistry, 2006, 4, 3044-3047
7151231 CIFC10 H11 N O2P 21 21 215.9454; 8.1078; 18.0676
90; 90; 90
870.93Davies, Stephen G.; Garner, A. Christopher; Roberts, Paul M.; Smith, Andrew D.; Sweet, Miles J.; Thomson, James E.
Oxazinanones as chiral auxiliaries: synthesis and evaluation in enolate alkylations and aldol reactions.
Organic & biomolecular chemistry, 2006, 4, 2753-2768
7151232 CIFC12 H15 N O2P 21 21 219.2401; 10.581; 46.9695
90; 90; 90
4592.18Davies, Stephen G.; Garner, A. Christopher; Roberts, Paul M.; Smith, Andrew D.; Sweet, Miles J.; Thomson, James E.
Oxazinanones as chiral auxiliaries: synthesis and evaluation in enolate alkylations and aldol reactions.
Organic & biomolecular chemistry, 2006, 4, 2753-2768
7151239 CIFC36 H40 Br Cl4 N3 O2P 21 21 219.7318; 18.078; 20.751
90; 90; 90
3650.8Dálaigh, Ciarán O; Hynes, Stephen J.; O'Brien, John E; McCabe, Thomas; Maher, Declan J.; Watson, Graeme W.; Connon, Stephen J.
Asymmetric acyl-transfer promoted by readily assembled chiral 4-N,N-dialkylaminopyridine derivatives.
Organic & biomolecular chemistry, 2006, 4, 2785-2793
7151244 CIFC13 H18 O2 SP 21 21 217.69; 9.26; 17.15
90; 90; 90
1221Okuma, Kentaro; Koda, Masahiro; Maekawa, Shinobu; Shioji, Kosei; Inoue, Tohru; Kurisaki, Tsutomu; Wakita, Hisanobu; Yokomori, Yoshinobu
Reaction of thioketones with propiolic acids.
Organic & biomolecular chemistry, 2006, 4, 2745-2752
7151246 CIFC17 H25 N O3P 21 21 217.2402; 11.8197; 18.467
90; 90; 90
1580.35Bull, Steven D.; Davies, Stephen G.; Garner, A. Christopher; Kruchinin, Dennis; Key, Min-Suk; Roberts, Paul M.; Savory, Edward D.; Smith, Andrew D.; Thomson, James E.
SuperQuat 5,5-dimethyl-4-iso-propyloxazolidin-2-one as a mimic of Evans 4-tert-butyloxazolidin-2-one.
Organic & biomolecular chemistry, 2006, 4, 2945-2964
7151261 CIFC18 H16 N4 O2P 21 21 218.7353; 9.81; 18.0556
90; 90; 90
1547.2Zhang, Xuejun; Hsung, Richard P.; You, Lingfeng
Tandem azidination- and hydroazidination-Huisgen [3 + 2] cycloadditions of ynamides. Synthesis of chiral amide-substituted triazoles.
Organic & biomolecular chemistry, 2006, 4, 2679-2682
7151264 CIFC29 H27 O3 PP 21 21 215.9419; 14.361; 26.6529
90; 90; 90
2274.34Fox, David J.; Parris, Sean; Pedersen, Daniel Sejer; Tyzack, Charles R.; Warren, Stuart
Asymmetric synthesis of cyclopropanes and dihydrofurans based on phosphine oxide chemistry.
Organic & biomolecular chemistry, 2006, 4, 3108-3112
7151267 CIFC27 H30 Cl O4 PP 21 21 215.8203; 11.4038; 37.8022
90; 90; 90
2509.1Fox, David J.; Pedersen, Daniel Sejer; Petersen, Asger B.; Warren, Stuart
Diphenylphosphinoyl chloride as a chlorinating agent–the selective double activation of 1,2-diols.
Organic & biomolecular chemistry, 2006, 4, 3117-3119
7151274 CIFC29 H32 F12 N4 O3P 21 21 2110.0545; 15.0943; 21.3967
90; 90; 90
3247.3Berkessel, Albrecht; Mukherjee, Santanu; Müller, Thomas N; Cleemann, Felix; Roland, Katrin; Brandenburg, Marc; Neudörfl, Jörg-M; Lex, Johann
Structural optimization of thiourea-based bifunctional organocatalysts for the highly enantioselective dynamic kinetic resolution of azlactones.
Organic & biomolecular chemistry, 2006, 4, 4319-4330
7151277 CIFC18 H29 N3 OP 21 21 2111.8168; 16.6626; 18.2008
90; 90; 90
3583.71Berkessel, Albrecht; Mukherjee, Santanu; Müller, Thomas N; Cleemann, Felix; Roland, Katrin; Brandenburg, Marc; Neudörfl, Jörg-M; Lex, Johann
Structural optimization of thiourea-based bifunctional organocatalysts for the highly enantioselective dynamic kinetic resolution of azlactones.
Organic & biomolecular chemistry, 2006, 4, 4319-4330
7151278 CIFC10 H21 N3 SP 21 21 2111.5762; 12.734; 16.3923
90; 90; 90
2416.41Berkessel, Albrecht; Mukherjee, Santanu; Müller, Thomas N; Cleemann, Felix; Roland, Katrin; Brandenburg, Marc; Neudörfl, Jörg-M; Lex, Johann
Structural optimization of thiourea-based bifunctional organocatalysts for the highly enantioselective dynamic kinetic resolution of azlactones.
Organic & biomolecular chemistry, 2006, 4, 4319-4330
7151280 CIFC17 H27 N3 OP 21 21 219.1661; 11.3191; 15.5757
90; 90; 90
1616.01Berkessel, Albrecht; Mukherjee, Santanu; Müller, Thomas N; Cleemann, Felix; Roland, Katrin; Brandenburg, Marc; Neudörfl, Jörg-M; Lex, Johann
Structural optimization of thiourea-based bifunctional organocatalysts for the highly enantioselective dynamic kinetic resolution of azlactones.
Organic & biomolecular chemistry, 2006, 4, 4319-4330
7151295 CIFC11 H22 I N OP 21 21 217.1485; 13.16; 14.239
90; 90; 90
1339.5Gawley, Robert E.; Eddings, Daniel B.; Santiago, Marcelina; Vicic, Davic A.
Diastereoselectivity of polar and radical couplings in electrophilic substitutions of rigid 2-lithio-N-methylpyrrolidines.
Organic & biomolecular chemistry, 2006, 4, 4285-4291
7151298 CIFC23 H20 Br N O2P 21 21 2112.865; 15.761; 19.557
90; 90; 90
3965Booker, James E. M.; Boto, Alicia; Churchill, Gwydion H.; Green, Clive P.; Ling, Matthew; Meek, Graham; Prabhakaran, Jaya; Sinclair, David; Blake, Alexander J.; Pattenden, Gerald
Approaches to the quaternary stereocentre and to the heterocyclic core in diazonamide A using the Heck reaction and related coupling reactions
Organic & Biomolecular Chemistry, 2006, 4, 4193
7151299 CIFC27 H35 N O5P 21 21 219.5722; 11.5881; 23.044
90; 90; 90
2556.1Booker, James E. M.; Boto, Alicia; Churchill, Gwydion H.; Green, Clive P.; Ling, Matthew; Meek, Graham; Prabhakaran, Jaya; Sinclair, David; Blake, Alexander J.; Pattenden, Gerald
Approaches to the quaternary stereocentre and to the heterocyclic core in diazonamide A using the Heck reaction and related coupling reactions
Organic & Biomolecular Chemistry, 2006, 4, 4193
7151305 CIFC14 H27 N3 O4P 21 21 216.297; 11.589; 22.503
90; 90; 90
1642.2Sengupta, Anindita; Aravinda, Subrayashastry; Shamala, Narayanaswamy; Raja, K. Muruga Poopathi; Balaram, Padmanabhan
Structural studies of model peptides containing ?-, ?- and ?-amino acids
Organic & Biomolecular Chemistry, 2006, 4, 4214
7151306 CIFC14 H26 N2 O5P 21 21 216.157; 11.547; 23.404
90; 90; 90
1663.9Sengupta, Anindita; Aravinda, Subrayashastry; Shamala, Narayanaswamy; Raja, K. Muruga Poopathi; Balaram, Padmanabhan
Structural studies of model peptides containing ?-, ?- and ?-amino acids
Organic & Biomolecular Chemistry, 2006, 4, 4214
7151322 CIFC63.53 H64.29 Cl N7.76 O6P 21 21 219.2512; 19.807; 34.048
90; 90; 90
6238.9Zhang, Weicheng; Wu, Shulin; Zhang, Zhaoguo; Yennawar, Hemant; Zhang, Xumu
Practical synthesis of chiral 9,9'-spirobixanthene-1,1'-diol.
Organic & biomolecular chemistry, 2006, 4, 4474-4477
7151345 CIFC13 H15 Cl O5 SP 21 21 216.853; 9.6726; 21.2802
90; 90; 90
1410.59Alonso, A. Mateo; Horcajada, Roberto; Motevalli, Majid; Utley, James H. P.; Wyatt, Peter B.
The reactivity, as electrogenerated bases, of chiral and achiral phenazine radical-anions, including application in asymmetric deprotonation.
Organic & biomolecular chemistry, 2005, 3, 2842-2847
7151357 CIFC19 H30 O3P 21 21 215.5947; 9.6504; 31.93
90; 90; 90
1723.9Sorensen, John L.; Auclair, Karine; Kennedy, Jonathan; Richard Hutchinson, C.; Vederas, John C.
Transformations of cyclic nonaketides by Aspergillus terreus mutants blocked for lovastatin biosynthesis at the lovA and lovC genes
Organic & Biomolecular Chemistry, 2003, 1, 50
7151358 CIFC19 H30 O4P 21 21 215.5318; 9.7123; 32.163
90; 90; 90
1728Sorensen, John L.; Auclair, Karine; Kennedy, Jonathan; Richard Hutchinson, C.; Vederas, John C.
Transformations of cyclic nonaketides by Aspergillus terreus mutants blocked for lovastatin biosynthesis at the lovA and lovC genes
Organic & Biomolecular Chemistry, 2003, 1, 50
7151363 CIFC29 H24 N2 O2 S2P 21 21 217.7426; 12.4048; 24.867
90; 90; 90
2388.36van Delden, Richard A.; Koumura, Nagatoshi; Schoevaars, Annemarie; Meetsma, Auke; Feringa, Ben L.
A donor–acceptor substituted molecular motor: unidirectional rotation driven by visible light
Organic & Biomolecular Chemistry, 2003, 1, 33-35
7151365 CIFC63.5 H119.8 N11 O14.9P 21 21 2112.3997; 20.171; 30.6428
90; 90; 90
7664.2Potter, Brian; Palmer, Rex A.; Withnall, Robert; Jenkins, Terence C.; Chowdhry, Babur Z.
Two new cyclosporin folds observed in the structures of the immunosuppressant cyclosporin G and the formyl peptide receptor antagonist cyclosporin H at ultra-high resolution
Organic & Biomolecular Chemistry, 2003, 1, 1466
7151366 CIFC64 H121.8 N11 O15.4P 21 21 2112.43; 20.256; 30.617
90; 90; 90
7708.8Potter, Brian; Palmer, Rex A.; Withnall, Robert; Jenkins, Terence C.; Chowdhry, Babur Z.
Two new cyclosporin folds observed in the structures of the immunosuppressant cyclosporin G and the formyl peptide receptor antagonist cyclosporin H at ultra-high resolution
Organic & Biomolecular Chemistry, 2003, 1, 1466
7151367 CIFC62 H123 N11 O18P 21 21 2117.2986; 19.69; 24.137
90; 90; 90
8221.3Potter, Brian; Palmer, Rex A.; Withnall, Robert; Jenkins, Terence C.; Chowdhry, Babur Z.
Two new cyclosporin folds observed in the structures of the immunosuppressant cyclosporin G and the formyl peptide receptor antagonist cyclosporin H at ultra-high resolution
Organic & Biomolecular Chemistry, 2003, 1, 1466
7151368 CIFC62 H123.8 N11 O18.4P 21 21 2117.358; 19.515; 23.225
90; 90; 90
7867.3Potter, Brian; Palmer, Rex A.; Withnall, Robert; Jenkins, Terence C.; Chowdhry, Babur Z.
Two new cyclosporin folds observed in the structures of the immunosuppressant cyclosporin G and the formyl peptide receptor antagonist cyclosporin H at ultra-high resolution
Organic & Biomolecular Chemistry, 2003, 1, 1466
7151372 CIFC54 H50 N4P 21 21 2111.4989; 14.7712; 25.141
90; 90; 90
4270.3Mathias Düggeli; Catherine Goujon-Ginglinger; Sarah Richard Ducotterd; David Mauron; Christophe Bonte; Alexander von Zelewsky; Helen Stoeckli-Evans; Antonia Neels
Synthetic routes for a new family of chiral tetradentate ligands containing pyridine rings
Org. Biomol. Chem., 2003, 1, 1894-1899
7151374 CIFC17 H17 Br N2P 21 21 216.1546; 13.5496; 17.5877
90; 90; 90
1466.7Mathias Düggeli; Catherine Goujon-Ginglinger; Sarah Richard Ducotterd; David Mauron; Christophe Bonte; Alexander von Zelewsky; Helen Stoeckli-Evans; Antonia Neels
Synthetic routes for a new family of chiral tetradentate ligands containing pyridine rings
Org. Biomol. Chem., 2003, 1, 1894-1899
7151376 CIFC17 H17 Br N2P 21 21 216.5403; 11.3397; 20.395
90; 90; 90
1512.6Mathias Düggeli; Catherine Goujon-Ginglinger; Sarah Richard Ducotterd; David Mauron; Christophe Bonte; Alexander von Zelewsky; Helen Stoeckli-Evans; Antonia Neels
Synthetic routes for a new family of chiral tetradentate ligands containing pyridine rings
Org. Biomol. Chem., 2003, 1, 1894-1899
7151398 CIFC49 H48 N4 O6 Si ZnP 21 21 2112.3217; 15.4829; 22.9369
90; 90; 90
4375.8Felber, Beatrice; Calle, Carlos; Seiler, Paul; Schweiger, Arthur; Diederich, François
Dendritic metalloporphyrins with a distal H-bond donor as mimics of haemoglobinElectronic supplementary information (ESI) available: procedures for the synthesis of 1 and 5 and iron(ii) insertion into the dendritic porphyrins including full spectral characterisation and complete EPR characterisation of the complex 22·Co(dmim) and the corresponding oxygenated complex. See http://www.rsc.org/suppdata/ob/b2/b212468h/
Organic & Biomolecular Chemistry, 2003, 1, 1090
7151412 CIFC15 H24 O4 SP 21 21 218.519; 9.782; 18.631
90; 90; 90
1552.6Andrés García-Granados; María C. Gutiérrez; Francisco Rivas
Improved microbiological hydroxylation of sesquiterpenoids: semisynthesis, structural determination and biotransformation studies of cyclic sulfite eudesmane derivatives
Org. Biomol. Chem., 2003, 1, 2314-2320
7151440 CIFC29 H26 Cl2 Cu N2 O2P 21 21 2110.066; 12.92; 19.424
90; 90; 90
2526.1Hester L. van Lingen; Wei Zhuang; Tore Hansen; Floris P. J. T. Rutjes; Karl Anker Jørgensen
Formation of optically active chromanes by catalytic asymmetric tandem oxa-Michael addition‒Friedel‒Crafts alkylation reactions
Org. Biomol. Chem., 2003, 1, 1953-1958
7151441 CIFC29 H26 Br2 Cu N2 O2P 21 21 2110.2389; 13.089; 19.466
90; 90; 90
2608.8Hester L. van Lingen; Wei Zhuang; Tore Hansen; Floris P. J. T. Rutjes; Karl Anker Jørgensen
Formation of optically active chromanes by catalytic asymmetric tandem oxa-Michael addition‒Friedel‒Crafts alkylation reactions
Org. Biomol. Chem., 2003, 1, 1953-1958
7151467 CIFC21 H27 N O7P 21 21 2111.559; 11.8196; 15.3885
90; 90; 90
2102.42Hussaini, Syed Raziullah; Moloney, Mark G.
2,5-Disubstituted pyrrolidines: versatile regioselective and diastereoselective synthesis by enamine reduction and subsequent alkylation
Organic & Biomolecular Chemistry, 2003, 1, 1838
7151468 CIFC22 H29 N O7P 21 21 215.8063; 16.1078; 22.717
90; 90; 90
2124.65Hussaini, Syed Raziullah; Moloney, Mark G.
2,5-Disubstituted pyrrolidines: versatile regioselective and diastereoselective synthesis by enamine reduction and subsequent alkylation
Organic & Biomolecular Chemistry, 2003, 1, 1838
7151469 CIFC10 H15 Br Cl N O4P 21 21 216.9448; 20.84; 30.325
90; 90; 90
4388.9Paul J. Dransfield; Paul M. Gore; Ivan Prokeš; Michael Shipman; Alexandra M. Z. Slawin
Preparation and reactivity of imino glycals: stereocontrolled, divergent approach to imino sugars
Org. Biomol. Chem., 2003, 1, 2723-2733
7151470 CIFC26 H26 N2 O4 SP 21 21 2114.089; 6.305; 25.875
90; 90; 90
2298.5Anwar, Muhammed; Bailey, Jonathan H.; Dickinson, Laura C.; Edwards, Hermia J.; Goswami, Rajesh; Moloney, Mark G.
Pyrrolidinones derived from (S)-pyroglutamic acid: penmacric acid and analoguesPart V. For parts I?IV see refs. 20?22, 24
Organic & Biomolecular Chemistry, 2003, 1, 2364
7151474 CIFC15 H25 N3 O5P 21 21 2110.2189; 15.3206; 27.7208
90; 90; 90
4340Hitchcock, Peter B.; Papadopoulos, Konstantinos; Young, Douglas W.
?-Lactams as versatile synthons for homochiral ibotenate analogues with potential for activity at glutamate receptors1
Organic & Biomolecular Chemistry, 2003, 1, 2670
7151477 CIFC16 H26 O2P 21 21 216.8589; 10.727; 20.398
90; 90; 90
1500.8Anderson, James C.; Blake, Alexander J.; Graham, Jonathan P.; Wilson, Claire
Investigation of the asymmetric ionic Diels?Alder reaction for the synthesis of cis-decalins
Organic & Biomolecular Chemistry, 2003, 1, 2877
7151478 CIFC16 H26 O3P 21 21 215.9429; 12.548; 20.128
90; 90; 90
1501Anderson, James C.; Blake, Alexander J.; Graham, Jonathan P.; Wilson, Claire
Investigation of the asymmetric ionic Diels?Alder reaction for the synthesis of cis-decalins
Organic & Biomolecular Chemistry, 2003, 1, 2877
7151479 CIFC23 H34 O4P 21 21 216.1489; 14.787; 23.008
90; 90; 90
2092Anderson, James C.; Blake, Alexander J.; Graham, Jonathan P.; Wilson, Claire
Investigation of the asymmetric ionic Diels?Alder reaction for the synthesis of cis-decalins
Organic & Biomolecular Chemistry, 2003, 1, 2877
7151488 CIFC37 H30 F6 N O P Pd SbP 21 21 2117.6824; 17.9641; 11.6546
90; 90; 90
3702.07Hatano, Manabu; Mikami, Koichi
Highly enantioselective alkaloid synthesis via ene-type cyclizations catalyzed by cationic chiral palladium(ii) complexes of PN-ligands with an achiral oxazoline unitElectronic supplementary information (ESI) available: spectral data of substrates, cyclized products and PN-ligands and crystallographic data of Pd complexes. See http://www.rsc.org/suppdata/ob/b3/b305865b/
Organic & Biomolecular Chemistry, 2003, 1, 3871
7151492 CIFC28 H34 N2 O7 SiP 21 21 217.5858; 8.444; 43.4801
90; 90; 90
2785.1Fleming, Ian; Maiti, Pranab; Ramarao, Chandrashekar
Stereocontrol of 1,5-related stereocentres using an intermediate silyl group?the diastereoselectivity of nucleophilic attack on a double bond adjacent to a stereogenic centre carrying a silyl group
Organic & Biomolecular Chemistry, 2003, 1, 3989
7151493 CIFC27 H32 N2 O7 SiP 21 21 217.1067; 14.8638; 26.2267
90; 90; 90
2770.39Fleming, Ian; Maiti, Pranab; Ramarao, Chandrashekar
Stereocontrol of 1,5-related stereocentres using an intermediate silyl group?the diastereoselectivity of nucleophilic attack on a double bond adjacent to a stereogenic centre carrying a silyl group
Organic & Biomolecular Chemistry, 2003, 1, 3989
7151504 CIFC16 H18 O4P 21 21 215.8009; 13.1214; 18.5666
90; 90; 90
1413.21Godage, H. Yasmin; Chambers, David J.; Evans, Graham R.; Fairbanks, Antony J.
Stereoselective synthesis of C-glycosides from carboxylic acids: the tandem Tebbe?Claisen approachThis is one of a number of contributions from the current members of the Dyson Perrins Laboratory to mark the end of almost 90 years of organic chemistry research in that building, as all its current academic staff move across South Parks Road to a new purpose-built laboratory.
Organic & Biomolecular Chemistry, 2003, 1, 3772
7151505 CIFC16 H18 O4P 21 21 215.1126; 14.2991; 19.1347
90; 90; 90
1398.85Godage, H. Yasmin; Chambers, David J.; Evans, Graham R.; Fairbanks, Antony J.
Stereoselective synthesis of C-glycosides from carboxylic acids: the tandem Tebbe?Claisen approachThis is one of a number of contributions from the current members of the Dyson Perrins Laboratory to mark the end of almost 90 years of organic chemistry research in that building, as all its current academic staff move across South Parks Road to a new purpose-built laboratory.
Organic & Biomolecular Chemistry, 2003, 1, 3772
7151508 CIFC44 H70 N2 O12P 21 21 218.6168; 9.3641; 56.595
90; 90; 90
4566.6Critchley, P.; Clarkson, G. J.
Carbohydrate-protein interactions at interfaces: comparison of the binding of Ricinus communis lectin to two series of synthetic glycolipids using surface plasmon resonance studies.
Organic & biomolecular chemistry, 2003, 1, 4148-4159
7151517 CIFC31 H39 N3 O6 S3P 21 21 2122.981; 13.623; 10.142
90; 90; 90
3175.2Pulacchini, Sonia; Nasser, Rima; Sibbons, Kevin F.; Motevalli, Majid; Hawkes, Geoffrey E.; Kroemer, Romano T.; Bento, Edson S.; Watkinson, Michael
Structure, modelling and dynamic behaviour of aza- and azaoxamacrocyclic ligands derived from (R,R)-1,2-diaminocyclohexaneElectronic supplementary information (ESI) available: different views of compounds 6, 6a and 6b. See http://www.rsc.org/suppdata/ob/b3/b306963j/
Organic & Biomolecular Chemistry, 2003, 1, 4058
7151522 CIFC15 H19 N O5 SP 21 21 218.385; 11.271; 16.603
90; 90; 90
1569.1Heaney, Frances; Fenlon, Julie; O'Mahony, Colm; McArdle, Patrick; Cunningham, Desmond
Alpha-oximono-esters as precursors to heterocycles–generation of oxazinone N-oxides and cycloaddition to alkene dipolarophiles.
Organic & biomolecular chemistry, 2003, 1, 4302-4316
7151540 CIFC23 H33 N O3 SiP 21 21 2119.214; 16.341; 7.1838
90; 90; 90
2255.5Tromp, Reynier A.; Brussee, Johannes; van der Gen, Arne
Stereochemistry of intramolecular Diels?Alder furan (IMDAF) reactions of furyl-substituted chiral ethanolamides
Organic & Biomolecular Chemistry, 2003, 1, 3592
7151544 CIFC19 H24 N2 O9 SP 21 21 219.939; 12.907; 20.16
90; 90; 90
2586Marietta Tóth; Katalin E. Kövér; Attila Bényei; László Somsák
C-Glycosylmethylene carbenes: synthesis of anhydro-aldose tosylhydrazones as precursors; generation and a new synthetic route to exo-glycals
Org. Biomol. Chem., 2003, 1, 4039-4046
7151561 CIFC13 H20 N2 O3P 21 21 217.9103; 9.9556; 15.8702
90; 90; 90
1249.81Jean-Paul R. Hermet; David W. Porter; Michael J. Dearden; Justin R. Harrison; Tobias Koplin; Peter O'Brien; Jérôme Parmene; Vladimir Tyurin; Adrian C. Whitwood; John Gilday; Neil M. Smith
Synthesis of sparteine-like chiral diamines and evaluation in the enantioselective lithiation–substitution of N-(tert-butoxycarbonyl)pyrrolidine
Org. Biomol. Chem., 2003, 1, 3977-3988
7151565 CIFC19 H28 O2P 21 21 218.5195; 10.0386; 19.37
90; 90; 90
1656.6Dang, Hai-Shan; Roberts, Brian P.; Tocher, Derek A.
Thiol-catalysed radical-chain redox rearrangement reactions of benzylidene acetals derived from terpenoid diols
Organic & Biomolecular Chemistry, 2003, 1, 4073
7151566 CIFC34 H42 O4P 21 21 2110.6743; 16.4346; 16.6813
90; 90; 90
2926.4Dang, Hai-Shan; Roberts, Brian P.; Tocher, Derek A.
Thiol-catalysed radical-chain redox rearrangement reactions of benzylidene acetals derived from terpenoid diols
Organic & Biomolecular Chemistry, 2003, 1, 4073
7151567 CIFC19 H28 O2P 21 21 218.804; 10.274; 18.428
90; 90; 90
1666.9Dang, Hai-Shan; Roberts, Brian P.; Tocher, Derek A.
Thiol-catalysed radical-chain redox rearrangement reactions of benzylidene acetals derived from terpenoid diols
Organic & Biomolecular Chemistry, 2003, 1, 4073
7151568 CIFC17 H25 N O6 SP 21 21 219.9643; 11.133; 17.3159
90; 90; 90
1920.9Foresti, Elisabetta; Palmieri, Gianni; Petrini, Marino; Profeta, Roberto
Highly diastereoselective addition of nitromethane anion to chiral alpha-amidoalkylphenyl sulfones. Synthesis of optically active alpha-amino acid derivatives.
Organic & biomolecular chemistry, 2003, 1, 4275-4281
7151578 CIFC13 H31 Br2 N3P 21 21 217.511; 12.0412; 19.598
90; 90; 90
1772.47Argouarch, Gilles; Stones, Graham; Gibson, Colin L.; Kennedy, Alan R.; Sherrington, David C.
Bifurcated, modular syntheses of chiral annulet triazacyclononanes
Organic & Biomolecular Chemistry, 2003, 1, 4408
7151584 CIFC10 H10 Cl F5 OP 21 21 217.979; 9.742; 14.053
90; 90; 90
1092.4DiMartino, Gianluca; Hursthouse, Michael B.; Light, Mark E.; Percy, Jonathan M.; Spencer, Neil S.; Tolley, Malcolm
Syntheses of selectively fluorinated cyclodecenones: the first deployment of the neutral oxy-Cope rearrangement in organofluorine chemistry
Organic & Biomolecular Chemistry, 2003, 1, 4423
7151593 CIFC19 H23 Cl F NP 21 21 219.21; 12.66; 14.89
90; 90; 90
1736Briggs, Caroline R. S.; Allen, Mark J.; O'Hagan, David; Tozer, David J.; Slawin, Alexandra M. Z.; Goeta, Andrés E; Howard, Judith A. K.
The observation of a large gauche preference when 2-fluoroethylamine and 2-fluoroethanol become protonated.
Organic & biomolecular chemistry, 2004, 2, 732-740
7151598 CIFC15 H20 Cl N O2P 21 21 217.2507; 12.939; 15.788
90; 90; 90
1481.2Kodato, Shinichi; Linders, Joannes T. M.; Gu, Xiao-Hui; Yamada, Koichiro; Flippen-Anderson, Judith L; Deschamps, Jeffrey R.; Jacobson, Arthur E.; Rice, Kenner C.
Synthesis of rac-(1R,4aR,9aR)-2-methyl-1,3,4,9a-tetrahydro-2H-1,4a-propanobenzofuro[2,3-c]pyridin-6-ol. An unusual double rearrangement leading to the ortho- and para-f oxide-bridged phenylmorphan isomers.
Organic & biomolecular chemistry, 2004, 2, 330-336
7151600 CIFC25 H31 N O4P 21 21 2118.064; 13.961; 9.143
90; 90; 90
2305.8Urones, Julio G.; Garrido, Narciso M.; Díez, David; El Hammoumi, Mohamed M.; Dominguez, Sara H.; Antonio Casaseca, J.; Davies, Stephen G.; Smith, Andrew D.
Asymmetric synthesis of the stereoisomers of 2-amino-5-carboxymethyl-cyclopentane-1-carboxylate.
Organic & biomolecular chemistry, 2004, 2, 364-372
7151607 CIFC11 H19 N O5P 21 21 216.4668; 10.4584; 19.4553
90; 90; 90
1315.81Charrier, Jean-Damien; Hadfield, David S.; Hitchcock, Peter B.; Young, Douglas W.
Synthesis of (2S,3S)-3'-fluoroisoleucine.
Organic & biomolecular chemistry, 2004, 2, 797-802
7151616 CIFC8 H3 F2 N OP 21 21 213.7369; 6.2036; 28.8526
90; 90; 90
668.87Olsen, Jacob; Seiler, Paul; Wagner, Björn; Fischer, Holger; Tschopp, Thomas; Obst-Sander, Ulrike; Banner, David W.; Kansy, Manfred; Müller, Klaus; Diederich, François
A fluorine scan of the phenylamidinium needle of tricyclic thrombin inhibitors: effects of fluorine substitution on pKa and binding affinity and evidence for intermolecular C-F...CN interactions.
Organic & biomolecular chemistry, 2004, 2, 1339-1352
7151657 CIFC14 H18 F3 N O2 SP 21 21 2110.9351; 11.7459; 24.978
90; 90; 90
3208.2Mei, Haibo; Xiong, Yiwen; Han, Jianlin; Pan, Yi
A facile process for the asymmetric synthesis of β-trifluoromethylated β-amino ketones via addition of ketone enolates to sulfinylimine.
Organic & biomolecular chemistry, 2011, 9, 1402-1406
7151683 CIFC20 H17 N3 O8P 21 21 219.7745; 9.7915; 20.5118
90; 90; 90
1963.12Sen, Subhabrata; Potti, Venkata R.; Surakanti, Ramu; Murthy, Y. L. N.; Pallepogu, Raghavaiah
Enantioselective synthesis of spirooxoindoles via chiral auxiliary (bicyclic lactam) controlled SNAr reactions.
Organic & biomolecular chemistry, 2011, 9, 358-360
7151684 CIFC16 H12 N2 O3P 21 21 217.471; 8.305; 21.194
90; 90; 90
1315.02Sunderland, Peter T.; Dhami, Archana; Mahon, Mary F.; Jones, Louise A.; Tully, Sophie R.; Lloyd, Matthew D.; Thompson, Andrew S.; Javaid, Hashim; Martin, Niall M. B.; Threadgill, Michael D.
Synthesis of 4-alkyl-, 4-aryl- and 4-arylamino-5-aminoisoquinolin-1-ones and identification of a new PARP-2 selective inhibitor.
Organic & biomolecular chemistry, 2011, 9, 881-891
7151688 CIFC24 H25 F3 N2 O2 SP 21 21 219.6263; 14.1765; 16.473
90; 90; 90
2248Grellepois, Fabienne; Nonnenmacher, Jean; Lachaud, Fabien; Portella, Charles
Enantiomerically pure 2-aryl(alkyl)-2-trifluoromethylaziridines: synthesis and ring opening with selected O- and N-nucleophiles.
Organic & biomolecular chemistry, 2011, 9, 1160-1168
7151691 CIFC25 H33 N O9P 21 21 2110.7328; 12.0282; 19.7768
90; 90; 90
2553.1Kurhade, Suresh E.; Mengawade, Tanaji; Bhuniya, Debnath; Palle, Venkata P.; Reddy, D. Srinivasa
Synthesis of novel sugar-lactam conjugates using the Aubé reaction.
Organic & biomolecular chemistry, 2011, 9, 744-747
7151709 CIFC12 H12 Br N O4P 21 21 216.8992; 6.9979; 24.978
90; 90; 90
1205.9Hong, Bor-Cherng; Kotame, Prakash; Liao, Ju-Hsiou
Enantioselective organocatalytic domino Michael-acetalization-Henry reactions of 2-hydroxynitrostyrene and aldehyde for the synthesis of tetrahydro-6H-benzo[c]chromenones.
Organic & biomolecular chemistry, 2011, 9, 382-386
7151719 CIFC25 H21 Cl N2 O3P 21 21 2110.27; 11.202; 18.897
90; 90; 90
2174Liu, Tang-Lin; Xue, Zhi-Yong; Tao, Hai-Yan; Wang, Chun-Jiang
Catalytic asymmetric 1,3-dipolar cycloaddition of N-unprotected 2-oxoindolin-3-ylidene derivatives and azomethine ylides for the construction of spirooxindole-pyrrolidines.
Organic & biomolecular chemistry, 2011, 9, 1980-1986
7151725 CIFC20 H16 SiP 21 21 218.3831; 11.7677; 15.012
90; 90; 90
1480.9Tanikawa, Tomoharu; Saito, Masaichi; Guo, Jing Dong; Nagase, Shigeru
Synthesis, structures and optical properties of trisilasumanene and its related compounds.
Organic & biomolecular chemistry, 2011, 9, 1731-1735
7151727 CIFC30 H30 Br2 N2 O4P 21 21 219.5861; 14.757; 19.402
90; 90; 90
2744.6Franklin, Andrew I.; Bensa, David; Adams, Harry; Coldham, Iain
Transannular dipolar cycloaddition as an approach towards the synthesis of the core ring system of the sarain alkaloids.
Organic & biomolecular chemistry, 2011, 9, 1901-1907
7151742 CIFC14 H16 O4P 21 21 215.4822; 8.8469; 24.9538
90; 90; 90
1210.27Nesbitt, Caroline L.; McErlean, Christopher S. P.
Total synthesis of C19 lipid diols containing a 2,5-disubstituted-3-oxygenated tetrahydrofuran.
Organic & biomolecular chemistry, 2011, 9, 2198-2208
7151756 CIFC20 H25 N O4 SP 21 21 215.3188; 12.594; 29.209
90; 90; 90
1956.6Kissane, Marie; Murphy, Maureen; O'Brien, Elisabeth; Chopra, Jay; Murphy, Linda; Collins, Stuart G.; Lawrence, Simon E.; Maguire, Anita R.
Addition-substitution reactions of 2-thio-3-chloroacrylamides with carbon, nitrogen, oxygen, sulfur and selenium nucleophiles.
Organic & biomolecular chemistry, 2011, 9, 2452-2472
7151759 CIFC12 H11 N O5P 21 21 215.6366; 12.6433; 16.9777
90; 90; 90
1209.92Ramachary, Dhevalapally B.; Prasad, M. Shiva; Madhavachary, R.
A general approach to high-yielding asymmetric synthesis of chiral 3-alkyl-4-nitromethylchromans via cascade Barbas-Michael and acetalization reactions.
Organic & biomolecular chemistry, 2011, 9, 2715-2721
7151774 CIFC16 H22 O5P 21 21 216.7923; 11.6086; 20.037
90; 90; 90
1579.9Schanderl, Martin; Jeong, Won Boo; Schwarz, Michael; Reiser, Oliver
Stereoselective rearrangement of guaianolides to tricyclic δ-valerolactones.
Organic & biomolecular chemistry, 2011, 9, 2543-2547
7151775 CIFC16 H22 O4P 21 21 216.9797; 11.9507; 17.3512
90; 90; 90
1447.3Schanderl, Martin; Jeong, Won Boo; Schwarz, Michael; Reiser, Oliver
Stereoselective rearrangement of guaianolides to tricyclic δ-valerolactones.
Organic & biomolecular chemistry, 2011, 9, 2543-2547
7151782 CIFC31 H32 N3 O4.5P 21 21 219.102; 18.341; 32.012
90; 90; 90
5344Amat, Mercedes; Arróniz, Carlos; Molins, Elies; Escolano, Carmen; Bosch, Joan
Highly stereoselective double (R)-phenylglycinol-induced cyclocondensation reactions of symmetric aryl bis(oxoacids).
Organic & biomolecular chemistry, 2011, 9, 2175-2184
7151785 CIFC30 H30 N2 O4P 21 21 219.737; 10.015; 26.408
90; 90; 90
2575Amat, Mercedes; Arróniz, Carlos; Molins, Elies; Escolano, Carmen; Bosch, Joan
Highly stereoselective double (R)-phenylglycinol-induced cyclocondensation reactions of symmetric aryl bis(oxoacids).
Organic & biomolecular chemistry, 2011, 9, 2175-2184
7151801 CIFC42 H62 N2 OP 21 21 2110.2181; 19.3153; 19.5555
90; 90; 90
3859.6Giffin, Nick A.; Makramalla, Miller; Hendsbee, Arthur D.; Robertson, Katherine N.; Sherren, Cody; Pye, Cory C.; Masuda, Jason D.; Clyburne, Jason A. C.
Anhydrous TEMPO-H: reactions of a good hydrogen atom donor with low-valent carbon centres.
Organic & biomolecular chemistry, 2011, 9, 3672-3680
7151809 CIFC20 H30 N2 O5P 21 21 215.1057; 10.2051; 40.956
90; 90; 90
2134Maity, Sibaprasad; Kumar, Pankaj; Haldar, Debasish
An amyloid-like fibril-forming supramolecular cross-β-structure of a model peptide: a crystallographic insight.
Organic & biomolecular chemistry, 2011, 9, 3787-3791
7151814 CIFC13 H25 I O2 SiP 21 21 2111.5224; 11.6757; 12.5624
90; 90; 90
1690Qi, Xian-Liang; Zhang, Jun-Tao; Feng, Jian-Peng; Cao, Xiao-Ping
Total synthesis and absolute configuration of malyngamide W.
Organic & biomolecular chemistry, 2011, 9, 3817-3824
7151822 CIFC28 H29 N O3P 21 21 216.0368; 13.398; 29.789
90; 90; 90
2409.4Wu, Yan-Chao; Li, Hui-Jing; Liu, Li; Liu, Zhe; Wang, Dong; Chen, Yong-Jun
Cascade reaction of β,γ-unsaturated α-ketoesters with phenols in trityl chloride/TFA system. Highly selective synthesis of 4-aryl-2H-chromenes and their applications.
Organic & biomolecular chemistry, 2011, 9, 2868-2877
7151834 CIFC20 H22 O6P 21 21 219.3443; 11.4954; 16.1665
90; 90; 90
1736.5Zhou, Bing; Li, Xiaomei; Tang, Huanyu; Miao, Zehong; Feng, Huijin; Li, Yuanchao
Total synthesis of novel D-ring-modified triptolide analogues: structure-cytotoxic activity relationship studies on the D-ring of triptolide.
Organic & biomolecular chemistry, 2011, 9, 3176-3179
7151838 CIFC23 H22 Br N O3P 21 21 2110.5465; 13.646; 14.694
90; 90; 90
2114.7Yang, Yuan-Liang; Pei, Cheng-Kui; Shi, Min
Multifunctional chiral phosphines-catalyzed highly diastereoselective and enantioselective substitution of Morita-Baylis-Hillman adducts with oxazolones.
Organic & biomolecular chemistry, 2011, 9, 3349-3358
7151840 CIFC33 H33 N5 O5P 21 21 219.261; 16.4271; 19.8316
90; 90; 90
3017.01Yang, Li; Yang, Fei; Lan, Jingbo; Gao, Ge; You, Jingsong; Su, Xiaoyu
Rational design of BINOL-based diimidazolyl ligands: homochiral channel-like mono-component organic frameworks by hydrogen-bond-directed self-assembly.
Organic & biomolecular chemistry, 2011, 9, 2618-2621
7151860 CIFC13 H16 O4P 21 21 215.9224; 11.4859; 17.6998
90; 90; 90
1204.01Macabeo, Allan Patrick G.; Kreuzer, Andreas; Reiser, Oliver
Stereoselective routes to aryl substituted γ-butyrolactones and their application towards the synthesis of highly oxidised furanocembranoids.
Organic & biomolecular chemistry, 2011, 9, 3146-3150
7151864 CIFC14 H13 Br Fe O7P 21 21 218.6252; 8.6773; 43.7286
90; 90; 90
3272.8Griffen, Julia A.; Le Coz, Amélie M; Kociok-Köhn, Gabriele; Khan, Monika Ali; Stewart, Alan J. W.; Lewis, Simon E.
Expanding the chiral pool: oxidation of meta-bromobenzoic acid by R. eutrophus B9 allows access to new reaction manifolds.
Organic & biomolecular chemistry, 2011, 9, 3920-3928
7151870 CIFC31 H33 Cl N2 O2 Ru SP 21 21 218.39707; 9.14896; 35.0858
90; 90; 90
2695.45Soni, Rina; Cheung, Fung Kei; Clarkson, Guy C.; Martins, Jose E. D.; Graham, Mark A.; Wills, Martin
The importance of the N-H bond in Ru/TsDPEN complexes for asymmetric transfer hydrogenation of ketones and imines.
Organic & biomolecular chemistry, 2011, 9, 3290-3294
7151875 CIFC22 H22 N2 OP 21 21 216.2211; 14.25; 19.7004
90; 90; 90
1746.45Nagaraj, Muthupandi; Boominathan, Muthusamy; Muthusubramanian, Shanmugam; Bhuvanesh, Nattamai
Synthesis of novel N-hydroxy heterocycles via intramolecular reductive cyclization of diketoximes by NaBH3CN
Organic & Biomolecular Chemistry, 2011, 9, 4642
7151891 CIFC40 H36 Br N O7P 21 21 2113.323; 15.987; 17.448
90; 90; 90
3716.3Xue, Zhi-Yong; Fang, Xin; Wang, Chun-Jiang
Asymmetric construction of 3-vinylidene-pyrrolidine derivatives containing allene moiety via Ag(I)/TF-BiphamPhos-catalyzed 1,3-dipolar cycloaddition of azomethine ylides with diethyl 2-(3,3-diphenylpropa-1,2-dienylidene) malonate.
Organic & biomolecular chemistry, 2011, 9, 3622-3624
7151893 CIFC25 H31 Br O3P 21 21 2110.3869; 13.1736; 15.8519
90; 90; 90
2169.1Stastna, Eva; Rath, Nigam P.; Covey, Douglas F.
The use of symmetry in enantioselective synthesis: Four pairs of chrysene enantiomers prepared from 19-nortestosterone
Organic & Biomolecular Chemistry, 2011, 9, 4685
7151901 CIFC19.5 H28 O8.5P 21 21 219.6172; 14.543; 27.025
90; 90; 90
3779.8Zhang, Mei; Zhang, Yangming; Lu, Wei; Nan, Fa-Jun
Synthesis and revision of stereochemistry of rubescensin S
Organic & Biomolecular Chemistry, 2011, 9, 4436
7151904 CIFC19 H36 Cl3 N3 O5P 21 21 2110.578; 11.206; 23.306
90; 90; 90
2762.6Jadhav, Sandip V.; Bandyopadhyay, Anupam; Benke, Sushil N.; Mali, Sachitanand M.; Gopi, Hosahudya N.
A facile synthesis and crystallographic analysis of N-protected β-amino alcohols and short peptaibols.
Organic & biomolecular chemistry, 2011, 9, 4182-4187
7151905 CIFC13 H26 N2 O4P 21 21 219.704; 13.077; 25.661
90; 90; 90
3256.4Jadhav, Sandip V.; Bandyopadhyay, Anupam; Benke, Sushil N.; Mali, Sachitanand M.; Gopi, Hosahudya N.
A facile synthesis and crystallographic analysis of N-protected β-amino alcohols and short peptaibols.
Organic & biomolecular chemistry, 2011, 9, 4182-4187
7151911 CIFC20 H14 Cl N OP 21 21 217.272; 11.909; 17.041
90; 90; 90
1475.8Wang, Ren; Lu, Shen-Ci; Zhang, Yi-Ming; Shi, Zong-Jun; Zhang, Wei
One-pot synthesis of benzo[f]quinolin-3-ones and benzo[a]phenanthridein-5-ones by the photoanuulation of 6-chloropyridin-2-ones and 3-chloroisoquinolin-1-ones to phenylacetylene.
Organic & biomolecular chemistry, 2011, 9, 5802-5808
7151913 CIFC11 H12 B F4 N3P 21 21 216.7538; 10.5562; 17.047
90; 90; 90
1215.4Campbell, Craig D.; Collett, Christopher J.; Thomson, Jennifer E.; Slawin, Alexandra M. Z.; Smith, Andrew D.
Organic base effects in NHC promoted O- to C-carboxyl transfer; chemoselectivity profiles, mechanistic studies and domino catalysis.
Organic & biomolecular chemistry, 2011, 9, 4205-4218
7151927 CIFC22 H19 N5 O2P 21 21 214.8025; 11.5872; 33.05
90; 90; 90
1839.15Gemma, Sandra; Colombo, Laura; Forloni, Gianluigi; Savini, Luisa; Fracasso, Claudia; Caccia, Silvio; Salmona, Mario; Brindisi, Margherita; Joshi, Bhupendra P.; Tripaldi, Pierangela; Giorgi, Gianluca; Taglialatela-Scafati, Orazio; Novellino, Ettore; Fiorini, Isabella; Campiani, Giuseppe; Butini, Stefania
Pyrroloquinoxaline hydrazones as fluorescent probes for amyloid fibrils.
Organic & biomolecular chemistry, 2011, 9, 5137-5148
7151936 CIFC12 H16 O3P 21 21 2110.396; 10.88; 19.224
90; 90; 90
2174.4Iqbal, Mudassar; Black, Richard J. G.; Winn, Joby; Reeder, Andrew T.; Blake, Alexander J.; Clarke, Paul A.
Studies on transannulation reactions across a nine-membered ring: the synthesis of natural product-like structures.
Organic & biomolecular chemistry, 2011, 9, 5062-5078
7151949 CIFC21 H39 N5 O8P 21 21 219.0917; 9.8531; 29.228
90; 90; 90
2618.3Srinivas, Deekonda; Vijayadas, Kuruppanthara N.; Gonnade, Rajesh; Phalgune, Usha D.; Rajamohanan, Pattuparambil R.; Sanjayan, Gangadhar J.
Concurrent display of both α- and β-turns in a model peptide.
Organic & biomolecular chemistry, 2011, 9, 5762-5765
7151951 CIFC21 H39 N5 O8P 21 21 219.056; 9.842; 29.153
90; 90; 90
2598Srinivas, Deekonda; Vijayadas, Kuruppanthara N.; Gonnade, Rajesh; Phalgune, Usha D.; Rajamohanan, Pattuparambil R.; Sanjayan, Gangadhar J.
Concurrent display of both α- and β-turns in a model peptide.
Organic & biomolecular chemistry, 2011, 9, 5762-5765
7151953 CIFC23 H43 N O8 SiP 21 21 219.0593; 15.3579; 19.9706
90; 90; 90
2778.55Kobayashi, Kenichi; Okamoto, Iwao; Morita, Nobuyoshi; Kiyotani, Tamiko; Tamura, Osamu
Synthesis of the proposed structure of phaeosphaeride A.
Organic & biomolecular chemistry, 2011, 9, 5825-5832
7151960 CIFC26 H35 N5 O11 SP 21 21 218.5748; 14.9184; 23.0172
90; 90; 90
2944.4Shen, Fengjuan; Li, Xiaoliu; Zhang, Xiaoyuan; Yin, Qingmei; Qin, Zhanbin; Chen, Hua; Zhang, Jinchao; Ma, Zhaipu
Microwave-assisted synthesis of dinucleoside analogues containing a thiazolidin-4-one linkage via one-pot tandem Staudinger/aza-Wittig/cyclization.
Organic & biomolecular chemistry, 2011, 9, 5766-5772
7151965 CIFC24 H23 N3 O4P 21 21 219.903; 10.8311; 19.231
90; 90; 90
2062.7Coote, Susannah C.; Quenum, Seidjolo; Procter, David J.
Exploiting Sm(ii) and Sm(iii) in SmI(2)-initiated reaction cascades: application in a tag removal-cyclisation approach to spirooxindole scaffolds.
Organic & biomolecular chemistry, 2011, 9, 5104-5108
7151966 CIFC20 H28 N2 O6P 21 21 2111.3829; 12.3833; 13.4311
90; 90; 90
1893.2Chen, Jia; Chen, Jian-Jun; Yao, Xiaojun; Gao, Kun
Kopsihainanines A and B, two unusual alkaloids from Kopsia hainanensis.
Organic & biomolecular chemistry, 2011, 9, 5334-5336
7151967 CIFC37 H69 N5 O6 Si4P 21 21 219.84534; 13.7667; 35.643
90; 90; 90
4830.98Meng, Xiangtai; Moriuchi, Toshiyuki; Tohnai, Norimitsu; Miyata, Mikiji; Kawahata, Masatoshi; Yamaguchi, Kentaro; Hirao, Toshikazu
Synthesis and assembling properties of bioorganometallic cyclometalated Au(iii) alkynyls bearing guanosine moieties.
Organic & biomolecular chemistry, 2011, 9, 5633-5636
7151980 CIFC32 H33 N O2 SP 21 21 217.4163; 14.0432; 25.9274
90; 90; 90
2700.3Ni, Cheng-Yan; Kan, Sha-Sha; Liu, Quan-Zhong; Kang, Tai-Ran
Diastereoselective and enantioselective capture of chiral zinc enolate using nitroolefins: a rapid access to chiral γ-nitro carbonyl compounds.
Organic & biomolecular chemistry, 2011, 9, 6211-6214
7151984 CIFC33 H42 Cl2 O17P 21 21 2111.2799; 15.1788; 21.4815
90; 90; 90
3678Nepogodiev, Sergey A.; Fais, Margherita; Hughes, David L.; Field, Robert A.
Synthesis of apiose-containing oligosaccharide fragments of the plant cell wall: fragments of rhamnogalacturonan-II side chains A and B, and apiogalacturonan.
Organic & biomolecular chemistry, 2011, 9, 6670-6684
7151993 CIFC15 H27 N O4P 21 21 2110.153; 10.273; 16.191
90; 90; 90
1688.7Mali, Sachitanand M.; Bandyopadhyay, Anupam; Jadhav, Sandip V.; Kumar, Mothukuri Ganesh; Gopi, Hosahudya N.
Synthesis of α, β-unsaturated γ-amino esters with unprecedented high (E)-stereoselectivity and their conformational analysis in peptides.
Organic & biomolecular chemistry, 2011, 9, 6566-6574
7151995 CIFC14 H25 N O4P 21 21 219.978; 10.083; 16.904
90; 90; 90
1700.7Mali, Sachitanand M.; Bandyopadhyay, Anupam; Jadhav, Sandip V.; Kumar, Mothukuri Ganesh; Gopi, Hosahudya N.
Synthesis of α, β-unsaturated γ-amino esters with unprecedented high (E)-stereoselectivity and their conformational analysis in peptides.
Organic & biomolecular chemistry, 2011, 9, 6566-6574
7152016 CIFC26 H37 N O6P 21 21 2110.4445; 14.899; 16.596
90; 90; 90
2582.5Fichtler, Robert; Neudörfl, Jörg-M; Jacobi von Wangelin, Axel
Practical three-component synthesis of crowded arenes with donor-acceptor substitution.
Organic & biomolecular chemistry, 2011, 9, 7224-7236
7152033 CIFC19 H23 N3 O3P 21 21 219.7941; 10.3009; 17.223
90; 90; 90
1737.6Liu, Shouxin; Mu, Yun; Han, Jianrong; Zhen, Xiaoli; Yang, Yihua; Tian, Xia; Whiting, Andrew
Stereoselective synthesis and rearrangement-fragmentation of arylidene N-alkoxydiketopiperazines.
Organic & biomolecular chemistry, 2011, 9, 7476-7481
7152048 CIFC19 H16 O2P 21 21 215.935; 14.0588; 17.2947
90; 90; 90
1443.05Chen, Jung-Hsuan; Chang, Chihliang; Chang, Hui-Ju; Chen, Kwunmin
Synthesis of 2,3,5,6-tetrahydro-1-alkyl/aryl-1H-benzo[f]chromen-3-ol derivatives from β-tetralones and α,β-unsaturated aldehydes.
Organic & biomolecular chemistry, 2011, 9, 7510-7516
7152055 CIFC20 H32 N2 O5P 21 21 218.1131; 10.109; 25.357
90; 90; 90
2079.7Aitken, David J.; Drouin, Ludovic; Goretta, Sarah; Guillot, Régis; Ollivier, Jean; Spiga, Marco
Stereoselective preparation of β,γ-methano-GABA derivatives.
Organic & biomolecular chemistry, 2011, 9, 7517-7524
7152058 CIFC25 H31 Br N2 O8P 21 21 2110.5256; 12.1392; 20.3601
90; 90; 90
2601.46Ramachary, Dhevalapally B.; Reddy, Y. Vijayendar; Banerjee, Atoshi; Banerjee, Sharmistha
Design, synthesis and biological evaluation of optically pure functionalized spiro[5,5]undecane-1,5,9-triones as HIV-1 inhibitors.
Organic & biomolecular chemistry, 2011, 9, 7282-7286
7152060 CIFC28 H38 O8P 21 21 217.1487; 13.2022; 28.639
90; 90; 90
2702.9Wang, Jian-Rong; Liu, Hai-Li; Kurtán, Tibor; Mándi, Attila; Antus, Sándor; Li, Jia; Zhang, Hai-Yan; Guo, Yue-Wei
Protolimonoids and norlimonoids from the stem bark of Toona ciliata var. pubescens.
Organic & biomolecular chemistry, 2011, 9, 7685-7696
7152061 CIFC31 H50 O4P 21 21 2110.208; 15.3825; 17.7371
90; 90; 90
2785.2Wang, Jian-Rong; Liu, Hai-Li; Kurtán, Tibor; Mándi, Attila; Antus, Sándor; Li, Jia; Zhang, Hai-Yan; Guo, Yue-Wei
Protolimonoids and norlimonoids from the stem bark of Toona ciliata var. pubescens.
Organic & biomolecular chemistry, 2011, 9, 7685-7696
7152076 CIFC19 H17 N OP 21 21 217.6826; 12.2144; 15.2964
90; 90; 90
1435.39Martínez, R Fernando; Avalos, Martín; Babiano, Reyes; Cintas, Pedro; Jiménez, José L; Light, Mark E.; Palacios, Juan C.
Tautomerism in Schiff bases. The cases of 2-hydroxy-1-naphthaldehyde and 1-hydroxy-2-naphthaldehyde investigated in solution and the solid state.
Organic & biomolecular chemistry, 2011, 9, 8268-8275
7152086 CIFC25 H45 N O3P 21 21 214.9152; 9.6665; 50.7258
90; 90; 90
2410.12Rives, Arnaud; Baudoin-Dehoux, Cécile; Saffon, Nathalie; Andrieu-Abadie, Nathalie; Génisson, Yves
Asymmetric synthesis and cytotoxic activity of isomeric phytosphingosine derivatives.
Organic & biomolecular chemistry, 2011, 9, 8163-8170
7152089 CIFC42 H36 Cl4 N4 O10P 21 21 2110.019; 16.372; 49.573
90; 90; 90
8132Lemouchi, Cyprien; Simonov, Sergey; Zorina, Leokadiya; Gautier, Christelle; Hudhomme, Piétrick; Batail, Patrick
Amino acid derivatives of perylenediimide and their N-HO peptide bond dipoles-templated solid state assembly into stacks.
Organic & biomolecular chemistry, 2011, 9, 8096-8101
7152090 CIFC14 H21 N OP 21 21 216.3355; 7.439; 26.291
90; 90; 90
1239.1Gálvez, José A; Díaz de Villegas, María D; Badorrey, Ramón; López-Ram-de-Víu, Pilar
Switch in regioselectivity of epoxide ring-opening by changing the organometallic reagent.
Organic & biomolecular chemistry, 2011, 9, 8155-8162
7152094 CIFC24 H22 O6 S2P 21 21 215.919; 14.531; 25.735
90; 90; 90
2213.4Companyó, Xavier; Valero, Guillem; Ceban, Victor; Calvet, Teresa; Font-Bardía, Mercé; Moyano, Albert; Rios, Ramon
Enantioselective organocatalytic asymmetric allylic alkylation. Bis(phenylsulfonyl)methane addition to MBH carbonates.
Organic & biomolecular chemistry, 2011, 9, 7986-7989
7152095 CIFC16 H20 O9P 21 21 217.1296; 9.0495; 27.5442
90; 90; 90
1777.13Leaver, David J.; Dawson, Raymond M.; White, Jonathan M.; Polyzos, Anastasios; Hughes, Andrew B.
Synthesis of 1,2,3-triazole linked galactopyranosides and evaluation of cholera toxin inhibition.
Organic & biomolecular chemistry, 2011, 9, 8465-8474
7152099 CIFC13 H13 I OP 21 21 215.4376; 9.7637; 22.815
90; 90; 90
1211.3Duce, Sara; Jorge, María; Alonso, Inés; Ruano, José Luis García; Cid, M Belén
An organocatalytic approach to enantiomerically enriched α-arylcyclohexenones and cyclohexanones.
Organic & biomolecular chemistry, 2011, 9, 8253-8260
7152114 CIFC6 H8 O4P 21 21 216.2773; 9.4898; 10.1036
90; 90; 90
601.87Karban, Jindřich; Císařová, Ivana; Strašák, Tomáš; Šťastná, Lucie Červenková; Sýkora, Jan
Skeletal rearrangements resulting from reactions of 1,6:2,3- and 1,6:3,4-dianhydro-β-D-hexopyranoses with diethylaminosulphur trifluoride.
Organic & biomolecular chemistry, 2012, 10, 394-403
7152115 CIFC6 H8 O4P 21 21 216.7114; 10.2593; 17.4506
90; 90; 90
1201.55Karban, Jindřich; Císařová, Ivana; Strašák, Tomáš; Šťastná, Lucie Červenková; Sýkora, Jan
Skeletal rearrangements resulting from reactions of 1,6:2,3- and 1,6:3,4-dianhydro-β-D-hexopyranoses with diethylaminosulphur trifluoride.
Organic & biomolecular chemistry, 2012, 10, 394-403
7152117 CIFC6 H8 O4P 21 21 215.6736; 9.5781; 10.7239
90; 90; 90
582.76Karban, Jindřich; Císařová, Ivana; Strašák, Tomáš; Šťastná, Lucie Červenková; Sýkora, Jan
Skeletal rearrangements resulting from reactions of 1,6:2,3- and 1,6:3,4-dianhydro-β-D-hexopyranoses with diethylaminosulphur trifluoride.
Organic & biomolecular chemistry, 2012, 10, 394-403
7152118 CIFC6 H8 O4P 21 21 216.4573; 9.4912; 10.0281
90; 90; 90
614.6Karban, Jindřich; Císařová, Ivana; Strašák, Tomáš; Šťastná, Lucie Červenková; Sýkora, Jan
Skeletal rearrangements resulting from reactions of 1,6:2,3- and 1,6:3,4-dianhydro-β-D-hexopyranoses with diethylaminosulphur trifluoride.
Organic & biomolecular chemistry, 2012, 10, 394-403
7152119 CIFC6 H8 O4P 21 21 216.1219; 8.5353; 11.8539
90; 90; 90
619.39Karban, Jindřich; Císařová, Ivana; Strašák, Tomáš; Šťastná, Lucie Červenková; Sýkora, Jan
Skeletal rearrangements resulting from reactions of 1,6:2,3- and 1,6:3,4-dianhydro-β-D-hexopyranoses with diethylaminosulphur trifluoride.
Organic & biomolecular chemistry, 2012, 10, 394-403
7152124 CIFC6 H7 F O3P 21 21 216.3628; 9.2072; 10.1628
90; 90; 90
595.37Karban, Jindřich; Císařová, Ivana; Strašák, Tomáš; Šťastná, Lucie Červenková; Sýkora, Jan
Skeletal rearrangements resulting from reactions of 1,6:2,3- and 1,6:3,4-dianhydro-β-D-hexopyranoses with diethylaminosulphur trifluoride.
Organic & biomolecular chemistry, 2012, 10, 394-403
7152125 CIFC6 H7 F O3P 21 21 215.7591; 6.2197; 16.2984
90; 90; 90
583.81Karban, Jindřich; Císařová, Ivana; Strašák, Tomáš; Šťastná, Lucie Červenková; Sýkora, Jan
Skeletal rearrangements resulting from reactions of 1,6:2,3- and 1,6:3,4-dianhydro-β-D-hexopyranoses with diethylaminosulphur trifluoride.
Organic & biomolecular chemistry, 2012, 10, 394-403
7152127 CIFC6 H7 F O3P 21 21 216.271; 7.6812; 12.1999
90; 90; 90
587.65Karban, Jindřich; Císařová, Ivana; Strašák, Tomáš; Šťastná, Lucie Červenková; Sýkora, Jan
Skeletal rearrangements resulting from reactions of 1,6:2,3- and 1,6:3,4-dianhydro-β-D-hexopyranoses with diethylaminosulphur trifluoride.
Organic & biomolecular chemistry, 2012, 10, 394-403
7152128 CIFC6 H7 F O3P 21 21 216.3457; 7.8536; 12.1288
90; 90; 90
604.46Karban, Jindřich; Císařová, Ivana; Strašák, Tomáš; Šťastná, Lucie Červenková; Sýkora, Jan
Skeletal rearrangements resulting from reactions of 1,6:2,3- and 1,6:3,4-dianhydro-β-D-hexopyranoses with diethylaminosulphur trifluoride.
Organic & biomolecular chemistry, 2012, 10, 394-403
7152129 CIFC6 H7 F O3P 21 21 217.2178; 8.7675; 9.5
90; 90; 90
601.18Karban, Jindřich; Císařová, Ivana; Strašák, Tomáš; Šťastná, Lucie Červenková; Sýkora, Jan
Skeletal rearrangements resulting from reactions of 1,6:2,3- and 1,6:3,4-dianhydro-β-D-hexopyranoses with diethylaminosulphur trifluoride.
Organic & biomolecular chemistry, 2012, 10, 394-403
7152131 CIFC6 H7 F O3P 21 21 216.7058; 8.1556; 10.7504
90; 90; 90
587.94Karban, Jindřich; Císařová, Ivana; Strašák, Tomáš; Šťastná, Lucie Červenková; Sýkora, Jan
Skeletal rearrangements resulting from reactions of 1,6:2,3- and 1,6:3,4-dianhydro-β-D-hexopyranoses with diethylaminosulphur trifluoride.
Organic & biomolecular chemistry, 2012, 10, 394-403
7152145 CIFC18 H13 N3 O2P 21 21 216.1634; 11.2748; 19.9532
90; 90; 90
1386.6Iaroshenko, Viktor O.; Mkrtchyan, Satenik; Gevorgyan, Ashot; Miliutina, Mariia; Villinger, Alexander; Volochnyuk, Dmytro; Sosnovskikh, Vyacheslav Ya; Langer, Peter
2,3-unsubstituted chromones and their enaminone precursors as versatile reagents for the synthesis of fused pyridines.
Organic & biomolecular chemistry, 2012, 10, 890-894
7152150 CIFC18 H19 N3 O SP 21 21 216.3395; 7.8493; 31.3577
90; 90; 90
1560.38Iaroshenko, Viktor O.; Mkrtchyan, Satenik; Gevorgyan, Ashot; Miliutina, Mariia; Villinger, Alexander; Volochnyuk, Dmytro; Sosnovskikh, Vyacheslav Ya; Langer, Peter
2,3-unsubstituted chromones and their enaminone precursors as versatile reagents for the synthesis of fused pyridines.
Organic & biomolecular chemistry, 2012, 10, 890-894
7152152 CIFC15 H14 N2 O2P 21 21 2110.021; 12.749; 10.714
90; 90; 90
1368.8Companyó, Xavier; Valero, Guillem; Pineda, Oriol; Calvet, Teresa; Font-Bardía, Mercè; Moyano, Albert; Rios, Ramon
Enantioselective organocatalytic oxyamination of unprotected 3-substituted oxindoles.
Organic & biomolecular chemistry, 2012, 10, 431-439
7152183 CIFC32 H37 B O3 P2P 21 21 219.31; 12.038; 27.103
90; 90; 90
3037.5Boyd, Derek R.; Bell, Mark; Dunne, Katherine S.; Kelly, Brian; Stevenson, Paul J.; Malone, John F.; Allen, Christopher C. R.
Chemoenzymatic synthesis of a mixed phosphine-phosphine oxide catalyst and its application to asymmetric allylation of aldehydes and hydrogenation of alkenes.
Organic & biomolecular chemistry, 2012, 10, 1388-1395
7152188 CIFC10 H12 Br N O2P 21 21 215.812; 6.7788; 25.807
90; 90; 90
1016.75Clerici, Paolo; Wennemers, Helma
Mono thiomalonates as thioester enolate equivalents–enantioselective 1,4-addition reactions to nitroolefins under mild conditions.
Organic & biomolecular chemistry, 2012, 10, 110-113
7152190 CIFC16 H13 Br N2 OP 21 21 218.581; 9.4511; 18.265
90; 90; 90
1481.3Huang, Long; Wei, Yin; Shi, Min
Asymmetric substitutions of O-Boc-protected Morita-Baylis-Hillman adducts with pyrrole and indole derivatives.
Organic & biomolecular chemistry, 2012, 10, 1396-1405
7152194 CIFC20 H25 N3 O3P 21 21 219.681; 12.864; 14.899
90; 90; 90
1855.5Znabet, Anass; Blanken, Sara; Janssen, Elwin; de Kanter, Frans J. J.; Helliwell, Madeleine; Turner, Nicholas J.; Ruijter, Eelco; Orru, Romano V. A.
Stereoselective synthesis of N-aryl proline amides by biotransformation-Ugi-Smiles sequence.
Organic & biomolecular chemistry, 2012, 10, 941-944
7152201 CIFC22 H17 F3 N2 O5 SP 21 21 2110.02411; 10.34453; 20.23764
90; 90; 90
2098.54Levy, Jean-Noël; Latham, Christopher M.; Roisin, Loïc; Kandziora, Nadine; Di Fruscia, Paolo; White, Andrew J. P.; Woodward, Simon; Fuchter, Matthew J.
The design and synthesis of novel IBiox N-heterocyclic carbene ligands derived from substituted amino-indanols.
Organic & biomolecular chemistry, 2012, 10, 512-515
7152212 CIFC18 H26 N2 O2P 21 21 216.43; 11.207; 21.269
90; 90; 90
1532.7Ruff, Bettina M.; Zhong, Sabilla; Nieger, Martin; Bräse, Stefan
Thiolation of symmetrical and unsymmetrical diketopiperazines.
Organic & biomolecular chemistry, 2012, 10, 935-940
7152213 CIFC18 H24 N2 O2 S2P 21 21 216.4416; 10.8045; 24.627
90; 90; 90
1714Ruff, Bettina M.; Zhong, Sabilla; Nieger, Martin; Bräse, Stefan
Thiolation of symmetrical and unsymmetrical diketopiperazines.
Organic & biomolecular chemistry, 2012, 10, 935-940
7152246 CIFC45 H72 N4 O17P 21 21 2113.8494; 17.4243; 20.0324
90; 90; 90
4834.1Pyta, Krystian; Przybylski, Piotr; Wicher, Barbara; Gdaniec, Maria; Stefańska, Joanna
Intramolecular proton transfer impact on antibacterial properties of ansamycin antibiotic rifampicin and its new amino analogues.
Organic & biomolecular chemistry, 2012, 10, 2385-2388
7152252 CIFC58 H90 N8 O11P 21 21 2111.312; 19.868; 28.099
90; 90; 90
6315Chandrappa, Siddappa; Aravinda, Subrayashastry; Raghothama, Srinivasarao; Sonti, Rajesh; Rai, Rajkishor; Harini, Veldore V.; Shamala, Narayanaswamy; Balaram, Padmanabhan
Helix and hairpin nucleation in short peptides using centrally positioned conformationally constrained dipeptide segments.
Organic & biomolecular chemistry, 2012, 10, 2815-2823
7152277 CIFC14 H22 O3P 21 21 218.0156; 8.4956; 19.4087
90; 90; 90
1321.68Schäfer, Christian; Miesch, Michel; Miesch, Laurence
Intramolecular reductive ketone-alkynoate coupling reaction promoted by (η(2)-propene)titanium.
Organic & biomolecular chemistry, 2012, 10, 3253-3257
7152278 CIFC13 H18 O2P 21 21 218.3229; 11.3609; 11.8761
90; 90; 90
1122.95Schäfer, Christian; Miesch, Michel; Miesch, Laurence
Intramolecular reductive ketone-alkynoate coupling reaction promoted by (η(2)-propene)titanium.
Organic & biomolecular chemistry, 2012, 10, 3253-3257
7152279 CIFC15 H24 O3P 21 21 217.2735; 9.0784; 21.1524
90; 90; 90
1396.73Schäfer, Christian; Miesch, Michel; Miesch, Laurence
Intramolecular reductive ketone-alkynoate coupling reaction promoted by (η(2)-propene)titanium.
Organic & biomolecular chemistry, 2012, 10, 3253-3257
7152286 CIFC29 H26 Br2 N2 O9P 21 21 216.64749; 13.2825; 33.3205
90; 90; 90
2942.04Komatsu, Yoshiyuki; Watanabe, Riki; Ikishima, Hideaki; Nakano, Keiji; Ichikawa, Yoshiyasu; Kotsuki, Hiyoshizo
Aminohydroxyacetone synthons: versatile intermediates for the organocatalytic asymmetric aldol reaction.
Organic & biomolecular chemistry, 2012, 10, 2993-3001
7152289 CIFC105 H152 F18 N8 O43 Pd4 S6 Sm2P 21 21 2113.4805; 20.3239; 24.982
90; 90; 90
6844.5Zhang, Guoqi
A heterotrimetallic Pd-Sm-Pd complex for asymmetric Friedel-Crafts alkylations of pyrroles with nitroalkenes.
Organic & biomolecular chemistry, 2012, 10, 2534-2536
7152294 CIFC18 H19 F2 N O2P 21 21 218.402; 9.71; 19.088
90; 90; 90
1557.3Fornalczyk, Michal; Singh, Kuldip; Stuart, Alison M.
Enantioselective Reformatsky reaction of ethyl iododifluoroacetate with ketones.
Organic & biomolecular chemistry, 2012, 10, 3332-3342
7152295 CIFC19 H21 F2 N O2P 21 21 218.8405; 9.7476; 19.684
90; 90; 90
1696.2Fornalczyk, Michal; Singh, Kuldip; Stuart, Alison M.
Enantioselective Reformatsky reaction of ethyl iododifluoroacetate with ketones.
Organic & biomolecular chemistry, 2012, 10, 3332-3342
7152296 CIFC20 H21 F2 N O2P 21 21 218.5802; 9.972; 19.406
90; 90; 90
1660.4Fornalczyk, Michal; Singh, Kuldip; Stuart, Alison M.
Enantioselective Reformatsky reaction of ethyl iododifluoroacetate with ketones.
Organic & biomolecular chemistry, 2012, 10, 3332-3342
7152299 CIFC20 H18 O5P 21 21 217.298; 13.566; 17.045
90; 90; 90
1687.5Mijangos, Marco V.; González-Marrero, Joaquin; Miranda, Luis D.; Vincent-Ruz, Paulette; Lujan-Montelongo, Armando; Olivera-Díaz, Diana; Bautista, Elhiu; Ortega, Alfredo; de la Luz Campos-González, María; Gamez-Montaño, Rocio
Microwave-assisted C-3 selective oxidative radical alkylation of flavones.
Organic & biomolecular chemistry, 2012, 10, 2946-2949
7152302 CIFC10 H17 N O6P 21 21 218.4697; 10.1103; 13.868
90; 90; 90
1187.53Angelov, Plamen; Chau, Yui Kwan Sonia; Fryer, Paul J.; Moloney, Mark G.; Thompson, Amber L.; Trippier, Paul C.
Biomimetic synthesis, antibacterial activity and structure-activity properties of the pyroglutamate core of oxazolomycin.
Organic & biomolecular chemistry, 2012, 10, 3472-3485
7152321 CIFC17 H15 N O4P 21 21 214.2571; 14.425; 23.481
90; 90; 90
1441.9Sun, Zhong-Xin; Cheng, Ying
N-Heterocyclic carbene-catalyzed cascade annulation reaction of o-vinylarylaldehydes with nitrosoarenes: one-step assembly of functionalized 2,3-benzoxazin-4-ones
Organic & Biomolecular Chemistry, 2012, 10, 4088
7152326 CIFC32 H31 Fe N O2 P2P 21 21 2112.0764; 13.3216; 17.3013
90; 90; 90
2783.4Martins, Nelson; Mateus, Nuno; Vinci, Daniele; Saidi, Ourida; Brigas, Amadeu; Bacsa, John; Xiao, Jianliang
Another side of the oxazaphospholidine oxide chiral ortho-directing group
Organic & Biomolecular Chemistry, 2012, 10, 4036
7152327 CIFC20 H22 Fe N O2 PP 21 21 2110.1623; 12.0052; 14.5445
90; 90; 90
1774.4Martins, Nelson; Mateus, Nuno; Vinci, Daniele; Saidi, Ourida; Brigas, Amadeu; Bacsa, John; Xiao, Jianliang
Another side of the oxazaphospholidine oxide chiral ortho-directing group
Organic & Biomolecular Chemistry, 2012, 10, 4036
7152328 CIFC20 H22 Fe N O2 PP 21 21 215.817; 12.8442; 23.6728
90; 90; 90
1768.71Martins, Nelson; Mateus, Nuno; Vinci, Daniele; Saidi, Ourida; Brigas, Amadeu; Bacsa, John; Xiao, Jianliang
Another side of the oxazaphospholidine oxide chiral ortho-directing group
Organic & Biomolecular Chemistry, 2012, 10, 4036
7152334 CIFC16 H15 Br N2 O4 SP 21 21 217.5614; 11.1691; 20.0521
90; 90; 90
1693.48Chen, Jie; Zhou, Ling; Yeung, Ying-Yeung
A highly enantioselective approach towards 2-substituted 3-bromopyrrolidines
Organic & Biomolecular Chemistry, 2012, 10, 3808
7152335 CIFC14 H13 Br N2 O4 S2P 21 21 217.4711; 11.1765; 19.4619
90; 90; 90
1625.1Chen, Jie; Zhou, Ling; Yeung, Ying-Yeung
A highly enantioselective approach towards 2-substituted 3-bromopyrrolidines
Organic & Biomolecular Chemistry, 2012, 10, 3808
7152336 CIFC14 H15 N O6P 21 21 216.5782; 8.7302; 21.2398
90; 90; 90
1219.78Ahmad, Sajjad; Swift, Michael D.; Farrugia, Louis J.; Senn, Hans Martin; Sutherland, Andrew
Stereoselective synthesis of functionalised carbocyclic amides: construction of the syn-(4aS,10bS)-phenanthridone skeleton
Organic & Biomolecular Chemistry, 2012, 10, 3937
7152337 CIFC36 H20 N4 O6 SP 21 21 219.5048; 18.9754; 19.2401
90; 90; 90
3470.1Leermann, Timo; Broutin, Pierre-Emmanuel; Leroux, Frédéric R.; Colobert, Françoise
Construction of the biaryl-part of vancomycin aglycon via atropo-diastereoselective Suzuki‒Miyaura coupling
Organic & Biomolecular Chemistry, 2012, 10, 4095
7152343 CIFC21 H26 O3 SP 21 21 219.1092; 10.189; 20.517
90; 90; 90
1904.3Gao, YuZhe; Wang, Xue; Sun, LiDong; Xie, LongGuan; Xu, XiaoHua
Zinc or indium-mediated Barbier-type allylation of aldehydes with 3-bromomethyl-5H-furan-2-one in aqueous media: an efficient synthesis method for α-methylene-γ-butyrolactone
Organic & Biomolecular Chemistry, 2012, 10, 3991
7152349 CIFC16 H18 N O3P 21 21 217.3012; 9.1671; 21.9003
90; 90; 90
1465.81Tchabanenko, Kirill; Sloan, Colleen; Bunetel, Yves-Mael; Mullen, Philip
Diastereoselective 1,3-dipolar cycloaddition of pyrylium ylides with chiral enamides.
Organic & biomolecular chemistry, 2012, 10, 4215-4219
7152351 CIFC30 H37 N O2 S SiP 21 21 2111.241; 13.09; 19.226
90; 90; 90
2829Narhe, Bharat D.; Sriramurthy, Vardhineedi; Yadav, Veejendra K.
A smooth rearrangement of N-p-toluenesulfonyl 2-tert-butyldiphenylsilylmethyl-substituted azetidines into N-p-toluenesulfonyl 3-tert-butyldiphenylsilyl-substituted pyrrolidines.
Organic & biomolecular chemistry, 2012, 10, 4390-4399
7152352 CIFC34 H39 N O2 S SiP 21 21 2110.1607; 13.0737; 22.9043
90; 90; 90
3042.6Narhe, Bharat D.; Sriramurthy, Vardhineedi; Yadav, Veejendra K.
A smooth rearrangement of N-p-toluenesulfonyl 2-tert-butyldiphenylsilylmethyl-substituted azetidines into N-p-toluenesulfonyl 3-tert-butyldiphenylsilyl-substituted pyrrolidines.
Organic & biomolecular chemistry, 2012, 10, 4390-4399
7152353 CIFC34 H39 N O2 S SiP 21 21 2110.158; 13.071; 22.898
90; 90; 90
3040Narhe, Bharat D.; Sriramurthy, Vardhineedi; Yadav, Veejendra K.
A smooth rearrangement of N-p-toluenesulfonyl 2-tert-butyldiphenylsilylmethyl-substituted azetidines into N-p-toluenesulfonyl 3-tert-butyldiphenylsilyl-substituted pyrrolidines.
Organic & biomolecular chemistry, 2012, 10, 4390-4399
7152354 CIFC33 H36 F N O2 S SiP 21 21 219.969; 10.025; 29.109
90; 90; 90
2909Narhe, Bharat D.; Sriramurthy, Vardhineedi; Yadav, Veejendra K.
A smooth rearrangement of N-p-toluenesulfonyl 2-tert-butyldiphenylsilylmethyl-substituted azetidines into N-p-toluenesulfonyl 3-tert-butyldiphenylsilyl-substituted pyrrolidines.
Organic & biomolecular chemistry, 2012, 10, 4390-4399
7152359 CIFC14 H14 Br N O4P 21 21 216.9084; 14.098; 14.21
90; 90; 90
1384Li, Wenyi; Liu, Xiaodong; Mao, Zhifeng; Chen, Qiao; Wang, Rui
New approach to the preparation of bicyclo octane derivatives via the enantioselective cascade reaction catalyzed by chiral diamine-Ni(OAc)(2) complex.
Organic & biomolecular chemistry, 2012, 10, 4767-4773
7152379 CIFC17 H13 Br N2 O3P 21 21 219.315; 10.631; 15.819
90; 90; 90
1566.5Jia, Yang; Yang, Wen; Du, Da-Ming
Asymmetric Friedel-Crafts alkylation of indoles with 3-nitro-2H-chromenes catalyzed by diphenylamine-linked bis(oxazoline) and bis(thiazoline) Zn(II) complexes.
Organic & biomolecular chemistry, 2012, 10, 4739-4746
7152382 CIFC10 H15 N O6P 21 21 217.4247; 9.3395; 16.7423
90; 90; 90
1160.96Kamimura, Akio; Miyazaki, Koichiro; Suzuki, Shuzo; Ishikawa, Shingo; Uno, Hidemitsu
Total synthesis of ent-calystegine B4 via nitro-Michael/aldol reaction.
Organic & biomolecular chemistry, 2012, 10, 4362-4366
7152390 CIFC18 H22 O5 SP 21 21 215.5779; 10.4276; 31.686
90; 90; 90
1843Pei, Cheng-Kui; Jiang, Yu; Shi, Min
Synthesis of optically active dihydropyrans from asymmetric [4 + 2] cycloaddition of β,γ-unsaturated α-ketoesters with allenic esters.
Organic & biomolecular chemistry, 2012, 10, 4355-4361
7152400 CIFC23 H19 F N2P 21 21 215.3015; 12.8502; 25.7032
90; 90; 90
1751.04Borkin, Dmitry A.; Puscau, Mirela; Carlson, Alena; Solan, Agnes; Wheeler, Kraig A.; Török, Béla; Dembinski, Roman
Synthesis of diversely 1,3,5-trisubstituted pyrazoles via 5-exo-dig cyclization.
Organic & biomolecular chemistry, 2012, 10, 4505-4508
7152401 CIFC12 H17 N O3P 21 21 217.5034; 12.2919; 13.0178
90; 90; 90
1200.65Warren, Sarah A.; Stokes, Stephen; Frampton, Christopher S.; White, Andrew J. P.; Spivey, Alan C.
Synthesis of anti and syn hydroxy-iso-evoninic acids.
Organic & biomolecular chemistry, 2012, 10, 4685-4688
7152402 CIFC12 H17 N O3P 21 21 215.97836; 12.6707; 15.76352
90; 90; 90
1194.09Warren, Sarah A.; Stokes, Stephen; Frampton, Christopher S.; White, Andrew J. P.; Spivey, Alan C.
Synthesis of anti and syn hydroxy-iso-evoninic acids.
Organic & biomolecular chemistry, 2012, 10, 4685-4688
7152405 CIFC14 H24 O8P 21 21 2110.0094; 12.121; 12.9524
90; 90; 90
1571.4Jaiswal, Rakesh; Dickman, Michael H.; Kuhnert, Nikolai
First diastereoselective synthesis of methyl caffeoyl- and feruloyl-muco-quinates.
Organic & biomolecular chemistry, 2012, 10, 5266-5277
7152408 CIFC20 H30 O4P 21 21 216.6246; 16.0121; 16.5233
90; 90; 90
1752.69Zou, Juan; Pan, Lutai; Li, Qiji; Pu, Jianxin; Yao, Ping; Zhu, Min; Banas, Jeffrey A.; Zhang, Hongjie; Sun, Handong
Rubesanolides C-E: abietane diterpenoids isolated from Isodon rubescens and evaluation of their anti-biofilm activity.
Organic & biomolecular chemistry, 2012, 10, 5039-5044
7152412 CIFC20 H30 Cl2 N2 O2P 21 21 215.7182; 12.0175; 30.1828
90; 90; 90
2074.1Ortiz, Adrian; Young, Ian S.; Sawyer, James R.; Hsiao, Yi; Singh, Amarjit; Sugiyama, Masano; Corbett, R. Michael; Chau, Melissa; Shi, Zhongping; Conlon, David A.
Synthetic approaches to a chiral 4-amino-3-hydroxy piperidine with pharmaceutical relevance.
Organic & biomolecular chemistry, 2012, 10, 5253-5257
7152425 CIFC21 H18 O3P 21 21 215.771; 10.93; 28.102
90; 90; 90
1772.6Ramachary, Dhevalapally B.; Mondal, Rumpa; Madhavachary, R.
Direct catalytic asymmetric synthesis of highly functionalized (2-ethynylphenyl)alcohols via Barbas-List aldol reaction: scope and synthetic applications.
Organic & biomolecular chemistry, 2012, 10, 5094-5101
7152426 CIFC22 H15 Br N4 O3P 21 21 219.26806; 13.0043; 16.2697
90; 90; 90
1960.9Wei, Wen-Tao; Chen, Chun-Xia; Lu, Rui-Jiong; Wang, Jin-Jia; Zhang, Xue-Jing; Yan, Ming
Enantioselective synthesis of 3,3'-dihydropyrryl-spirooxindoles via an organocatalytic three-component reaction.
Organic & biomolecular chemistry, 2012, 10, 5245-5252
7152431 CIFC40 H62 Cl2 Fe2 N2 O4P 21 21 219.4738; 17.4767; 26.9117
90; 90; 90
4455.8Muthupandi, Pandi; Sekar, Govindasamy
Synthesis of an unusual dinuclear chiral iron complex and its application in asymmetric hydrophosphorylation of aldehydes.
Organic & biomolecular chemistry, 2012, 10, 5347-5352
7152437 CIFC12 H10 Br2 O4P 21 21 2113.574; 17.699; 21.533
90; 90; 90
5173Siva Swaroop, Pandrangi; Raut, Gajanan N.; Gonnade, Rajesh G.; Verma, Priyanka; Gokhale, Rajesh S.; Srinivasa Reddy, D.
Antituberculosis agent diaportheone B: synthesis, absolute configuration assignment, and anti-TB activity of its analogues.
Organic & biomolecular chemistry, 2012, 10, 5385-5394
7152439 CIFC40 H32 Cl2 N10 O8P 21 21 2110.5103; 13.662; 25.537
90; 90; 90
3666.9Zhou, Feng; Fu, Haoliang; Ong, Wei Qiang; Ye, Ruijuan; Yuan, Weixing; Lu, Yu-Jing; Huo, Yan-Ping; Zhang, Kun; Su, Haibin; Zeng, Huaqiang
Locking high energy 1D chain of dichloromethane molecules containing abnormally short ClCl contacts of 2.524 Å inside organic crystals.
Organic & biomolecular chemistry, 2012, 10, 5525-5528
7152440 CIFC40 H32 Cl2 N10 O8P 21 21 2110.5003; 13.6695; 25.51
90; 90; 90
3661.5Zhou, Feng; Fu, Haoliang; Ong, Wei Qiang; Ye, Ruijuan; Yuan, Weixing; Lu, Yu-Jing; Huo, Yan-Ping; Zhang, Kun; Su, Haibin; Zeng, Huaqiang
Locking high energy 1D chain of dichloromethane molecules containing abnormally short ClCl contacts of 2.524 Å inside organic crystals.
Organic & biomolecular chemistry, 2012, 10, 5525-5528
7152446 CIFC18 H13 Br F3 N OP 21 21 218.2256; 11.0205; 18.212
90; 90; 90
1650.9Ye, Ke-Yin; Dai, Li-Xin; You, Shu-Li
Enantioselective synthesis of 2,5-dihydrobenzo[b]azepine derivatives via iridium-catalyzed asymmetric allylic amination with 2-allylanilines and ring-closing-metathesis reaction.
Organic & biomolecular chemistry, 2012, 10, 5932-5939
7152447 CIFC14 H13 N O5P 21 21 216.0553; 13.8095; 15.5347
90; 90; 90
1299.02Ramachary, Dhevalapally B.; Madhavachary, R.; Prasad, M. Shiva
Observation of neighboring ortho-hydroxyl group participation in organocatalytic asymmetric sequential Michael-lactonization reactions: synthesis of highly substituted chiral spirodihydrocoumarins.
Organic & biomolecular chemistry, 2012, 10, 5825-5829
7152448 CIFC43 H62 N2 O6P 21 21 219.2659; 14.2973; 29.1661
90; 90; 90
3863.8Sasaki, Toshiyuki; Shizuki, Norie; Hiraishi, Eri; Hisaki, Ichiro; Tohnai, Norimitsu; Miyata, Mikiji
Construction of multi-component supramolecular architectures of bile acids and cinchona alkaloids through helical-pitch-synchronized crystallization.
Organic & biomolecular chemistry, 2012, 10, 5985-5992
7152449 CIFC43 H62 N2 O5P 21 21 219.3208; 14.1964; 29.1726
90; 90; 90
3860.2Sasaki, Toshiyuki; Shizuki, Norie; Hiraishi, Eri; Hisaki, Ichiro; Tohnai, Norimitsu; Miyata, Mikiji
Construction of multi-component supramolecular architectures of bile acids and cinchona alkaloids through helical-pitch-synchronized crystallization.
Organic & biomolecular chemistry, 2012, 10, 5985-5992
7152453 CIFC7 H9 F O3P 21 21 214.641; 10.535; 15.936
90; 90; 90
779.2Boyd, Derek R.; Sharma, Narain D.; Malone, John F.; McIntyre, Peter B. A.; Stevenson, Paul J.; Allen, Christopher C. R.; Kwit, Marcin; Gawronski, Jacek
Structure, stereochemistry and synthesis of enantiopure cyclohexenone cis-diol bacterial metabolites derived from phenols.
Organic & biomolecular chemistry, 2012, 10, 6217-6229
7152457 CIFC20 H21 N O4P 21 21 219.681; 28.33; 6.26
90; 90; 90
1716.9Hallett, David J.; Tanikkul, Nongluk; Thomas, Eric J.
Remote stereocontrol in reactions between 4- and 5-alkoxyalk-2-enylstannanes and 1-alkoxycarbonylimines and analogues: stereoselective approaches to novel α-amino acids.
Organic & biomolecular chemistry, 2012, 10, 6130-6158
7152461 CIFC28 H39 N O4P 21 21 219.326; 13.7383; 20.3169
90; 90; 90
2603.07Davies, Stephen G.; Foster, Emma M.; Frost, Aileen B.; Lee, James A.; Roberts, Paul M.; Thomson, James E.
On the origins of diastereoselectivity in the conjugate additions of the antipodes of lithium N-benzyl-(N-α-methylbenzyl)amide to enantiopure cis- and trans-dioxolane containing α,β-unsaturated esters.
Organic & biomolecular chemistry, 2012, 10, 6186-6200
7152463 CIFC24 H21 N3 O5 SP 21 21 216.95676; 12.7545; 24.6435
90; 90; 90
2186.62Tsukano, Chihiro; Yokouchi, Shinsuke; Girard, Anne-Lise; Kuribayashi, Toshifumi; Sakamoto, Shota; Enomoto, Taro; Takemoto, Yoshiji
Platinum catalyzed 7-endo cyclization of internal alkynyl amides and its application to synthesis of the caprazamycin core.
Organic & biomolecular chemistry, 2012, 10, 6074-6086
7152478 CIFC88 H81 Br2 Cu2 Fe2 N3 P4P 21 21 219.3018; 16.8469; 25.9616
90; 90; 90
4068.4Ou, Jun; Wong, Wing-Tak; Chiu, Pauline
Desymmetrizing reductive aldol cyclizations of enethioate derivatives of 1,3-diones catalyzed by a chiral copper hydride.
Organic & biomolecular chemistry, 2012, 10, 5971-5978
7152482 CIFC18 H15 N3 O2P 21 21 214.9211; 12.5759; 23.0138
90; 90; 90
1424.26Cao, Liming; Maciejewski, John P.; Elzner, Stephan; Amantini, David; Wipf, Peter
Synthesis of 1,2,4-triazines and the triazinoisoquinolinedione DEF ring system of noelaquinone.
Organic & biomolecular chemistry, 2012, 10, 5811-5814
7152484 CIFC11 H9 N3 O2P 21 21 214.9819; 6.5576; 28.039
90; 90; 90
916.01Cao, Liming; Maciejewski, John P.; Elzner, Stephan; Amantini, David; Wipf, Peter
Synthesis of 1,2,4-triazines and the triazinoisoquinolinedione DEF ring system of noelaquinone.
Organic & biomolecular chemistry, 2012, 10, 5811-5814
7152497 CIFC14 H20 O4P 21 21 218.8972; 12.2375; 12.7413
90; 90; 90
1387.27Gregg, Claire; Perkins, Michael V.
Total synthesis and structural elucidation of ent-micropyrone and (+)-ascosalipyrone.
Organic & biomolecular chemistry, 2012, 10, 6547-6553
7152498 CIFC14 H20 O4P 21 21 218.1642; 12.0184; 14.2772
90; 90; 90
1400.89Gregg, Claire; Perkins, Michael V.
Total synthesis and structural elucidation of ent-micropyrone and (+)-ascosalipyrone.
Organic & biomolecular chemistry, 2012, 10, 6547-6553
7152506 CIFC17 H21 B N2P 21 21 217.4473; 9.7852; 20.4386
90; 90; 90
1489.43Son, Jung-Ho; Hoefelmeyer, James D.
1,2-Nucleophilic addition of 2-(picolyl)organoboranes to nitrile, aldehyde, ketone, and amide.
Organic & biomolecular chemistry, 2012, 10, 6656-6664
7152509 CIFC23 H26 B N OP 21 21 218.6575; 14.9677; 14.9962
90; 90; 90
1943.3Son, Jung-Ho; Hoefelmeyer, James D.
1,2-Nucleophilic addition of 2-(picolyl)organoboranes to nitrile, aldehyde, ketone, and amide.
Organic & biomolecular chemistry, 2012, 10, 6656-6664
7152528 CIFC15 H18 Br N3 O2P 21 21 218.8707; 10.082; 18.499
90; 90; 90
1654.4Zhao, Fei; Wang, Yang; Zhang, Wen-Xiong; Xi, Zhenfeng
Metal-free synthesis of cyclic di-oxoguanidines via one-pot sequential transformation of amines, carbodiimides and acyl dichlorides.
Organic & biomolecular chemistry, 2012, 10, 6266-6270
7152547 CIFC22 H20 Br N OP 21 21 215.7061; 17.048; 18.4614
90; 90; 90
1795.9Liu, Xin-Yuan; Xiao, Ya-Ping; Siu, Fung-Ming; Ni, Li-Chen; Chen, Yong; Wang, Lin; Che, Chi-Ming
Highly regio-, diastereo- and enantioselective one-pot gold/chiral Brønsted acid-catalysed cascade synthesis of bioactive diversely substituted tetrahydroquinolines.
Organic & biomolecular chemistry, 2012, 10, 7208-7219
7152552 CIFC34 H52 O8 Si2P 21 21 2114.316; 15.96; 16.397
90; 90; 90
3746.4Díaz-Oltra, Santiago; Ruiz, Purificación; Falomir, Eva; Murga, Juan; Carda, Miguel; Marco, J. Alberto
Double diastereoselection in anti aldol reactions mediated by dicyclohexylchloroborane between an l-erythrulose derivative and chiral aldehydes.
Organic & biomolecular chemistry, 2012, 10, 6937-6944
7152553 CIFC41 H59 N O7 Si2P 21 21 2114.2378; 16.4937; 19.1231
90; 90; 90
4490.8Díaz-Oltra, Santiago; Ruiz, Purificación; Falomir, Eva; Murga, Juan; Carda, Miguel; Marco, J. Alberto
Double diastereoselection in anti aldol reactions mediated by dicyclohexylchloroborane between an l-erythrulose derivative and chiral aldehydes.
Organic & biomolecular chemistry, 2012, 10, 6937-6944
7152558 CIFC32 H32 N2 O3P 21 21 2110.0288; 15.96; 16.609
90; 90; 90
2658.4Barry, Sarah M.; Mueller-Bunz, Helge; Rutledge, Peter J.
Investigating the oxidation of alkenes by non-heme iron enzyme mimics.
Organic & biomolecular chemistry, 2012, 10, 7372-7381
7152592 CIFC11 H12 Br N O3 SP 21 21 215.276; 14.278; 17.698
90; 90; 90
1333.2Yang, Wen; Du, Da-Ming
Squaramide-catalysed enantio- and diastereoselective sulfa-Michael addition of thioacetic acid to α,β-disubstituted nitroalkenes.
Organic & biomolecular chemistry, 2012, 10, 6876-6884
7152594 CIFC28 H24 F6 O6 SP 21 21 2110.026; 12.876; 21.444
90; 90; 90
2768.3Boyd, Derek R.; Sharma, Narain D.; Brannigan, Ian N.; Evans, Timothy A.; Haughey, Simon A.; McMurray, Brian T.; Malone, John F.; McIntyre, Peter B. A.; Stevenson, Paul J.; Allen, Christopher C. R.
Toluene dioxygenase-catalyzed cis-dihydroxylation of benzo[b]thiophenes and benzo[b]furans: synthesis of benzo[b]thiophene 2,3-oxide.
Organic & biomolecular chemistry, 2012, 10, 7292-7304
7152596 CIFC28 H22 F6 O7P 21 21 216.783; 16.637; 23.581
90; 90; 90
2661.1Boyd, Derek R.; Sharma, Narain D.; Brannigan, Ian N.; Evans, Timothy A.; Haughey, Simon A.; McMurray, Brian T.; Malone, John F.; McIntyre, Peter B. A.; Stevenson, Paul J.; Allen, Christopher C. R.
Toluene dioxygenase-catalyzed cis-dihydroxylation of benzo[b]thiophenes and benzo[b]furans: synthesis of benzo[b]thiophene 2,3-oxide.
Organic & biomolecular chemistry, 2012, 10, 7292-7304
7152605 CIFC25 H24 O2 SP 21 21 215.9235; 8.7289; 41.0305
90; 90; 90
2121.51Kitanosono, Taku; Sakai, Masaru; Ueno, Masaharu; Kobayashi, Shū
Chiral-Sc catalyzed asymmetric Michael addition/protonation of thiols with enones in water.
Organic & biomolecular chemistry, 2012, 10, 7134-7147
7152606 CIFC17 H18 O SP 21 21 215.7153; 7.9637; 32.145
90; 90; 90
1463.1Kitanosono, Taku; Sakai, Masaru; Ueno, Masaharu; Kobayashi, Shū
Chiral-Sc catalyzed asymmetric Michael addition/protonation of thiols with enones in water.
Organic & biomolecular chemistry, 2012, 10, 7134-7147
7152612 CIFC19 H15 N O3P 21 21 215.551; 11.084; 24.666
90; 90; 90
1517.6Yang, Lihua; Xie, Peizhong; Li, Erqing; Li, Xin; Huang, You; Chen, Ruyu
Phosphine-catalyzed domino reaction: an efficient method for the synthesis of highly functionalized spirooxazolines.
Organic & biomolecular chemistry, 2012, 10, 7628-7634
7152637 CIFC30 H43 N O11 P2P 21 21 218.8403; 11.1099; 35.459
90; 90; 90
3482.6Zhao, Mei-Xin; Dai, Tong-Lei; Liu, Ran; Wei, Deng-Ke; Zhou, Hao; Ji, Fei-Hu; Shi, Min
Enantioselective Michael addition of 3-aryloxindoles to a vinyl bisphosphonate ester catalyzed by a cinchona alkaloid derived thiourea catalyst.
Organic & biomolecular chemistry, 2012, 10, 7970-7979
7152655 CIFC18 H20 Cl N O8P 21 21 219.7433; 11.3443; 18.273
90; 90; 90
2019.73Guo, Zhi-Wei; Xie, Jian-Wu; Chen, Ce; Zhu, Wei-Dong
Asymmetric catalytic [4 + 1] annulations catalyzed by quinidine: enantioselective synthesis of multi-functionalized isoxazoline N-oxides.
Organic & biomolecular chemistry, 2012, 10, 8471-8477
7152657 CIFC28 H42 Cl2 Pd2P 21 21 217.2879; 18.6931; 21.3386
90; 90; 90
2907.03Fernandes, Rodney A.; Nallasivam, Jothi L.
Enantioselective allylation of imines catalyzed by newly developed (-)-β-pinene-based π-allylpalladium catalyst: an efficient synthesis of (R)-α-propylpiperonylamine and (R)-pipecolic acid.
Organic & biomolecular chemistry, 2012, 10, 7789-7800
7152696 CIFC22 H22 Cl F4 NP 21 21 217.271; 13.0197; 22.3322
90; 90; 90
2114.11Chia, Poh Wai; Brennan, Sarah C.; Slawin, Alexandra M. Z.; Riccardi, Daniela; O'Hagan, David
Allosteric agonists of the calcium receptor (CaR): fluorine and SF5 analogues of cinacalcet.
Organic & biomolecular chemistry, 2012, 10, 7922-7927
7152699 CIFC20 H24 Br N O8P 21 21 2110.122; 10.799; 20.017
90; 90; 90
2188Wang, Yao; Luo, Yong-Chun; Zhang, Hong-Bo; Xu, Peng-Fei
Concise construction of the tetracyclic core of lycorine-type alkaloids and the formal synthesis of α-lycorane based on asymmetric bifunctional thiourea-catalyzed cascade reaction.
Organic & biomolecular chemistry, 2012, 10, 8211-8215
7152706 CIFC14 H10 N2 O3P 21 21 216.355; 8.01; 24.798
90; 90; 90
1262.31Bentabed-Ababsa, Ghenia; Hamza-Reguig, Samira; Derdour, Aïcha; Domingo, Luis R.; Sáez, José A; Roisnel, Thierry; Dorcet, Vincent; Nassar, Ekhlass; Mongin, Florence
Experimental and theoretical study of the [3 + 2] cycloaddition of carbonyl ylides with alkynes.
Organic & biomolecular chemistry, 2012, 10, 8434-8444
7152714 CIFC6 H14 Cl N OP 21 21 218.2735; 9.7455; 9.7543
90; 90; 90
786.48Wang, Qi-Qiang; Begum, Rowshan Ara; Day, Victor W.; Bowman-James, Kristin
Sulfur, oxygen, and nitrogen mustards: stability and reactivity.
Organic & biomolecular chemistry, 2012, 10, 8786-8793
7152745 CIFC20 H25 F3 N2 O5P 21 21 216.3446; 16.7461; 19.6159
90; 90; 90
2084.14Erdbrink, Holger; Peuser, Ilona; Gerling, Ulla I. M.; Lentz, Dieter; Koksch, Beate; Czekelius, Constantin
Conjugate hydrotrifluoromethylation of α,β-unsaturated acyl-oxazolidinones: synthesis of chiral fluorinated amino acids.
Organic & biomolecular chemistry, 2012, 10, 8583-8586
7152746 CIFC21 H27 F3 N2 O5P 21 21 216.3032; 17.505; 19.677
90; 90; 90
2171.1Erdbrink, Holger; Peuser, Ilona; Gerling, Ulla I. M.; Lentz, Dieter; Koksch, Beate; Czekelius, Constantin
Conjugate hydrotrifluoromethylation of α,β-unsaturated acyl-oxazolidinones: synthesis of chiral fluorinated amino acids.
Organic & biomolecular chemistry, 2012, 10, 8583-8586
7152747 CIFC15 H16 F3 N O3P 21 21 215.409; 11.831; 22.811
90; 90; 90
1459.8Erdbrink, Holger; Peuser, Ilona; Gerling, Ulla I. M.; Lentz, Dieter; Koksch, Beate; Czekelius, Constantin
Conjugate hydrotrifluoromethylation of α,β-unsaturated acyl-oxazolidinones: synthesis of chiral fluorinated amino acids.
Organic & biomolecular chemistry, 2012, 10, 8583-8586
7152767 CIFC26 H36 N6 O6P 21 21 214.9166; 13.1195; 42.105
90; 90; 90
2715.9Pehere, Ashok D.; Sumby, Christopher J.; Abell, Andrew D.
New cylindrical peptide assemblies defined by extended parallel β-sheets.
Organic & biomolecular chemistry, 2013, 11, 425-429
7152789 CIFC29 H45 O5 P SP 21 21 219.4027; 13.097; 24.592
90; 90; 90
3028.4Wu, Zong-Ze; Jang, Yeong-Jiunn; Lee, Chia-Jui; Lee, Yen-Te; Lin, Wenwei
A versatile and practical method for regioselective synthesis of polysubstituted furanonaphthoquinones.
Organic & biomolecular chemistry, 2013, 11, 828-834
7152804 CIFC15 H27 N O4P 21 21 2110.153; 10.273; 16.191
90; 90; 90
1688.7Ganesh Kumar, Mothukuri; Mali, Sachitanand M.; Gopi, Hosahudya N.
Synthesis and stereochemical analysis of β-nitromethane substituted γ-amino acids and peptides.
Organic & biomolecular chemistry, 2013, 11, 803-813
7152809 CIFC27 H22 Br Cl N2 O2P 21 21 218.258; 11.699; 23.879
90; 90; 90
2307Liang, Jinyan; Chen, Qiao; Liu, Luping; Jiang, Xianxing; Wang, Rui
An organocatalytic asymmetric double Michael cascade reaction of unsaturated ketones and unsaturated pyrazolones: highly efficient synthesis of spiropyrazolone derivatives.
Organic & biomolecular chemistry, 2013, 11, 1441-1445
7152814 CIFC32 H40 O8P 21 21 216.248; 14.246; 32.517
90; 90; 90
2894.3Song, Qiu-Yan; Jiang, Kan; Zhao, Qian-Qian; Gao, Kun; Jin, Xiao-Jie; Yao, Xiao-Jun
Eleven new highly oxygenated triterpenoids from the leaves and stems of Schisandra chinensis.
Organic & biomolecular chemistry, 2013, 11, 1251-1258
7152822 CIFC28 H21 Br N2 O3P 21 21 219.098; 15.524; 17.674
90; 90; 90
2496.2Qin, Tian-You; Liao, Wei-Wei; Zhang, Yan-Jing; Zhang, Sean Xiao-An
Asymmetric organocatalytic allylic alkylation of Reissert compounds: a facile access to chiral 1,1-disubstituted 1,2-dihydroisoquinolines.
Organic & biomolecular chemistry, 2013, 11, 984-990
7152823 CIFC16 H12 Br N O3P 21 21 219.801; 10.969; 14.07
90; 90; 90
1512.6De Fusco, Claudia; Meninno, Sara; Tedesco, Consiglia; Lattanzi, Alessandra
Enantioselective α-hydroxylation of β-ketoamides.
Organic & biomolecular chemistry, 2013, 11, 896-899
7152828 CIFC12 H11 N3 O SP 21 21 217.0809; 7.6178; 21.146
90; 90; 90
1140.6Xie, Zengyang; Zhu, Xiaojun; Guan, Yangfan; Zhu, Dunru; Hu, Hongwen; Lin, Chen; Pan, Yi; Jiang, Juli; Wang, Leyong
Cu-catalyzed direct C-H bond functionalization: a regioselective protocol to 5-aryl thiazolo[3,2-b]-1,2,4-triazoles.
Organic & biomolecular chemistry, 2013, 11, 1390-1398
7152832 CIFC16 H16 O3P 21 21 218.0469; 20.6366; 32.852
90; 90; 90
5455.4Bonancía, Paula; Vayá, Ignacio; Markovitsi, Dimitra; Gustavsson, Thomas; Jiménez, M Consuelo; Miranda, Miguel A.
Stereodifferentiation in the intramolecular singlet excited state quenching of hydroxybiphenyl-tryptophan dyads.
Organic & biomolecular chemistry, 2013, 11, 1958-1963
7152833 CIFC27 H26 N2 O4P 21 21 2110.6549; 12.0512; 17.2822
90; 90; 90
2219.11Bonancía, Paula; Vayá, Ignacio; Markovitsi, Dimitra; Gustavsson, Thomas; Jiménez, M Consuelo; Miranda, Miguel A.
Stereodifferentiation in the intramolecular singlet excited state quenching of hydroxybiphenyl-tryptophan dyads.
Organic & biomolecular chemistry, 2013, 11, 1958-1963
7152849 CIFC27 H43 N O4P 21 21 219.862; 10.08; 27.249
90; 90; 90
2708.8Shankar, Sreejith P.; Jagodzinska, Monika; Malpezzi, Luciana; Lazzari, Paolo; Manca, Ilaria; Greig, Iain R.; Sani, Monica; Zanda, Matteo
Synthesis and structure-activity relationship studies of novel tubulysin U analogues - effect on cytotoxicity of structural variations in the tubuvaline fragment.
Organic & biomolecular chemistry, 2013, 11, 2273-2287
7152851 CIFC29 H39 F6 N3 O8P 21 21 2114.698; 14.698; 15.598
90; 90; 90
3369.7Bellucci, Maria Cristina; Terraneo, Giancarlo; Volonterio, Alessandro
Multi-component synthesis of peptide-sugar conjugates.
Organic & biomolecular chemistry, 2013, 11, 2421-2444
7152860 CIFC14 H11 Br SP 21 21 216.0206; 10.2488; 20.3688
90; 90; 90
1256.83Yang, Zhaozhen; Chen, Xiaoyi; Kong, Wei; Xia, Siyuan; Zheng, Renwei; Luo, Fang; Zhu, Gangguo
An operationally simple approach to (E)-α-halo vinyl sulfides and their applications for accessing stereodefined trisubstituted alkenes.
Organic & biomolecular chemistry, 2013, 11, 2175-2185
7152870 CIFC16 H23 N O4 SP 21 21 219.829; 9.8991; 16.3718
90; 90; 90
1592.95Yeh, Ming-Chang P; Liang, Chia-Jung; Liu, Cheng-Yuan; Shih, Ya-Fon; Lee, I-Chen; Liu, Hsiang-Fang; Wang, Jeng-Long
Diastereoselective synthesis of vicinal cis-dihydroxyheterospirocycles by one-pot epoxidation/spirocyclization of C(3)-functionalized cyclohex-2-en-1-ols.
Organic & biomolecular chemistry, 2013, 11, 3393-3399
7152873 CIFC17 H24 N4 O2P 21 21 218.53; 12.4076; 15.1863
90; 90; 90
1607.27Rowley, Julian H.; Yau, Sze Chak; Kariuki, Benson M.; Kennedy, Alan R.; Tomkinson, Nicholas C. O.
Readily accessible chiral at nitrogen cage structures.
Organic & biomolecular chemistry, 2013, 11, 2198-2205
7152879 CIFC15 H28 N4 O2P 21 21 2114.0399; 8.1422; 14.4418
90; 90; 90
1650.92Rowley, Julian H.; Yau, Sze Chak; Kariuki, Benson M.; Kennedy, Alan R.; Tomkinson, Nicholas C. O.
Readily accessible chiral at nitrogen cage structures.
Organic & biomolecular chemistry, 2013, 11, 2198-2205
7152889 CIFC30 H36 O7 S2P 21 21 219.6394; 13.2527; 22.5332
90; 90; 90
2878.57Sreedharan, Dinesh T.; Clive, Derrick L. J.
Asymmetric synthesis of carbocycles: use of intramolecular conjugate displacement.
Organic & biomolecular chemistry, 2013, 11, 3128-3144
7152891 CIFC38 H46 F O7.5 S2P 21 21 2112.4942; 13.9308; 40.8485
90; 90; 90
7109.9Sreedharan, Dinesh T.; Clive, Derrick L. J.
Asymmetric synthesis of carbocycles: use of intramolecular conjugate displacement.
Organic & biomolecular chemistry, 2013, 11, 3128-3144
7152892 CIFC40 H48 F O9 S2P 21 21 218.2366; 12.8102; 37.2684
90; 90; 90
3932.28Sreedharan, Dinesh T.; Clive, Derrick L. J.
Asymmetric synthesis of carbocycles: use of intramolecular conjugate displacement.
Organic & biomolecular chemistry, 2013, 11, 3128-3144
7152893 CIFC37 H42 F O7.5 S2P 21 21 2112.3385; 13.7101; 41.224
90; 90; 90
6973.54Sreedharan, Dinesh T.; Clive, Derrick L. J.
Asymmetric synthesis of carbocycles: use of intramolecular conjugate displacement.
Organic & biomolecular chemistry, 2013, 11, 3128-3144
7152898 CIFC8 H15 N O3P 21 21 216.9174; 9.4363; 14.0634
90; 90; 90
917.98Brock, E. Anne; Davies, Stephen G.; Lee, James A.; Roberts, Paul M.; Thomson, James E.
Polyhydroxylated pyrrolizidine alkaloids from transannular iodoaminations: application to the asymmetric syntheses of (-)-hyacinthacine A1, (-)-7a-epi-hyacinthacine A1, (-)-hyacinthacine A2, and (-)-1-epi-alexine.
Organic & biomolecular chemistry, 2013, 11, 3187-3202
7152899 CIFC25 H37 N O6P 21 21 219.0523; 11.9795; 22.5183
90; 90; 90
2441.93Brock, E. Anne; Davies, Stephen G.; Lee, James A.; Roberts, Paul M.; Thomson, James E.
Polyhydroxylated pyrrolizidine alkaloids from transannular iodoaminations: application to the asymmetric syntheses of (-)-hyacinthacine A1, (-)-7a-epi-hyacinthacine A1, (-)-hyacinthacine A2, and (-)-1-epi-alexine.
Organic & biomolecular chemistry, 2013, 11, 3187-3202
7152916 CIFC15 H23 N2 O7 PP 21 21 219.992; 10.278; 17.851
90; 90; 90
1833.3Fan, Weidong; Kong, Shasha; Cai, Yan; Wu, Guiping; Miao, Zhiwei
Diastereo- and enantioselective nitro-Mannich reaction of α-substituted nitroacetates to N-phosphoryl imines catalyzed by cinchona alkaloid thiourea organocatalysts.
Organic & biomolecular chemistry, 2013, 11, 3223-3229
7152936 CIFC70.5 H130 O42P 21 21 2115.4853; 23.2543; 27.7178
90; 90; 90
9981.2Jouffroy, Matthieu; Armspach, Dominique; Matt, Dominique; Toupet, Loïc
Regioselective di- and tetra-functionalisation of γ-cyclodextrin using capping methodology.
Organic & biomolecular chemistry, 2013, 11, 3699-3705
7152954 CIFC25 H29 N3 O2P 21 21 217.9993; 12.1497; 21.7198
90; 90; 90
2110.93Sinha, Mantosh K.; Khoury, Kareem; Herdtweck, Eberhardt; Dömling, Alexander
Various cyclization scaffolds by a truly Ugi 4-CR.
Organic & biomolecular chemistry, 2013, 11, 4792-4796
7152969 CIFC16 H30 O3P 21 21 2133.5085; 6.1892; 8.0369
90; 90; 90
1666.78Liao, Cang-Song; Tang, Chun-Ping; Yao, Sheng; Ye, Yang
Humulane-type sesquiterpenoids from Pilea cavaleriei subsp. crenata.
Organic & biomolecular chemistry, 2013, 11, 4840-4846
7152979 CIFC54 H78 N8 O12P 21 21 2118.7511; 23.3396; 28.1926
90; 90; 90
12338.3Aravinda, Subrayashastry; Raghavender, Upadhyayula S.; Rai, Rajkishor; Harini, Veldore V.; Shamala, Narayanaswamy; Balaram, Padmanabhan
Analysis of designed β-hairpin peptides: molecular conformation and packing in crystals.
Organic & biomolecular chemistry, 2013, 11, 4220-4231
7152980 CIFC58 H88 N8 O12.5P 21 21 2118.88; 24.579; 28.78
90; 90; 90
13355Aravinda, Subrayashastry; Raghavender, Upadhyayula S.; Rai, Rajkishor; Harini, Veldore V.; Shamala, Narayanaswamy; Balaram, Padmanabhan
Analysis of designed β-hairpin peptides: molecular conformation and packing in crystals.
Organic & biomolecular chemistry, 2013, 11, 4220-4231
7152985 CIFC56 H83.5 N8 O13.5P 21 21 2119.086; 26.216; 28.015
90; 90; 90
14018Aravinda, Subrayashastry; Raghavender, Upadhyayula S.; Rai, Rajkishor; Harini, Veldore V.; Shamala, Narayanaswamy; Balaram, Padmanabhan
Analysis of designed β-hairpin peptides: molecular conformation and packing in crystals.
Organic & biomolecular chemistry, 2013, 11, 4220-4231
7152989 CIFC24 H40 N3 O4P 21 21 216.8433; 18.424; 20.221
90; 90; 90
2549.5Frantz, Marie-Céline; Skoda, Erin M.; Sacher, Joshua R.; Epperly, Michael W.; Goff, Julie P.; Greenberger, Joel S.; Wipf, Peter
Synthesis of analogs of the radiation mitigator JP4-039 and visualization of BODIPY derivatives in mitochondria.
Organic & biomolecular chemistry, 2013, 11, 4147-4153
7153001 CIFC25 H27 NP 21 21 218.1508; 17.5996; 28.8453
90; 90; 90
4137.9Jennings, W. Brian; O'Connell, Niamh; Malone, John F.; Boyd, Derek R.
An evaluation of substituent effects on aromatic edge-to-face interactions and CF-π versus CH-π interactions using an imino torsion balance model.
Organic & biomolecular chemistry, 2013, 11, 5278-5291
7153004 CIFC21 H25 N O3P 21 21 219.746; 17.508; 25.813
90; 90; 90
4404.5Jennings, W. Brian; O'Connell, Niamh; Malone, John F.; Boyd, Derek R.
An evaluation of substituent effects on aromatic edge-to-face interactions and CF-π versus CH-π interactions using an imino torsion balance model.
Organic & biomolecular chemistry, 2013, 11, 5278-5291
7153017 CIFC12 H20 O6P 21 21 215.6971; 11.5145; 19.4201
90; 90; 90
1273.94Vidyasagar, Adiyala; Pathigoolla, Atchutarao; Sureshan, Kana M.
Chemoselective alcoholysis/acetolysis of trans-ketals over cis-ketals and its application in the total synthesis of the cellular second messenger, d-myo-inositol-1,4,5-trisphosphate.
Organic & biomolecular chemistry, 2013, 11, 5443-5453
7153030 CIFC13 H16 O3P 21 21 215.1378; 6.7876; 32.299
90; 90; 90
1126.37Asta, Chimène; Schmidt, Dietmar; Conrad, Jürgen; Frey, Wolfgang; Beifuss, Uwe
Combination of enzyme- and Lewis acid-catalyzed reactions: a new method for the synthesis of 6,7-dihydrobenzofuran-4(5H)-ones starting from 2,5-dimethylfuran and 1,3-cyclohexanediones.
Organic & biomolecular chemistry, 2013, 11, 5692-5701
7153033 CIFC21 H25 N3 O2P 21 21 2111.2588; 11.763; 12.8358
90; 90; 90
1699.94Simpkins, Nigel S.; Pavlakos, Ilias; Weller, Michael D.; Male, Louise
The cascade radical cyclisation approach to prenylated alkaloids: synthesis of stephacidin A and notoamide B.
Organic & biomolecular chemistry, 2013, 11, 4957-4970
7153034 CIFC22 H29 N3 O3P 21 21 218.047; 10.678; 22.331
90; 90; 90
1918.8Simpkins, Nigel S.; Pavlakos, Ilias; Weller, Michael D.; Male, Louise
The cascade radical cyclisation approach to prenylated alkaloids: synthesis of stephacidin A and notoamide B.
Organic & biomolecular chemistry, 2013, 11, 4957-4970
7153035 CIFC41 H49 N3 O6 SP 21 21 2110.6567; 13.9156; 24.7451
90; 90; 90
3669.56Simpkins, Nigel S.; Pavlakos, Ilias; Weller, Michael D.; Male, Louise
The cascade radical cyclisation approach to prenylated alkaloids: synthesis of stephacidin A and notoamide B.
Organic & biomolecular chemistry, 2013, 11, 4957-4970
7153044 CIFC20 H22 O3 SP 21 21 2110.3509; 11.7545; 15.0554
90; 90; 90
1831.79Aitken, Harry R. M.; Furkert, Daniel P.; Hubert, Jonathan G.; Wood, James M.; Brimble, Margaret A.
Enantioselective access to benzannulated spiroketals using a chiral sulfoxide auxiliary.
Organic & biomolecular chemistry, 2013, 11, 5147-5155
7153057 CIFC27 H25 F2 N O7 S2P 21 21 218.2718; 13.6799; 23.831
90; 90; 90
2696.7Dou, Xiaowei; Lu, Yixin
Enantioselective conjugate addition of 3-fluoro-oxindoles to vinyl sulfone: an organocatalytic access to chiral 3-fluoro-3-substituted oxindoles.
Organic & biomolecular chemistry, 2013, 11, 5217-5221
7153058 CIFC24 H22 N2 O5P 21 21 218.4338; 15.4596; 15.6357
90; 90; 90
2038.63Hardman, Andrea M.; So, Sonia S.; Mattson, Anita E.
Urea-catalyzed construction of oxazinanes.
Organic & biomolecular chemistry, 2013, 11, 5793-5797
7153061 CIFC24 H21 Cl N2 O5P 21 21 218.5784; 15.2797; 16.5909
90; 90; 90
2174.66Hardman, Andrea M.; So, Sonia S.; Mattson, Anita E.
Urea-catalyzed construction of oxazinanes.
Organic & biomolecular chemistry, 2013, 11, 5793-5797
7153078 CIFC31 H36 N2 O4P 21 21 218.6627; 13.7443; 23.277
90; 90; 90
2771.4Liu, Gang; Li, Jian; Qiu, Lin; Liu, Li; Xu, Guangyang; Ma, Bing; Sun, Jiangtao
Palladium-catalyzed carbenoid based N-H bond insertions: application to the synthesis of chiral α-amino esters.
Organic & biomolecular chemistry, 2013, 11, 5998-6002
7153082 CIFC27 H34 N2 O4P 21 21 218.046; 14.28; 22.646
90; 90; 90
2602Jones, Raymond C. F.; Howard, Kevin J.; Snaith, John S.; Blake, Alexander J.; Li, Wang-Shei; Steel, Peter J.
Cycloaddition of homochiral dihydroimidazoles: a 1,3-dipolar cycloaddition route to optically active pyrrolo[1,2-a]imidazoles.
Organic & biomolecular chemistry, 2011, 9, 297-306
7153090 CIFC23 H30 O3P 21 21 217.2458; 7.571; 34.793
90; 90; 90
1908.7Wan, Wen; Ma, Guobin; Gao, Wei; Wang, Jing; Li, Lei; Rao, Shangqin; Zheng, Chunfang; Jiang, Haizhen; Deng, Hongmei; Hao, Jian
A facile total synthesis of drospirenone isomers containing 14β-hydrogen configuration.
Organic & biomolecular chemistry, 2013, 11, 6597-6603
7153091 CIFC23 H30 O3P 21 21 216.2123; 14.7435; 20.723
90; 90; 90
1898Wan, Wen; Ma, Guobin; Gao, Wei; Wang, Jing; Li, Lei; Rao, Shangqin; Zheng, Chunfang; Jiang, Haizhen; Deng, Hongmei; Hao, Jian
A facile total synthesis of drospirenone isomers containing 14β-hydrogen configuration.
Organic & biomolecular chemistry, 2013, 11, 6597-6603
7153107 CIFC13 H19 N3 O6P 21 21 217.36955; 8.40431; 24.1914
90; 90; 90
1498.32Glawar, Andreas F. G.; Jenkinson, Sarah F.; Newberry, Scott J.; Thompson, Amber L.; Nakagawa, Shinpei; Yoshihara, Akihide; Akimitsu, Kazuya; Izumori, Ken; Butters, Terry D.; Kato, Atsushi; Fleet, George W. J.
An approach to 8 stereoisomers of homonojirimycin from d-glucose via kinetic & thermodynamic azido-γ-lactones.
Organic & biomolecular chemistry, 2013, 11, 6886-6899
7153117 CIFC23 H22 Br N O5 SP 21 21 217.7952; 13.733; 21.171
90; 90; 90
2266.4Zou, Gong-Feng; Pan, Feng; Liao, Wei-Wei
Lewis base catalyzed asymmetric substitution/Diels-Alder cascade reaction: a rapid and efficient construction of enantioenriched diverse tricyclic heterocycles.
Organic & biomolecular chemistry, 2013, 11, 7080-7083
7153120 CIFC20 H26 N4 O6P 21 21 219.7965; 10.618; 21.199
90; 90; 90
2205.1Vangala, Madhuri; Dhokale, Snehal A.; Gawade, Rupesh L.; Pattuparambil, Rajamohanan R.; Puranik, Vedavati G.; Dhavale, Dilip D.
Sugar furanoid trans-vicinal diacid as a γ-turn inducer: synthesis and conformational study.
Organic & biomolecular chemistry, 2013, 11, 6874-6878
7153123 CIFC24 H21 N3P 21 21 216.7467; 12.811; 21.6174
90; 90; 90
1868.43Kinthada, Lakshmana K.; Ghosh, Santanu; De, Subhadip; Bhunia, Subhajit; Dey, Dhananjay; Bisai, Alakesh
Acid-catalyzed reactions of 3-hydroxy-2-oxindoles with electron-rich substrates: synthesis of 2-oxindoles with all-carbon quaternary center.
Organic & biomolecular chemistry, 2013, 11, 6984-6993
7153124 CIFC9 H0 N8 O4P 21 21 218.7505; 10.8915; 15.6217
90; 90; 90
1488.84Wang, Wenjing; Xue, Jijun; Tian, Tian; Jiao, Yingdong; Li, Ying
The first asymmetric total synthesis of (+)-coriandrone A and B.
Organic & biomolecular chemistry, 2013, 11, 6686-6690
7153131 CIFC18 H18 O6P 21 21 219.0858; 10.4482; 17.2738
90; 90; 90
1639.81Guo, Rui; Li, Kang-Nan; Gong, Liu-Zhu
Catalytic cascade hydroalkoxylation/isomerization/[4 + 2] cycloaddition using enyne alcohols as latent dienes or dienophiles.
Organic & biomolecular chemistry, 2013, 11, 6707-6712
7153132 CIFC18 H18 O6P 21 21 219.0802; 10.4402; 17.2659
90; 90; 90
1636.79Guo, Rui; Li, Kang-Nan; Gong, Liu-Zhu
Catalytic cascade hydroalkoxylation/isomerization/[4 + 2] cycloaddition using enyne alcohols as latent dienes or dienophiles.
Organic & biomolecular chemistry, 2013, 11, 6707-6712
7153161 CIFC18 H19 O6 PP 21 21 219.7943; 10.0856; 17.1604
90; 90; 90
1695.13Schiessl, Katharina; Roller, Alexander; Hammerschmidt, Friedrich
Determination of absolute configuration of the phosphonic acid moiety of fosfazinomycins.
Organic & biomolecular chemistry, 2013, 11, 7420-7426
7153181 CIFC19 H22 N2 O3P 21 21 217.735; 14.242; 16.353
90; 90; 90
1801.5Gould, Eoin; Lebl, Tomas; Slawin, Alexandra M. Z.; Reid, Mark; Davies, Tony; Smith, Andrew D.
The development of highly active acyclic chiral hydrazides for asymmetric iminium ion organocatalysis.
Organic & biomolecular chemistry, 2013, 11, 7877-7892
7153184 CIFC18 H18 Cl F3 N3 O S2P 21 21 217.392; 10.7494; 25.7003
90; 90; 90
2042.1Mei, Haibo; Xie, Chen; Wu, Lingmin; Soloshonok, Vadim A.; Han, Jianlin; Pan, Yi
Asymmetric Mannich reactions of imidazo[2,1-b]thiazole-derived nucleophiles with (SS)-N-tert-butanesulfinyl (3,3,3)-trifluoroacetaldimine.
Organic & biomolecular chemistry, 2013, 11, 8018-8021
7153204 CIFC23 H32 N4 O5P 21 21 218.9732; 10.4292; 25.653
90; 90; 90
2400.7Vijayadas, Kuruppanthara N.; Nair, Roshna V.; Gawade, Rupesh L.; Kotmale, Amol S.; Prabhakaran, Panchami; Gonnade, Rajesh G.; Puranik, Vedavadi G.; Rajamohanan, Pattuparambil R.; Sanjayan, Gangadhar J.
Ester vs. amide on folding: a case study with a 2-residue synthetic peptide.
Organic & biomolecular chemistry, 2013, 11, 8348-8356
7153205 CIFC21 H22 Br N3 O4P 21 21 217.1599; 11.846; 25.16
90; 90; 90
2134Vijayadas, Kuruppanthara N.; Nair, Roshna V.; Gawade, Rupesh L.; Kotmale, Amol S.; Prabhakaran, Panchami; Gonnade, Rajesh G.; Puranik, Vedavadi G.; Rajamohanan, Pattuparambil R.; Sanjayan, Gangadhar J.
Ester vs. amide on folding: a case study with a 2-residue synthetic peptide.
Organic & biomolecular chemistry, 2013, 11, 8348-8356
7153208 CIFC18 H24 N2 O5P 21 21 218.547; 9.694; 22.943
90; 90; 90
1900.9Vijayadas, Kuruppanthara N.; Nair, Roshna V.; Gawade, Rupesh L.; Kotmale, Amol S.; Prabhakaran, Panchami; Gonnade, Rajesh G.; Puranik, Vedavadi G.; Rajamohanan, Pattuparambil R.; Sanjayan, Gangadhar J.
Ester vs. amide on folding: a case study with a 2-residue synthetic peptide.
Organic & biomolecular chemistry, 2013, 11, 8348-8356
7153209 CIFC24 H28 N2 O5P 21 21 2110.6231; 10.9569; 19.528
90; 90; 90
2273Vijayadas, Kuruppanthara N.; Nair, Roshna V.; Gawade, Rupesh L.; Kotmale, Amol S.; Prabhakaran, Panchami; Gonnade, Rajesh G.; Puranik, Vedavadi G.; Rajamohanan, Pattuparambil R.; Sanjayan, Gangadhar J.
Ester vs. amide on folding: a case study with a 2-residue synthetic peptide.
Organic & biomolecular chemistry, 2013, 11, 8348-8356
7153210 CIFC16 H20 N2 O5P 21 21 218.111; 9.756; 20.126
90; 90; 90
1592.6Vijayadas, Kuruppanthara N.; Nair, Roshna V.; Gawade, Rupesh L.; Kotmale, Amol S.; Prabhakaran, Panchami; Gonnade, Rajesh G.; Puranik, Vedavadi G.; Rajamohanan, Pattuparambil R.; Sanjayan, Gangadhar J.
Ester vs. amide on folding: a case study with a 2-residue synthetic peptide.
Organic & biomolecular chemistry, 2013, 11, 8348-8356
7153211 CIFC25 H34 N2 O5P 21 21 217.4115; 16.548; 19.3577
90; 90; 90
2374.1Vijayadas, Kuruppanthara N.; Nair, Roshna V.; Gawade, Rupesh L.; Kotmale, Amol S.; Prabhakaran, Panchami; Gonnade, Rajesh G.; Puranik, Vedavadi G.; Rajamohanan, Pattuparambil R.; Sanjayan, Gangadhar J.
Ester vs. amide on folding: a case study with a 2-residue synthetic peptide.
Organic & biomolecular chemistry, 2013, 11, 8348-8356
7153212 CIFC18 H24 N2 O5P 21 21 218.3515; 9.6398; 22.979
90; 90; 90
1850Vijayadas, Kuruppanthara N.; Nair, Roshna V.; Gawade, Rupesh L.; Kotmale, Amol S.; Prabhakaran, Panchami; Gonnade, Rajesh G.; Puranik, Vedavadi G.; Rajamohanan, Pattuparambil R.; Sanjayan, Gangadhar J.
Ester vs. amide on folding: a case study with a 2-residue synthetic peptide.
Organic & biomolecular chemistry, 2013, 11, 8348-8356
7153213 CIFC20 H20 N2 O4P 21 21 218.173; 13.001; 17.35
90; 90; 90
1844Vijayadas, Kuruppanthara N.; Nair, Roshna V.; Gawade, Rupesh L.; Kotmale, Amol S.; Prabhakaran, Panchami; Gonnade, Rajesh G.; Puranik, Vedavadi G.; Rajamohanan, Pattuparambil R.; Sanjayan, Gangadhar J.
Ester vs. amide on folding: a case study with a 2-residue synthetic peptide.
Organic & biomolecular chemistry, 2013, 11, 8348-8356
7153233 CIFC19 H28 Cl N O2 SP 21 21 219.5924; 12.9905; 15.0218
90; 90; 90
1871.87Dobbs, Adrian P.; Guesné, Sebastien J J; Parker, Robert J.; Skidmore, John; Stephenson, Richard A.; Hursthouse, Mike B.
A detailed investigation of the aza-Prins reaction.
Organic & biomolecular chemistry, 2010, 8, 1064-1080
7153260 CIFC7 H7 N O4 SeP 21 21 214.9234; 9.5712; 17.319
90; 90; 90
816.12Yu, Sun-Chol; Kuhn, Hartmut; Daniliuc, Constantin-Gabriel; Ivanov, Igor; Jones, Peter G.; du Mont, Wolf-Walther
5-Selenization of salicylic acid derivatives yielded isoform-specific 5-lipoxygenase inhibitors.
Organic & biomolecular chemistry, 2010, 8, 828-834
7153271 CIFC26 H32 N2 O5P 21 21 2114.072; 14.218; 22.889
90; 90; 90
4579.53Boyd, D. R.; Sharma, N. D.; Sbircea, L.; Murphy, D.; Malone, J. F.; James, S. L.; Allen, C. C. R.; Hamilton, J. T. G.
Chemoenzymatic synthesis of chiral 2,2'-bipyridine ligands and their N-oxide derivatives: applications in the asymmetric aminolysis of epoxides and asymmetric allylation of aldehydes.
Organic & biomolecular chemistry, 2010, 8, 1081-1090
7153272 CIFC26 H32 N2 O6P 21 21 2114.1616; 14.2969; 22.8822
90; 90; 90
4632.89Boyd, D. R.; Sharma, N. D.; Sbircea, L.; Murphy, D.; Malone, J. F.; James, S. L.; Allen, C. C. R.; Hamilton, J. T. G.
Chemoenzymatic synthesis of chiral 2,2'-bipyridine ligands and their N-oxide derivatives: applications in the asymmetric aminolysis of epoxides and asymmetric allylation of aldehydes.
Organic & biomolecular chemistry, 2010, 8, 1081-1090
7153277 CIFC14 H18 O3P 21 21 216.3882; 10.3973; 18.3495
90; 90; 90
1218.77Austin, Kerrie A. B.; Elsworth, Jon D.; Banwell, Martin G.; Willis, Anthony C.
Chemoenzymatic and enantiodivergent routes to 1,2-ring-fused bicyclo[2.2.2]octane and related tricyclic frameworks.
Organic & biomolecular chemistry, 2010, 8, 751-754
7153278 CIFC14 H18 O3P 21 21 216.205; 11.5001; 17.0648
90; 90; 90
1217.71Austin, Kerrie A. B.; Elsworth, Jon D.; Banwell, Martin G.; Willis, Anthony C.
Chemoenzymatic and enantiodivergent routes to 1,2-ring-fused bicyclo[2.2.2]octane and related tricyclic frameworks.
Organic & biomolecular chemistry, 2010, 8, 751-754
7153279 CIFC18 H18 O3P 21 21 219.7159; 9.7758; 14.8253
90; 90; 90
1408.12Austin, Kerrie A. B.; Elsworth, Jon D.; Banwell, Martin G.; Willis, Anthony C.
Chemoenzymatic and enantiodivergent routes to 1,2-ring-fused bicyclo[2.2.2]octane and related tricyclic frameworks.
Organic & biomolecular chemistry, 2010, 8, 751-754
7153282 CIFC14 H20 O3P 21 21 216.3638; 12.4427; 15.6175
90; 90; 90
1236.64Austin, Kerrie A. B.; Elsworth, Jon D.; Banwell, Martin G.; Willis, Anthony C.
Chemoenzymatic and enantiodivergent routes to 1,2-ring-fused bicyclo[2.2.2]octane and related tricyclic frameworks.
Organic & biomolecular chemistry, 2010, 8, 751-754
7153287 CIFC18 H17 N O4P 21 21 216.4808; 15.236; 15.7084
90; 90; 90
1551.1Dungan, Victoria J.; Ortin, Yannick; Mueller-Bunz, Helge; Rutledge, Peter J.
Design and synthesis of a tetradentate '3-amine-1-carboxylate' ligand to mimic the metal binding environment at the non-heme iron(II) oxidase active site.
Organic & biomolecular chemistry, 2010, 8, 1666-1673
7153295 CIFC14 H20 O3P 21 21 217.4309; 10.1138; 16.7778
90; 90; 90
1260.9Hayashi, Nobuyuki; Yamamoto, Kentaro; Minowa, Nobuto; Mitomi, Masaaki; Nakada, Masahisa
Synthesis of NH006–a photostable fungicide effective against Botrytis cinerea–according to the asymmetric total synthesis of MK8383.
Organic & biomolecular chemistry, 2010, 8, 1821-1825
7153310 CIFC29 H20 O4P 21 21 216.3113; 8.5733; 39.914
90; 90; 90
2159.7Xie, Fuchun; Pan, Xuan; Lin, Shijun; Hu, Youhong
A base-promoted desalicyloylative dimerization of 3-(1-alkynyl)chromones: an unusual approach to 2-alkynyl xanthones.
Organic & biomolecular chemistry, 2010, 8, 1378-1381
7153319 CIFC14 H18 N2 OP 21 21 218.7304; 8.9046; 16.6172
90; 90; 90
1291.83Fuentes de Arriba, Angel L.; Simón, Luis; Raposo, César; Alcázar, Victoria; Sanz, Francisca; Muñiz, Francisco M; Morán, Joaquín R
Imidazolidinone intermediates in prolinamide-catalyzed aldol reactions.
Organic & biomolecular chemistry, 2010, 8, 2979-2985
7153321 CIFC18 H17 N3 O3P 21 21 216.6712; 14.9403; 15.7482
90; 90; 90
1569.62Fuentes de Arriba, Angel L.; Simón, Luis; Raposo, César; Alcázar, Victoria; Sanz, Francisca; Muñiz, Francisco M; Morán, Joaquín R
Imidazolidinone intermediates in prolinamide-catalyzed aldol reactions.
Organic & biomolecular chemistry, 2010, 8, 2979-2985
7153326 CIFC24 H19 Cl O2P 21 21 2112.5855; 14.0795; 21.9701
90; 90; 90
3893Wu, Chunlin; Li, Wenjun; Yang, Juanjuan; Liang, Xinmiao; Ye, Jinxing
Asymmetric organocatalytic Michael addition of anthrone to enone.
Organic & biomolecular chemistry, 2010, 8, 3244-3250
7153328 CIFC33 H25 N O2P 21 21 2112.4729; 13.3772; 13.8882
90; 90; 90
2317.3Kohmoto, Shigeo; Hisamatsu, Shugo; Mitsuhashi, Hakuei; Takahashi, Masahiro; Masu, Hyuma; Azumaya, Isao; Yamaguchi, Kentaro; Kishikawa, Keiki
Reversal of regioselectivity (straight vs. cross ring closure) in the intramolecular [2+2] photocycloaddition of phenanthrene derivatives.
Organic & biomolecular chemistry, 2010, 8, 2174-2179
7153339 CIFC31 H50 O5P 21 21 218.165; 13.02; 26.83
90; 90; 90
2852Yang, Xian-Wen; Li, Su-Mei; Wu, Liang; Li, Yong-Li; Feng, Lin; Shen, Yun-Heng; Tian, Jun-Mian; Tang, Jian; Wang, Ning; Liu, Yonghong; Zhang, Wei-Dong
Abiesatrines A-J: anti-inflammatory and antitumor triterpenoids from Abies georgei Orr.
Organic & biomolecular chemistry, 2010, 8, 2609-2616
7153341 CIFC16 H18 Cl N O3P 21 21 215.53; 8.5175; 34.0903
90; 90; 90
1605.71Li, Zhao-Bo; Luo, Shu-Ping; Guo, Yi; Xia, Ai-Bao; Xu, Dan-Qian
The highly enantioselective Michael addition of ketones to nitrodienes catalyzed by the efficient organocatalyst system of pyrrolidinyl-thioimidazole and chiral thioureido acid.
Organic & biomolecular chemistry, 2010, 8, 2505-2508
7153350 CIFC13 H12 N2 OP 21 21 216.286; 8.661; 19.599
90; 90; 90
1067Butin, Alexander V.; Nevolina, Tatyana A.; Shcherbinin, Vitaly A.; Trushkov, Igor V.; Cheshkov, Dmitry A.; Krapivin, Gennady D.
Furan ring opening-pyrrole ring closure: a new synthetic route to aryl(heteroaryl)-annulated pyrrolo[1,2-a][1,4]diazepines.
Organic & biomolecular chemistry, 2010, 8, 3316-3327
7153352 CIFC9 H12 Cl N SP 21 21 215.3436; 6.2291; 29.214
90; 90; 90
972.4Mercey, Guillaume; Legay, Remi; Lohier, Jean-François; Santos, Jana Sopkova-de Oliveira; Levillain, Jocelyne; Gaumont, Annie-Claude; Gulea, Mihaela
Synthesis of 3-amino-thiochromanes from 4-benzyl 2-thiazolines, via an unprecedented intramolecular electrophilic aromatic substitution.
Organic & biomolecular chemistry, 2010, 8, 2520-2521
7153353 CIFC9 H12 Cl N SP 21 21 215.3668; 6.2152; 29.035
90; 90; 90
968.5Mercey, Guillaume; Legay, Remi; Lohier, Jean-François; Santos, Jana Sopkova-de Oliveira; Levillain, Jocelyne; Gaumont, Annie-Claude; Gulea, Mihaela
Synthesis of 3-amino-thiochromanes from 4-benzyl 2-thiazolines, via an unprecedented intramolecular electrophilic aromatic substitution.
Organic & biomolecular chemistry, 2010, 8, 2520-2521
7153366 CIFC15 H15 F3 N2 O4P 21 21 2110.0807; 19.0872; 22.99
90; 90; 90
4423.56Stewart, Scott G.; Ghisalberti, Emilio L.; Skelton, Brian W.; Heath, Charles H.
Formation and reactions of azepino[4,5-b]indoles: an unprecedented ozone reaction in the formation of novel benzo[c]naphthyridinones.
Organic & biomolecular chemistry, 2010, 8, 3563-3570
7153374 CIFC40.71 H42.42 Cl1.42 N3 O5P 21 21 2110.949; 14.354; 24.633
90; 90; 90
3871.4Wright, Karen; Moretto, Alessandro; Crisma, Marco; Wakselman, Michel; Mazaleyrat, Jean-Paul; Formaggio, Fernando; Toniolo, Claudio
A new tool for photoaffinity labeling studies: a partially constrained, benzophenone based, alpha-amino acid.
Organic & biomolecular chemistry, 2010, 8, 3281-3286
7153389 CIFC14 H11 N O4P 21 21 216.778; 8.5059; 19.6445
90; 90; 90
1132.56Sar, Anobick; Lindeman, Sergey; Donaldson, William A.
De novo synthesis of polyhydroxyl aminocyclohexanes.
Organic & biomolecular chemistry, 2010, 8, 3908-3917
7153395 CIFC23 H15 BrP 21 21 216.1828; 9.6681; 27.58
90; 90; 90
1648.6Banide, Emilie V.; O'Connor, Crystal; Fortune, Natasha; Ortin, Yannick; Milosevic, Sandra; Müller-Bunz, Helge; McGlinchey, Michael J.
Syntheses, X-ray crystal structures and reactivity of fluorenylidene- and dibenzosuberenylidene-allenes: convenient precursors to dispirotetracenes, di-indenotetracenes and 2-phenyl-11bH-dibenz[cd,h]azulene.
Organic & biomolecular chemistry, 2010, 8, 3997-4010
7153396 CIFC23 H16P 21 21 216.8227; 9.1562; 25.406
90; 90; 90
1587.1Banide, Emilie V.; O'Connor, Crystal; Fortune, Natasha; Ortin, Yannick; Milosevic, Sandra; Müller-Bunz, Helge; McGlinchey, Michael J.
Syntheses, X-ray crystal structures and reactivity of fluorenylidene- and dibenzosuberenylidene-allenes: convenient precursors to dispirotetracenes, di-indenotetracenes and 2-phenyl-11bH-dibenz[cd,h]azulene.
Organic & biomolecular chemistry, 2010, 8, 3997-4010
7153426 CIFC18 H35 B K N3 O7P 21 21 218.5561; 15.6585; 17.715
90; 90; 90
2373.38Pitchumony, Tamil Selvi; Spingler, Bernhard; Motterlini, Roberto; Alberto, Roger
Syntheses, structural characterization and CO releasing properties of boranocarbonate [H3BCO2H]- derivatives.
Organic & biomolecular chemistry, 2010, 8, 4849-4854
7153442 CIFC37 H34 N2 OP 21 21 2110.9909; 13.0053; 20.0553
90; 90; 90
2866.7Gabbutt, Christopher D.; Heron, B. Mark; Kilner, Colin; Kolla, Suresh B.
The influence of a 1,1-diarylvinyl moiety on the photochromism of naphthopyrans.
Organic & biomolecular chemistry, 2010, 8, 4874-4883
7153443 CIFC14 H14 Br N O3P 21 21 216.607; 10.212; 20.641
90; 90; 90
1392.7Yu, Feng; Jin, Zhichao; Huang, Huicai; Ye, Tingting; Liang, Xinmiao; Ye, Jinxing
A highly efficient asymmetric Michael addition of α,α-disubstituted aldehydes to maleimides catalyzed by primary amine thiourea salt.
Organic & biomolecular chemistry, 2010, 8, 4767-4774
7153455 CIFC7 H10 I N O2P 21 21 216.634; 9.052; 14.778
90; 90; 90
887.4Leng, Dong-Hui; Wang, De-Xian; Huang, Zhi-Tang; Wang, Mei-Xiang
Highly efficient and enantioselective biotransformations of β-lactam carbonitriles and carboxamides and their synthetic applications.
Organic & biomolecular chemistry, 2010, 8, 4736-4743
7153459 CIFC18 H16 N4 OP 21 21 218.459; 9.484; 18.978
90; 90; 90
1522.5Chowdhury, Chinmay; Sasmal, Anup Kumar; Achari, Basudeb
An expedient and facile route for the general synthesis of 3-aryl substituted 1,2,3-triazolo[1,5-a][1,4]benzodiazepin-6-ones and 1,2,3-triazolo[1,5-a][1,5]benzodiazocin-7-ones.
Organic & biomolecular chemistry, 2010, 8, 4971-4977
7153460 CIFC20 H18 Cl N3 O SP 21 21 217.2935; 12.373; 20.6291
90; 90; 90
1861.62Kumar, Varun; Raghavaiah, Pallepogu; Mobin, Shaikh M.; Nair, Vipin A.
Diastereoselective syntheses of 3-aryl-5-(arylalkyl)-6-methyl-1-(1-phenylethyl)thioxotetrahydropyrimidin-4(1H)-ones: a stereochemical perspective from endo and exocyclic chiral centres.
Organic & biomolecular chemistry, 2010, 8, 4960-4970
7153461 CIFC20 H18 Cl N3 O SP 21 21 217.5879; 10.1912; 24.2981
90; 90; 90
1878.97Kumar, Varun; Raghavaiah, Pallepogu; Mobin, Shaikh M.; Nair, Vipin A.
Diastereoselective syntheses of 3-aryl-5-(arylalkyl)-6-methyl-1-(1-phenylethyl)thioxotetrahydropyrimidin-4(1H)-ones: a stereochemical perspective from endo and exocyclic chiral centres.
Organic & biomolecular chemistry, 2010, 8, 4960-4970
7153481 CIFC26 H28 F6 N2 O4P 21 21 2111.001; 11.945; 20.385
90; 90; 90
2678.7Madelaine, Claire; Buriez, Olivier; Crousse, Benoît; Florent, Isabelle; Grellier, Philippe; Retailleau, Pascal; Six, Yvan
Aminocyclopropanes as precursors of endoperoxides with antimalarial activity.
Organic & biomolecular chemistry, 2010, 8, 5591-5601
7153491 CIFC20 H15 N O2P 21 21 216.03265; 14.26965; 16.47322
90; 90; 90
1418.08Chamas, Zein el abidine; Dietz, Olivier; Aubert, Emmanuel; Fort, Yves; Mamane, Victor
Synthesis of new pentacyclic chromophores through a highly regio- and diastereoselective cascade process.
Organic & biomolecular chemistry, 2010, 8, 4815-4818
7153492 CIFC20 H15 N O2P 21 21 214.0331; 15.7754; 22.1253
90; 90; 90
1407.69Chamas, Zein el abidine; Dietz, Olivier; Aubert, Emmanuel; Fort, Yves; Mamane, Victor
Synthesis of new pentacyclic chromophores through a highly regio- and diastereoselective cascade process.
Organic & biomolecular chemistry, 2010, 8, 4815-4818
7153497 CIFC13 H17 N3 O6P 21 21 216.837; 10.47; 18.506
90; 90; 90
1324.7Xie, Yun; Maxson, Tucker; Tor, Yitzhak
Fluorescent nucleoside analogue displays enhanced emission upon pairing with guanine.
Organic & biomolecular chemistry, 2010, 8, 5053-5055
7153517 CIFC8 H16 N2 O5P 21 21 215.804; 11.033; 15.991
90; 90; 90
1024Davies, Stephen G.; Haggitt, Jane R.; Ichihara, Osamu; Kelly, Richard J.; Leech, Michael A.; Price Mortimer, Anne J.; Roberts, Paul M.; Smith, Andrew D.
Asymmetric total synthesis of sperabillins B and D via lithium amide conjugate addition
Organic & Biomolecular Chemistry, 2004, 2, 2630-2649
7153518 CIFC19 H26 I N O4P 21 21 218.2499; 13.392; 18.48
90; 90; 90
2041.7Davies, Stephen G.; Haggitt, Jane R.; Ichihara, Osamu; Kelly, Richard J.; Leech, Michael A.; Price Mortimer, Anne J.; Roberts, Paul M.; Smith, Andrew D.
Asymmetric total synthesis of sperabillins B and D via lithium amide conjugate addition
Organic & Biomolecular Chemistry, 2004, 2, 2630-2649
7153519 CIFC16 H16 N3 O6 TcP 21 21 219.0094; 13.0282; 15.5661
90; 90; 90
1827.1van Staveren, Dave R.; Mundwiler, Stefan; Hoffmanns, Ulrich; Pak, Jae Kyoung; Spingler, Bernhard; Metzler-Nolte, Nils; Alberto, Roger
Conjugation of a novel histidine derivative to biomolecules and labelling with [99mTc(OH2)3(CO)3]+Electronic supplementary information (ESI) available: complete 1H and 13C NMR spectra of 14, 15, 16 and 19. See http://www.rsc.org/suppdata/ob/b4/b405575f/
Organic & Biomolecular Chemistry, 2004, 2, 2593-2603
7153531 CIFC17 H23 N O4 SP 21 21 218.23; 9.09; 22.57
90; 90; 90
1688Wang, Libo; Nakamura, Shuichi; Toru, Takeshi
Highly enantioselective reaction of lithiated N-Boc-thiazolidine: a new chiral formyl anion equivalent
Organic & Biomolecular Chemistry, 2004, 2, 2168-2169
7153533 CIFC30 H36 N4 O3P 21 21 2111.1668; 11.7777; 20.32
90; 90; 90
2672.47El Drubi Vega, Ismael; Gale, Philip A.; Hursthouse, Michael B.; Light, Mark E.
Anion binding properties of 5,5?-dicarboxamido-dipyrrolylmethanes
Organic & Biomolecular Chemistry, 2004, 2, 2935-2941
7153536 CIFC28 H41 N3 O5 S2P 21 21 217.476; 14.31; 26.388
90; 90; 90
2823.03Scheuermann, J. Erik W.; Sibbons, Kevin F.; Benoit, David M.; Motevalli, Majid; Watkinson, Michael
The synthesis of unsymmetrically N-substituted chiral 1,4,7-triazacyclononanesElectronic supplementary information (ESI) available: Molecular modelling methodology. Figs. S1?S4: Lowest energy conformation calculated for the protonated form of 6b, 6b�HOAc, the protonated form of 6a and 6a�HOAc. Figs. S5 and S6: Charge distribution calculated for the protonated forms of 6a and 6b. See http://www.rsc.org/suppdata/ob/b4/b409259g/
Organic & Biomolecular Chemistry, 2004, 2, 2664-2670
7153537 CIFC24 H37 N3 O4 S2P 21 21 2110.752; 11.183; 21.829
90; 90; 90
2624.7Scheuermann, J. Erik W.; Sibbons, Kevin F.; Benoit, David M.; Motevalli, Majid; Watkinson, Michael
The synthesis of unsymmetrically N-substituted chiral 1,4,7-triazacyclononanesElectronic supplementary information (ESI) available: Molecular modelling methodology. Figs. S1?S4: Lowest energy conformation calculated for the protonated form of 6b, 6b�HOAc, the protonated form of 6a and 6a�HOAc. Figs. S5 and S6: Charge distribution calculated for the protonated forms of 6a and 6b. See http://www.rsc.org/suppdata/ob/b4/b409259g/
Organic & Biomolecular Chemistry, 2004, 2, 2664-2670
7153548 CIFC18 H31 N O4P 21 21 215.5694; 10.414; 30.935
90; 90; 90
1794.2Lin, Geng-Jie; Huang, Pei-Qiang
A concise and fully selective synthesis of the ant venom alkaloid (3S,5R,8S,9S)-3-butyl-5-propyl-8-hydroxyindolizidine
Organic & Biomolecular Chemistry, 2009, 7, 4491-4495
7153587 CIFC25 H25 N2 O6 PP 21 21 218.901; 12.206; 22.343
90; 90; 90
2427.5George, Jimil; Sridhar, B.; Reddy, B. V. Subba
First example of quinine-squaramide catalyzed enantioselective addition of diphenyl phosphite to ketimines derived from isatins.
Organic & biomolecular chemistry, 2014, 12, 1595-1602
7153591 CIFC18 H17 N O3P 21 21 219.3972; 16.1308; 19.6022
90; 90; 90
2971.39Nandakumar, Avanashiappan; Kiruthika, Selvarangam E.; Naveen, Kanagaraj; Perumal, Paramasivan Thirumalai
Pd(0)-catalyzed regio- and stereoselective cyclization of alkynes: selective synthesis of (E)-4-(isobenzofuran-1(3H)-ylidene)-1,2,3,4-tetrahydroisoquinolines and aze/oxepinoindoles.
Organic & biomolecular chemistry, 2014, 12, 876-880
7153601 CIFC17 H14 O4P 21 21 218.85; 12.001; 12.727
90; 90; 90
1351.7Zhang, Hongrui; Li, Haifeng; Xue, Jijun; Chen, Rui; Li, Ying; Tang, Yu; Li, Chunxin
New facile enantio- and diastereo-selective syntheses of (-)-triptonide and (-)-triptolide.
Organic & biomolecular chemistry, 2014, 12, 732-736
7153604 CIFC34 H46 Br N5 O6P 21 21 219.6704; 9.8238; 38.263
90; 90; 90
3635Nair, Roshna V.; Kotmale, Amol S.; Dhokale, Snehal A.; Gawade, Rupesh L.; Puranik, Vedavadi G.; Rajamohanan, Pattuparambil R.; Sanjayan, Gangadhar J.
Formation of a pseudo-β-hairpin motif utilizing the Ant-Pro reverse turn: consequences of stereochemical reordering.
Organic & biomolecular chemistry, 2014, 12, 774-782
7153618 CIFC19 H16 Cl O4 PP 21 21 216.2873; 12.402; 22.054
90; 90; 90
1719.7Alegre-Requena, Juan V; Marqués-López, Eugenia; Sanz Miguel, Pablo J.; Herrera, Raquel P.
Organocatalytic enantioselective hydrophosphonylation of aldehydes.
Organic & biomolecular chemistry, 2014, 12, 1258-1264
7153619 CIFC28 H29 N3 O2 SeP 21 21 219.29; 16.2681; 16.8894
90; 90; 90
2552.5Balkrishna, Shah Jaimin; Kumar, Shailesh; Azad, Gajendra Kumar; Bhakuni, Bhagat Singh; Panini, Piyush; Ahalawat, Navjeet; Tomar, Raghuvir Singh; Detty, Michael R.; Kumar, Sangit
An ebselen like catalyst with enhanced GPx activity via a selenol intermediate.
Organic & biomolecular chemistry, 2014, 12, 1215-1219
7153629 CIFC12 H7 I2 N3P 21 21 214.4884; 12.4932; 22.191
90; 90; 90
1244.35Nagaradja, Elisabeth; Chevallier, Floris; Roisnel, Thierry; Dorcet, Vincent; Halauko, Yury S.; Ivashkevich, Oleg A.; Matulis, Vadim E.; Mongin, Florence
Deproto-metallation using a mixed lithium-zinc base and computed CH acidity of 1-aryl 1H-benzotriazoles and 1-aryl 1H-indazoles.
Organic & biomolecular chemistry, 2014, 12, 1475-1487
7153652 CIFC14 H14 Cl4 OP 21 21 218.8558; 12.1899; 12.9536
90; 90; 90
1398.36Olbrich, Martin; Mayer, Peter; Trauner, Dirk
A step toward polytwistane: synthesis and characterization of C2-symmetric tritwistane.
Organic & biomolecular chemistry, 2014, 12, 108-112
7153662 CIFC13 H13 Br N2 O4 SP 21 21 219.5461; 9.6709; 15.4442
90; 90; 90
1425.8Jiang, Jianbing; Vairaprakash, Pothiappan; Reddy, Kanumuri Ramesh; Sahin, Tuba; Pavan, M. Phani; Lubian, Elisa; Lindsey, Jonathan S.
Hydrophilic tetracarboxy bacteriochlorins for photonics applications.
Organic & biomolecular chemistry, 2014, 12, 86-103
7153665 CIFC6 H7 Cl2 I O3 SP 21 21 215.9357; 8.96; 20.683
90; 90; 90
1100Boyd, Derek R.; Sharma, Narain D.; Kaik, Magdalena; McIntyre, Peter B. A.; Malone, John F.; Stevenson, Paul J.
Reactions of enantiopure cyclic diols with sulfuryl chloride.
Organic & biomolecular chemistry, 2014, 12, 2128-2136
7153667 CIFC6 H7 Cl O4 SP 21 21 216.6774; 10.9657; 11.0176
90; 90; 90
806.73Boyd, Derek R.; Sharma, Narain D.; Kaik, Magdalena; McIntyre, Peter B. A.; Malone, John F.; Stevenson, Paul J.
Reactions of enantiopure cyclic diols with sulfuryl chloride.
Organic & biomolecular chemistry, 2014, 12, 2128-2136
7153671 CIFC16 H17 F3 N4 O S2P 21 21 2110.499; 11.042; 16.3
90; 90; 90
1890Mei, Haibo; Xiong, Yiwen; Xie, Chen; Soloshonok, Vadim A.; Han, Jianlin; Pan, Yi
Concise and scalable asymmetric synthesis of 5-(1-amino-2,2,2-trifluoroethyl)thiazolo[3,2-b][1,2,4]triazoles.
Organic & biomolecular chemistry, 2014, 12, 2108-2113
7153695 CIFC18 H20 Cl3 N O3P 21 21 216.4986; 7.2522; 40.288
90; 90; 90
1898.7Jia, Wen-Qiang; Chen, Xiang-Yu; Sun, Li-Hui; Ye, Song
Organocatalytic [4 + 2] cyclocondensation of α,β-unsaturated acyl chlorides with imines: highly enantioselective synthesis of dihydropyridinone and piperidine derivatives.
Organic & biomolecular chemistry, 2014, 12, 2167-2171
7153696 CIFC22 H23 N O6 SP 21 21 215.8326; 8.921; 40.497
90; 90; 90
2107.2Jia, Wen-Qiang; Chen, Xiang-Yu; Sun, Li-Hui; Ye, Song
Organocatalytic [4 + 2] cyclocondensation of α,β-unsaturated acyl chlorides with imines: highly enantioselective synthesis of dihydropyridinone and piperidine derivatives.
Organic & biomolecular chemistry, 2014, 12, 2167-2171
7153697 CIFC12 H12 Cl3 N OP 21 21 219.4908; 11.747; 23.965
90; 90; 90
2671.8Jia, Wen-Qiang; Chen, Xiang-Yu; Sun, Li-Hui; Ye, Song
Organocatalytic [4 + 2] cyclocondensation of α,β-unsaturated acyl chlorides with imines: highly enantioselective synthesis of dihydropyridinone and piperidine derivatives.
Organic & biomolecular chemistry, 2014, 12, 2167-2171
7153727 CIFC16 H25 N O2P 21 21 218.66504; 9.9818; 18.4067
90; 90; 90
1592.05Davies, Stephen G.; Fletcher, Ai M.; Lee, James A.; Roberts, Paul M.; Souleymanou, Myriam Y.; Thomson, James E.; Zammit, Charlotte M.
Diastereoselective Ireland-Claisen rearrangements of substituted allyl β-amino esters: applications in the asymmetric synthesis of C(5)-substituted transpentacins.
Organic & biomolecular chemistry, 2014, 12, 2702-2728
7153732 CIFC34.5 H36 N O2.5P 21 21 2112.315; 15.4817; 29.8308
90; 90; 90
5687.45Davies, Stephen G.; Fletcher, Ai M.; Lee, James A.; Roberts, Paul M.; Souleymanou, Myriam Y.; Thomson, James E.; Zammit, Charlotte M.
Diastereoselective Ireland-Claisen rearrangements of substituted allyl β-amino esters: applications in the asymmetric synthesis of C(5)-substituted transpentacins.
Organic & biomolecular chemistry, 2014, 12, 2702-2728
7153749 CIFC15 H27 N O6 SP 21 21 219.2379; 10.1214; 19.9426
90; 90; 90
1864.64Callebaut, Gert; Colpaert, Filip; Nonn, Melinda; Kiss, Loránd; Sillanpää, Reijo; Törnroos, Karl W; Fülöp, Ferenc; De Kimpe, Norbert; Mangelinckx, Sven
Asymmetric synthesis of chloroisothreonine derivatives via syn-stereoselective Mannich-type additions across N-sulfinyl-α-chloroimines.
Organic & biomolecular chemistry, 2014, 12, 3393-3405
7153755 CIFC18 H13 N O3P 21 21 218.954; 9.455; 17.176
90; 90; 90
1454.1Zhang, Yu; Lu, Yingyan; Tang, Weifang; Lu, Tao; Du, Ding
Cooperative N-heterocyclic carbene (NHC)-Lewis acid-mediated regioselective umpolung formal [3 + 2] annulations of alkynyl aldehydes with isatins.
Organic & biomolecular chemistry, 2014, 12, 3009-3015
7153776 CIFC26 H22 N6 S4P 21 21 216.7025; 19.621; 20.267
90; 90; 90
2665.3Biet, Thomas; Avarvari, Narcis
Tetrathiafulvalene mono- and bis-1,2,3-triazole precursors by click chemistry: structural diversity and reactivity.
Organic & biomolecular chemistry, 2014, 12, 3167-3174
7153786 CIFC14 H23 B N3 PP 21 21 219.85; 11.141; 14.4209
90; 90; 90
1582.53Veillard, Romain; Bernoud, Elise; Abdellah, Ibrahim; Lohier, Jean-François; Alayrac, Carole; Gaumont, Annie-Claude
Silyl alkynylphosphine-boranes: key precursors of triazolylphosphines via tandem desilylation-Click chemistry.
Organic & biomolecular chemistry, 2014, 12, 3635-3640
7153788 CIFC12 H22 N4 O3P 21 21 219.2345; 10.4403; 15.8938
90; 90; 90
1532.34Pike, Sarah J.; Raftery, James; Webb, Simon J.; Clayden, Jonathan
Conformational analysis of helical aminoisobutyric acid (Aib) oligomers bearing C-terminal ester Schellman motifs.
Organic & biomolecular chemistry, 2014, 12, 4124-4131
7153796 CIFC11 H13 F N2 O2P 21 21 218.1246; 9.2109; 14.8139
90; 90; 90
1108.6Ramachary, Dhevalapally B.; Shruthi, Kodambahalli S.
Asymmetric synthesis of tetrahydroquinolines through supramolecular organocatalysis.
Organic & biomolecular chemistry, 2014, 12, 4300-4304
7153806 CIFC16 H11 N O2P 21 21 214.896; 11.351; 21.44
90; 90; 90
1191.52Edeson, Steven J.; Jiang, Julong; Swanson, Stephen; Procopiou, Panayiotis A.; Adams, Harry; Meijer, Anthony J. H. M.; Harrity, Joseph P. A.
Studies on the stereochemical assignment of 3-acylidene 2-oxindoles.
Organic & biomolecular chemistry, 2014, 12, 3201-3210
7153813 CIFC17 H19 N O4P 21 21 219.1314; 12.4725; 12.8711
90; 90; 90
1465.9Liu, Dandan; Ai, Long; Li, Fan; Zhao, Annan; Chen, Jingbo; Zhang, Hongbin; Liu, Jianping
Total synthesis of lycorine-type alkaloids by cyclopropyl ring-opening rearrangement.
Organic & biomolecular chemistry, 2014, 12, 3191-3200
7153815 CIFC18 H16 N2 OP 21 21 214.9093; 14.694; 19.032
90; 90; 90
1372.9Prasad, Karothu Durga; Trinath, Jamma; Biswas, Ansuman; Sekar, Kanagaraj; Balaji, Kithiganahalli N.; Guru Row, Tayur N.
Alkyl chain substituted 1,9-pyrazoloanthrones exhibit prominent inhibitory effect on c-Jun N-terminal kinase (JNK).
Organic & biomolecular chemistry, 2014, 12, 4656-4662
7153817 CIFC17 H14 N2 OP 21 21 215.4152; 15.1404; 15.678
90; 90; 90
1285.41Prasad, Karothu Durga; Trinath, Jamma; Biswas, Ansuman; Sekar, Kanagaraj; Balaji, Kithiganahalli N.; Guru Row, Tayur N.
Alkyl chain substituted 1,9-pyrazoloanthrones exhibit prominent inhibitory effect on c-Jun N-terminal kinase (JNK).
Organic & biomolecular chemistry, 2014, 12, 4656-4662
7153823 CIFC30 H54 O5P 21 21 2110.5637; 13.2734; 20.6274
90; 90; 90
2892.3Yu, Jin-Hai; Shen, Yu; Liu, Hong-Bing; Leng, Ying; Zhang, Hua; Yue, Jian-Min
Dammarane-type triterpenoids as 11β-HSD1 inhibitors from Homonoia riparia.
Organic & biomolecular chemistry, 2014, 12, 4716-4722
7153828 CIFC17 H17 N O2P 21 21 218.6589; 10.1791; 15.9766
90; 90; 90
1408.17Zhu, Xu; Chiba, Shunsuke
TEMPO-mediated allylic C-H amination with hydrazones.
Organic & biomolecular chemistry, 2014, 12, 4567-4570
7153837 CIFC18 H25 N O4P 21 21 215.5701; 9.012; 33.683
90; 90; 90
1690.81Su, Cunxiang; Xie, Ying; Pan, Hongjie; Liu, Mao; Tian, Hua; Shi, Yian
Organocatalytic synthesis of optically active β-branched α-amino esters via asymmetric biomimetic transamination.
Organic & biomolecular chemistry, 2014, 12, 5856-5860
7153848 CIFC10 H8 N2 O2P 21 21 215.6964; 12.6163; 12.8565
90; 90; 90
923.96Pratap Reddy Gajulapalli, V.; Vinayagam, Poopathy; Kesavan, Venkitasamy
Organocatalytic asymmetric decarboxylative cyanomethylation of isatins using l-proline derived bifunctional thiourea.
Organic & biomolecular chemistry, 2014, 12, 4186-4191
7153857 CIFC21 H20 N2 O6 SP 21 21 218.534; 15.242; 16.014
90; 90; 90
2083Huynh, Thi Ngoc Tram; Retailleau, Pascal; Denhez, Clément; Nguyen, Kim Phi Phung; Guillaume, Dom
Regioselective synthesis of 3,4,5-trisubstituted 2-aminofurans.
Organic & biomolecular chemistry, 2014, 12, 5098-5101
7153861 CIFC20.25 H20.25 N2.25 O4.5 S0P 21 21 219.259; 13.478; 15.399
90; 90; 90
1921.7Srivastava, Abhijeet; Shukla, Gaurav; Nagaraju, Anugula; Verma, Girijesh Kumar; Raghuvanshi, Keshav; Jones, Raymond C. F.; Singh, Maya Shankar
In(OTf)3-catalysed one-pot versatile pyrrole synthesis through domino annulation of α-oxoketene-N,S-acetals with nitroolefins.
Organic & biomolecular chemistry, 2014, 12, 5484-5491
7153863 CIFC7 H10 O6P 21 21 216.7699; 8.2068; 15.1001
90; 90; 90
838.95Sudhakar, Gangarajula; Bayya, Shruthi; Kadam, Vilas D.; Nanubolu, Jagadeesh Babu
Total synthesis of gonytolides C and G, lachnone C, and formal synthesis of blennolide C and diversonol.
Organic & biomolecular chemistry, 2014, 12, 5601-5610
7153875 CIFC29 H37 N3 O3P 21 21 215.9134; 19.9075; 23.6392
90; 90; 90
2782.83Kotovshchikov, Yury N.; Latyshev, Gennadij V.; Lukashev, Nikolay V.; Beletskaya, Irina P.
Synthesis of novel 1,2,3-triazolyl derivatives of pregnane, androstane and d-homoandrostane. Tandem "click" reaction/Cu-catalyzed d-homo rearrangement.
Organic & biomolecular chemistry, 2014, 12, 3707-3720
7153880 CIFC14 H21 N O5P 21 21 215.51; 13.604; 19.941
90; 90; 90
1495Tian, Xiang-Yin; Han, Jian-Wei; Zhao, Qiong; Wong, Henry N. C.
Asymmetric synthesis of 3,3,5,5-tetrasubstituted 1,2-dioxolanes: total synthesis of epiplakinic acid F.
Organic & biomolecular chemistry, 2014, 12, 3686-3700
7153887 CIFC21 H15 Cl N2 O2P 21 21 218.8826; 9.7822; 20.8708
90; 90; 90
1813.5Mandha, Santhosh Reddy; Alla, Manjula; Nanubolu, Jagadeesh Babu
"One-pot" access to dihydrofurans via tandem oxidative difunctionalization and ring contraction of aminopyrans.
Organic & biomolecular chemistry, 2014, 12, 4412-4420
7153889 CIFC17 H16 N2 O3P 21 21 219.3671; 9.5385; 17.0984
90; 90; 90
1527.71Roca-López, David; Marqués-López, Eugenia; Alcaine, Ana; Merino, Pedro; Herrera, Raquel P.
A Friedel-Crafts alkylation mechanism using an aminoindanol-derived thiourea catalyst.
Organic & biomolecular chemistry, 2014, 12, 4503-4510
7153899 CIFC30 H30 Cl2 N2 O3P 21 21 218.9169; 17.351; 17.602
90; 90; 90
2723.3Weber, Anna K.; Schachtner, Josef; Fichtler, Robert; Leermann, Timo M.; Neudörfl, Jörg M; Jacobi von Wangelin, Axel
Modular synthesis of cyclic cis- and trans-1,2-diamine derivatives.
Organic & biomolecular chemistry, 2014, 12, 5267-5277
7153909 CIFC24 H16 O3 SeP 21 21 219.96379; 10.04828; 19.6441
90; 90; 90
1966.75Wu, Xiangfei; Shirakawa, Seiji; Maruoka, Keiji
Efficient asymmetric synthesis of spiro-2(3H)-furanones via phase-transfer-catalyzed alkynylation.
Organic & biomolecular chemistry, 2014, 12, 5388-5392
7153929 CIFC24 H25 N O6 SP 21 21 2110.6; 12.434; 16.898
90; 90; 90
2227.2Bera, Kalisankar; Namboothiri, Irishi N. N.
Enantioselective synthesis of γ-tetrasubstituted nitrosulfonyl carboxylates and amides vial-tert-leucine-derived-squaramide catalyzed conjugate addition of nitrosulfones to acrylates and acrylamides.
Organic & biomolecular chemistry, 2014, 12, 6425-6431
7153941 CIFC21 H27 N3 O3P 21 21 219.167; 13.2568; 15.2701
90; 90; 90
1855.7Li, Fuying; Cheng, Kejun; Antoline, Joshua F. G.; Iyer, Malliga R.; Matyas, Gary R.; Torres, Oscar B.; Jalah, Rashmi; Beck, Zoltan; Alving, Carl R.; Parrish, Damon A.; Deschamps, Jeffrey R.; Jacobson, Arthur E.; Rice, Kenner C.
Synthesis and immunological effects of heroin vaccines.
Organic & biomolecular chemistry, 2014, 12, 7211-7232
7153942 CIFC17 H17 Cl N2 O4P 21 21 217.3581; 9.136; 23.005
90; 90; 90
1546.5Li, Fuying; Cheng, Kejun; Antoline, Joshua F. G.; Iyer, Malliga R.; Matyas, Gary R.; Torres, Oscar B.; Jalah, Rashmi; Beck, Zoltan; Alving, Carl R.; Parrish, Damon A.; Deschamps, Jeffrey R.; Jacobson, Arthur E.; Rice, Kenner C.
Synthesis and immunological effects of heroin vaccines.
Organic & biomolecular chemistry, 2014, 12, 7211-7232
7153943 CIFC18 H23 N O2P 21 21 216.8411; 12.9417; 16.7006
90; 90; 90
1478.6Li, Fuying; Cheng, Kejun; Antoline, Joshua F. G.; Iyer, Malliga R.; Matyas, Gary R.; Torres, Oscar B.; Jalah, Rashmi; Beck, Zoltan; Alving, Carl R.; Parrish, Damon A.; Deschamps, Jeffrey R.; Jacobson, Arthur E.; Rice, Kenner C.
Synthesis and immunological effects of heroin vaccines.
Organic & biomolecular chemistry, 2014, 12, 7211-7232
7153948 CIFC20 H21 Br O2P 21 21 2111.211; 16.7616; 18.3398
90; 90; 90
3446.3Subba Reddy, B. V.; Ramana Reddy, M.; Sridhar, B.; Singarapu, Kiran Kumar
Acetal-initiated Prins bicyclization for the synthesis of hexahydrofuro-[3,4-c]furan lignans and octahydropyrano[3,4-c]pyran derivatives.
Organic & biomolecular chemistry, 2014, 12, 4754-4762
7153974 CIFC21 H31 N O7 SP 21 21 216.7501; 17.4344; 19.5104
90; 90; 90
2296.1Tiwari, Dipak Kumar; Bharadwaj, Kishor Chandra; Puranik, Vedavati G.; Tiwari, Dharmendra Kumar
Divergent total synthesis of 1,6,8a-tri-epi-castanospermine and 1-deoxy-6,8a-di-epi-castanospermine from substituted azetidin-2-one (β-lactam), involving a cascade sequence of reactions as a key step.
Organic & biomolecular chemistry, 2014, 12, 7389-7396
7153986 CIFC26 H38 Cl3 N O5P 21 21 2111.8362; 12.2518; 19.0137
90; 90; 90
2757.27Kong, Lili; Rao, Mingjin; Ou, Jinjie; Yin, Jun; Lu, Weiqiang; Liu, Mingyao; Pang, Xiufeng; Gao, Shuanhu
Total synthesis and biological studies of cryptocin and derivatives of equisetin and fusarisetin A.
Organic & biomolecular chemistry, 2014, 12, 7591-7597
7153987 CIFC25 H37 N O4P 21 21 216.8794; 14.9305; 22.2706
90; 90; 90
2287.5Kong, Lili; Rao, Mingjin; Ou, Jinjie; Yin, Jun; Lu, Weiqiang; Liu, Mingyao; Pang, Xiufeng; Gao, Shuanhu
Total synthesis and biological studies of cryptocin and derivatives of equisetin and fusarisetin A.
Organic & biomolecular chemistry, 2014, 12, 7591-7597
7153992 CIFC13 H15 N3 O3P 21 21 217.028; 12.5922; 14.037
90; 90; 90
1242.2Putapatri, Siddamal Reddy; Kanwal, Abhinav; Sridhar, Balasubramanian; Banerjee, Sanjay K.; Kantevari, Srinivas
Synthesis of l-rhamnose derived chiral bicyclic triazoles as novel sodium-glucose transporter (SGLT) inhibitors.
Organic & biomolecular chemistry, 2014, 12, 8415-8421
7153993 CIFC14 H17 N3 O3P 21 21 217.555; 11.987; 15.0918
90; 90; 90
1366.74Putapatri, Siddamal Reddy; Kanwal, Abhinav; Sridhar, Balasubramanian; Banerjee, Sanjay K.; Kantevari, Srinivas
Synthesis of l-rhamnose derived chiral bicyclic triazoles as novel sodium-glucose transporter (SGLT) inhibitors.
Organic & biomolecular chemistry, 2014, 12, 8415-8421
7153997 CIFC19 H18 Cl N O4P 21 21 216.627; 7.9739; 32.9949
90; 90; 90
1743.55Takahashi, Masaki; Murata, Yusuke; Ishida, Masahiro; Yagishita, Fumitoshi; Sakamoto, Masami; Sengoku, Tetsuya; Yoda, Hidemi
Catalytic amide allylation of α-ketoesters: extremely high enantioselective synthesis of ester functionalised α-methylene-γ-butyrolactones.
Organic & biomolecular chemistry, 2014, 12, 7686-7689
7154007 CIFC14 H19 N O3 SP 21 21 217.681; 12.525; 14.693
90; 90; 90
1413.5Clarke, Leslie Ann; Ring, Aoife; Ford, Alan; Sinha, Abhijeet S.; Lawrence, Simon E.; Maguire, Anita R.
Enantioselective copper catalysed C-H insertion reaction of 2-sulfonyl-2-diazoacetamides to form γ-lactams.
Organic & biomolecular chemistry, 2014, 12, 7612-7628
7154008 CIFC23 H25 N5 O5P 21 21 215.5457; 8.9659; 42.4254
90; 90; 90
2109.48Kovaliov, Marina; Wachtel, Chaim; Yavin, Eylon; Fischer, Bilha
Synthesis and evaluation of a photoresponsive quencher for fluorescent hybridization probes.
Organic & biomolecular chemistry, 2014, 12, 7844-7858
7154012 CIFC19 H10 B F2 N3 OP 21 21 216.4067; 7.2419; 32.409
90; 90; 90
1503.7Liu, Hui; Lu, Hua; Wu, Fan; Li, Zhifang; Kobayashi, Nagao; Shen, Zhen
Synthesis and spectroscopic properties of novel meso-cyano boron-pyridyl-isoindoline dyes.
Organic & biomolecular chemistry, 2014, 12, 8223-8229
7154027 CIFC43 H60 O16P 21 21 2110.054; 16.853; 23.794
90; 90; 90
4031.7Ding, Chunyong; Wang, Lili; Chen, Haijun; Wild, Christopher; Ye, Na; Ding, Ye; Wang, Tianzhi; White, Mark A.; Shen, Qiang; Zhou, Jia
ent-Kaurane-based regio- and stereoselective inverse electron demand hetero-Diels-Alder reactions: synthesis of dihydropyran-fused diterpenoids.
Organic & biomolecular chemistry, 2014, 12, 8442-8452
7154028 CIFC28 H37 Cl O7P 21 21 219.4979; 13.0601; 21.0823
90; 90; 90
2615.1Ding, Chunyong; Wang, Lili; Chen, Haijun; Wild, Christopher; Ye, Na; Ding, Ye; Wang, Tianzhi; White, Mark A.; Shen, Qiang; Zhou, Jia
ent-Kaurane-based regio- and stereoselective inverse electron demand hetero-Diels-Alder reactions: synthesis of dihydropyran-fused diterpenoids.
Organic & biomolecular chemistry, 2014, 12, 8442-8452
7154029 CIFC15 H19 F3 N2 O2 SP 21 21 215.7933; 15.9715; 18.559
90; 90; 90
1717.2Qian, Ping; Xie, Chen; Wu, Lingmin; Mei, Haibo; Soloshonok, Vadim A.; Han, Jianlin; Pan, Yi
Asymmetric synthesis of (3S,1'S)-3-(1-amino-2,2,2-trifluoroethyl)-1-(alkyl)-indolin-2-one derivatives by addition of (S)-N-t-butylsulfinyl-3,3,3-trifluoroacetaldimine to 1-(alkyl)-indolin-2-ones.
Organic & biomolecular chemistry, 2014, 12, 7909-7913
7154075 CIFC18 H37 Cl N O4P 21 21 215.3932; 7.7138; 49.332
90; 90; 90
2052.3Désiré, J; Mondon, M.; Fontelle, N.; Nakagawa, S.; Hirokami, Y.; Adachi, I.; Iwaki, R.; Fleet, G. W. J.; Alonzi, D. S.; Twigg, G.; Butters, T. D.; Bertrand, J.; Cendret, V.; Becq, F.; Norez, C.; Marrot, J.; Kato, A.; Blériot, Y
N- and C-alkylation of seven-membered iminosugars generates potent glucocerebrosidase inhibitors and F508del-CFTR correctors.
Organic & biomolecular chemistry, 2014, 12, 8977-8996
7154077 CIFC18 H24 N4 O5P 21 21 219.0217; 13.8727; 15.2216
90; 90; 90
1905.1Majer, Roberta; Konechnaya, Olga; Delso, Ignacio; Tejero, Tomas; Attanasi, Orazio A.; Santeusanio, Stefania; Merino, Pedro
Highly diastereoselective 1,3-dipolar cycloadditions of chiral non-racemic nitrones to 1,2-diaza-1,3-dienes: an experimental and computational investigation.
Organic & biomolecular chemistry, 2014, 12, 8888-8901
7154080 CIFC28 H27 N O3P 21 21 218.9295; 13.0992; 19.384
90; 90; 90
2267.3Ariyarathna, Yamuna; Tunge, Jon A.
Decarboxylative allylations of ester enolate equivalents.
Organic & biomolecular chemistry, 2014, 12, 8386-8389
7154086 CIFC25 H23 F N2 O2P 21 21 218.2975; 11.26; 21.17
90; 90; 90
1977.9Aillard, Boris; Robertson, Naomi S.; Baldwin, Adam R.; Robins, Siobhan; Jamieson, Andrew G.
Robust asymmetric synthesis of unnatural alkenyl amino acids for conformationally constrained α-helix peptides.
Organic & biomolecular chemistry, 2014, 12, 8775-8782
7154087 CIFC28 H26 Cl2 F N3 Ni O3P 21 21 219.38; 16.703; 16.766
90; 90; 90
2627Aillard, Boris; Robertson, Naomi S.; Baldwin, Adam R.; Robins, Siobhan; Jamieson, Andrew G.
Robust asymmetric synthesis of unnatural alkenyl amino acids for conformationally constrained α-helix peptides.
Organic & biomolecular chemistry, 2014, 12, 8775-8782
7154088 CIFC30 H30 Cl4 F N3 Ni O3P 21 21 219.1183; 14.255; 23.374
90; 90; 90
3038.2Aillard, Boris; Robertson, Naomi S.; Baldwin, Adam R.; Robins, Siobhan; Jamieson, Andrew G.
Robust asymmetric synthesis of unnatural alkenyl amino acids for conformationally constrained α-helix peptides.
Organic & biomolecular chemistry, 2014, 12, 8775-8782
7154090 CIFC35 H38 F N3 Ni O3P 21 21 219.165; 13.957; 23.73
90; 90; 90
3035Aillard, Boris; Robertson, Naomi S.; Baldwin, Adam R.; Robins, Siobhan; Jamieson, Andrew G.
Robust asymmetric synthesis of unnatural alkenyl amino acids for conformationally constrained α-helix peptides.
Organic & biomolecular chemistry, 2014, 12, 8775-8782
7154092 CIFC26 H38 O6P 21 21 2111.4718; 12.9514; 15.8446
90; 90; 90
2354.13Zhang, Rong-Rong; Tian, Hai-Yan; Tan, Ya-Fang; Chung, Tse-Yu; Sun, Xiao-Hui; Xia, Xue; Ye, Wen-Cai; Middleton, David A.; Fedosova, Natalya; Esmann, Mikael; Tzen, Jason T. C.; Jiang, Ren-Wang
Structures, chemotaxonomic significance, cytotoxic and Na(+),K(+)-ATPase inhibitory activities of new cardenolides from Asclepias curassavica.
Organic & biomolecular chemistry, 2014, 12, 8919-8929
7154093 CIFC26 H38 N O6P 21 21 2110.4301; 11.8072; 18.744
90; 90; 90
2308.33Zhang, Rong-Rong; Tian, Hai-Yan; Tan, Ya-Fang; Chung, Tse-Yu; Sun, Xiao-Hui; Xia, Xue; Ye, Wen-Cai; Middleton, David A.; Fedosova, Natalya; Esmann, Mikael; Tzen, Jason T. C.; Jiang, Ren-Wang
Structures, chemotaxonomic significance, cytotoxic and Na(+),K(+)-ATPase inhibitory activities of new cardenolides from Asclepias curassavica.
Organic & biomolecular chemistry, 2014, 12, 8919-8929
7154109 CIFC10 H10 Cl N O4 SP 21 21 217.3279; 14.173; 22.626
90; 90; 90
2349.9Wang, You-Qing; Cui, Xiao-Yu; Ren, Yuan-Yuan; Zhang, Yongna
A highly enantioselective and regioselective organocatalytic direct Mannich reaction of methyl alkyl ketones with cyclic imines benzo[e][1,2,3]oxathiazine 2,2-dioxides.
Organic & biomolecular chemistry, 2014, 12, 9101-9104
7154110 CIFC12 H16 O3P 21 21 216.687; 19.034; 35.511
90; 90; 90
4520Shing, Tony K. M.; Wong, Anthony W. H.; Li, Huiyan; Liu, Z. F.; Chan, Paul K. S.
Conformationally locked bicyclo[4.3.0]nonane carbanucleosides: synthesis and bio-evaluation.
Organic & biomolecular chemistry, 2014, 12, 9439
7154111 CIFC14 H19.5 N5 O3.5P 21 21 218.5282; 10.7576; 41.024
90; 90; 90
3763.7Shing, Tony K. M.; Wong, Anthony W. H.; Li, Huiyan; Liu, Z. F.; Chan, Paul K. S.
Conformationally locked bicyclo[4.3.0]nonane carbanucleosides: synthesis and bio-evaluation.
Organic & biomolecular chemistry, 2014, 12, 9439
7154128 CIFC36 H30 N2 O6P 21 21 2112.2096; 13.7443; 18.0044
90; 90; 90
3021.4Yagishita, Fumitoshi; Baba, Nozomi; Ueda, Yuki; Katabira, Satoshi; Kasashima, Yoshio; Mino, Takashi; Sakamoto, Masami
Diastereoselective photodimerization reactions of chromone-2-carboxamides to construct a C2-chiral scaffold.
Organic & biomolecular chemistry, 2014, 12, 9644-9649
7154129 CIFC36 H30 N2 O6P 21 21 219.7337; 13.9495; 22.104
90; 90; 90
3001.3Yagishita, Fumitoshi; Baba, Nozomi; Ueda, Yuki; Katabira, Satoshi; Kasashima, Yoshio; Mino, Takashi; Sakamoto, Masami
Diastereoselective photodimerization reactions of chromone-2-carboxamides to construct a C2-chiral scaffold.
Organic & biomolecular chemistry, 2014, 12, 9644-9649
7154130 CIFC32 H38 N2 O6P 21 21 217.704; 14.23; 26.5
90; 90; 90
2905Yagishita, Fumitoshi; Baba, Nozomi; Ueda, Yuki; Katabira, Satoshi; Kasashima, Yoshio; Mino, Takashi; Sakamoto, Masami
Diastereoselective photodimerization reactions of chromone-2-carboxamides to construct a C2-chiral scaffold.
Organic & biomolecular chemistry, 2014, 12, 9644-9649
7154131 CIFC28 H26 N2 O10P 21 21 218.021; 15.273; 21.484
90; 90; 90
2631.9Yagishita, Fumitoshi; Baba, Nozomi; Ueda, Yuki; Katabira, Satoshi; Kasashima, Yoshio; Mino, Takashi; Sakamoto, Masami
Diastereoselective photodimerization reactions of chromone-2-carboxamides to construct a C2-chiral scaffold.
Organic & biomolecular chemistry, 2014, 12, 9644-9649
7154133 CIFC32 H36 Cl N OP 21 21 2110.084; 10.408; 26.571
90; 90; 90
2788.7Liu, Yilin; Feng, Xiangqing; Du, Haifeng
Asymmetric synthesis of axially chiral anilides by Pd-catalyzed allylic substitutions with P/olefin ligands.
Organic & biomolecular chemistry, 2015, 13, 125-132
7154134 CIFC30 H40 Cl N OP 21 21 219.779; 10.66; 26.314
90; 90; 90
2743.1Liu, Yilin; Feng, Xiangqing; Du, Haifeng
Asymmetric synthesis of axially chiral anilides by Pd-catalyzed allylic substitutions with P/olefin ligands.
Organic & biomolecular chemistry, 2015, 13, 125-132
7154144 CIFC33 H33 N O5P 21 21 2111.012; 13.289; 18.958
90; 90; 90
2774.3Zanato, Chiara; Watson, Sonia; Bewick, Guy S.; Harrison, William T. A.; Zanda, Matteo
Synthesis and biological evaluation of (-)-kainic acid analogues as phospholipase D-coupled metabotropic glutamate receptor ligands.
Organic & biomolecular chemistry, 2014, 12, 9638-9643
7154154 CIFC24 H33 N O5 PP 21 21 215.8926; 18.289; 22.043
90; 90; 90
2375.6Sun, Yong-Ming; Xin, Nana; Xu, Zhong-Yuan; Liu, Li-Juan; Meng, Fan-Jie; Zhang, He; Fu, Bao-Ci; Liang, Qiu-Ju; Zheng, Hong-Xing; Sun, Li-Jun; Zhao, Chang-Qiu; Han, Li-Biao
Addition of optically pure H-phosphinate to ketones: selectivity, stereochemistry and mechanism.
Organic & biomolecular chemistry, 2014, 12, 9457
7154158 CIFC15 H11 Cl2 N5P 21 21 216.5036; 12.9729; 17.9702
90; 90; 90
1516.2Dai, Zhi-Cheng; Chen, Yong-Fei; Zhang, Mao; Li, Sheng-Kun; Yang, Ting-Ting; Shen, Li; Wang, Jian-Xin; Qian, Shao-Song; Zhu, Hai-Liang; Ye, Yong-Hao
Synthesis and antifungal activity of 1,2,3-triazole phenylhydrazone derivatives.
Organic & biomolecular chemistry, 2015, 13, 477-486
7154162 CIFC39 H26 Cl2 N2 OP 21 21 217.1928; 13.3215; 32.7007
90; 90; 90
3133.3Li, Wei; Fan, Zhoulong; Geng, Kaijun; Xu, Youjun; Zhang, Ao
Late-stage diversification of biologically active pyridazinones via a direct C-H functionalization strategy.
Organic & biomolecular chemistry, 2015, 13, 539-548
7154180 CIFC15 H16 N2 O3P 21 21 215.6153; 14.7482; 16.9257
90; 90; 90
1401.71Łukasik, Beata; Mikołajczyk, Marian; Bujacz, Grzegorz; Żurawiński, Remigiusz
Synthesis and the absolute configuration of both enantiomers of 4,5-dihydroxy-3-(formyl)cyclopent-2-enone acetonide as a new chiral building block for prostanoid synthesis.
Organic & biomolecular chemistry, 2015, 13, 807-816
7154183 CIFC24 H15 N O4P 21 21 214.9114; 9.9314; 36.687
90; 90; 90
1789.5Savych, Iryna; Gläsel, Tim; Villinger, Alexander; Sosnovskikh, Vyacheslav Ya; Iaroshenko, Viktor O.; Langer, Peter
Synthesis of functionalized 2-salicyloylfurans, furo[3,2-b]chromen-9-ones and 2-benzoyl-8H-thieno[2,3-b]indoles by one-pot cyclizations of 3-halochromones with β-ketoamides and 1,3-dihydroindole-2-thiones.
Organic & biomolecular chemistry, 2015, 13, 729-750
7154190 CIFC14 H18 N4 O5 SP 21 21 215.7297; 16.224; 17.5243
90; 90; 90
1629.04Denoël, Thibaut; Zervosen, Astrid; Lemaire, Christian; Joris, Bernard; Hervé, Mireille; Blanot, Didier; Zaragoza, Guillermo; Luxen, André
Enantioselective synthesis of α-benzylated lanthionines and related tripeptides for biological incorporation into E. coli peptidoglycan.
Organic & biomolecular chemistry, 2014, 12, 9853-9863
7154192 CIFC79 H84 Cl N2 O10 RhP 21 21 2115.0756; 15.9328; 28.2582
90; 90; 90
6787.5Henderson, Alexander S.; Bower, John F.; Galan, M. Carmen
Carbohydrate-based N-heterocyclic carbenes for enantioselective catalysis.
Organic & biomolecular chemistry, 2014, 12, 9180-9183
7154196 CIFC19 H16 Br N O2P 21 21 2117.158; 6.001; 15.681
90; 90; 90
1614.6Guo, Jiajia; Yu, Shouyun
Enantioselective synthesis of benzoindolizidine derivatives using chiral phase-transfer catalytic intramolecular domino aza-Michael addition/alkylation.
Organic & biomolecular chemistry, 2015, 13, 1179-1186
7154201 CIFC70.15 H81.65 Cl15.44 F1.5 N12 O19 S6P 21 21 2117.1143; 20.8803; 26.8416
90; 90; 90
9591.9Wu, Haifan; She, Fengyu; Gao, Wenyang; Prince, Austin; Li, Yaqiong; Wei, Lulu; Mercer, Allison; Wojtas, Lukasz; Ma, Shengqian; Cai, Jianfeng
The synthesis of head-to-tail cyclic sulfono-γ-AApeptides.
Organic & biomolecular chemistry, 2015, 13, 672-676
7154210 CIFC22 H24 N2 O6P 21 21 219.4466; 12.186; 18.704
90; 90; 90
2153.1Alcaide, Benito; Almendros, Pedro; Aragoncillo, Cristina; Callejo, Ricardo; Pilar Ruiz, M.; Rosario Torres, M.
Investigation of the Passerini and Ugi reactions in β-lactam aldehydes. Synthetic applications.
Organic & biomolecular chemistry, 2015, 13, 1387-1394
7154220 CIFC21 H20 O5P 21 21 219.095; 11.415; 17.22
90; 90; 90
1787.8Cheng, Jin-Tang; Chen, Xiang-Yu; Ye, Song
N-heterocyclic carbene-catalyzed cyclocondensation of 2-aryl carboxylic acids and enones: highly enantioselective synthesis of δ-lactones.
Organic & biomolecular chemistry, 2015, 13, 1313-1316
7154234 CIFC20 H21 N O3P 21 21 217.4058; 12.3833; 18.9412
90; 90; 90
1737.1Pichler, Mathias; Novacek, Johanna; Robiette, Raphaël; Poscher, Vanessa; Himmelsbach, Markus; Monkowius, Uwe; Müller, Norbert; Waser, Mario
Asymmetric syntheses of three-membered heterocycles using chiral amide-based ammonium ylides.
Organic & biomolecular chemistry, 2015, 13, 2092-2099
7154235 CIFC25 H29 Br N2 O4P 21 21 217.8797; 12.465; 25.404
90; 90; 90
2495.2Pichler, Mathias; Novacek, Johanna; Robiette, Raphaël; Poscher, Vanessa; Himmelsbach, Markus; Monkowius, Uwe; Müller, Norbert; Waser, Mario
Asymmetric syntheses of three-membered heterocycles using chiral amide-based ammonium ylides.
Organic & biomolecular chemistry, 2015, 13, 2092-2099
7154237 CIFC18 H16 N2 O8P 21 21 215.83; 9.556; 31.119
90; 90; 90
1733.7Jana, Anupam; Mondal, Sujit; Ghosh, Subrata
Studies towards the synthesis of bielschowskysin. Construction of the highly functionalized bicyclo[3.2.0]heptane segment.
Organic & biomolecular chemistry, 2015, 13, 1846-1859
7154266 CIFC17 H31 Cl2 N P2 PdP 21 21 217.2904; 10.5177; 31.1288
90; 90; 90
2386.9Yang, Zehua; Xia, Chao; Liu, Delong; Liu, Yangang; Sugiya, Masashi; Imamoto, Tsuneo; Zhang, Wanbin
P-stereogenic PNP pincer-Pd catalyzed intramolecular hydroamination of amino-1,3-dienes.
Organic & biomolecular chemistry, 2015, 13, 2694-2702
7154274 CIFC15 H17 N O4P 21 21 216.046; 10.17; 24.25
90; 90; 90
1491Targel, Tom A.; Kumar, Jayprakash N.; Shneider, O. Svetlana; Bar, Sukanta; Fridman, Natalia; Maximenko, Shimon; Szpilman, Alex M.
Oxidative asymmetric umpolung alkylation of Evans' β-ketoimides using dialkylzinc nucleophiles.
Organic & biomolecular chemistry, 2015, 13, 2546-2549
7154278 CIFC12 H13 F N2 O6P 21 21 215.5351; 11.2034; 21.678
90; 90; 90
1344.3Kwiatkowski, Jacek; Lu, Yixin
Asymmetric Michael addition of α-fluoro-α-nitro esters to nitroolefins: towards synthesis of α-fluoro-α-substituted amino acids.
Organic & biomolecular chemistry, 2015, 13, 2350-2359
7154289 CIFC27 H33 Br N4 O5 SP 21 21 216.7186; 15.8096; 26.5176
90; 90; 90
2816.66Vijayadas, Kuruppanthara N.; Kotmale, Amol S.; Thorat, Shridhar H.; Gonnade, Rajesh G.; Nair, Roshna V.; Rajamohanan, Pattuparambil R.; Sanjayan, Gangadhar J.
Reversal of H-bonding direction by N-sulfonation in a synthetic reverse-turn peptide motif.
Organic & biomolecular chemistry, 2015, 13, 3064-3069
7154292 CIFC17 H26 N4 O6 S2P 21 21 219.5896; 14.7665; 14.7848
90; 90; 90
2093.6Vijayadas, Kuruppanthara N.; Kotmale, Amol S.; Thorat, Shridhar H.; Gonnade, Rajesh G.; Nair, Roshna V.; Rajamohanan, Pattuparambil R.; Sanjayan, Gangadhar J.
Reversal of H-bonding direction by N-sulfonation in a synthetic reverse-turn peptide motif.
Organic & biomolecular chemistry, 2015, 13, 3064-3069
7154294 CIFC19 H20 Br N3 O4 SP 21 21 219.2942; 13.9119; 15.3096
90; 90; 90
1979.5Vijayadas, Kuruppanthara N.; Kotmale, Amol S.; Thorat, Shridhar H.; Gonnade, Rajesh G.; Nair, Roshna V.; Rajamohanan, Pattuparambil R.; Sanjayan, Gangadhar J.
Reversal of H-bonding direction by N-sulfonation in a synthetic reverse-turn peptide motif.
Organic & biomolecular chemistry, 2015, 13, 3064-3069
7154321 CIFC14 H15 Br N4 O4 SP 21 21 218.079; 11.113; 18.417
90; 90; 90
1653.5Huang, Hu; Pan, Hongjie; Cai, Yudong; Liu, Mao; Tian, Hua; Shi, Yian
Enantioselective 6-endo bromoaminocyclization of 2,4-dienyl N-tosylcarbamates catalyzed by a chiral phosphine oxide-Sc(OTf)3 complex. A dramatic additive effect.
Organic & biomolecular chemistry, 2015, 13, 3566-3570
7154326 CIFC20 H24 Br N O5 S2P 21 21 215.6597; 15.69; 24.567
90; 90; 90
2181.6Huang, Hu; Pan, Hongjie; Cai, Yudong; Liu, Mao; Tian, Hua; Shi, Yian
Enantioselective 6-endo bromoaminocyclization of 2,4-dienyl N-tosylcarbamates catalyzed by a chiral phosphine oxide-Sc(OTf)3 complex. A dramatic additive effect.
Organic & biomolecular chemistry, 2015, 13, 3566-3570
7154328 CIFC19 H18 Br N O4 SP 21 21 217.963; 11.336; 20.402
90; 90; 90
1841.7Huang, Hu; Pan, Hongjie; Cai, Yudong; Liu, Mao; Tian, Hua; Shi, Yian
Enantioselective 6-endo bromoaminocyclization of 2,4-dienyl N-tosylcarbamates catalyzed by a chiral phosphine oxide-Sc(OTf)3 complex. A dramatic additive effect.
Organic & biomolecular chemistry, 2015, 13, 3566-3570
7154334 CIFC26 H18 Br N3 OP 21 21 2111.7456; 13.5528; 13.0646
90; 90; 90
2079.7Fang, Fang; Hua, Genghong; Shi, Feng; Li, Pengfei
Organocatalytic enantioselective Friedel-Crafts reaction: an efficient access to chiral isoindolo-β-carboline derivatives.
Organic & biomolecular chemistry, 2015, 13, 4395-4398
7154353 CIFC35 H33 N O6 SP 21 21 2110.5513; 13.4479; 21.737
90; 90; 90
3084.3Pandey, Ganesh; Varkhedkar, Rajesh; Tiwari, Divya
Efficient access to enantiopure 1,3-disubstituted isoindolines from selective catalytic fragmentation of an original desymmetrized rigid overbred template.
Organic & biomolecular chemistry, 2015, 13, 4438-4448
7154356 CIFC69 H74 N12 O7P 21 21 2115.5903; 18.0794; 25.8875
90; 90; 90
7296.7Chavez-Acevedo, Lizbeth; Miranda, Luis D.
Synthesis of novel tryptamine-based macrocycles using an Ugi 4-CR/microwave assisted click-cycloaddition reaction protocol.
Organic & biomolecular chemistry, 2015, 13, 4408-4412
7154373 CIFC13 H14 O2P 21 21 218.1768; 9.01871; 14.2224
90; 90; 90
1048.82Fan, Lulu; Takizawa, Shinobu; Takeuchi, Yoshiki; Takenaka, Kazuhiro; Sasai, Hiroaki
Pd-catalyzed enantioselective intramolecular α-arylation of α-substituted cyclic ketones: facile synthesis of functionalized chiral spirobicycles.
Organic & biomolecular chemistry, 2015, 13, 4837-4840
7154376 CIFC18 H18 Br N O5 SP 21 21 219.3617; 13.1822; 14.7459
90; 90; 90
1819.76Takechi, Ryosuke; Nishimura, Takahiro
Rhodium-catalyzed asymmetric addition of arylboronic acids to cyclic N-sulfonyl ketimines towards the synthesis of α,α-diaryl-α-amino acid derivatives.
Organic & biomolecular chemistry, 2015, 13, 4918-4924
7154392 CIFC20 H23 N O5P 21 21 219.1967; 10.3931; 19.4118
90; 90; 90
1855.42Shashank, Adluri B.; Ramachary, Dhevalapally B.
Organocatalytic diastereoselective synthesis of chiral decalines through the domino Claisen-Schmidt/Henry reaction.
Organic & biomolecular chemistry, 2015, 13, 5110-5114
7154394 CIFC8 H18 N2 O9 S2P 21 21 217.9598; 9.8111; 17.7241
90; 90; 90
1384.15Miller, Duncan C.; Carbain, Benoit; Beale, Gary S.; Alhasan, Sari F.; Reeves, Helen L.; Baisch, Ulrich; Newell, David R.; Golding, Bernard T.; Griffin, Roger J.
Regioselective sulfamoylation at low temperature enables concise syntheses of putative small molecule inhibitors of sulfatases.
Organic & biomolecular chemistry, 2015, 13, 5279-5284
7154405 CIFC25 H25 Cl N2 O6P 21 21 217.5714; 15.502; 20.241
90; 90; 90
2375.7Sun, Jing; Chen, Liang; Gong, Hui; Yan, Chao-Guo
Convenient synthesis of functionalized spiro[indoline-3,2'-pyrrolizines] or spiro[indoline-3,3'-pyrrolidines] via multicomponent reactions.
Organic & biomolecular chemistry, 2015, 13, 5905-5917
7154407 CIFC33 H32 N2 O7 SP 21 21 2118.95; 13.964; 11.122
90; 90; 90
2943Sun, Jing; Chen, Liang; Gong, Hui; Yan, Chao-Guo
Convenient synthesis of functionalized spiro[indoline-3,2'-pyrrolizines] or spiro[indoline-3,3'-pyrrolidines] via multicomponent reactions.
Organic & biomolecular chemistry, 2015, 13, 5905-5917
7154408 CIFC30 H33 Cl N2 O7 SP 21 21 2110.504; 16.482; 16.712
90; 90; 90
2893.3Sun, Jing; Chen, Liang; Gong, Hui; Yan, Chao-Guo
Convenient synthesis of functionalized spiro[indoline-3,2'-pyrrolizines] or spiro[indoline-3,3'-pyrrolidines] via multicomponent reactions.
Organic & biomolecular chemistry, 2015, 13, 5905-5917
7154418 CIFC19 H16 F4 O2P 21 21 218.7578; 10.8532; 18.2457
90; 90; 90
1734.26Wang, Jingjing; Kong, Wei-Guang; Li, Feng; Liu, Jie; Shen, Qin; Liu, Lantao; Zhao, Wen-Xian
Silver salts and DBU cooperatively catalyzed nucleophilic addition/cyclization of propargylic alcohols with trifluoromethyl ketones.
Organic & biomolecular chemistry, 2015, 13, 5399-5406
7154425 CIFC14 H16 N4 O4P 21 21 218.1008; 9.745; 18.18
90; 90; 90
1435.2de la Fuente, Alex; Mena-Barragán, Teresa; Farrar-Tobar, Ronald A; Verdaguer, Xavier; García Fernández, José M; Ortiz Mellet, Carmen; Riera, Antoni
Stereoselective synthesis of 2-acetamido-1,2-dideoxynojirimycin (DNJNAc) and ureido-DNJNAc derivatives as new hexosaminidase inhibitors.
Organic & biomolecular chemistry, 2015, 13, 6500-6510
7154426 CIFC14 H16 N4 O4P 21 21 219.6858; 9.9838; 15.1087
90; 90; 90
1461.03de la Fuente, Alex; Mena-Barragán, Teresa; Farrar-Tobar, Ronald A; Verdaguer, Xavier; García Fernández, José M; Ortiz Mellet, Carmen; Riera, Antoni
Stereoselective synthesis of 2-acetamido-1,2-dideoxynojirimycin (DNJNAc) and ureido-DNJNAc derivatives as new hexosaminidase inhibitors.
Organic & biomolecular chemistry, 2015, 13, 6500-6510
7154427 CIFC25 H17 Cl O3P 21 21 215.8099; 21.073; 32.234
90; 90; 90
3946.5Chen, Kun-Quan; Zhang, Han-Ming; Wang, Dong-Ling; Sun, De-Qun; Ye, Song
Enantioselective N-heterocyclic carbene-catalyzed synthesis of indenopyrones.
Organic & biomolecular chemistry, 2015, 13, 6694-6697
7154443 CIFC24 H24 Br2 N2 O3 SP 21 21 219.181; 9.395; 27.281
90; 90; 90
2353.1Gui, Yong-Yuan; Yang, Jian; Qi, Liang-Wen; Wang, Xiao; Tian, Fang; Li, Xiao-Nian; Peng, Lin; Wang, Li-Xin
A cinchona alkaloid catalyzed enantioselective sulfa-Michael/aldol cascade reaction of isoindigos: construction of chiral bispirooxindole tetrahydrothiophenes with vicinal quaternary spirocenters.
Organic & biomolecular chemistry, 2015, 13, 6371-6379
7154446 CIFC7 H7 Cl2 N OP 21 21 215.9311; 10.5722; 13.4606
90; 90; 90
844.04Essa, Ali H.; Lerrick, Reinner I.; Çiftçi, Eçe; Harrington, Ross W.; Waddell, Paul G.; Clegg, William; Hall, Michael J.
Grignard-mediated reduction of 2,2,2-trichloro-1-arylethanones.
Organic & biomolecular chemistry, 2015, 13, 5793-5803
7154453 CIFC23 H18 Cl2 N2 O7P 21 21 218.4445; 15.4187; 17.2259
90; 90; 90
2242.87Essa, Ali H.; Lerrick, Reinner I.; Çiftçi, Eçe; Harrington, Ross W.; Waddell, Paul G.; Clegg, William; Hall, Michael J.
Grignard-mediated reduction of 2,2,2-trichloro-1-arylethanones.
Organic & biomolecular chemistry, 2015, 13, 5793-5803
7154471 CIFC15 H10 Cl N3 O2P 21 21 217.052; 19.594; 19.706
90; 90; 90
2722.9Li, Gen; Feng, Xiangqing; Du, Haifeng
Palladium-catalyzed asymmetric allylic amination of racemic butadiene monoxide with isatin derivatives.
Organic & biomolecular chemistry, 2015, 13, 5826-5830
7154492 CIFC15 H13 Br N2 O2P 21 21 215.947; 7.118; 32.87
90; 90; 90
1391.4Maity, Rajendra; Pan, Subhas Chandra
Organocatalytic asymmetric intramolecular aza-Henry reaction: facile synthesis of trans-2,3-disubstituted tetrahydroquinolines.
Organic & biomolecular chemistry, 2015, 13, 6825-6831
7154493 CIFC6 H13 N O6 SP 21 21 215.14008; 9.60877; 18.4697
90; 90; 90
912.216Suthagar, Kajitha; Polson, Matthew I. J.; Fairbanks, Antony J.
Unexpected furanose/pyranose equilibration of N-glycosyl sulfonamides, sulfamides and sulfamates.
Organic & biomolecular chemistry, 2015, 13, 6573-6579
7154502 CIFC19 H18 N2 O2P 21 21 217.9192; 14.304; 14.6004
90; 90; 90
1653.88Quick, Matthias P.; Fröhlich, Roland; Schepmann, Dirk; Wünsch, Bernhard
Asymmetric synthesis of 3-substituted tetrahydro-2-benzazepines.
Organic & biomolecular chemistry, 2015, 13, 7265-7281
7154516 CIFC26 H28 N2 O6P 21 21 216.59; 14.579; 25.484
90; 90; 90
2448.4Lenci, Elena; Innocenti, Riccardo; Menchi, Gloria; Faggi, Cristina; Trabocchi, Andrea
Two-step one-pot synthesis of dihydropyrazinones as Xaa-Ser dipeptide isosteres through morpholine acetal rearrangement.
Organic & biomolecular chemistry, 2015, 13, 7013-7019
7154518 CIFC17 H14 Br N O5 SP 21 21 2110.476; 8.883; 18.154
90; 90; 90
1689.38De Munck, Lode; Monleón, Alicia; Vila, Carlos; Muñoz, M Carmen; Pedro, José R
Enantioselective alkynylation of benzo[e][1,2,3]-oxathiazine 2,2-dioxides catalysed by (R)-VAPOL-Zn complexes: synthesis of chiral propargylic cyclic sulfamidates.
Organic & biomolecular chemistry, 2015, 13, 7393-7396
7154522 CIFC18 H27 N O4P 21 21 215.7917; 15.4852; 18.6976
90; 90; 90
1676.91Jimenez-Aleman, Guillermo H; Machado, Ricardo A. R.; Görls, Helmar; Baldwin, Ian T.; Boland, Wilhelm
Synthesis, structural characterization and biological activity of two diastereomeric JA-Ile macrolactones.
Organic & biomolecular chemistry, 2015, 13, 5885-5893
7154529 CIFC20 H24 Br N O2P 21 21 217.77818; 13.158; 16.9759
90; 90; 90
1737.4Ishida, Hiroaki; Kimura, Shinya; Kogure, Noriyuki; Kitajima, Mariko; Takayama, Hiromitsu
The first asymmetric total synthesis of lycoposerramine-R.
Organic & biomolecular chemistry, 2015, 13, 7762-7771
7154530 CIFC20 H24 Br N O2P 21 21 217.63463; 11.4385; 19.919
90; 90; 90
1739.5Ishida, Hiroaki; Kimura, Shinya; Kogure, Noriyuki; Kitajima, Mariko; Takayama, Hiromitsu
The first asymmetric total synthesis of lycoposerramine-R.
Organic & biomolecular chemistry, 2015, 13, 7762-7771
7154545 CIFC34 H38 N4 O3 SP 21 21 218.7342; 12.9336; 27.4037
90; 90; 90
3095.65Saura, A. Vanessa; Marín, María J; Burguete, M. Isabel; Russell, David A.; Galindo, Francisco; Luis, Santiago V.
The synthesis of new fluorescent bichromophoric compounds as ratiometric pH probes for intracellular measurements.
Organic & biomolecular chemistry, 2015, 13, 7736-7749
7154556 CIFC29 H34 O5P 21 21 219.3233; 10.2871; 26.846
90; 90; 90
2574.8Salamone, Stéphane; Clement, Lise L.; Viuff, Agnete H.; Andersen, Ole Juul; Jensen, Frank; Jensen, Henrik H.
Synthesis and evaluation of galacto-noeurostegine and its 2-deoxy analogue as glycosidase inhibitors.
Organic & biomolecular chemistry, 2015, 13, 7979-7992
7154557 CIFC17 H16 I O4 SiP 21 21 217.4496; 11.1966; 26.6185
90; 90; 90
2220.25Lu, Hai-Hua; Hinkelmann, Bettina; Tautz, Thomas; Li, Jun; Sasse, Florenz; Franke, Raimo; Kalesse, Markus
Paleo-soraphens: chemical total syntheses and biological studies.
Organic & biomolecular chemistry, 2015, 13, 8029-8036
7154558 CIFC15 H22 O3P 21 21 217.73264; 8.92045; 20.1079
90; 90; 90
1387.02Ma, Jiang-Hao; Zhao, Feng; Wang, Ying; Liu, Yue; Gao, Su-Yu; Ding, Li-Qin; Chen, Li-Xia; Qiu, Feng
Natural nitric oxide (NO) inhibitors from the rhizomes of Curcuma phaeocaulis.
Organic & biomolecular chemistry, 2015, 13, 8349-8358
7154563 CIFC14 H21 Br N2 O2P 21 21 217.0938; 11.5502; 18.1965
90; 90; 90
1490.93Ozeryanskii, Valery A.; Gorbacheva, Anastasia Yu; Pozharskii, Alexander F.; Vlasenko, Marina P.; Tereznikov, Alexander Yu; Chernov'yants, Margarita S.
The first proton sponge-based amino acids: synthesis, acid-base properties and some reactivity.
Organic & biomolecular chemistry, 2015, 13, 8524-8532
7154602 CIFC28 H37 N O2 SeP 21 21 218.5898; 10.768; 28.159
90; 90; 90
2604.6Nieto, Javier; Andrés, Celia; Pérez-Encabo, Alfonso
7-endo selenocyclization reactions on chiral 3-prenyl and 3-cinnamyl-2-hydroxymethylperhydro-1,3-benzoxazine derivatives. A way to enantiopure 1,4-oxazepanes.
Organic & biomolecular chemistry, 2015, 13, 9118-9126
7154603 CIFC26 H41 N O2 SeP 21 21 2112.295; 13.5593; 15.728
90; 90; 90
2622Nieto, Javier; Andrés, Celia; Pérez-Encabo, Alfonso
7-endo selenocyclization reactions on chiral 3-prenyl and 3-cinnamyl-2-hydroxymethylperhydro-1,3-benzoxazine derivatives. A way to enantiopure 1,4-oxazepanes.
Organic & biomolecular chemistry, 2015, 13, 9118-9126
7154605 CIFC22 H32 Cl N O2P 21 21 218.8571; 15.0597; 15.5921
90; 90; 90
2079.8Nieto, Javier; Andrés, Celia; Pérez-Encabo, Alfonso
7-endo selenocyclization reactions on chiral 3-prenyl and 3-cinnamyl-2-hydroxymethylperhydro-1,3-benzoxazine derivatives. A way to enantiopure 1,4-oxazepanes.
Organic & biomolecular chemistry, 2015, 13, 9118-9126
7154610 CIFC34 H36 N O9 P SP 21 21 2116.3644; 15.9689; 12.8284
90; 90; 90
3352.3D'Onofrio, A; Copey, L.; Jean-Gérard, L; Goux-Henry, C; Pilet, G.; Andrioletti, B.; Framery, E.
d-Glucosamine as a novel chiral auxiliary for the stereoselective synthesis of P-stereogenic phosphine oxides.
Organic & biomolecular chemistry, 2015, 13, 9029-9034
7154612 CIFC27 H28 N O8 P SP 21 21 2111.8008; 14.3566; 16.6799
90; 90; 90
2825.9D'Onofrio, A; Copey, L.; Jean-Gérard, L; Goux-Henry, C; Pilet, G.; Andrioletti, B.; Framery, E.
d-Glucosamine as a novel chiral auxiliary for the stereoselective synthesis of P-stereogenic phosphine oxides.
Organic & biomolecular chemistry, 2015, 13, 9029-9034
7154614 CIFC17 H28 N2 O5 Se SiP 21 21 217.621; 13.163; 23.299
90; 90; 90
2337.2Kogami, Masakazu; Koketsu, Mamoru
An efficient method for the synthesis of selenium modified nucleosides: its application in the synthesis of Se-adenosyl-l-selenomethionine (SeAM).
Organic & biomolecular chemistry, 2015, 13, 9405-9417
7154623 CIFC21 H20 Br N O3P 21 21 216.4981; 11.985; 23.813
90; 90; 90
1854.5Chen, Min; Huang, Zhi-Tang; Zheng, Qi-Yu
Organic base-promoted enantioselective electrophilic cyanation of β-keto esters by using chiral phase-transfer catalysts.
Organic & biomolecular chemistry, 2015, 13, 8812-8816
7154642 CIFC18 H25 N2 O7 P S2P 21 21 216.3711; 12.1422; 27.2294
90; 90; 90
2106.44Jastrzębska, Katarzyna; Maciaszek, Anna; Dolot, Rafał; Bujacz, Grzegorz; Guga, Piotr
Thermal stability and conformation of antiparallel duplexes formed by P-stereodefined phosphorothioate DNA/LNA chimeric oligomers with DNA and RNA matrices.
Organic & biomolecular chemistry, 2015, 13, 10032-10040
7154700 CIFC20 H16 O2 SP 21 21 217.467; 13.272; 16.898
90; 90; 90
1674.6Boufroura, H.; Souibgui, A.; Gaucher, A.; Marrot, J.; Pieters, G.; Aloui, F.; Ben Hassine, B.; Clavier, G.; Prim, D.
3D shapes of aryl(dihydro)naphthothiophenes: a comprehensive and structural study.
Organic & biomolecular chemistry, 2015, 13, 10844-10851
7154725 CIFC18 H23 N O2P 21 21 215.2823; 10.763; 27.6349
90; 90; 90
1571.14Luo, Lan; Yamamoto, Hisashi
Synthesis of virtually enantiopure aminodiols with three adjacent stereogenic centers by epoxidation and ring-opening.
Organic & biomolecular chemistry, 2015, 13, 10466-10470
7154730 CIFC17 H19 N3 O5P 21 21 217.0673; 14.647; 15.48
90; 90; 90
1602.4Disetti, Paolo; Moccia, Maria; Salazar Illera, Diana; Suresh, Surisetti; Adamo, Mauro F. A.
Catalytic enantioselective addition of isocyanoacetate to 3-methyl-4-nitro-5-styrylisoxazoles under phase transfer catalysis conditions.
Organic & biomolecular chemistry, 2015, 13, 10609-10612
7154735 CIFC17 H23 N O9P 21 21 219.123; 14.399; 15.26
90; 90; 90
2004.6Thomas, Baptiste; Pifferi, Carlo; Daskhan, Gour Chand; Fiore, Michele; Berthet, Nathalie; Renaudet, Olivier
Divergent and convergent synthesis of GalNAc-conjugated dendrimers using dual orthogonal ligations.
Organic & biomolecular chemistry, 2015, 13, 11529-11538
7154739 CIFC24 H18 Cl N3 O3 SP 21 21 219.398; 9.776; 24.059
90; 90; 90
2210.4Bakthadoss, Manickam; Vinayagam, Varathan
A novel protocol for the facile construction of tetrahydroquinoline fused tricyclic frameworks via an intramolecular 1,3-dipolar nitrile oxide cycloaddition reaction.
Organic & biomolecular chemistry, 2015, 13, 10007-10014
7154754 CIFC27 H24 F3 N O4 SP 21 21 218.8259; 14.64; 19.755
90; 90; 90
2552.6Zhao, Yingying; Wang, Haolong; Li, Xincheng; Wang, Dongping; Xin, Xiaoyi; Wan, Boshun
Selective synthesis of functionalized pyrroles from 3-aza-1,5-enynes.
Organic & biomolecular chemistry, 2015, 14, 526-541
7154773 CIFC11 H19 N O6P 21 21 215.206; 14.978; 16.033
90; 90; 90
1250.2Johnson, Sherida; Tanaka, Fujie
Direct synthesis of C-glycosides from unprotected 2-N-acyl-aldohexoses via aldol condensation-oxa-Michael reactions with unactivated ketones.
Organic & biomolecular chemistry, 2016, 14, 259-264
7154782 CIFC104 H102 Cl8 N6 O4P 21 21 2114.177; 21.094; 32.557
90; 90; 90
9736Janiak, Agnieszka; Petryk, Małgorzata; Barbour, Leonard J.; Kwit, Marcin
Readily prepared inclusion forming chiral calixsalens.
Organic & biomolecular chemistry, 2015, 14, 669-673
7154783 CIFC100.5 H92.25 N6.75 O3P 21 21 2115.145; 21.42; 25.216
90; 90; 90
8180.2Janiak, Agnieszka; Petryk, Małgorzata; Barbour, Leonard J.; Kwit, Marcin
Readily prepared inclusion forming chiral calixsalens.
Organic & biomolecular chemistry, 2015, 14, 669-673
7154789 CIFC14 H24 F2 O2P 21 21 215.3073; 10.169; 26.061
90; 90; 90
1406.5Corr, Michael J.; Cormanich, Rodrigo A.; von Hahmann, Cortney N.; Bühl, Michael; Cordes, David B.; Slawin, Alexandra M. Z.; O'Hagan, David
Fluorine in fragrances: exploring the difluoromethylene (CF2) group as a conformational constraint in macrocyclic musk lactones.
Organic & biomolecular chemistry, 2016, 14, 211-219
7154800 CIFC23 H22 N2P 21 21 216.9535; 8.5937; 30.8423
90; 90; 90
1843.02Kim, Byeong Hyo; Bae, Seolhee; Go, Ahra; Lee, Hyunseung; Gong, Cheoloh; Lee, Byung Min
Synthesis of two distinct pyrrole moiety-containing arenes from nitroanilines using Paal-Knorr followed by an indium-mediated reaction.
Organic & biomolecular chemistry, 2015, 14, 265-276
7154801 CIFC10 H20 Cl N O3P 21 21 216.82581; 12.0234; 14.6468
90; 90; 90
1202.06Malinowski, Maciej; Rowicki, Tomasz; Guzik, Patrycja; Gryszel, Maciej; Łapczyński, Sebastian; Wielechowska, Monika; Czerwińska, Karolina; Madura, Izabela; Sas, Wojciech
[1,4]-sigmatropic rearrangement of chiral nitrones and their utilization in the synthesis of new iminosugars.
Organic & biomolecular chemistry, 2015, 14, 470-482
7154802 CIFC23 H43 N O7 SiP 21 21 217.96665; 10.06647; 31.833
90; 90; 90
2552.88Malinowski, Maciej; Rowicki, Tomasz; Guzik, Patrycja; Gryszel, Maciej; Łapczyński, Sebastian; Wielechowska, Monika; Czerwińska, Karolina; Madura, Izabela; Sas, Wojciech
[1,4]-sigmatropic rearrangement of chiral nitrones and their utilization in the synthesis of new iminosugars.
Organic & biomolecular chemistry, 2015, 14, 470-482
7154803 CIFC19 H24 N2 O8P 21 21 217.824; 13.359; 20.5454
90; 90; 90
2147.42Suresh Kumar, A.; Prabhakar Reddy, T.; Madhavachary, R.; Ramachary, Dhevalapally B.
Rawal's catalyst as an effective stimulant for the highly asymmetric Michael addition of β-keto esters to functionally rich nitro-olefins.
Organic & biomolecular chemistry, 2016, 14, 5494-5499
7154815 CIFC15 H16 N4 O4 SP 21 21 215.8334; 10.9763; 24.922
90; 90; 90
1595.7Simlandy, Amit K.; Mukherjee, Santanu
Catalytic asymmetric formal γ-allylation of deconjugated butenolides.
Organic & biomolecular chemistry, 2016, 14, 5659-5664
7154832 CIFC25 H28 F4 N2 O3P 21 21 219.768; 10.296; 22.978
90; 90; 90
2310.9Bykova, Tetiana; Al-Maharik, Nawaf; Slawin, Alexandra M. Z.; O'Hagan, David
Multicomponent reactions of methyl substituted all-cis tetrafluorocyclohexane aldehydes.
Organic & biomolecular chemistry, 2016, 14, 1117-1123
7154843 CIFC20 H25 N O2P 21 21 2111.71049; 11.80555; 52.7036
90; 90; 90
7286.21Wu, Shaotong; Yin, Qianqian; Zhao, Liang; Fan, Ningning; Tang, Xiaowan; Zhao, Jianxiong; Sheng, Tao; Guo, Ying; Tian, Chao; Zhang, Zhili; Xu, Weisi; Liu, Zhenming; Jiang, Shibo; Ma, Liying; Liu, Junyi; Wang, Xiaowei
A stereo configuration-activity study of 3-iodo-4-(2-methylcyclohexyloxy)-6-phenethylpyridin-2(2H)-ones as potency inhibitors of HIV-1 variants.
Organic & biomolecular chemistry, 2016, 14, 1413-1420
7154848 CIFC28 H38 O11P 21 21 2110.0374; 12.6398; 21.0812
90; 90; 90
2674.59An, Fa-Liang; Luo, Jun; Wang, Xiao-Bing; Yang, Ming-Hua; Kong, Ling-Yi
Trichiconlides A and B: two novel limonoids from the fruits of Trichilia connaroides.
Organic & biomolecular chemistry, 2016, 14, 1231-1235
7154855 CIFC20 H16 Br N O4P 21 21 219.7918; 10.8744; 17.136
90; 90; 90
1824.6Zhu, Ling; Yu, Chenxia; Li, Tuanjie; Wang, Yuhong; Lu, Yinan; Wang, Wenjing; Yao, Changsheng
N-Heterocyclic carbene-catalyzed [4 + 2] cyclization of α,β-unsaturated carboxylic acids bearing γ-H with isatins: an enantioselective synthesis of spirocyclic oxindole-dihydropyranones.
Organic & biomolecular chemistry, 2016, 14, 1485-1491
7154856 CIFC27 H46 O4P 21 21 216.8943; 11.6898; 32.2785
90; 90; 90
2601.42Kulesza, Urszula; Plum, Lori A.; DeLuca, Hector F.; Mouriño, Antonio; Sicinski, Rafal R.
A new suprasterol by photochemical reaction of 1α,25-dihydroxy-9-methylene-19-norvitamin D3.
Organic & biomolecular chemistry, 2016, 14, 1646-1652
7154873 CIFC50 H68 N12 O15 S2P 21 21 2115.515; 17.783; 22.102
90; 90; 90
6098Hattori, Kozo; Koike, Kota; Okuda, Kensuke; Hirayama, Tasuku; Ebihara, Masahiro; Takenaka, Mei; Nagasawa, Hideko
Solution-phase synthesis and biological evaluation of triostin A and its analogues.
Organic & biomolecular chemistry, 2016, 14, 2090-2111
7154894 CIFC11 H12 O3P 21 21 214.7902; 12.6722; 16.8843
90; 90; 90
1024.92Rast, Slavko; Modec, Barbara; Stephan, Michel; Mohar, Barbara
γ-Sultam-cored N,N-ligands in the ruthenium(ii)-catalyzed asymmetric transfer hydrogenation of aryl ketones.
Organic & biomolecular chemistry, 2016, 14, 2112-2120
7154902 CIFC30 H24 N2 OP 21 21 215.8608; 13.688; 27.498
90; 90; 90
2206De Los Santos, Zeus A.; Ding, Ransheng; Wolf, Christian
Quantitative chirality sensing of amines and amino alcohols via Schiff base formation with a stereodynamic UV/CD probe.
Organic & biomolecular chemistry, 2016, 14, 1934-1939
7154913 CIFC19.35 H24.7 N2 O8P 21 21 217.1213; 8.9288; 29.9909
90; 90; 90
1906.96Giacometti, Robert D.; Salinas, Juan C.; Østergaard, Michael E; Swayze, Eric E.; Seth, Punit P.; Hanessian, Stephen
Design, synthesis, and duplex-stabilizing properties of conformationally constrained tricyclic analogues of LNA.
Organic & biomolecular chemistry, 2016, 14, 2034-2040
7154917 CIFC14 H11 Br O S2P 21 21 215.9198; 8.4943; 26.9054
90; 90; 90
1352.93Yu, Jin-Sheng; Wu, Wen-Biao; Zhou, Feng
The first catalytic asymmetric thioacetalization by chiral phosphoric acid catalysis.
Organic & biomolecular chemistry, 2016, 14, 2205-2209
7154921 CIFC16 H20 I N O5P 21 21 216.4983; 10.457; 27.274
90; 90; 90
1853.3Forbes, Christina R.; Pandey, Anil K.; Ganguly, Himal K.; Yap, Glenn P. A.; Zondlo, Neal J.
4R- and 4S-iodophenyl hydroxyproline, 4R-pentynoyl hydroxyproline, and S-propargyl-4-thiolphenylalanine: conformationally biased and tunable amino acids for bioorthogonal reactions.
Organic & biomolecular chemistry, 2016, 14, 2327-2346
7154924 CIFC28 H27 N O5 SP 21 21 219.9601; 10.8355; 23.6278
90; 90; 90
2550Li, Ji-Yao; Li, Zhi-Long; Zhao, Wei-Wei; Liu, Yan-Kai; Tong, Zhi-Ping; Tan, Rui
One-pot, highly efficient, asymmetric synthesis of ring-fused piperidine derivatives bearing N,O- or N,N-acetal moieties.
Organic & biomolecular chemistry, 2016, 14, 2444-2453
7154925 CIFC28 H31 N O5 SP 21 21 2110.0985; 14.8716; 17.4835
90; 90; 90
2625.7Li, Ji-Yao; Li, Zhi-Long; Zhao, Wei-Wei; Liu, Yan-Kai; Tong, Zhi-Ping; Tan, Rui
One-pot, highly efficient, asymmetric synthesis of ring-fused piperidine derivatives bearing N,O- or N,N-acetal moieties.
Organic & biomolecular chemistry, 2016, 14, 2444-2453
7154926 CIFC20 H22 N2 OP 21 21 216.3758; 10.5378; 23.8709
90; 90; 90
1603.81Xu, Xin; Chen, Jingchao; He, Zhenxiu; Zhou, Yongyun; Fan, Baomin
Rhodium-catalyzed asymmetric ring opening reaction of oxabenzonorbornadienes with amines using ZnI2 as the activator.
Organic & biomolecular chemistry, 2016, 14, 2480-2486
7154936 CIFC20 H27 Cl F6 N4 P RhP 21 21 217.7291; 15.0891; 21.358
90; 90; 90
2490.9Zhao, Shixian; Wu, Feifei; Ma, Yuyu; Chen, Wanzhi; Liu, Miaochang; Wu, Huayue
Enhancement of N-heterocyclic carbenes on rhodium catalyzed olefination of triazoles.
Organic & biomolecular chemistry, 2016, 14, 2550-2555
7154946 CIFC43 H49 N3 O4P 21 21 2112.5755; 16.641; 17.7068
90; 90; 90
3705.5Khanvilkar, Aditya N.; Bedekar, Ashutosh V.
Synthesis and characterization of chiral aza-macrocycles and study of their enantiomer recognition ability for organo-phosphoric acid and phosphonic acid derivatives by (31)P NMR and fluorescence spectroscopy.
Organic & biomolecular chemistry, 2016, 14, 2742-2748
7154947 CIFC43 H49 N3 O4P 21 21 2112.8516; 13.959; 21.1978
90; 90; 90
3802.79Khanvilkar, Aditya N.; Bedekar, Ashutosh V.
Synthesis and characterization of chiral aza-macrocycles and study of their enantiomer recognition ability for organo-phosphoric acid and phosphonic acid derivatives by (31)P NMR and fluorescence spectroscopy.
Organic & biomolecular chemistry, 2016, 14, 2742-2748
7154950 CIFC15 H14 O3 SP 21 21 215.4884; 11.4294; 19.5736
90; 90; 90
1227.83Boyd, Derek R.; Sharma, Narain D.; Malone, John F.; Ljubez, Vera; Murphy, Deirdre; Shepherd, Steven D.; Allen, Christopher C. R.
Chemoenzymatic synthesis of enantiopure hydroxy sulfoxides derived from substituted arenes.
Organic & biomolecular chemistry, 2016, 14, 2651-2664
7154951 CIFC15 H14 O3 SP 21 21 217.292; 11.75; 14.698
90; 90; 90
1259.3Boyd, Derek R.; Sharma, Narain D.; Malone, John F.; Ljubez, Vera; Murphy, Deirdre; Shepherd, Steven D.; Allen, Christopher C. R.
Chemoenzymatic synthesis of enantiopure hydroxy sulfoxides derived from substituted arenes.
Organic & biomolecular chemistry, 2016, 14, 2651-2664
7154952 CIFC12 H12 O3 SP 21 21 218.108; 11.284; 24.513
90; 90; 90
2242.7Boyd, Derek R.; Sharma, Narain D.; Malone, John F.; Ljubez, Vera; Murphy, Deirdre; Shepherd, Steven D.; Allen, Christopher C. R.
Chemoenzymatic synthesis of enantiopure hydroxy sulfoxides derived from substituted arenes.
Organic & biomolecular chemistry, 2016, 14, 2651-2664
7154968 CIFC29 H35 F N2 O5P 21 21 219.7463; 11.9704; 24.3772
90; 90; 90
2844Marques, A.-S.; Giardinetti, M.; Marrot, J.; Coeffard, V.; Moreau, X.; Greck, C.
Construction of enantioenriched polysubstituted hexahydropyridazines via a sequential multicatalytic process merging palladium catalysis and aminocatalysis.
Organic & biomolecular chemistry, 2016, 14, 2828-2832
7154980 CIFC17 H14 O6 SP 21 21 218.5357; 12.3308; 14.9954
90; 90; 90
1578.3Cornaggia, Claudio; Gundala, Sivaji; Manoni, Francesco; Gopalasetty, Nagaraju; Connon, Stephen J.
Catalytic formal cycloadditions between anhydrides and ketones: excellent enantio and diastereocontrol, controllable decarboxylation and the formation of adjacent quaternary stereocentres.
Organic & biomolecular chemistry, 2016, 14, 3040-3046
7154991 CIFC21 H16 O2 SP 21 21 2110.2816; 10.436; 15.0467
90; 90; 90
1614.49Wong, Yuk Fai; Wang, Zhaobin; Sun, Jianwei
Chiral phosphoric acid catalyzed asymmetric addition of naphthols to para-quinone methides.
Organic & biomolecular chemistry, 2016, 14, 5751-5754
7154995 CIFC18 H17 N O5 SP 21 21 218.2474; 11.1326; 18.0136
90; 90; 90
1653.92Luridiana, Alberto; Frongia, Angelo; Aitken, David J.; Guillot, Regis; Sarais, Giorgia; Secci, Francesco
Deracemizing organocatalyzed Michael addition reactions of 2-(arylthio)cyclobutanones with β-nitrostyrenes.
Organic & biomolecular chemistry, 2016, 14, 3394-3403
7155017 CIFC15 H11 F4 N O3P 21 21 218.7967; 9.2428; 17.2636
90; 90; 90
1403.64Liu, Wei; Lai, Xiaoyan; Zha, Gaofeng; Xu, Yan; Sun, Panpan; Xia, Tao; Shen, Yongcun
The squaramide-catalyzed asymmetric Michael/cyclization tandem reaction for the synthesis of chiral trifluoromethylated hydroxyimino tetrahydrobenzofuranones.
Organic & biomolecular chemistry, 2016, 14, 3603-3607
7155018 CIFC11 H13 N5 O4P 21 21 217.4773; 8.2931; 20.419
90; 90; 90
1266.2Zhang, Hu; Liu, Peng-Fei; Chen, Qiong; Wu, Qiong-You; Seville, Anne; Gu, Yu-Cheng; Clough, John; Zhou, Shao-Lin; Yang, Guang-Fu
Synthesis and absolute configuration assignment of albucidin: a late-stage reductive deiodination by visible light photocatalysis.
Organic & biomolecular chemistry, 2016, 14, 3482-3485
7155032 CIFC31 H32 N O3 RhP 21 21 219.7915; 10.0496; 33.148
90; 90; 90
3261.8Zhao, Yi-Shuang; Liu, Jian-Kang; He, Zhi-Tao; Tao, Jing-Chao; Tian, Ping; Lin, Guo-Qiang
Two phenyls are better than one or three: synthesis and application of terminal olefin-oxazoline (TOlefOx) ligands.
Organic & biomolecular chemistry, 2016, 14, 3686-3689
7155033 CIFC37 H36 N O3 RhP 21 21 2110.8993; 13.2135; 21.2588
90; 90; 90
3061.6Zhao, Yi-Shuang; Liu, Jian-Kang; He, Zhi-Tao; Tao, Jing-Chao; Tian, Ping; Lin, Guo-Qiang
Two phenyls are better than one or three: synthesis and application of terminal olefin-oxazoline (TOlefOx) ligands.
Organic & biomolecular chemistry, 2016, 14, 3686-3689
7155041 CIFC15 H16 Al Br O2 SP 21 21 218.0842; 12.4461; 16.7654
90; 90; 90
1686.88Tang, Yani; Sun, Yuji; Liu, Jiyong; Duttwyler, Simon
Facile synthesis of enantioenriched phenol-sulfoxides and their aluminum complexes.
Organic & biomolecular chemistry, 2016, 14, 5580-5585
7155044 CIFC13 H11 Br O2 SP 21 21 219.1301; 10.89; 13.3698
90; 90; 90
1329.32Tang, Yani; Sun, Yuji; Liu, Jiyong; Duttwyler, Simon
Facile synthesis of enantioenriched phenol-sulfoxides and their aluminum complexes.
Organic & biomolecular chemistry, 2016, 14, 5580-5585
7155050 CIFC19 H19 N O2 S2P 21 21 2110.846; 11.5153; 14.8533
90; 90; 90
1855.1Wu, Shanchao; Li, Yu; Zhang, Yongqiang; Fang, Kun; Dong, Guoqiang; Liu, Na; Miao, Zhenyuan; Yao, Jianzhong; Wang, Wei; Zhang, Wannian; Sheng, Chunquan
Enantioselective organocatalytic Michael addition of isorhodanines to α,β-unsaturated aldehydes.
Organic & biomolecular chemistry, 2016, 14, 3926-3933
7155055 CIFC20 H19 Cl N2 OP 21 21 216.684; 11.847; 22.594
90; 90; 90
1789.1Kuznetsov, N. Yu; Tikhov, R. M.; Godovikov, I. A.; Khrustalev, V. N.; Bubnov, Yu N.
New enolate-carbodiimide rearrangement in the concise synthesis of 6-amino-2,3-dihydro-4-pyridinones from homoallylamines.
Organic & biomolecular chemistry, 2016, 14, 4283-4298
7155061 CIFC16 H18 N2 O3P 21 21 215.7178; 10.4187; 24.9522
90; 90; 90
1486.45Sontakke, Vyankat A.; Lawande, Pravin P.; Kate, Anup N.; Khan, Ayesha; Joshi, Rakesh; Kumbhar, Anupa A.; Shinde, Vaishali S.
Antiproliferative activity of bicyclic benzimidazole nucleosides: synthesis, DNA-binding and cell cycle analysis.
Organic & biomolecular chemistry, 2016, 14, 4136-4145
7155078 CIFC38 H34 B2 N4 O6P 21 21 2111.3239; 12.888; 25.7528
90; 90; 90
3758.4Liu, Bowen; Novikova, Nina; Simpson, M. Cather; Timmer, Mattie S. M.; Stocker, Bridget L.; Söhnel, Tilo; Ware, David C.; Brothers, Penelope J.
Lighting up sugars: fluorescent BODIPY-gluco-furanose and -septanose conjugates linked by direct B-O-C bonds.
Organic & biomolecular chemistry, 2016, 14, 5205-5209
7155080 CIFC14 H19 N O6P 21 21 215.6525; 7.679; 32.488
90; 90; 90
1410.2Qian, Bao-Chen; Kamori, Akiko; Kinami, Kyoko; Kato, Atsushi; Li, Yi-Xian; Fleet, George W. J.; Yu, Chu-Yi
Epimerization of C5 of an N-hydroxypyrrolidine in the synthesis of swainsonine related iminosugars.
Organic & biomolecular chemistry, 2016, 14, 4488-4498
7155081 CIFC9 H13 N O6 SP 21 21 215.5868; 6.1938; 31.33
90; 90; 90
1084.13Wuttke, André; Fischer, Sebastian Nils; Nebel, Annika; Marsch, Michael; Geyer, Armin
Improved δ-valerolactam templates for the assembly of Aβ-miniamyloids by boronic ester formation.
Organic & biomolecular chemistry, 2016, 14, 5032-5048
7155084 CIFC9 H12 N4 O5 SP 21 21 216.2462; 9.5487; 20.1585
90; 90; 90
1202.32Wuttke, André; Fischer, Sebastian Nils; Nebel, Annika; Marsch, Michael; Geyer, Armin
Improved δ-valerolactam templates for the assembly of Aβ-miniamyloids by boronic ester formation.
Organic & biomolecular chemistry, 2016, 14, 5032-5048
7155085 CIFC17 H19 B N2 O7 SP 21 21 216.4782; 9.8389; 28.471
90; 90; 90
1814.69Wuttke, André; Fischer, Sebastian Nils; Nebel, Annika; Marsch, Michael; Geyer, Armin
Improved δ-valerolactam templates for the assembly of Aβ-miniamyloids by boronic ester formation.
Organic & biomolecular chemistry, 2016, 14, 5032-5048
7155086 CIFC20 H32 O4P 21 21 2111.8465; 23.7593; 6.5189
90; 90; 90
1834.84Xiong, Juan; Hong, Zhi-Lai; Xu, Peng; Zou, Yike; Yu, Shang-Bo; Yang, Guo-Xun; Hu, Jin-Feng
ent-Abietane diterpenoids with anti-neuroinflammatory activity from the rare Chloranthaceae plant Chloranthus oldhamii.
Organic & biomolecular chemistry, 2016, 14, 4678-4689
7155090 CIFC13 H14 N4 O5P 21 21 216.4456; 9.8102; 21.821
90; 90; 90
1379.8Bag, Subhendu Sekhar; Talukdar, Sangita; Das, Suman Kalyan; Pradhan, Manoj Kumar; Mukherjee, Soumen
Donor/acceptor chromophores-decorated triazolyl unnatural nucleosides: synthesis, photophysical properties and study of interaction with BSA.
Organic & biomolecular chemistry, 2016, 14, 5088-5108
7155105 CIFC27 H20 O4P 21 21 2110.0372; 13.0997; 15.0079
90; 90; 90
1973.3Han, Xiaoyu; Ni, Huanzhen; Chan, Wai-Lun; Gai, Xikun; Wang, Yongjiang; Lu, Yixin
Highly enantioselective synthesis of dihydrocoumarin-fused dihydropyrans via the phosphine-catalyzed [4 + 2] annulation of allenones with 3-aroylcoumarins.
Organic & biomolecular chemistry, 2016, 14, 5059-5064
7155107 CIFC14 H11 I N2P 21 21 218.2657; 14.1996; 21.2896
90; 90; 90
2498.75Samanta, Sadhanendu; Jana, Sourav; Mondal, Susmita; Monir, Kamarul; Chandra, Swapan K.; Hajra, Alakananda
Switching the regioselectivity in the copper-catalyzed synthesis of iodoimidazo[1,2-a]pyridines.
Organic & biomolecular chemistry, 2016, 14, 5073-5078
7155123 CIFC18 H16 O SP 21 21 215.7389; 11.4338; 22.2456
90; 90; 90
1459.7Fu, Xuan; Lin, Lili; Xia, Yong; Zhou, Pengfei; Liu, Xiaohua; Feng, Xiaoming
Catalytic asymmetric [3 + 3] annulation of cyclopropanes with mercaptoacetaldehyde.
Organic & biomolecular chemistry, 2016, 14, 5914-5917
7155124 CIFC17 H21 N O5 SP 21 21 217.5608; 13.1579; 16.9471
90; 90; 90
1686Fu, Jian-Guo; Shan, Yi-Fan; Sun, Wang-Bin; Lin, Guo-Qiang; Sun, Bing-Feng
An asymmetric approach to bicyclo[2.2.1]heptane-1-carboxylates via a formal [4 + 2] cycloaddition reaction enabled by organocatalysis.
Organic & biomolecular chemistry, 2016, 14, 5229-5232
7155129 CIFC11 H12 N2 O3P 21 21 215.4617; 8.2109; 23.4585
90; 90; 90
1052.01You, Zhi-Hao; Chen, Ying-Han; Liu, Yan-Kai
From racemic precursors to fully stereocontrolled products: one-pot synthesis of chiral α-amino lactones and lactams.
Organic & biomolecular chemistry, 2016, 14, 6316-6327
7155147 CIFC17 H26 F N O3 SP 21 21 219.6078; 18.11; 21.537
90; 90; 90
3747.4Li, Xiang; Li, Ya; Shang, Huaqi
A diastereoselective Mannich-type reaction of α-fluorinated carboxylate esters: synthesis of β-amino acids containing α-quaternary fluorinated carbon centers.
Organic & biomolecular chemistry, 2016, 14, 6457-6462
7155149 CIFC24 H15 Cl O3P 21 21 2110.5258; 11.7582; 14.4254
90; 90; 90
1785.4Jiang, Yu; Fu, Jun-Hao; Li, Tian-Ze; Sha, Feng; Wu, Xin-Yan
Enantioselective direct vinylogous aldol-cyclization cascade reaction between β,γ-unsaturated amides and o-quinones.
Organic & biomolecular chemistry, 2016, 14, 6435-6441
7155153 CIFC21 H22 N2 O4 SP 21 21 218.291; 10.918; 22.462
90; 90; 90
2033.3Wang, Zhen-Hua; Wu, Zhi-Jun; Yue, Deng-Feng; You, Yong; Xu, Xiao-Ying; Zhang, Xiao-Mei; Yuan, Wei-Cheng
Enantioselective synthesis of chiral α,β-unsaturated γ-substituted butyrolactams by organocatalyzed direct asymmetric vinylogous Michael addition of α,β-unsaturated γ-butyrolactam to 2-enoylpyridines.
Organic & biomolecular chemistry, 2016, 14, 6568-6576
7155155 CIFC24 H19 N O3 SP 21 21 2111.908; 12.416; 13.154
90; 90; 90
1944.8Liang, Zhi-Qin; Wang, Dong-Ling; Zhang, Chun-Lin; Ye, Song
Enantioselective N-heterocyclic carbene-catalyzed synthesis of saccharine-derived dihydropyridinones with cis-selectivity.
Organic & biomolecular chemistry, 2016, 14, 6422-6425
7155157 CIFC24 H20 N4 O2 SP 21 21 214.9002; 16.6369; 25.4887
90; 90; 90
2077.9Wang, Yanxin J.; Szantai-Kis, D Miklos; Petersson, E. James
Chemoselective modifications for the traceless ligation of thioamide-containing peptides and proteins.
Organic & biomolecular chemistry, 2016, 14, 6262-6269
7155159 CIFC15 H24 O2P 21 21 217.49844; 10.97341; 16.2847
90; 90; 90
1339.96Huang, David; Schuppe, Alexander W.; Liang, Michael Z.; Newhouse, Timothy R.
Scalable procedure for the fragmentation of hydroperoxides mediated by copper and iron tetrafluoroborate salts.
Organic & biomolecular chemistry, 2016, 14, 6197-6200
7155169 CIFC17 H16 F3 N SP 21 21 219.8932; 15.009; 21.27
90; 90; 90
3158.3Zhou, Ji; Zhang, Qian-Fan; Zhao, Wei-Hao; Jiang, Guo-Fang
Chiral phosphoric acid-catalyzed asymmetric transfer hydrogenation of 3-trifluoromethylthioquinolines.
Organic & biomolecular chemistry, 2016, 14, 6937-6941
7155170 CIFC24 H20 N2 O2P 21 21 217.6135; 13.282; 18.5374
90; 90; 90
1874.5He, Liwenze; Liu, Lin; Han, Runfeng; Zhang, Weiwei; Xie, Xingang; She, Xuegong
Thermal 1,3-dipolar cycloaddition reaction of azomethine imines with active esters.
Organic & biomolecular chemistry, 2016, 14, 6757-6761
7155171 CIFC11 H16 O S2P 21 21 218.4952; 9.1213; 14.963
90; 90; 90
1159.44Diebler, J.; Spannenberg, A.; Werner, T.
Atom economical synthesis of di- and trithiocarbonates by the lithium tert-butoxide catalyzed addition of carbon disulfide to epoxides and thiiranes.
Organic & biomolecular chemistry, 2016, 14, 7480-7489
7155194 CIFC18 H12 Cl F O3P 21 21 217.958; 9.449; 19.866
90; 90; 90
1493.8Sha, Wanxing; Zhang, Lijun; Zhang, Wenzhong; Mei, Haibo; Soloshonok, Vadim A.; Han, Jianlin; Pan, Yi
Catalytic cascade aldol-cyclization of tertiary ketone enolates for enantioselective synthesis of keto-esters with a C-F quaternary stereogenic center.
Organic & biomolecular chemistry, 2016, 14, 7295-7303
7155196 CIFC30 H46 O3P 21 21 2111.82201; 19.9887; 23.1114
90; 90; 90
5461.38Liu, Hong-Xin; Chen, Kai; Yuan, Yao; Xu, Zhi-Fang; Tan, Hai-Bo; Qiu, Sheng-Xiang
Rhodomentones A and B, novel meroterpenoids with unique NMR characteristics from Rhodomyrtus tomentosa.
Organic & biomolecular chemistry, 2016, 14, 7354-7360
7155198 CIFC38 H40 N PP 21 21 2110.5138; 14.5405; 19.6851
90; 90; 90
3009.38Mino, Takashi; Nishikawa, Kenji; Asano, Moeko; Shima, Yamato; Ebisawa, Toshibumi; Yoshida, Yasushi; Sakamoto, Masami
Chiral N-1-adamantyl-N-trans-cinnamylaniline type ligands: synthesis and application to palladium-catalyzed asymmetric allylic alkylation of indoles.
Organic & biomolecular chemistry, 2016, 14, 7509-7519
7155199 CIFC41 H40 N PP 21 21 2110.6196; 22.1572; 26.8016
90; 90; 90
6306.43Mino, Takashi; Nishikawa, Kenji; Asano, Moeko; Shima, Yamato; Ebisawa, Toshibumi; Yoshida, Yasushi; Sakamoto, Masami
Chiral N-1-adamantyl-N-trans-cinnamylaniline type ligands: synthesis and application to palladium-catalyzed asymmetric allylic alkylation of indoles.
Organic & biomolecular chemistry, 2016, 14, 7509-7519
7155200 CIFC41 H42 N PP 21 21 2110.5997; 14.5202; 21.027
90; 90; 90
3236.26Mino, Takashi; Nishikawa, Kenji; Asano, Moeko; Shima, Yamato; Ebisawa, Toshibumi; Yoshida, Yasushi; Sakamoto, Masami
Chiral N-1-adamantyl-N-trans-cinnamylaniline type ligands: synthesis and application to palladium-catalyzed asymmetric allylic alkylation of indoles.
Organic & biomolecular chemistry, 2016, 14, 7509-7519
7155202 CIFC21 H22 O3P 21 21 219.2519; 9.9263; 18.4119
90; 90; 90
1690.9Barrios Antúnez, Diego-Javier; Greenhalgh, Mark D.; Fallan, Charlene; Slawin, Alexandra M. Z.; Smith, Andrew D.
Enantioselective synthesis of 2,3-disubstituted trans-2,3-dihydrobenzofurans using a Brønsted base/thiourea bifunctional catalyst.
Organic & biomolecular chemistry, 2016, 14, 7268-7274
7155211 CIFC17 H16 Br N O3P 21 21 217.5275; 13.374; 15.278
90; 90; 90
1538.1Stark, Daniel G.; Williamson, Patrick; Gayner, Emma R.; Musolino, Stefania F.; Kerr, Ryan W. F.; Taylor, James E.; Slawin, Alexandra M. Z.; O'Riordan, Timothy J C; Macgregor, Stuart A.; Smith, Andrew D.
Isothiourea-catalysed enantioselective pyrrolizine synthesis: synthetic and computational studies.
Organic & biomolecular chemistry, 2016, 14, 8957-8965
7155212 CIFC16 H15 Cl N4 OP 21 21 218.0275; 11.093; 17.321
90; 90; 90
1542.4Chen, Long; Xing, Haotian; Zhang, Huaibin; Jiang, Zhong-Xing; Yang, Zhigang
Copper-catalyzed intermolecular chloroazidation of α,β-unsaturated amides.
Organic & biomolecular chemistry, 2016, 14, 7463-7467
7155219 CIFC9 H10 Br Cl OP 21 21 215.3545; 11.656; 15.876
90; 90; 90
990.9Huang, Wei-Sheng; Chen, Li; Zheng, Zhan-Jiang; Yang, Ke-Fang; Xu, Zheng; Cui, Yu-Ming; Xu, Li-Wen
Catalytic asymmetric bromochlorination of aromatic allylic alcohols promoted by multifunctional Schiff base ligands.
Organic & biomolecular chemistry, 2016, 14, 7927-7932
7155223 CIFC33 H48 Cl N O4 S SnP 21 21 219.403; 10.4777; 36.3472
90; 90; 90
3581Kamimura, Akio; Tanaka, Toshiyuki; So, Masahiro; Itaya, Tomoyuki; Matsuda, Kantaro; Kawamoto, Takuji
A regioselective double Stille coupling reaction of bicyclic stannolanes.
Organic & biomolecular chemistry, 2016, 14, 8109-8122
7155234 CIFC37 H42 N3 O3 PP 21 21 2114.6046; 18.958; 23.9068
90; 90; 90
6619.2Yang, Bing; Ji, Xiaozhou; Xue, Yunsheng; Zhang, Haowei; Shen, Minxing; Jiang, Bo; Li, Guigen
Asymmetric aza-Morita-Baylis-Hillman reactions of chiral N-phosphonyl imines with acrylates via GAP chemistry/technology.
Organic & biomolecular chemistry, 2016, 14, 6024-6035
7155237 CIFC20 H35 N O3P 21 21 216.7242; 15.1813; 19.2667
90; 90; 90
1966.79Philkhana, Satish Chandra; Mehrotra, Suneet; Murray, Thomas F.; Reddy, D. Srinivasa
Synthesis and biological evaluation of palmyrolide A macrocycles as sodium channel blockers towards neuroprotection.
Organic & biomolecular chemistry, 2016, 14, 8457-8473
7155239 CIFC21 H37 N O3P 21 21 215.615; 10.654; 35.955
90; 90; 90
2150.9Philkhana, Satish Chandra; Mehrotra, Suneet; Murray, Thomas F.; Reddy, D. Srinivasa
Synthesis and biological evaluation of palmyrolide A macrocycles as sodium channel blockers towards neuroprotection.
Organic & biomolecular chemistry, 2016, 14, 8457-8473
7155245 CIFC11 H8 O Se2P 21 21 214.6505; 13.4476; 16.1385
90; 90; 90
1009.27Mondal, Santanu; Mugesh, Govindasamy
Biomimetic deiodination of thyroid hormones and iodothyronamines - a structure-activity relationship study.
Organic & biomolecular chemistry, 2016, 14, 9490-9500
7155249 CIFC27 H44 N4 O9P 21 21 2110.4185; 15.6536; 18.156
90; 90; 90
2961Lee, Jaeyeon; Jang, Geunhyeok; Kang, Philjae; Choi, Moon-Gun; Choi, Soo Hyuk
Helical α/β-depsipeptides with alternating residue types: conformational change from the 11-helix to the 14/15-helix.
Organic & biomolecular chemistry, 2016, 14, 8438-8442
7155253 CIFC15 H20 Br N O4 SP 21 21 215.168; 10.0269; 32.073
90; 90; 90
1662Feng, Bo-Xu; Wang, Bin; Li, Xin
Asymmetric additions of thioglycolates and N-Boc aldimines catalyzed by a bifunctional tertiary-amine squaramide.
Organic & biomolecular chemistry, 2016, 14, 9206-9209
7155260 CIFC17 H28 O3P 21 21 214.672; 5.359; 67.02
90; 90; 90
1678Kuilya, Tapan Kumar; Goswami, Rajib Kumar
Total synthesis of cananginone C and structural revision of debilisone A.
Organic & biomolecular chemistry, 2016, 14, 8789-8799
7155267 CIFC13 H10 Cl F5 O SP 21 21 215.1495; 9.3429; 27.7278
90; 90; 90
1334.02Desroches, Justine; Tremblay, Ariane; Paquin, Jean-François
Racemic and enantioselective metal-catalyzed synthesis of SF5-containing diarylmethanols.
Organic & biomolecular chemistry, 2016, 14, 8764-8780
7155272 CIFC43 H31 B N4 O2P 21 21 219.4858; 16.647; 20.977
90; 90; 90
3312.5Brittain, William D. G.; Chapin, Brette M.; Zhai, Wenlei; Lynch, Vincent M.; Buckley, Benjamin R.; Anslyn, Eric V.; Fossey, John S.
The Bull-James assembly as a chiral auxiliary and shift reagent in kinetic resolution of alkyne amines by the CuAAC reaction.
Organic & biomolecular chemistry, 2016, 14, 10778-10782
7155290 CIFC25 H26 N2 O6 SP 21 21 217.4819; 12.1332; 25.226
90; 90; 90
2290Mondal, Pravat; Argade, Narshinha P.
Stereoselective synthesis of (-)-desethyleburnamonine, (-)-vindeburnol and (-)-3-epitacamonine: observation of a substrate dependent diastereoselectivity reversal of an aldol reaction.
Organic & biomolecular chemistry, 2016, 14, 10394-10406
7155291 CIFC25 H28 N2 O5 SP 21 21 219.0934; 10.9932; 25.0614
90; 90; 90
2505.3Mondal, Pravat; Argade, Narshinha P.
Stereoselective synthesis of (-)-desethyleburnamonine, (-)-vindeburnol and (-)-3-epitacamonine: observation of a substrate dependent diastereoselectivity reversal of an aldol reaction.
Organic & biomolecular chemistry, 2016, 14, 10394-10406
7155298 CIFC24 H23 N2 O3 PP 21 21 2110.0376; 11.6437; 18.2329
90; 90; 90
2130.97Lin, Shaoquan; Kumagai, Naoya; Shibasaki, Masakatsu
Enantioselective synthesis of α,α-disubstituted α-amino acids via direct catalytic asymmetric addition of acetonitrile to α-iminoesters.
Organic & biomolecular chemistry, 2016, 14, 9725-9730
7155308 CIFC31 H23 Cl3 N2 O3 SP 21 21 218.0194; 16.8849; 20.7855
90; 90; 90
2814.5Kayal, Satavisha; Mukherjee, Santanu
Catalytic enantioselective cascade Michael/cyclization reaction of 3-isothiocyanato oxindoles with exocyclic α,β-unsaturated ketones en route to 3,2'-pyrrolidinyl bispirooxindoles.
Organic & biomolecular chemistry, 2016, 14, 10175-10179
7155312 CIFC16 H13 Cl N2 OP 21 21 214.7439; 16.18; 18.262
90; 90; 90
1401.7Zhou, Hui; Deng, Xin Zhao; Zhang, Ai Hua; Tan, Ren Xiang
Visible-light-promoted synthesis of phenanthridines via an intermolecular isocyanide insertion reaction.
Organic & biomolecular chemistry, 2016, 14, 10407-10414
7155321 CIFC22 H19 Cl N O3P 21 21 217.367; 12.1881; 21.7372
90; 90; 90
1951.78Chi, Yongjian; Qiu, Lihua; Xu, Xinfang
Highly enantioselective synthesis of spirocyclopropyloxindoles via a Rh(ii)-catalyzed asymmetric cyclopropanation reaction.
Organic & biomolecular chemistry, 2016, 14, 10357-10361
7155322 CIFC21 H20 Cl N O3P 21 21 2111.3609; 11.3606; 14.5605
90; 90; 90
1879.27Chi, Yongjian; Qiu, Lihua; Xu, Xinfang
Highly enantioselective synthesis of spirocyclopropyloxindoles via a Rh(ii)-catalyzed asymmetric cyclopropanation reaction.
Organic & biomolecular chemistry, 2016, 14, 10357-10361
7155334 CIFC12 H8 F N3P 21 21 216.5842; 10.527; 14.581
90; 90; 90
1010.6Inturi, Surendra Babu; Kalita, Biswajit; Ahamed, A. Jafar
I2-TBHP-catalyzed one-pot highly efficient synthesis of 4,3-fused 1,2,4-triazoles from N-tosylhydrazones and aromatic N-heterocycles via intermolecular formal 1,3-dipolar cycloaddition.
Organic & biomolecular chemistry, 2016, 14, 11061-11064
7155337 CIFC21 H24 O5 SP 21 21 2110.2408; 11.0014; 17.5608
90; 90; 90
1978.5Wang, Xuan; Sun, Wangbin; Zou, Jian-Ping; lin, guoqiang; Sun, Bingfeng
Asymmetric Total Synthesis of Hedyosumin E aglycon, 7,10-Epoxyhedyosminolide and ent-Zedolactone A
Org. Biomol. Chem., 2016
7155339 CIFC40 H57 N15 O8.35 S5P 21 21 219.3172; 18.6791; 29.1423
90; 90; 90
5071.84Mungalpara, Disha; Kelm, Harald; Valkonen, Arto; Rissanen, Kari; Keller, Sandro; Kubik, Stefan
Oxoanion binding to a cyclic pseudopeptide containing 1,4-disubstituted 1,2,3-triazole moieties.
Organic & biomolecular chemistry, 2016, 15, 102-113
7155340 CIFC31 H36 N2 O6P 21 21 219.9835; 12.2707; 23.46
90; 90; 90
2874Tan, Yu; Feng, Er-Lu; Sun, Qiang-Sheng; Lin, Hua; Sun, Xun; Lin, Guo-Qiang; Sun, Xing-Wen
Enantioselective synthesis of spirooxindole benzoquinolizines via organo-catalyzed cascade reactions.
Organic & biomolecular chemistry, 2017, 15, 778-781
7155344 CIFC10 H18 O5P 21 21 215.3124; 7.0459; 29.215
90; 90; 90
1093.54Zhang, Chenxi; Wang, Chengcheng; Wang, Zihao; Tanabe, Genzoh; Muraoka, Osamu; Lin, Aijun; Xu, Jinyi; Wu, Xiaoming; Wu, Liang; Xie, Weijia
Total synthesis, structural elucidation and anti-inflammatory activity evaluation of 2-deoxy-3,6-anhydro hexofuranoside derivatives isolated from Sauropus rostratus.
Organic & biomolecular chemistry, 2016, 14, 10906-10913
7155349 CIFC32 H54 O4P 21 21 2112.104; 34.297; 7.195
90; 90; 90
2986.9Chen, Dongyin; Zhang, Pu; Sun, Yan; Wang, Pengfei; Zhang, Can; Kong, Lingyi; Zhang, Ji; Sun, Hongbin; Wen, Xiaoan
Protonated montmorillonite-mediated highly specific isomerization of oleanolic acid esters: application to the synthesis of Δ(13(18))-CDDO-Me.
Organic & biomolecular chemistry, 2016, 14, 11154-11161
7155359 CIFC28 H35 Br N2 O7 SP 21 21 219.05634; 11.2038; 30.5045
90; 90; 90
3095.15Chowdhury, Raghunath; Kumar, Mukesh; Ghosh, Sunil K.
Organocatalyzed enantioselective Michael addition/cyclization cascade reaction of 3-isothiocyanato oxindoles with arylidene malonates.
Organic & biomolecular chemistry, 2016, 14, 11250-11260
7155360 CIFC29 H46 O4 SiP 21 21 217.1072; 13.7421; 27.891
90; 90; 90
2724.1Dethe, Dattatraya H.; Dherange, Balu D.; Ali, Saghir; Parsutkar, Mahesh M.
Enantiospecific total syntheses of meroterpenoids (-)-F1839-I and (-)-corallidictyals B and D.
Organic & biomolecular chemistry, 2016, 15, 65-68
7155364 CIFC15 H14 Br N O2P 21 21 215.4842; 15.284; 16.885
90; 90; 90
1415.3Li, Ruikun; Wen, Zhongqing; Wu, Na
A nordehydroabietyl amide-containing chiral diene for rhodium-catalysed asymmetric arylation to nitroolefins.
Organic & biomolecular chemistry, 2016, 14, 11080-11084
7155376 CIFC14 H21 N O5P 21 21 217.4821; 13.9447; 14.9797
90; 90; 90
1562.92Zhang, Zhijiang; Liu, Bo
Total synthesis and confirmation of the revised structures of jiangrines A, C and D.
Organic & biomolecular chemistry, 2016, 15, 207-212
7155380 CIFC12 H24 O2P 21 21 216.3617; 10.0016; 20.4847
90; 90; 90
1303.38Roldán, Steven; Cardona, Adrià; Conesa, Laura; Murga, Juan; Falomir, Eva; Carda, Miguel; Marco, J. Alberto
Synthesis and biological evaluation of simplified pironetin analogues with modifications in the side chain and the lactone ring.
Organic & biomolecular chemistry, 2016, 15, 220-232
7155381 CIFC12 H24 O2P 21 21 216.35866; 9.99503; 20.4733
90; 90; 90
1301.18Roldán, Steven; Cardona, Adrià; Conesa, Laura; Murga, Juan; Falomir, Eva; Carda, Miguel; Marco, J. Alberto
Synthesis and biological evaluation of simplified pironetin analogues with modifications in the side chain and the lactone ring.
Organic & biomolecular chemistry, 2016, 15, 220-232
7155385 CIFC28.15 H54.38 O4 Si2P 21 21 2116.5936; 16.0072; 12.75162
90; 90; 90
3387.05Roldán, Steven; Cardona, Adrià; Conesa, Laura; Murga, Juan; Falomir, Eva; Carda, Miguel; Marco, J. Alberto
Synthesis and biological evaluation of simplified pironetin analogues with modifications in the side chain and the lactone ring.
Organic & biomolecular chemistry, 2016, 15, 220-232
7155398 CIFC11 H17 N5 O2P 21 21 2112.7749; 10.4901; 9.508
90; 90; 90
1274.2Van Mileghem, Seger; Egle, Brecht; Gilles, Philippe; Veryser, Cedrick; Van Meervelt, Luc; De Borggraeve, Wim M.
Carbonylation as a novel method for the assembly of pyrazine based oligoamide alpha-helix mimetics.
Organic & biomolecular chemistry, 2017, 15, 373-378
7155402 CIFC15 H11 N O4 SP 21 21 2110.8402; 10.9776; 11.4168
90; 90; 90
1358.6Wu, Hongxiang; Liu, Tingting; Cui, Ming; Li, Yue; Jian, Junsheng; Wang, Hui; Zeng, Zhuo
Rhodium-catalyzed C-H functionalization with N-acylsaccharins.
Organic & biomolecular chemistry, 2017, 15, 536-540
7155412 CIFC12 H19 N O3P 21 21 217.0321; 8.4501; 40.7561
90; 90; 90
2421.81Kubyshkin, Vladimir; Budisa, Nediljko
Construction of a polyproline structure with hydrophobic exterior using octahydroindole-2-carboxylic acid.
Organic & biomolecular chemistry, 2017, 15, 619-627
7155414 CIFC13 H23 N O4P 21 21 216.2188; 9.282; 25.561
90; 90; 90
1475.5Si, Chang-Mei; Shao, Lu-Ping; Mao, Zhuo-Ya; Zhou, Wen; Wei, Bang-Guo
An efficient approach to trans-4-hydroxy-5-substituted 2-pyrrolidinones through a stereoselective tandem Barbier process: divergent syntheses of (3R,4S)-statines, (+)-preussin and (-)-hapalosin.
Organic & biomolecular chemistry, 2017, 15, 649-661
7155437 CIFC16 H19 N O2P 21 21 218.8657; 11.708; 13.548
90; 90; 90
1406.3Chen, Pengquan; Zhu, Chuanle; Zhu, Rui; Lin, Zhiming; Wu, Wanqing; Jiang, Huanfeng
Synthesis of 3-azabicyclo[3.1.0]hexane derivatives via palladium-catalyzed cyclopropanation of maleimides with N-tosylhydrazones: practical and facile access to CP-866,087.
Organic & biomolecular chemistry, 2017, 15, 1228-1235
7155438 CIFC25 H15 NP 21 21 217.25647; 13.0278; 17.2343
90; 90; 90
1629.26Matsumoto, Arimasa; Yonemitsu, Kento; Ozaki, Hanae; Míšek, Jiří; Starý, Ivo; Stará, Irena G; Soai, Kenso
Reversal of the sense of enantioselectivity between 1- and 2-aza[6]helicenes used as chiral inducers of asymmetric autocatalysis.
Organic & biomolecular chemistry, 2017, 15, 1321-1324
7155439 CIFC25 H15 NP 21 21 217.29278; 12.9794; 17.3679
90; 90; 90
1643.97Matsumoto, Arimasa; Yonemitsu, Kento; Ozaki, Hanae; Míšek, Jiří; Starý, Ivo; Stará, Irena G; Soai, Kenso
Reversal of the sense of enantioselectivity between 1- and 2-aza[6]helicenes used as chiral inducers of asymmetric autocatalysis.
Organic & biomolecular chemistry, 2017, 15, 1321-1324
7155440 CIFC15 H13 Br O3P 21 21 215.2767; 8.2192; 29.2713
90; 90; 90
1269.5Ren, Qiao; Li, Muyao; Yuan, Lujiang
Expeditious assembly of fused dihydropyranones via N-heterocyclic carbene-catalyzed tandem Michael addition/lactonization.
Organic & biomolecular chemistry, 2017, 15, 1329-1333
7155462 CIFC10 H8 Cl N O4P 21 21 215.5571; 5.6305; 32.3624
90; 90; 90
1012.6Chen, Wei; Zhou, Zhao-Hui; Chen, Hong-Bin
Efficient synthesis of chiral benzofuryl β-amino alcohols via a catalytic asymmetric Henry reaction.
Organic & biomolecular chemistry, 2017, 15, 1530-1536
7155467 CIFC19 H16 Br N O5P 21 21 2110.415; 11.469; 15.047
90; 90; 90
1797.4Manoni, Francesco; Farid, Umar; Trujillo, Cristina; Connon, Stephen J.
Catalytic asymmetric Tamura cycloadditions involving nitroalkenes.
Organic & biomolecular chemistry, 2017, 15, 1463-1474
7155468 CIFC13 H8 O2P 21 21 214.8942; 13.6964; 14.1713
90; 90; 90
949.94Tang, Jing; Zhao, Shijun; Wei, Yuanyuan; Quan, Zhengjun; Huo, Congde
CBr4 promoted intramolecular aerobic oxidative dehydrogenative arylation of aldehydes: application in the synthesis of xanthones and fluorenones.
Organic & biomolecular chemistry, 2017, 15, 1589-1592
7155478 CIFC10 H13 N OP 21 21 215.9842; 9.104; 16.0223
90; 90; 90
872.9Li, Ke; Wang, Juxiang; Wu, Kailin; Zheng, Daijun; Zhou, Xiaojian; Han, Wenyong; Wan, Nanwei; Cui, Baodong; Chen, Yongzheng
Enantioselective synthesis of 1,2,3,4-tetrahydroquinoline-4-ols and 2,3-dihydroquinolin-4(1H)-ones via a sequential asymmetric hydroxylation/diastereoselective oxidation process using Rhodococcus equi ZMU-LK19.
Organic & biomolecular chemistry, 2017, 15, 3580-3584
7155488 CIFC18 H16 N2 O3P 21 21 214.87924; 14.43858; 20.3657
90; 90; 90
1434.75Verhasselt, Sigrid; Roman, Bart I.; De Wever, Olivier; Van Hecke, Kristof; Van Deun, Rik; Bracke, Marc E.; Stevens, Christian V.
Discovery of (S)-3'-hydroxyblebbistatin and (S)-3'-aminoblebbistatin: polar myosin II inhibitors with superior research tool properties.
Organic & biomolecular chemistry, 2017, 15, 2104-2118
7155489 CIFC18 H16 N2 O3P 21 21 214.88084; 14.45507; 20.3743
90; 90; 90
1437.47Verhasselt, Sigrid; Roman, Bart I.; De Wever, Olivier; Van Hecke, Kristof; Van Deun, Rik; Bracke, Marc E.; Stevens, Christian V.
Discovery of (S)-3'-hydroxyblebbistatin and (S)-3'-aminoblebbistatin: polar myosin II inhibitors with superior research tool properties.
Organic & biomolecular chemistry, 2017, 15, 2104-2118
7155512 CIFC17 H15 Br O3 SP 21 21 217.8117; 12.6388; 16.816
90; 90; 90
1660.3Shiely, Amy E.; Slattery, Catherine N.; Ford, Alan; Eccles, Kevin S.; Lawrence, Simon E.; Maguire, Anita R.
Enantioselective copper catalysed intramolecular C-H insertion reactions of α-diazo-β-keto sulfones, α-diazo-β-keto phosphine oxides and 2-diazo-1,3-diketones; the influence of the carbene substituent.
Organic & biomolecular chemistry, 2017, 15, 2609-2628
7155513 CIFC17 H15 Br O3 SP 21 21 217.8064; 12.6377; 16.783
90; 90; 90
1655.7Shiely, Amy E.; Slattery, Catherine N.; Ford, Alan; Eccles, Kevin S.; Lawrence, Simon E.; Maguire, Anita R.
Enantioselective copper catalysed intramolecular C-H insertion reactions of α-diazo-β-keto sulfones, α-diazo-β-keto phosphine oxides and 2-diazo-1,3-diketones; the influence of the carbene substituent.
Organic & biomolecular chemistry, 2017, 15, 2609-2628
7155517 CIFC11 H12 O2P 21 21 214.6462; 9.7488; 19.6719
90; 90; 90
891.04Ma, Fujie; Chen, Jingchao; Yang, Fan; Shinde, Madhuri Vikas; Zhou, Yongyun; Fan, Baomin
Palladium/zinc co-catalyzed asymmetric transfer hydrogenation of oxabenzonorbornadienes with alcohols as hydrogen sources.
Organic & biomolecular chemistry, 2017, 15, 2359-2362
7155528 CIFC15 H21 N O2P 21 21 216.953; 11.068; 16.703
90; 90; 90
1285.4Kuznetsov, Nikolai Yu; Tikhov, Rabdan M.; Godovikov, Ivan A.; Medvedev, Michael G.; Lyssenko, Konstantin A.; Burtseva, Elena I.; Kirillova, Elena S.; Bubnov, Yuri N.
Stereoselective synthesis of novel adamantane derivatives with high potency against rimantadine-resistant influenza A virus strains.
Organic & biomolecular chemistry, 2017, 15, 3152-3157
7155530 CIFC19 H30 Br N O2P 21 21 2110.6735; 11.9007; 14.2306
90; 90; 90
1807.6Kuznetsov, Nikolai Yu; Tikhov, Rabdan M.; Godovikov, Ivan A.; Medvedev, Michael G.; Lyssenko, Konstantin A.; Burtseva, Elena I.; Kirillova, Elena S.; Bubnov, Yuri N.
Stereoselective synthesis of novel adamantane derivatives with high potency against rimantadine-resistant influenza A virus strains.
Organic & biomolecular chemistry, 2017, 15, 3152-3157
7155533 CIFC12 H25 N O4P 21 21 218.2056; 11.9665; 13.8857
90; 90; 90
1363.47Zhang, Jing; Kolluri, Rao; Alvarez, Salvador G.; Irving, Mark M.; Singh, Rajinder; Duncton, Matthew A. J.
Enantioselective synthesis of an octahydroindolizine (indolizidine) alcohol using an enzymatic resolution.
Organic & biomolecular chemistry, 2017, 15, 2953-2961
7155553 CIFC20 H20 O5P 21 21 215.6783; 18.1808; 34.1983
90; 90; 90
3530.5Lian, Xiao-Lei; Adili, Alafate; Liu, Bin; Tao, Zhong-Lin; Han, Zhi-Yong
Enantioselective [4 + 1] cycloaddition of ortho-quinone methides and bromomalonates under phase-transfer catalysis.
Organic & biomolecular chemistry, 2017, 15, 3670-3673
7155560 CIFC21 H25 N O2 SP 21 21 2111.8441; 11.9103; 13.4579
90; 90; 90
1898.46Chung, Min-Ching; Chan, Yung-Hsiang; Chang, Wen-Jung; Hou, Duen-Ren
Synthesis of 2,3-dihydro-1H-pyrroles by intramolecular cyclization of N-(3-butynyl)-sulfonamides.
Organic & biomolecular chemistry, 2017, 15, 3783-3790
7155562 CIFC20 H16 N2 OP 21 21 217.199; 13.738; 30.836
90; 90; 90
3050Midya, Siba Prasad; Gopi, Elumalai; Satam, Nishikant; Namboothiri, Irishi N. N.
Synthesis of fused cyanopyrroles and spirocyclopropanes via addition of N-ylides to chalconimines.
Organic & biomolecular chemistry, 2017, 15, 3616-3627
7155567 CIFC22 H22 F3 N O6 SP 21 21 219.68066; 12.6194; 18.5137
90; 90; 90
2261.71Espinosa, Miguel; Herrera, Jorge; Blay, Gonzalo; Cardona, Luz; Muñoz, M Carmen; Pedro, Jose R.
Copper-Catalysed Enantioselective Michael Addition of Malonic Esters to β-Trifluoromethyl-α,β-Unsaturated Imines
Org. Biomol. Chem., 2017
7155570 CIFC27 H26 I N O3P 21 21 215.5901; 10.1207; 40.4585
90; 90; 90
2288.97Hodík, Tomáš; Schneider, Christoph
Brønsted acid-catalyzed, enantioselective synthesis of 1,4-dihydroquinoline-3-carboxylates via in situ generated ortho-quinone methide imines.
Organic & biomolecular chemistry, 2017, 15, 3706-3716
7155601 CIFC25 H33 Cl2 N3 O4P 21 21 219.0157; 14.404; 19.6135
90; 90; 90
2547.1Hernandez Rubio, Omayra; Borrego, Sara del Mazo; Marcos Monleon, Laura; Simon, Luis; Temprano, Álvaro G.; rodriguez moran, joaquin
A cleft type receptor which combines an oxyanion hole with electrostatic interactions
Org. Biomol. Chem., 2017
7155603 CIFC32 H37 Cl2 N3 O6P 21 21 218.4007; 14.3494; 26.2774
90; 90; 90
3167.6Hernandez Rubio, Omayra; Borrego, Sara del Mazo; Marcos Monleon, Laura; Simon, Luis; Temprano, Álvaro G.; rodriguez moran, joaquin
A cleft type receptor which combines an oxyanion hole with electrostatic interactions
Org. Biomol. Chem., 2017
7155604 CIFC34 H42 Cl2 N4 O7 SP 21 21 2110.7729; 23.4747; 28.9321
90; 90; 90
7316.7Hernandez Rubio, Omayra; Borrego, Sara del Mazo; Marcos Monleon, Laura; Simon, Luis; Temprano, Álvaro G.; rodriguez moran, joaquin
A cleft type receptor which combines an oxyanion hole with electrostatic interactions
Org. Biomol. Chem., 2017
7155613 CIFC17 H20 N2 O3P 21 21 215.8639; 8.5853; 29.2551
90; 90; 90
1472.8Sheth, Vishal M.; Hong, Bor-Cherng; Lee, Gene-Hsiang
Enantioselective total synthesis of (+)-arborescidine C and related tetracyclic indole alkaloids using organocatalysis.
Organic & biomolecular chemistry, 2017, 15, 3408-3412
7155627 CIFC31 H34 O2P 21 21 219.6403; 16.1153; 16.1214
90; 90; 90
2504.6Zhou, Tao; Li, Shenhuan; Huang, Ben; Li, Cao; Zhao, Yang; Chen, Jieqiong; Chen, Aoling; Xiao, Yuanjin; Liu, Lu; Zhang, Junliang
Phosphine-catalyzed Friedel–Crafts reaction of naphthols with para-quinone methides: expedient access to triarylmethanes
Org. Biomol. Chem., 2017
7155633 CIFC23 H19 N3 O2P 21 21 219.5443; 19.2006; 20.0739
90; 90; 90
3678.67Del Grosso, Alessandro; Galanopoulos, Lavrentis-Dimitrios; Chiu, Cookson K. C.; Clarkson, Guy J.; O′ Connor, Peter B.; Wills, Martin
Strained alkynes derived from 2,2′-dihydroxy-1,1′-biaryls; synthesis and copper-free cycloaddition with azides
Org. Biomol. Chem., 2017
7155646 CIFC17 H13 F4 N3 SP 21 21 215.3006; 8.666; 35.753
90; 90; 90
1642.3Voltrová, Svatava; Muselli, Mickaël; Filgas, Josef; Matoušek, Václav; Klepetářová, Blanka; Beier, Petr
Synthesis of tetrafluoroethylene- and tetrafluoroethyl-containing azides and their 1,3-dipolar cycloaddition as synthetic application
Org. Biomol. Chem., 2017
7155651 CIFC24 H17 Cl F3 N3 O7 SP 21 21 219.6118; 9.9839; 26.2874
90; 90; 90
2522.6Zhu, Yuanyuan; Li, Boyu; Wang, Cui; Dong, Zhenghao; Zhong, Xiaoling; Wang, Kairong; Yan, Wenjin; Wang, Rui
Asymmetric Synthesis of CF3-Containing Tetrahydroquinoline via Thiourea-Catalyzed Cascade Reaction
Org. Biomol. Chem., 2017
7155652 CIFC24 H17 Br F3 N3 O7 SP 21 21 219.9489; 10.0773; 51.389
90; 90; 90
5152.2Zhu, Yuanyuan; Li, Boyu; Wang, Cui; Dong, Zhenghao; Zhong, Xiaoling; Wang, Kairong; Yan, Wenjin; Wang, Rui
Asymmetric Synthesis of CF3-Containing Tetrahydroquinoline via Thiourea-Catalyzed Cascade Reaction
Org. Biomol. Chem., 2017
7155666 CIFC11 H11 F9 O4P 21 21 218.2625; 9.6405; 17.8895
90; 90; 90
1424.98Silvestri, Anthony Paul; Dawson, Philip Edward
Base-catalyzed Diastereoselective Trimerization of Trifluoroacetone
Org. Biomol. Chem., 2017
7155668 CIFC13 H19 N O5P 21 21 216.3866; 10.6043; 19.7027
90; 90; 90
1334.37Moloney, Mark G.; Josa-Cullere, Laia; Towers, Christopher; Willenbrock, Frances; Macauley, Valentine; Christensen, Kirsten
Synthesis and bioactivity of fused- and spiro–lactone-lactam systems
Org. Biomol. Chem., 2017
7155688 CIFC26 H17 Cl N2 O4P 21 21 218.624; 9.752; 26.737
90; 90; 90
2248.6Xia, Ai-Bao; Zhang, Xiao-Long; Tang, Chengke; Feng, Kai-Xiang; Du, Xiao-Hua; Xu, Danqian
One-pot Asymmetric Synthesis of Spiro[dihydrofurocoumarin/ pyrazolone] Scaffolds by Michael Addition/I2-Mediated Cyclization Sequence
Org. Biomol. Chem., 2017
7155690 CIFC27 H20 N2 O4P 21 21 218.3497; 9.7735; 27.653
90; 90; 90
2256.6Xia, Ai-Bao; Zhang, Xiao-Long; Tang, Chengke; Feng, Kai-Xiang; Du, Xiao-Hua; Xu, Danqian
One-pot Asymmetric Synthesis of Spiro[dihydrofurocoumarin/ pyrazolone] Scaffolds by Michael Addition/I2-Mediated Cyclization Sequence
Org. Biomol. Chem., 2017
7155692 CIFC15 H26 O3P 21 21 219.9836; 11.1199; 12.6582
90; 90; 90
1405.3Franco dos Santos, Gabriel; Moraga, Javier; Takahashi, Jacqueline A.; Viaud, Muriel; Hanson, James R.; Hern�ndez- Gal�n, Rosario; Collado, I. G.
The formation of sesquiterpenoid presilphiperfolane and cameroonane metabolites in the Bcbot4 null mutant of Botrytis cinerea
Org. Biomol. Chem., 2017
7155693 CIFC15 H20 F N O3 SP 21 21 218.8617; 13.1073; 28.6
90; 90; 90
3322Wei, qiaoling; Zhang, Feng; zhao, xiaofang; Wang, Chao; Xiao, Jianling; Tang, Weijun
Ru-catalyzed highly diastereoselective hydrogenation of N-tert-butylsulfinyl ketimines for the synthesis of aryl glycine derivatives
Org. Biomol. Chem., 2017
7155742 CIFC24 H18 Br N O3P 21 21 2110.585; 17.682; 21.378
90; 90; 90
4001.2Ming, Sheng; Zhao, Bo-Liang; Du, Da-Ming
Chiral squaramide-catalysed enantioselective Michael/cyclization cascade reaction of 3-hydroxyoxindoles with α,β-unsaturated N-acylated succinimides
Org. Biomol. Chem., 2017
7155779 CIFC28 H26 Cl N O3 SeP 21 21 218.269; 16.049; 18.529
90; 90; 90
2459Singha Roy, Soumya Jyoti; Mukherjee, Santanu
“On water” catalytic enantioselective sulfenylation of deconjugated butyrolactams
Org. Biomol. Chem., 2017
7155780 CIFC28 H26 Cl N O3 SP 21 21 218.373; 11.816; 25.567
90; 90; 90
2529Singha Roy, Soumya Jyoti; Mukherjee, Santanu
“On water” catalytic enantioselective sulfenylation of deconjugated butyrolactams
Org. Biomol. Chem., 2017
7155784 CIFC41 H46 B N O2P 21 21 2113.4025; 15.8388; 16.5989
90; 90; 90
3523.6Tayama, Eiji; Watanabe, Kazutoshi; Sotome, Sho
Structural and mechanistic studies of the base-induced Sommelet–Hauser rearrangement of N-α-branched benzylic azetidine-2-carboxylic acid-derived ammonium salts
Org. Biomol. Chem., 2017
7155798 CIFC15 H10 O3P 21 21 215.8423; 10.7141; 17.775
90; 90; 90
1112.63Cheng, Yuyu; Zhang, Pengfei; Jia, Yanwen; Fang, Zhiqiang; Li, Pengfei
Organocatalytic condensation–ring opening–annulation cascade reactions between N-Bocindolin-2-ones/benzofuran-2(3H)-ones and salicylaldehydes for synthesis of 3-arylcoumarins
Org. Biomol. Chem., 2017
7155813 CIFC25 H23 Cl O4P 21 21 215.8155; 11.5974; 31.3321
90; 90; 90
2113.18Kowalczyk, Dorota; Albrecht, Lukasz
Organocatalytic cis-Selective Approach to Bicyclic δ-Lactones
Org. Biomol. Chem., 2017
7155830 CIFC31 H58 O3 Si2P 21 21 217.4726; 20.1154; 23.4601
90; 90; 90
3526.4Guillade, Lucía; Gónzalez Pérez, Adán B; R. de LERA, Angel
Synthesis of the Octahydronaphthalene Core of Nahuoic Acid A via a B(C6F5)3-Catalyzed Intramolecular Diels-Alder (IMDA) Reaction
Org. Biomol. Chem., 2017
7155852 CIFC22 H23 N O6P 21 21 219.0736; 10.7768; 21.461
90; 90; 90
2098.6Prandi, Cristina; Lombardi, Chiara; Artuso, Emma; LOLLI, Marco Lucio Lucio; Grandi, Eleonora; Priola, Emanuele; Spyrakis, Francesca
Recent Advances in the Synthesis of Analogues of Phytohormones Strigolactones with Ring-Closing Metathesis as a Key Step
Org. Biomol. Chem., 2017
7155879 CIFC23 H23 Cl N2 O2P 21 21 215.9545; 12.1404; 28.388
90; 90; 90
2052.2Pan, Subhas Chandra; Maity, Rajendra
Enantioselective Aminocatalytic Synthesis of Tetrahydropyrano [2,3-c]Pyrazoles via Domino Michael-Hemiacetalization Reaction with Alkylidene Pyrazolones
Org. Biomol. Chem., 2017
7155885 CIFC21 H23 N O4P 21 21 218.75356; 8.85744; 24.746
90; 90; 90
1918.66Jackson, Mark; O'Broin, Calvin Quince; Müller-Bunz, Helge; Guiry, Patrick J.
Enantioselective synthesis of sterically hindered α-allyl–α-aryl oxindoles via palladium-catalysed decarboxylative asymmetric allylic alkylation
Org. Biomol. Chem., 2017
7155888 CIFC22 H23 N OP 21 21 215.8282; 12.018; 24.9007
90; 90; 90
1744.13Alvarez, Rosana; Vilar, Unai; Madich, Youssef; Aurrecoechea, Jose M.
On the Regiochemical Differences between Pd-Catalyzed Heterocyclization-Allylation and -Arylation Reactions of Alkynylbenzamides: Preparation of 4-Allyl-isochromen-1-imines and Computational Study
Org. Biomol. Chem., 2017
7155890 CIFC20 H28 O2P 21 21 2110.371; 11.8296; 13.3226
90; 90; 90
1634.48Uroos, Maliha; Pitt, Phillip; Harwood, Laurence Marius; Lewis, William; Blake, Alexander J.; Hayes, Christopher J. J
Total synthesis of (–)-aritasone via the ultra-high pressure hetero-Diels-Alder dimerisation of (–)-pinocarvone
Org. Biomol. Chem., 2017
7155891 CIFC20 H28 O2P 21 21 216.6086; 9.9529; 25.6799
90; 90; 90
1689.09Uroos, Maliha; Pitt, Phillip; Harwood, Laurence Marius; Lewis, William; Blake, Alexander J.; Hayes, Christopher J. J
Total synthesis of (–)-aritasone via the ultra-high pressure hetero-Diels-Alder dimerisation of (–)-pinocarvone
Org. Biomol. Chem., 2017
7155892 CIFC20 H28 O2P 21 21 216.2525; 10.9938; 24.717
90; 90; 90
1699Uroos, Maliha; Pitt, Phillip; Harwood, Laurence Marius; Lewis, William; Blake, Alexander J.; Hayes, Christopher J. J
Total synthesis of (–)-aritasone via the ultra-high pressure hetero-Diels-Alder dimerisation of (–)-pinocarvone
Org. Biomol. Chem., 2017
7155905 CIFC32 H36 Br N O4P 21 21 2110.3304; 11.1679; 24.5971
90; 90; 90
2837.7Li, Wenjun; Zhang, Lili; Liu, Yang; Liu, Kun; Liu, Zhantao; He, Ningning
Asymmetric synthesis of dihydrocoumarins via organocatalytic hetero-Diels-Alder reaction of ortho-quinone methides
Org. Biomol. Chem., 2017
7155920 CIFC19 H17 N3 O4P 21 21 218.962; 9.634; 20.046
90; 90; 90
1730.8Sen, Subhabrata; Chauhan, Jyoti; Luthra, Tania; Gundla, Rambabu; Ferraro, Antonio; Holzgrabe, Ulrike
A diversity oriented synthesis of natural product inspired molecular libraries
Org. Biomol. Chem., 2017
7155921 CIFC16 H22 O5P 21 21 215.7984; 7.8542; 33.8291
90; 90; 90
1540.64Mirabella, Stefania; Fibbi, Giulia; Matassini, Camilla; Faggi, Cristina; Goti, Andrea; Cardona, Francesca
Accessing 2-substituted piperidine iminosugars by organometallic addition/intramolecular reductive amination: aldehyde vs nitrone route
Org. Biomol. Chem., 2017
7155922 CIFC9 H17 N O3P 21 21 215.5; 9.816; 18.586
90; 90; 90
1003.42Mirabella, Stefania; Fibbi, Giulia; Matassini, Camilla; Faggi, Cristina; Goti, Andrea; Cardona, Francesca
Accessing 2-substituted piperidine iminosugars by organometallic addition/intramolecular reductive amination: aldehyde vs nitrone route
Org. Biomol. Chem., 2017
7155930 CIFC38 H41 N5 O8P 21 21 2110.8476; 17.322; 37.2345
90; 90; 90
6996.4Kicsák, Máté; Mándi, Attila; Varga, Szabolcs; Herczeg, Mihály; Batta, Gyula; Bényei, Attila; Borbás, Anikó; Herczegh, Pál
Tricyclanos: conformationally constrained nucleoside analogues with a new heterotricycle obtained from a d-ribofuranose unit.
Organic & biomolecular chemistry, 2018, 16, 393-401
7155931 CIFC17 H15 Br2 N O2P 21 21 216.1907; 15.2739; 17.2701
90; 90; 90
1632.99Jiang, Hua-Jie; Liu, Kun; Wang, Jing; Li, Na; Yu, Jie
Brønsted Acids of Anionic Chiral Co(III) Complexes as Catalysts for the Stereoselective Synthesis of cis-4-Aminofuranobenzopyrans
Org. Biomol. Chem., 2017
7155933 CIFC13 H12 N2 OP 21 21 217.4367; 11.0255; 13.3188
90; 90; 90
1092.05Liu, Shuai; Zu, Weisai; Zhang, Jinli; Xu, Liang
Chemoselective N-arylation of Aminobenzamides via Copper Catalysed Chan−Evans−Lam Reactions
Org. Biomol. Chem., 2017
7155934 CIFC20 H19 Cu F6 N3 O7 S2P 21 21 218.683; 10.2079; 27.0713
90; 90; 90
2399.47Wang, Yang; Liu, Haixiong; Zhang, Xiaofeng; Zhang, Zilong; Huang, Deguang
Experimental and mechanistic insights into copper(ii)–dioxygen catalyzed oxidative N-dealkylation of N-(2-pyridylmethyl)phenylamine and its derivatives
Org. Biomol. Chem., 2017
7155969 CIFC30 H44 N2 O10P 21 21 2110.3732; 16.8818; 35.8766
90; 90; 90
6282.6Chiu, Din-Chi; Lin, Tzu-Chen; Huang, Wen-I; Cheng, Ting-Jen R.; Tsai, Keng-Chang; Fang, Jim-Min
Peramivir analogues bearing hydrophilic side chains exhibit higher activities against H275Y mutant than wild-type influenza virus
Organic & Biomolecular Chemistry, 2017
7155971 CIFC15 H22 F3 N O2 SP 21 21 218.1745; 10.1237; 20.5314
90; 90; 90
1699.1Grellepois, Fabienne; Ben Jamaa, Abdelkhalek; Saraiva Rosa, Nathalie
α-Trifluoromethylated tertiary homoallylic amines: diastereoselective synthesis and conversion into β-aminoesters, γ- and δ-aminoalcohols, azetidines and pyrrolidines
Organic & Biomolecular Chemistry, 2017
7155974 CIFC11 H22 F3 N O SP 21 21 219.071; 16.862; 19.003
90; 90; 90
2907Grellepois, Fabienne; Ben Jamaa, Abdelkhalek; Saraiva Rosa, Nathalie
α-Trifluoromethylated tertiary homoallylic amines: diastereoselective synthesis and conversion into β-aminoesters, γ- and δ-aminoalcohols, azetidines and pyrrolidines
Organic & Biomolecular Chemistry, 2017
7155975 CIFC11 H20 F3 N O2 SP 21 21 2111.039; 12.316; 21.359
90; 90; 90
2903.9Grellepois, Fabienne; Ben Jamaa, Abdelkhalek; Saraiva Rosa, Nathalie
α-Trifluoromethylated tertiary homoallylic amines: diastereoselective synthesis and conversion into β-aminoesters, γ- and δ-aminoalcohols, azetidines and pyrrolidines
Organic & Biomolecular Chemistry, 2017
7155978 CIFC41 H67 O16P 21 21 217.9929; 9.2895; 54.987
90; 90; 90
4082.8Xia, Guiyang; Yao, Tie; Zhang, Bing-Yang; Li, Yang; Kang, Ning; Cao, Shijie; Ding, Liqin; Chen, Lixia; Qiu, Feng
Withapubesides A‒D, natural inducible nitric oxide synthase (iNOS) inhibitors from Physalis pubescens
Organic & Biomolecular Chemistry, 2017
7155979 CIFC6 H9 N O3P 21 21 218.5061; 15.9215; 9.6417
90; 90; 90
1305.77Alhifthi, Amani; Harris, Benjamin L.; Goerigk, Lars; White, Jonathan; Williams, Spencer J.
Structure-reactivity correlations of the abnormal Beckmann reaction of dihydrolevoglucosenone oxime
Organic & Biomolecular Chemistry, 2017
7155980 CIFC13 H12 N2 O6P 21 21 217.3112; 12.3133; 13.9596
90; 90; 90
1256.71Alhifthi, Amani; Harris, Benjamin L.; Goerigk, Lars; White, Jonathan; Williams, Spencer J.
Structure-reactivity correlations of the abnormal Beckmann reaction of dihydrolevoglucosenone oxime
Organic & Biomolecular Chemistry, 2017
7155982 CIFC12 H13 N O3P 21 21 215.9489; 8.1059; 22.3033
90; 90; 90
1075.49Alhifthi, Amani; Harris, Benjamin L.; Goerigk, Lars; White, Jonathan; Williams, Spencer J.
Structure-reactivity correlations of the abnormal Beckmann reaction of dihydrolevoglucosenone oxime
Organic & Biomolecular Chemistry, 2017
7155983 CIFC12 H12 N2 O5P 21 21 216.7738; 11.4773; 14.8982
90; 90; 90
1158.26Alhifthi, Amani; Harris, Benjamin L.; Goerigk, Lars; White, Jonathan; Williams, Spencer J.
Structure-reactivity correlations of the abnormal Beckmann reaction of dihydrolevoglucosenone oxime
Organic & Biomolecular Chemistry, 2017
7155985 CIFC8 H11 N O4P 21 21 215.6704; 15.6773; 9.7844
90; 90; 90
869.8Alhifthi, Amani; Harris, Benjamin L.; Goerigk, Lars; White, Jonathan; Williams, Spencer J.
Structure-reactivity correlations of the abnormal Beckmann reaction of dihydrolevoglucosenone oxime
Organic & Biomolecular Chemistry, 2017
7155986 CIFC13 H11 N3 O8P 21 21 216.27; 9.456; 23.6
90; 90; 90
1399.2Alhifthi, Amani; Harris, Benjamin L.; Goerigk, Lars; White, Jonathan; Williams, Spencer J.
Structure-reactivity correlations of the abnormal Beckmann reaction of dihydrolevoglucosenone oxime
Organic & Biomolecular Chemistry, 2017
7155991 CIFC14 H17 N O4P 21 21 216.32903; 8.54815; 23.7167
90; 90; 90
1283.11Osorio-Nieto, Urbano; Vázquez-Amaya, Laura Y; Höpfl, Herbert; Quintero, Leticia; Sartillo-Piscil, Fernando
The direct and highly diastereoselective synthesis of 3,4-epoxy-2-piperidones. Application to the total synthesis and absolute configurational assignment of 3α,4α-epoxy-5β-pipermethystine.
Organic & biomolecular chemistry, 2017, 16, 77-88
7155993 CIFC14 H17 N O4P 21 21 216.38939; 7.59037; 26.8562
90; 90; 90
1302.47Osorio-Nieto, Urbano; Vázquez-Amaya, Laura Y; Höpfl, Herbert; Quintero, Leticia; Sartillo-Piscil, Fernando
The direct and highly diastereoselective synthesis of 3,4-epoxy-2-piperidones. Application to the total synthesis and absolute configurational assignment of 3α,4α-epoxy-5β-pipermethystine.
Organic & biomolecular chemistry, 2017, 16, 77-88
7156003 CIFC17 H28 O4 SiP 21 21 217.2037; 10.9197; 23.762
90; 90; 90
1869.2Ojo, O. Stephen; Nardone, Brunello; Musolino, Stefania F.; Neal, Andrew R.; Wilson, Liam; Lebl, Tomas; Slawin, Alexandra M. Z.; Cordes, David B.; Taylor, James E.; Naismith, James H.; Smith, Andrew D.; Westwood, Nicholas J.
Synthesis of the natural product descurainolide and cyclic peptides from lignin-derived aromatics.
Organic & biomolecular chemistry, 2018, 16, 266-273
7156009 CIFC24 H20 Br N O2P 21 21 216.6297; 15.443; 20.287
90; 90; 90
2077Guo, Tao; Yuan, Bin-Hua; Liu, Wen-Jie
Highly efficient asymmetric construction of novel indolines and tetrahydroquinoline derivatives via aza-Barbier/C-N coupling reaction.
Organic & biomolecular chemistry, 2017, 16, 57-61
7156013 CIFC18 H15 N3 OP 21 21 215.5664; 8.8236; 28.6221
90; 90; 90
1405.79Ruvinskaya, Julia O.; Rostovskii, Nikolai V.; Filippov, Ilya P.; Khlebnikov, Alexander F.; Novikov, Mikhail S.
A novel approach to 5H-pyrazino[2,3-b]indoles via annulation of 3-diazoindolin-2-imines with 2H-azirines or 5-alkoxyisoxazoles under Rh(ii) catalysis.
Organic & biomolecular chemistry, 2017, 16, 38-42
7156022 CIFC33 H55 Cl6 N5 O8P 21 21 2110.1637; 17.2472; 25.5023
90; 90; 90
4470.4Lee, Jaeyeon; Shim, Jihyun; Kang, Philjae; Choi, Moon-Gun; Choi, Soo Hyuk
Side chain-specific 11/9-helix propensity of α/β-peptides with alternating residue types.
Organic & biomolecular chemistry, 2018, 16, 433-438
7156046 CIFC14 H23 N O2P 21 21 217.7672; 9.3611; 19.2665
90; 90; 90
1400.86Liu, Yi-Wen; Ma, Rui-Jun; Yan, Jia-Hang; Zhou, Zhu; Wei, Bang-Guo
Asymmetric synthesis of (-)-sedacryptine through a diastereoselective Mannich reaction of N,O-acetals with ketones.
Organic & biomolecular chemistry, 2018, 16, 771-779
7156052 CIFC54 H60 N4 O8P 21 21 2110.7257; 11.3249; 39.4835
90; 90; 90
4795.96Grajewski, J.; Piotrowska, K.; Zgorzelak, M.; Janiak, A.; Biniek-Antosiak, K; Rychlewska, U.; Gawronski, J.
Introduction of axial chirality at a spiro carbon atom in the synthesis of pentaerythritol-imine macrocycles.
Organic & biomolecular chemistry, 2018, 16, 981-987
7156054 CIFC31 H23 Br F N3 O4P 21 21 219.608; 9.984; 28.09
90; 90; 90
2695Wu, Shiqi; Zhu, Guodong; Wei, Shiqiang; Chen, Hongbo; Qu, Jingping; Wang, Baomin
Organocatalytic [3 + 2] cycloaddition of oxindole-based azomethine ylides with 3-nitrochromenes: a facile approach to enantioenriched polycyclic spirooxindole-chromane adducts.
Organic & biomolecular chemistry, 2018, 16, 807-815
7156055 CIFC43 H47 B N2 O3P 21 21 219.6421; 18.6118; 20.0924
90; 90; 90
3605.7Setner, B.; Wierzbicka, M.; Jerzykiewicz, L.; Lisowski, M.; Szewczuk, Z.
The unexpected racemization and hydrogen-deuterium exchange of the hydrogen at the α-carbon of proline analogs containing the 5-azoniaspiro[4.4]nonyl-group.
Organic & biomolecular chemistry, 2018, 16, 825-831
7156056 CIFC23 H30 N2 O4 SP 21 21 219.7197; 12.3037; 19.686
90; 90; 90
2354.2Castán, A; Badorrey, R.; Gálvez, J A; López-Ram-de-Víu, P; Díaz-de-Villegas, M D
Michael addition of carbonyl compounds to nitroolefins under the catalysis of new pyrrolidine-based bifunctional organocatalysts.
Organic & biomolecular chemistry, 2018, 16, 924-935
7156062 CIFC17 H11 Cl O2P 21 21 216.1663; 12.6929; 17.4233
90; 90; 90
1363.7Chehal, Navneet K.; Budzelaar, Peter H. M.; Hultin, Philip G.
E-Z isomerization in Suzuki cross-couplings of haloenones: ligand effects and evidence for a separate catalytic cycle.
Organic & biomolecular chemistry, 2018, 16, 1134-1143
7156076 CIFC20 H13 Cl N2 OP 21 21 216.3278; 13.3923; 18.8088
90; 90; 90
1593.9Kour, Dilpreet; Gupta, Annah; Kapoor, Kamal K.; Gupta, Vivek K.; Rajnikant, ?; Singh, Deepika; Das, Parthasarathi
Iodine-NH<sub>4</sub>OAc mediated regioselective synthesis of 2-aroyl-3-arylimidazo[1,2-a]pyridines from 1,3-diaryl-prop-2-en-1-ones.
Organic & biomolecular chemistry, 2018, 16, 1330-1336
7156081 CIFC24 H32 N4 O2P 21 21 218.83; 14.378; 17.669
90; 90; 90
2243.2Darapaneni, Chandra Mohan; Kaniraj, Prathap Jeya; Maayan, Galia
Water soluble hydrophobic peptoids via a minor backbone modification.
Organic & biomolecular chemistry, 2018, 16, 1480-1488
7156095 CIFC124.4 H156.62 N20 O25.4 S16.2P 21 21 2119.763; 21.594; 33.712
90; 90; 90
14387Cholewiak, Agnieszka; Dobrzycki, Łukasz; Jurczak, Janusz; Ulatowski, Filip
Disulphide bond exchange inhibited by air - kinetic and thermodynamic products in a library of macrocyclic cysteine derivatives.
Organic & biomolecular chemistry, 2018, 16, 2411-2420
7156116 CIFC17 H14 Cl N O5P 21 21 217.5946; 13.4938; 15.8269
90; 90; 90
1621.94Maity, Rajendra; Pan, Subhas Chandra
Organocatalytic asymmetric Michael/hemiacetalization/acyl transfer reaction of α-nitroketones with o-hydroxycinnamaldehydes: synthesis of 2,4-disubstituted chromans.
Organic & biomolecular chemistry, 2018, 16, 1598-1608
7156124 CIFC17 H22 O7P 21 21 218.16871; 8.25025; 23.3395
90; 90; 90
1572.94Zhang, Zhan-Xin; Wu, Pei-Qian; Li, Hui-Hong; Qi, Feng-Ming; Fei, Dong-Qing; Hu, Qiao-Ling; Liu, Ying-Hong; Huang, Xiao-Ling
Norcrassin A, a novel C<sub>16</sub> tetranorditerpenoid, and bicrotonol A, an unusual dimeric labdane-type diterpenoid, from the roots of Croton crassifolius.
Organic & biomolecular chemistry, 2018, 16, 1745-1750
7156139 CIFC27 H34 O3 SiP 21 21 218.2816; 11.7445; 25.888
90; 90; 90
2518Halder, Joydev; Das, Debabrata; Nanda, Samik
A distinctive transformation based diversity oriented synthesis of small ring carbocycles and heterocycles from biocatalytically derived enantiopure α-substituted-β-hydroxyesters.
Organic & biomolecular chemistry, 2018, 16, 2549-2575
7156141 CIFC19 H29 Cl O2P 21 21 217.5312; 20.9084; 21.2244
90; 90; 90
3342.1Kratena, Nicolas; Pilz, Sarah M.; Weil, Matthias; Gmeiner, Günter; Enev, Valentin S.; Gärtner, Peter
Synthesis and structural elucidation of a dehydrochloromethyltestosterone metabolite.
Organic & biomolecular chemistry, 2018, 16, 2508-2521
7156144 CIFC19 H27 Cl O2P 21 21 217.4333; 13.538; 16.411
90; 90; 90
1651.5Kratena, Nicolas; Pilz, Sarah M.; Weil, Matthias; Gmeiner, Günter; Enev, Valentin S.; Gärtner, Peter
Synthesis and structural elucidation of a dehydrochloromethyltestosterone metabolite.
Organic & biomolecular chemistry, 2018, 16, 2508-2521
7156145 CIFC33 H25 O2 PP 21 21 2111.149; 11.921; 18.456
90; 90; 90
2452.9Yin, Yao; Weng, Wei-Zhi; Sun, Jian-Guo; Zhang, Bo
Eosin Y-catalyzed, visible-light-promoted carbophosphinylation of allylic alcohols via a radical neophyl rearrangement.
Organic & biomolecular chemistry, 2018, 16, 2356-2361
7156160 CIFC16 H26 N2 O7P 21 21 218.5004; 12.8701; 16.4218
90; 90; 90
1796.56Josa-Culleré, Laia; Christensen, Kirsten E.; Moloney, Mark G.
Diastereoselective reduction of the tricarbonyl moiety in bicyclic tetramates giving pyroglutamates.
Organic & biomolecular chemistry, 2018, 16, 2705-2710
7156161 CIFC15 H23 I N2 O6P 21 21 218.5534; 13.2093; 16.1337
90; 90; 90
1822.86Josa-Culleré, Laia; Christensen, Kirsten E.; Moloney, Mark G.
Diastereoselective reduction of the tricarbonyl moiety in bicyclic tetramates giving pyroglutamates.
Organic & biomolecular chemistry, 2018, 16, 2705-2710
7156164 CIFC20 H17 Br O5P 21 21 216.3579; 12.657; 22.518
90; 90; 90
1812.1Shen, Yue; Yang, Peng-Fei; Yang, Gaosheng; Chen, Wen-Long; Chai, Zhuo
Lewis acid-catalyzed enantiospecific [3 + 2] annulations of γ-butyrolactone fused cyclopropanes with aromatic aldehydes: synthesis of chiral furanolignans.
Organic & biomolecular chemistry, 2018, 16, 2688-2696
7156165 CIFC21 H20 O7P 21 21 215.8248; 11.9048; 26.568
90; 90; 90
1842.3Shen, Yue; Yang, Peng-Fei; Yang, Gaosheng; Chen, Wen-Long; Chai, Zhuo
Lewis acid-catalyzed enantiospecific [3 + 2] annulations of γ-butyrolactone fused cyclopropanes with aromatic aldehydes: synthesis of chiral furanolignans.
Organic & biomolecular chemistry, 2018, 16, 2688-2696
7156183 CIFC10 H9 I N2P 21 21 218.7463; 9.1092; 13.1444
90; 90; 90
1047.24Das, Ranajit; Banerjee, Mainak; Rai, Rakesh Kumar; Karri, Ramesh; Roy, Gouriprasanna
Metal-free C(sp<sup>2</sup>)-H functionalization of azoles: K<sub>2</sub>CO<sub>3</sub>/I<sub>2</sub>-mediated oxidation, imination, and amination.
Organic & biomolecular chemistry, 2018, 16, 4243-4260
7156196 CIFC17 H17 N O5 S2P 21 21 215.8407; 14.9477; 19.3104
90; 90; 90
1685.9García de la Concepción, Juan; Ávalos, Martín; Cintas, Pedro; Jiménez, José L; Light, Mark E.
Mechanistic studies of 1,3-dipolar cycloadditions of bicyclic thioisomünchnones with alkenes. A computational rationale focused on donor-acceptor interactions.
Organic & biomolecular chemistry, 2018, 16, 3438-3452
7156204 CIFC93 H151 N25 O23P 21 21 219.2019; 33.434; 36.933
90; 90; 90
11362.7Ben Haj Salah, Khoubaib; Das, Sanjit; Ruiz, Nicolas; Andreu, Vanessa; Martinez, Jean; Wenger, Emmanuel; Amblard, Muriel; Didierjean, Claude; Legrand, Baptiste; Inguimbert, Nicolas
How are 1,2,3-triazoles accommodated in helical secondary structures?
Organic & biomolecular chemistry, 2018, 16, 3576-3583
7156207 CIFC71 H114 N18 O17P 21 21 2110.1857; 17.9944; 46.7774
90; 90; 90
8573.6Ben Haj Salah, Khoubaib; Das, Sanjit; Ruiz, Nicolas; Andreu, Vanessa; Martinez, Jean; Wenger, Emmanuel; Amblard, Muriel; Didierjean, Claude; Legrand, Baptiste; Inguimbert, Nicolas
How are 1,2,3-triazoles accommodated in helical secondary structures?
Organic & biomolecular chemistry, 2018, 16, 3576-3583
7156211 CIFC14 H19 N O12P 21 21 215.5311; 13.8941; 23.168
90; 90; 90
1780.5Wang, Tinghua; Nigudkar, Swati S.; Yasomanee, Jagodige P.; Rath, Nigam P.; Stine, Keith J.; Demchenko, Alexei V.
Glycosyl nitrates in synthesis: streamlined access to glucopyranose building blocks differentiated at C-2.
Organic & biomolecular chemistry, 2018, 16, 3596-3604
7156213 CIFC28 H22 Cl F3 N4 O3P 21 21 2110.3289; 13.752; 18.4669
90; 90; 90
2623.09Luo, Yuan; Xie, Ke-Xin; Yue, Deng-Feng; Zhang, Xiao-Mei; Xu, Xiao-Ying; Yuan, Wei-Cheng
An organocatalytic asymmetric Mannich reaction of pyrazoleamides with cyclic trifluoromethyl ketimines: enantioselective access to dihydroquinazolinone skeletons.
Organic & biomolecular chemistry, 2018, 16, 3372-3375
7156248 CIFC15 H11 N OP 21 21 216.4849; 7.9199; 21.9097
90; 90; 90
1125.28Wang, Zheng; Xu, Ming-Hua
Highly enantioselective synthesis of α-tertiary chiral amino acid derivatives through rhodium-catalyzed asymmetric arylation of cyclic N-sulfonyl α-ketimino esters.
Organic & biomolecular chemistry, 2018, 16, 4633-4640
7156260 CIFC23 H22 N2 O6P 21 21 219.6235; 13.3554; 16.7938
90; 90; 90
2158.4Chen, Jin-Quan; Mi, Yang; Shi, Zi-Fa; Cao, Xiao-Ping
Construction of the tetracyclic core of (±)-cycloclavine and 4-amino Uhle's ketone.
Organic & biomolecular chemistry, 2018, 16, 3801-3808
7156269 CIFC27 H39 N2 O4 PP 21 21 219.947; 15.743; 18.185
90; 90; 90
2847.7Gupta, Ashis Kumar; Ahamad, Shakir; Vaishanv, Narendra Kumar; Kant, Ruchir; Mohanan, Kishor
Base-mediated 1,6-conjugate addition of the Seyferth-Gilbert reagent to para-quinone methides.
Organic & biomolecular chemistry, 2018, 16, 4623-4627
7156281 CIFC28 H44 Br N O4 SP 21 21 215.6897; 11.2486; 45.457
90; 90; 90
2909.3Guerola, Marta; Escolano, Marcos; Alzuet-Piña, Gloria; Gómez-Bengoa, Enrique; Ramírez de Arellano, Carmen; Sánchez-Roselló, María; Del Pozo, Carlos
Synthesis of substituted piperidines by enantioselective desymmetrizing intramolecular aza-Michael reactions.
Organic & biomolecular chemistry, 2018, 16, 4650-4658
7156288 CIFC36 H40 Cl N3 Ni O4P 21 21 216.2383; 15.367; 32.9494
90; 90; 90
3158.66Takeda, Ryosuke; Kawamura, Akie; Kawashima, Aki; Sato, Tatsunori; Moriwaki, Hiroki; Izawa, Kunisuke; Abe, Hidenori; Soloshonok, Vadim A.
Second-order asymmetric transformation and its application for the practical synthesis of α-amino acids.
Organic & biomolecular chemistry, 2018, 16, 4968-4972
7156306 CIFC34 H46 N4 O3 S2P 21 21 2113.5505; 14.85; 16.762
90; 90; 90
3372.9Huang, Yin-Hui; Jin, Xian-Yi; Zhao, Yong-Yi; Cong, Hang; Tao, Zhu
A fluorescence-enhanced chemosensor based on multifarene[2,2] and its recognition of metal cations.
Organic & biomolecular chemistry, 2018, 16, 5343-5349
7156308 CIFC43 H38 N2 OP 21 21 218.7773; 16.6542; 21.9525
90; 90; 90
3209Wu, Jia-Le; Wang, Cong-Shuai; Wang, Jin-Rong; Mei, Guang-Jian; Shi, Feng
A catalytic asymmetric interrupted Nazarov-type cyclization of 2-indolylmethanols with cyclic enaminones.
Organic & biomolecular chemistry, 2018, 16, 5457-5464
7156326 CIFC24 H24 Br N3 O4 S2P 21 21 218.7914; 16.8836; 17.728
90; 90; 90
2631.4Xu, Han; Kang, Tian-Chen; Sha, Feng; Wu, Xin-Yan
Enantioselective Mannich reaction between rhodanines and isatin-derived ketimines to construct vicinal tetrasubstituted stereocenters.
Organic & biomolecular chemistry, 2018, 16, 5780-5787
7156329 CIFC21 H30 N2 O7P 21 21 218.5893; 11.638; 22.452
90; 90; 90
2244.4Niwetmarin, Worawat; Rego Campello, Hugo; Sparkes, Hazel A.; Aggarwal, Varinder K.; Gallagher, Timothy
(-)-Cytisine: Access to a stereochemically defined and functionally flexible piperidine scaffold.
Organic & biomolecular chemistry, 2018, 16, 5823-5832
7156350 CIFC42 H35.85 Cl4.15 N4 O8P 21 21 2110.5565; 14.9406; 25.9563
90; 90; 90
4093.84Butler, Nicholas M.; Hendra, Rudi; Bremner, John B.; Willis, Anthony C.; Lucantoni, Leonardo; Avery, Vicky M.; Keller, Paul A.
Cascade reactions of indigo with oxiranes and aziridines: efficient access to dihydropyrazinodiindoles and spiro-oxazocinodiindoles.
Organic & biomolecular chemistry, 2018, 16, 6006-6016
7156351 CIFC22 H18 N2 O4P 21 21 218.6464; 11.41283; 17.69376
90; 90; 90
1746.02Butler, Nicholas M.; Hendra, Rudi; Bremner, John B.; Willis, Anthony C.; Lucantoni, Leonardo; Avery, Vicky M.; Keller, Paul A.
Cascade reactions of indigo with oxiranes and aziridines: efficient access to dihydropyrazinodiindoles and spiro-oxazocinodiindoles.
Organic & biomolecular chemistry, 2018, 16, 6006-6016
7156354 CIFC55 H58 N2 O9 SP 21 21 2111.1611; 18.4375; 23.2735
90; 90; 90
4789.3Łęczycka-Wilk, Katarzyna; Ulatowski, Filip; Cmoch, Piotr; Jarosz, Sławomir
"Choose-a-size" control in the synthesis of sucrose based urea and thiourea macrocycles.
Organic & biomolecular chemistry, 2018, 16, 6063-6069
7156381 CIFC140 H160 N8 O24P 21 21 217.9683; 16.3532; 23.8547
90; 90; 90
3108.4Wu, Xiao-Na; You, Zhi-Hao; Liu, Yan-Kai
Different hybridized oxygen atoms controlled chemoselective formation of oxocarbenium ions: synthesis of chiral heterocyclic compounds.
Organic & biomolecular chemistry, 2018, 16, 6507-6520
7156386 CIFC45 H45 Cl N O7 P PdP 21 21 219.1935; 14.7832; 30.8543
90; 90; 90
4193.39Russell, David A.; Freudenreich, Julien J.; Stewart, Hannah L.; Bond, Andrew D.; Sore, Hannah F.; Spring, David R.
Semi-syntheses of the 11-hydroxyrotenoids sumatrol and villosinol.
Organic & biomolecular chemistry, 2018, 16, 6395-6398
7156407 CIFC14 H18 O6P 21 21 215.0069; 9.5409; 26.84
90; 90; 90
1282.16Verma, Ashish Kumar; Chennaiah, Ande; Dubbu, Sateesh; Vankar, Yashwant D.
Stereoselective synthesis of sugar-fused (or 1,2-annulated) isochromans and isochromanones by using oxa-Pictet-Spengler reaction.
Organic & biomolecular chemistry, 2018, 16, 8258-8262
7156430 CIFC26 H20 N2P 21 21 216.9592; 9.9148; 27.7881
90; 90; 90
1917.35Bulman Page, Philip C.; Kinsey, Francesca S.; Chan, Yohan; Strutt, Ian R.; Slawin, Alexandra M. Z.; Jones, Garth A.
Novel binaphthyl and biphenyl α- and β-amino acids and esters: organocatalysis of asymmetric Diels-Alder reactions. A combined synthetic and computational study.
Organic & biomolecular chemistry, 2018, 16, 7400-7416
7156431 CIFC19 H18 F3 N O4P 21 21 2110.5475; 20.671; 24.988
90; 90; 90
5448.1Bulman Page, Philip C.; Kinsey, Francesca S.; Chan, Yohan; Strutt, Ian R.; Slawin, Alexandra M. Z.; Jones, Garth A.
Novel binaphthyl and biphenyl α- and β-amino acids and esters: organocatalysis of asymmetric Diels-Alder reactions. A combined synthetic and computational study.
Organic & biomolecular chemistry, 2018, 16, 7400-7416
7156433 CIFC24 H19 N O2P 21 21 217.6334; 14.828; 15.793
90; 90; 90
1787.6Bulman Page, Philip C.; Kinsey, Francesca S.; Chan, Yohan; Strutt, Ian R.; Slawin, Alexandra M. Z.; Jones, Garth A.
Novel binaphthyl and biphenyl α- and β-amino acids and esters: organocatalysis of asymmetric Diels-Alder reactions. A combined synthetic and computational study.
Organic & biomolecular chemistry, 2018, 16, 7400-7416
7156436 CIFC11 H11 F O2P 21 21 215.605; 7.129; 24.013
90; 90; 90
959.5Minhas, Harsimran K.; Riley, William; Stuart, Alison M.; Urbonaite, Martyna
Activation of the hypervalent fluoroiodane reagent by hydrogen bonding to hexafluoroisopropanol.
Organic & biomolecular chemistry, 2018, 16, 7170-7173
7156437 CIFC26 H17 Br O5P 21 21 218.3403; 15.6568; 16.7849
90; 90; 90
2191.81Xu, Han; Sha, Feng; Li, Qiong; Wu, Xin-Yan
Catalytic asymmetric Tamura cycloaddition of homophthalic anhydrides with 2-arylidene-1,3-diones.
Organic & biomolecular chemistry, 2018, 16, 7214-7222
7156449 CIFC31 H28 F2 N2 O SP 21 21 219.0912; 17.553; 20.148
90; 90; 90
3215.2Liu, Feng; Zhao, Guoqing; Cai, Weiqi; Xu, Dongfang; Zhao, Baoguo
Aminative Umpolung cyclization for synthesis of chiral exocyclic vicinal diamines.
Organic & biomolecular chemistry, 2018, 16, 7498-7502
7156457 CIFC141 H157 Cl3 N8 O8P 21 21 2115.6212; 31.4079; 25.8937
90; 90; 90
12704.2Liu, Qiuhua; Zhang, Jinjin; Tang, Min; Yang, Yan; Zhang, Jian; Zhou, Zaichun
Geometric deconstruction of core and electron activation of a π-system in a series of deformed porphyrins: mimics of heme.
Organic & biomolecular chemistry, 2018, 16, 7725-7736
7156463 CIFC66 H70 N4 O4P 21 21 2116.2769; 18.6656; 19.3939
90; 90; 90
5892.2Liu, Qiuhua; Zhang, Jinjin; Tang, Min; Yang, Yan; Zhang, Jian; Zhou, Zaichun
Geometric deconstruction of core and electron activation of a π-system in a series of deformed porphyrins: mimics of heme.
Organic & biomolecular chemistry, 2018, 16, 7725-7736
7156490 CIFC29 H24 O3 SP 21 21 217.942; 16.844; 17.488
90; 90; 90
2339Jadhav, Sandip B.; Thopate, Satish B.; Nanubolu, Jagadeesh Babu; Chegondi, Rambabu
Rh-Catalyzed diastereoselective desymmetrization of enone tethered-cyclohexadienones via tandem arylative cyclization.
Organic & biomolecular chemistry, 2019, 17, 1937-1946
7156491 CIFC40 H62 O7P 21 21 2110.994; 17.4175; 19.4407
90; 90; 90
3722.66Guo, Yi; Zhang, Na; Sun, Weiguang; Duan, Xueyan; Zhang, Qing; Zhou, Qun; Chen, Chunmei; Zhu, Hucheng; Luo, Zengwei; Liu, Junjun; Li, Xiao-Nian; Xue, Yongbo; Zhang, Yonghui
Bioactive polycyclic polyprenylated acylphloroglucinols from Hypericum perforatum.
Organic & biomolecular chemistry, 2018, 16, 8130-8143
7156510 CIFC28 H30 F6 N4 O4 SP 21 21 2110.0847; 12.3157; 23.0056
90; 90; 90
2857.3Claveau, Romain; Twamley, Brendan; Connon, Stephen J.
Synthesis of α-alkylated γ-butyrolactones with concomitant anhydride kinetic resolution using a sulfamide-based catalyst.
Organic & biomolecular chemistry, 2018, 16, 7574-7578
7156518 CIFC25 H17 Br N4P 21 21 217.7966; 14.3031; 18.1018
90; 90; 90
2018.6Deka, Bhaskar; Baruah, Pranjal K.; Deb, Mohit L.
Multi-component synthesis of 3-substituted indoles and their cyclisation to α-carbolines via I<sub>2</sub>-promoted intramolecular C2 oxidative amination/aromatisation at room temperature.
Organic & biomolecular chemistry, 2018, 16, 7806-7810
7156519 CIFC35 H48 O7P 21 21 2111.2746; 16.1738; 18.2342
90; 90; 90
3325.06Hou, Ji-Qin; Wang, Bao-Lin; Han, Chao; Xu, Jian; Wang, Zhe; He, Qi-Wei; Zhang, Pei-Lin; Zhao, Shu-Min; Pei, Xin; Wang, Hao
Atropisomeric meroterpenoids with rare triketone-phloroglucinol-terpene hybrids from Baeckea frutescens.
Organic & biomolecular chemistry, 2018, 16, 8513-8524
7156523 CIFC16 H19 F3 I N OP 21 21 2111.6524; 15.998; 18.6279
90; 90; 90
3472.5Shi, Yingkun; Xiao, Hongqing; Xu, Xiu-Hua; Huang, Yangen
Transition metal free decarboxylative fluoroalkylation of N-acrylamides with 3,3,3-trifluoro-2,2-dimethylpropanoic acid (TFDMPA).
Organic & biomolecular chemistry, 2018, 16, 8472-8476
7156534 CIFC16 H23 N O2P 21 21 219.8834; 10.2262; 13.9008
90; 90; 90
1404.95Li, Tao; Wu, Guangmiao; Feng, Shangbiao; Wang, Zemin; Xie, Xingang; She, Xuegong
A rapid construction of the ABC tricyclic skeleton of malabanone A.
Organic & biomolecular chemistry, 2018, 16, 8491-8494
7156535 CIFC16 H23 N O2P 21 21 217.3868; 17.0662; 23.1039
90; 90; 90
2912.6Li, Tao; Wu, Guangmiao; Feng, Shangbiao; Wang, Zemin; Xie, Xingang; She, Xuegong
A rapid construction of the ABC tricyclic skeleton of malabanone A.
Organic & biomolecular chemistry, 2018, 16, 8491-8494
7156543 CIFC21 H32 O5P 21 21 218.8265; 21.615; 30.7813
90; 90; 90
5872.6Li, Fengli; Sun, Weiguang; Guan, Jiankun; Lu, Yuanyuan; Lin, Shuang; Zhang, Sitian; Gao, Weixi; Liu, Junjun; Du, Guang; Wang, Jianping; Zhu, Hucheng; Qi, Changxing; Hu, Zhengxi; Zhang, Yonghui
Anti-inflammatory fusicoccane-type diterpenoids from the phytopathogenic fungus Alternaria brassicicola.
Organic & biomolecular chemistry, 2018, 16, 8751-8760
7156546 CIFC19 H28 O2P 21 21 219.0892; 9.9719; 17.8361
90; 90; 90
1616.6Li, Fengli; Sun, Weiguang; Guan, Jiankun; Lu, Yuanyuan; Lin, Shuang; Zhang, Sitian; Gao, Weixi; Liu, Junjun; Du, Guang; Wang, Jianping; Zhu, Hucheng; Qi, Changxing; Hu, Zhengxi; Zhang, Yonghui
Anti-inflammatory fusicoccane-type diterpenoids from the phytopathogenic fungus Alternaria brassicicola.
Organic & biomolecular chemistry, 2018, 16, 8751-8760
7156548 CIFC46 H37 F2 N4 O4 S2P 21 21 218.434; 10.662; 44.27
90; 90; 90
3981Li, Weihua; Wang, Yifeng; Xu, Danqian
Asymmetric synthesis of β-amino ketones by using cinchona alkaloid-based chiral phase transfer catalysts.
Organic & biomolecular chemistry, 2018, 16, 8704-8709
7156552 CIFC68 H68 Cl4 F12 N4 O8 S4P 21 21 2115.1112; 15.5876; 31.4003
90; 90; 90
7396.3Qin, Tian; Jiang, Quanbin; Ji, Jieying; Luo, Jie; Zhao, Xiaodan
Chiral selenide-catalyzed enantioselective synthesis of trifluoromethylthiolated 2,5-disubstituted oxazolines.
Organic & biomolecular chemistry, 2019, 17, 1763-1766
7156554 CIFC23 H20 Cl F N2 O3 SP 21 21 219.5099; 9.7883; 23.6429
90; 90; 90
2200.82Zheng, Bu-Quan; Chen, Ling-Yan; Zhao, Jian-Bo; Ji, Jian; Qiu, Zi-Bin; Ren, Xinfeng; Li, Ya
Organocatalytic asymmetric syntheses of 3-fluorooxindoles containing vicinal fluoroamine motifs.
Organic & biomolecular chemistry, 2018, 16, 8989-8993
7156557 CIFC27 H38 O9P 21 21 2111.4298; 14.3863; 15.3115
90; 90; 90
2517.7Qi, Changxing; Qiao, Yuben; Gao, Weixi; Liu, Mengting; Zhou, Qun; Chen, Chunmei; Lai, Yongji; Xue, Yongbo; Zhang, Jinwen; Li, Dongyan; Wang, Jianping; Zhu, Hucheng; Hu, Zhengxi; Zhou, Yuan; Zhang, Yonghui
New 3,5-dimethylorsellinic acid-based meroterpenoids with BACE1 and AchE inhibitory activities from Aspergillus terreus.
Organic & biomolecular chemistry, 2018, 16, 9046-9052
7156562 CIFC15 H24 O3P 21 21 2110.44121; 11.19736; 11.7174
90; 90; 90
1369.93Wu, Pei-Qian; Yu, Yi-Fan; Zhao, Ye; Yu, Chun-Xue; Zhi, De-Juan; Qi, Feng-Ming; Fei, Dong-Qing; Zhang, Zhan-Xin
Four novel sesquiterpenoids with their anti-Alzheimer's disease activity from Nardostachys chinensis.
Organic & biomolecular chemistry, 2018, 16, 9038-9045
7156563 CIFC20 H20 Cl N O3P 21 21 215.32172; 11.65514; 28.13606
90; 90; 90
1745.15Huang, Yi; Li, Pan; Dong, Xiu-Qin; Zhang, Xumu
Synthesis of chiral seven-membered β-substituted lactams via Rh-catalyzed asymmetric hydrogenation.
Organic & biomolecular chemistry, 2018, 16, 8819-8823
7156564 CIFC41 H58 O7P 21 21 2112.9237; 15.5472; 39.6257
90; 90; 90
7961.9Wang, Wen-Li; Zhu, Dong-Rong; Luo, Jie; Liu, Fei-Yan; Chen, Chen; Zhu, Tian-Yu; Li, Ling-Nan; Han, Chao; Luo, Jian-Guang; Kong, Ling-Yi
Taiwanoids A-D, four dimeric diterpenoids featuring tetracyclic [7. 7<sup>5, 9</sup>. 4. 0<sup>5, 10</sup>. 0<sup>8, 9</sup>] octodecane from Taiwania cryptomerioidesim.
Organic & biomolecular chemistry, 2018, 16, 9059-9063
7156569 CIFC2.3 H2.15 N0.15 O0.44P 21 21 218.4217; 17.9017; 18.0406
90; 90; 90
2719.9Liu, Yuxin; Wang, Jingdong; Wei, Zhonglin; Cao, Jungang; Liang, Dapeng; Lin, Yingjie; Duan, Haifeng
Direct enantio- and diastereoselective Mannich reactions of isatin-derived ketimines with oxo-indanecarboxylates catalyzed by chiral thiourea derived from hydroquinidine.
Organic & biomolecular chemistry, 2018, 16, 8927-8932
7156587 CIFC26 H34 O5P 21 21 217.7671; 16.3554; 17.5789
90; 90; 90
2233.12Ma, Shuang-Jiang; Yu, Jie; Yan, Da-Wei; Wang, Da-Cheng; Gao, Jin-Ming; Zhang, Qiang
Meroterpene-like compounds derived from β-caryophyllene as potent α-glucosidase inhibitors
Organic & Biomolecular Chemistry, 2018
7156589 CIFC39 H53 N O6P 21 21 2113.9171; 18.5603; 27.189
90; 90; 90
7023.1Ma, Shuang-Jiang; Yu, Jie; Yan, Da-Wei; Wang, Da-Cheng; Gao, Jin-Ming; Zhang, Qiang
Meroterpene-like compounds derived from β-caryophyllene as potent α-glucosidase inhibitors
Organic & Biomolecular Chemistry, 2018
7156592 CIFC10 H7 F3 O3P 21 21 219.877; 11.908; 16.045
90; 90; 90
1887Yan, Weitao; Wang, Ruo; Zhang, Tesen; Deng, Hongtao; Chen, Jian; Wu, Wei; Weng, Zhiqiang
Synthesis of 4-trifluoromethyl 2-pyrones and pyridones through the Brønsted base-catalyzed Pechmann-type reaction with cyclic 1,3-diones.
Organic & biomolecular chemistry, 2018, 16, 9440-9445
7156606 CIFC20 H32 O11P 21 21 216.9268; 7.6212; 39.643
90; 90; 90
2092.8Wang, Junfeng; Qin, Li; Zhao, Biqing; Cai, Liang; Zhong, Zhenping; Liu, Yonghong; Zhou, Xiaojiang
Crotonols A and B, two rare tigliane diterpenoid derivatives against K562 cells from Croton tiglium.
Organic & biomolecular chemistry, 2018, 17, 195-202
7156607 CIFC15 H17 N OP 21 21 217.1064; 10.3163; 15.973
90; 90; 90
1171Xu, Dawen; Kaiser, Felix; Li, Han; Reich, Robert M.; Guo, Hao; Kühn, Fritz E
Highly selective AlCl<sub>3</sub> initiated intramolecular α-alkylation of α,β-unsaturated lactams and lactones.
Organic & biomolecular chemistry, 2018, 17, 49-52
7156619 CIFC13 H10 Br Cl N2 O2P 21 21 215.9701; 7.3338; 31.4408
90; 90; 90
1376.59Yu, Kun-Ming; Zhu, Hui-Kai; Zhao, Xiao-Li; Shi, Min; Zhao, Mei-Xin
Organocatalyzed asymmetric tandem conjugate addition-protonation of isocyanoacetates to 2-chloroacrylonitrile.
Organic & biomolecular chemistry, 2019, 17, 639-645
7156621 CIFC36 H49 N O3P 21 21 217.3603; 16.4621; 24.344
90; 90; 90
2949.7Khusnutdinova, Elmira F.; Kazakova, Oxana B.; Lobov, Alexander N.; Kukovinets, Olga S.; Suponitsky, Kyrill Yu; Meyers, Craig B.; Prichard, Mark N.
Synthesis of A-ring quinolones, nine-membered oxolactams and spiroindoles by oxidative transformations of 2,3-indolotriterpenoids.
Organic & biomolecular chemistry, 2019, 17, 585-597
7156625 CIFC35 H30 O5P 21 21 2111.362; 15.3627; 16.0741
90; 90; 90
2805.8Intakaew, Neeranuth; Rithchumpon, Puracheth; Prommin, Chanatkran; Yimklan, Saranphong; Kungwan, Nawee; Thavornyutikarn, Praput; Meepowpan, Puttinan
Synthesis and characterization of novel chiral derivatizing agents containing β-keto-anthracene adducts (KAAs) by <sup>1</sup>H-NMR: aromatic influence and chiral alcohol absolute configuration determination.
Organic & biomolecular chemistry, 2019, 17, 541-554
7156643 CIFC14 H9 Br O2P 21 21 216.1663; 11.1767; 16.5802
90; 90; 90
1142.69Carlos, Andressa M. M.; Stieler, Rafael; Lüdtke, Diogo S
Catalytic asymmetric synthesis of 3-aryl phthalides enabled by arylation-lactonization of 2-formylbenzoates.
Organic & biomolecular chemistry, 2019, 17, 283-289
7156654 CIFC42 H41 Cl3 N PP 21 21 2110.1412; 17.5089; 19.7319
90; 90; 90
3503.62Mino, Takashi; Yamaguchi, Daiki; Masuda, Chihiro; Youda, Junpei; Ebisawa, Toshibumi; Yoshida, Yasushi; Sakamoto, Masami
Synthesis and application of P,olefin type axially chiral ligands with sec-alkyl groups.
Organic & biomolecular chemistry, 2019, 17, 1455-1465
7156661 CIFC24 H22 O4 SP 21 21 216.7899; 16.6281; 18.1779
90; 90; 90
2052.3Zehra, Syeda Tazeen; Zhang, Guoxiang; Yang, Shuang; Fang, Xinqiang
Kinetic resolution of β-ketoesters with quaternary stereocenters via a carbene-catalyzed benzoin reaction.
Organic & biomolecular chemistry, 2019, 17, 2169-2173
7156673 CIFC31 H38 O10P 21 21 2111.8058; 12.6003; 19.4463
90; 90; 90
2892.8He, Jun; Xu, Jie-Kun; Zhang, Jia; Bai, Hong-Jin; Ma, Bing-Zhi; Cheng, Yung-Chi; Zhang, Wei-Ku
Fischeriana A, a meroterpenoid with an unusual 6/6/5/5/5/6/6 heptacyclic carbon skeleton from the roots of Euphorbia fischeriana.
Organic & biomolecular chemistry, 2019, 17, 2721-2724
7156677 CIFC17 H16 Cl N O4P 21 21 215.7177; 7.7029; 35.315
90; 90; 90
1555.4Sengoku, Tetsuya; Ikeda, Ikuhei; Ai, Keisuke; Takahashi, Masaki; Yoda, Hidemi
Indium- and zinc-catalyzed enantioselective amide propargylation of aldehydes with stannylated allenyl amides.
Organic & biomolecular chemistry, 2019, 17, 2614-2618
7156682 CIFC26 H26 O5P 21 21 218.2235; 15.8364; 17.2177
90; 90; 90
2242.3Khanvilkar, Aditya N.; Samanta, Sudeep G.; Bedekar, Ashutosh V.
Applications of chiral naphthyloxycyclohexanols in deracemization of α-substituted carboxylic acids by dynamic thermodynamic resolution.
Organic & biomolecular chemistry, 2019, 17, 2670-2683
7156684 CIFC26 H26 O5P 21 21 219.3173; 10.8597; 22.3122
90; 90; 90
2257.6Khanvilkar, Aditya N.; Samanta, Sudeep G.; Bedekar, Ashutosh V.
Applications of chiral naphthyloxycyclohexanols in deracemization of α-substituted carboxylic acids by dynamic thermodynamic resolution.
Organic & biomolecular chemistry, 2019, 17, 2670-2683
7156686 CIFC19 H21 Cl O3P 21 21 218.8657; 10.5557; 18.97
90; 90; 90
1775.3Khanvilkar, Aditya N.; Samanta, Sudeep G.; Bedekar, Ashutosh V.
Applications of chiral naphthyloxycyclohexanols in deracemization of α-substituted carboxylic acids by dynamic thermodynamic resolution.
Organic & biomolecular chemistry, 2019, 17, 2670-2683
7156688 CIFC20 H24 O8P 21 21 216.5026; 13.1145; 21.4093
90; 90; 90
1825.75Liu, Hong-Xin; Tan, Hai-Bo; Chen, Kai; Zhao, Li-Yun; Chen, Yu-Chan; Li, Sai-Ni; Li, Hao-Hua; Zhang, Wei-Min
Cytosporins A-D, novel benzophenone derivatives from the endophytic fungus Cytospora rhizophorae A761.
Organic & biomolecular chemistry, 2019, 17, 2346-2350
7156713 CIFC26 H22 Cl NP 21 21 2110.141; 10.4626; 19.267
90; 90; 90
2044.3Uruvakili, Anasuyamma; Kumara Swamy, K. C.
Gold catalysed transformation of 2-arylindoles to terphenyl amines via 3-dienyl indoles and Brønsted acid promoted formation of 2-carboxyindoles to 3-indenylindoles via 3-allenylindoles.
Organic & biomolecular chemistry, 2019, 17, 3275-3284
7156757 CIFC34 H28 Cl N3 O3P 21 21 216.2201; 12.705; 35.317
90; 90; 90
2791Hutskalova, Valeriia; Mykhailiuk, Pavel K.
Pd-Catalyzed directed CH-(hetero)arylation of cyclic α-amino acids: effects of substituents and the ring size.
Organic & biomolecular chemistry, 2019, 17, 4342-4349
7156769 CIFC17 H17 N O2P 21 21 217.21212; 15.4816; 26.0416
90; 90; 90
2907.68Ghosh, Arnab; Hegde, Rajeev; Makane, Vitthal B.; Sridhar, Balasubramanian; Rode, Haridas B.; Patil, Siddappa A.; Dateer, Ramesh B.
Transition metal-free functionalized hydration of alkynes: one-pot synthesis of fluorinated β-keto-imidates using Selectfluor.
Organic & biomolecular chemistry, 2019, 17, 4440-4445
7156810 CIFC30 H24 O2 SP 21 21 217.6174; 26.721; 34.0314
90; 90; 90
6926.9Feng, Ze-Nan; Luo, Jin-Yun; Zhang, Yang; Du, Guang-Fen; He, Lin
N-Heterocyclic carbene-catalyzed diastereoselective synthesis of sulfenylated indanes via sulfa-Michael-Michael (aldol) cascade reactions.
Organic & biomolecular chemistry, 2019, 17, 4700-4704
7156820 CIFC28 H16 N4 O16P 21 21 219.7079; 14.071; 20.822
90; 90; 90
2844.3Ma, Jiao-Xia; Fang, Xu; Xue, Min; Yang, Yong
Synthesis, structure, and anion binding of functional oxacalix[4]arenes.
Organic & biomolecular chemistry, 2019, 17, 5075-5085
7156841 CIFC22 H19 I N3 O2 PP 21 21 218.3026; 8.563; 30.125
90; 90; 90
2141.74Anitha, Mandala; Kumara Swamy, K. C.
Highly functionalised (γ-azido/γ-fluoro-β-iodo/)vinyl derivatives from phosphorus based allenes or allenoates: IO halogen bonding interactions.
Organic & biomolecular chemistry, 2019, 17, 5736-5748
7156849 CIFC21 H16 Cl I N3 O PP 21 21 2129.548; 8.3033; 8.5609
90; 90; 90
2100.4Anitha, Mandala; Kumara Swamy, K. C.
Highly functionalised (γ-azido/γ-fluoro-β-iodo/)vinyl derivatives from phosphorus based allenes or allenoates: IO halogen bonding interactions.
Organic & biomolecular chemistry, 2019, 17, 5736-5748
7156861 CIFC23 H24 Cl F N2 O3 SP 21 21 216.8998; 11.7197; 26.4465
90; 90; 90
2138.56Panduwawala, Tharindi D.; Iqbal, Sarosh; Thompson, Amber L.; Genov, Miroslav; Pretsch, Alexander; Pretsch, Dagmar; Liu, Shuang; Ebright, Richard H.; Howells, Alison; Maxwell, Anthony; Moloney, Mark G.
Functionalised bicyclic tetramates derived from cysteine as antibacterial agents.
Organic & biomolecular chemistry, 2019, 17, 5615-5632
7156862 CIFC21 H22 O4 SP 21 21 217.5793; 15.2528; 15.4509
90; 90; 90
1786.21Palange, Megha N.; Gonnade, Rajesh G.; Kontham, Ravindar
TiCl<sub>4</sub>-n-Bu<sub>3</sub>N-mediated cascade annulation of ketones with α-ketoesters: a facile synthesis of highly substituted fused γ-alkylidene-butenolides.
Organic & biomolecular chemistry, 2019, 17, 5749-5759
7156867 CIFC6 H8 F2 O3P 21 21 215.6134; 10.6394; 21.7983
90; 90; 90
1301.86Malassis, Julien; Vendeville, Jean-Baptiste; Nguyen, Qui-Hien; Boujon, Marie; Gaignard-Gaillard, Quentin; Light, Mark; Linclau, Bruno
Synthesis of vicinal dideoxy-difluorinated galactoses.
Organic & biomolecular chemistry, 2019, 17, 5331-5340
7156868 CIFC6 H10 F2 O4P 21 21 218.3866; 8.4182; 10.232
90; 90; 90
722.38Malassis, Julien; Vendeville, Jean-Baptiste; Nguyen, Qui-Hien; Boujon, Marie; Gaignard-Gaillard, Quentin; Light, Mark; Linclau, Bruno
Synthesis of vicinal dideoxy-difluorinated galactoses.
Organic & biomolecular chemistry, 2019, 17, 5331-5340
7156906 CIFC37 H47 N O11 SP 21 21 2110.2529; 11.3156; 39.0323
90; 90; 90
4528.44Wang, Kaiye; Xiang, Yanan; Shi, Zhujun; Wang, Hongyu; Li, Na; Tang, Bo
Asymmetric kinetic resolution of sulfides for the construction of unsymmetric sulfides and chiral 3,3-disubstituted oxindoles.
Organic & biomolecular chemistry, 2019, 17, 6351-6354
7156909 CIFC27 H25 N O5 SP 21 21 218.0766; 9.1009; 33.009
90; 90; 90
2426.3Zhao, Zi-Biao; Shi, Lei; Li, Yaming; Meng, Fan-Jie; Zhou, Yong-Gui
Facile synthesis of chiral ε-sultams via an organocatalytic aza-Friedel-Crafts reaction.
Organic & biomolecular chemistry, 2019, 17, 6364-6368
7156927 CIFC21 H19 N3 O2P 21 21 217.6371; 14.5261; 16.1757
90; 90; 90
1794.49Pilicer, Samantha L.; Mancinelli, Michele; Mazzanti, Andrea; Wolf, Christian
Predictive chirality sensing via Schiff base formation.
Organic & biomolecular chemistry, 2019, 17, 6699-6705
7156929 CIFC34 H35.51 N5 O7 SP 21 21 2110.6941; 16.3625; 18.2683
90; 90; 90
3196.63Chen, Shuang; Wang, Guan-Lian; Xu, Sheng-Wen; Tian, Min-Yi; Zhang, Min; Liu, Xiong-Li; Yuan, Wei-Cheng
Regio- and stereoselective [3 + 2] cycloaddition reaction: access to isoxazole-dispirobisoxindoles featuring three contiguous stereocenters.
Organic & biomolecular chemistry, 2019, 17, 6551-6556
7156930 CIFC33 H33 N5 O7 SP 21 21 2111.1703; 15.8824; 18.1124
90; 90; 90
3213.34Chen, Shuang; Wang, Guan-Lian; Xu, Sheng-Wen; Tian, Min-Yi; Zhang, Min; Liu, Xiong-Li; Yuan, Wei-Cheng
Regio- and stereoselective [3 + 2] cycloaddition reaction: access to isoxazole-dispirobisoxindoles featuring three contiguous stereocenters.
Organic & biomolecular chemistry, 2019, 17, 6551-6556
7156937 CIFC72 H58 B F24 N2 Na O8P 21 21 2118.8583; 19.3929; 19.5642
90; 90; 90
7155Homberg, Alexandre; Hrdina, Radim; Vishe, Mahesh; Guénée, Laure; Lacour, Jérôme
Stereoselective deconjugation of macrocyclic α,β-unsaturated esters by sequential amidation and olefin transposition: application to enantioselective phase-transfer catalysis.
Organic & biomolecular chemistry, 2019, 17, 6905-6910
7156940 CIFC24 H27 N O3P 21 21 219.7132; 14.1931; 14.3361
90; 90; 90
1976.38Houston, Sevan D.; Fahrenhorst-Jones, Tyler; Xing, Hui; Chalmers, Benjamin A.; Sykes, Melissa L.; Stok, Jeanette E.; Farfan Soto, Clementina; Burns, Jed M.; Bernhardt, Paul V.; De Voss, James J.; Boyle, Glen M.; Smith, Maree T.; Tsanaktsidis, John; Savage, G. Paul; Avery, Vicky M.; Williams, Craig M.
The cubane paradigm in bioactive molecule discovery: further scope, limitations and the cyclooctatetraene complement.
Organic & biomolecular chemistry, 2019, 17, 6790-6798
7156949 CIFC35 H14 F14 O2P 21 21 216.2739; 20.464; 23.723
90; 90; 90
3045.8Yamada, Shigeyuki; Nishizawa, Akito; Morita, Masato; Hosokai, Takuya; Okabayashi, Yusuke; Agou, Tomohiro; Hosoya, Takaaki; Kubota, Toshio; Konno, Tsutomu
Synthesis and characterization of bent fluorine-containing donor-π-acceptor molecules as intense luminophores with large Stokes shifts.
Organic & biomolecular chemistry, 2019, 17, 6911-6919
7156964 CIFC24 H25 N O6P 21 21 215.53; 12.216; 32.227
90; 90; 90
2177.1Luo, Jinghua; Chen, Rongshun; Fan, Xia; Gong, Junyu; Han, Jie; He, Zhengjie
Catalytic asymmetric (4 + 1) annulation of nitroalkenes with allylic acetates: stereoselective synthesis of isoxazoline N-oxides.
Organic & biomolecular chemistry, 2019, 17, 6989-6993
7156965 CIFC25 H20 Br F N4 O2P 21 21 216.4813; 16.177; 21.944
90; 90; 90
2300.8Zhang, Qing-Da; Zhao, Bo-Liang; Li, Bing-Yu; Du, Da-Ming
Squaramide-catalyzed asymmetric Mannich reactions between 3-fluorooxindoles and pyrazolinone ketimines.
Organic & biomolecular chemistry, 2019, 17, 7182-7191
7156969 CIFC46 H42 N6 O11P 21 21 2114.1242; 14.398; 20.2906
90; 90; 90
4126.3Miao, Yu-Hang; Hua, Yuan-Zhao; Wang, Min-Can
Dinuclear zinc cooperative catalytic three-component reactions for highly enantioselective synthesis of 3,3'-dihydrofuran spirooxindoles.
Organic & biomolecular chemistry, 2019, 17, 7172-7181
7156970 CIFC10 H19 Cl N O4P 21 21 217.9383; 8.9382; 16.392
90; 90; 90
1163.08Foucart, Quentin; Shimadate, Yuna; Marrot, Jérôme; Kato, Atsushi; Désiré, Jérôme; Blériot, Yves
Synthesis and glycosidase inhibition of conformationally locked DNJ and DMJ derivatives exploiting a 2-oxo-C-allyl iminosugar.
Organic & biomolecular chemistry, 2019, 17, 7204-7214
7156972 CIFC17 H12 N2 O2P 21 21 218.2455; 11.3533; 13.652
90; 90; 90
1278Ahire, Milind M.; Pol, Mahesh D.; Kavale, Dattatry S.; Gonnade, Rajesh G.; Mhaske, Santosh B.
Stereoselective construction of deoxy-cruciferane alkaloids by NHC-catalyzed intramolecular annulation of homoenolate with quinazolinone.
Organic & biomolecular chemistry, 2019, 17, 7135-7139
7156973 CIFC23 H23 N O6P 21 21 218.7557; 14.297; 16.454
90; 90; 90
2059.7Shahrestani, Naeimeh; Khosravi, Hormoz; Jadidi, Khosrow; Notash, Behrouz; Naderi, Soheila
Organocatalytic synthesis of enantiopure spiro acenaphthyl-pyrrolizidine/pyrrolidines: justifying the regioselectivity based on a distortion/interaction model.
Organic & biomolecular chemistry, 2019, 17, 7013-7024
7156974 CIFC28 H26 N2 O4P 21 21 218.1876; 14.121; 19.915
90; 90; 90
2302.5Shahrestani, Naeimeh; Khosravi, Hormoz; Jadidi, Khosrow; Notash, Behrouz; Naderi, Soheila
Organocatalytic synthesis of enantiopure spiro acenaphthyl-pyrrolizidine/pyrrolidines: justifying the regioselectivity based on a distortion/interaction model.
Organic & biomolecular chemistry, 2019, 17, 7013-7024
7156975 CIFC30 H28 N2 O4P 21 21 218.5232; 13.562; 21.283
90; 90; 90
2460.1Shahrestani, Naeimeh; Khosravi, Hormoz; Jadidi, Khosrow; Notash, Behrouz; Naderi, Soheila
Organocatalytic synthesis of enantiopure spiro acenaphthyl-pyrrolizidine/pyrrolidines: justifying the regioselectivity based on a distortion/interaction model.
Organic & biomolecular chemistry, 2019, 17, 7013-7024
7156978 CIFC37 H48 O10P 21 21 219.751; 16.7972; 20.8431
90; 90; 90
3413.9Salin, Alexey V.; Islamov, Daut R.
Phosphine-catalyzed Michael additions to α-methylene-γ-butyrolactones.
Organic & biomolecular chemistry, 2019, 17, 7293-7299
7156981 CIFC27 H29 O4 PP 21 21 216.0344; 31.7014; 12.0302
90; 90; 90
2301.36Salin, Alexey V.; Islamov, Daut R.
Phosphine-catalyzed Michael additions to α-methylene-γ-butyrolactones.
Organic & biomolecular chemistry, 2019, 17, 7293-7299
7156993 CIFC35 H31 Br N2 O4 SP 21 21 217.2208; 16.3286; 27.1076
90; 90; 90
3196.1Franc, Michael; Urban, Michal; Císařová, Ivana; Veselý, Jan
Highly enantioselective addition of sulfur-containing heterocycles to isatin-derived ketimines.
Organic & biomolecular chemistry, 2019, 17, 7309-7314
7157005 CIFC28 H32 N2 SP 21 21 219.6029; 10.57062; 23.0787
90; 90; 90
2342.69Prusinowska, Natalia; Czapik, Agnieszka; Wojciechowska, Martika; Kwit, Marcin
Dynamic optical activity induction in the N-alkyl-N'-trityl ureas and thioureas.
Organic & biomolecular chemistry, 2019, 17, 7782-7793
7157031 CIFC30 H37 N O7P 21 21 2110.9844; 12.425; 19.6238
90; 90; 90
2678.28Wang, Wen-Xuan; Cheng, Gui-Guang; Li, Zheng-Hui; Ai, Hong-Lian; He, Juan; Li, Jing; Feng, Tao; Liu, Ji-Kai
Curtachalasins, immunosuppressive agents from the endophytic fungus Xylaria cf. curta.
Organic & biomolecular chemistry, 2019, 17, 7985-7994
7157032 CIFC47 H45 N O13P 21 21 2111.2462; 16.3107; 25.345
90; 90; 90
4649.1Lu, Kui; Li, Ming; Huang, Yuna; Sun, Yuanyuan; Gong, Zhi; Wei, Qijun; Zhao, Xia; Zhang, Yongmin; Yu, Peng
Total synthesis of wikstrol A and wikstrol B.
Organic & biomolecular chemistry, 2019, 17, 8206-8213
7157037 CIFC31 H45 O6P 21 21 219.97968; 10.81315; 27.7238
90; 90; 90
2991.72Duan, Yulin; Xie, Shuangshuang; Guo, Yi; Qiao, Yuben; Shi, Zhengyi; Tao, Li; Deng, Mengyi; Cao, Yunfang; Xue, Yongbo; Qi, Changxing; Zhang, Yonghui
Przewalcyrones A-F, epoxychromene-containing polycyclic polyprenylated acylphloroglucinols with immunosuppressive activity from Hypericum przewalskii Maxim.
Organic & biomolecular chemistry, 2019, 17, 8234-8242
7157044 CIFC38 H25 Cl N4 O4P 21 21 217.50014; 16.7058; 22.9329
90; 90; 90
2873.4Pozharskii, Alexander F.; Ozeryanskii, Valery A.; Mikshiev, Vladimir Y.; Chernyshev, Anatoly V.; Metelitsa, Anatoly V.; Antonov, Alexander S.
Proton-induced fluorescence in modified quino[7,8-h]quinolines: dual sensing for protons and π-donors.
Organic & biomolecular chemistry, 2019, 17, 8221-8233
7157049 CIFC22 H22 Br N5 O3P 21 21 2110.238; 10.6914; 19.2761
90; 90; 90
2109.93Zhang, Chen; Shang, Xinye; Cheng, Yuyu; Li, Fushuai; Zhao, Hanhui; Li, Pengfei; Li, Wenjun
Enantioselective construction of 3-substituted 3-amino-2-oxindoles containing an N,N-ketal skeleton via organocatalyzed aza-addition of isatin imines.
Organic & biomolecular chemistry, 2019, 17, 8374-8378
7157057 CIFC22 H32 O8P 21 21 2111.34869; 12.79403; 14.62274
90; 90; 90
2123.16Chen, Heng-Ye; Liu, Ting-Kai; Yang, Jian; Yang, Xiao-Long
Emerones A-C: three novel merosesquiterpenoids with unprecedented skeletons from Emericella sp. XL029.
Organic & biomolecular chemistry, 2019, 17, 8450-8455
7157058 CIFC21 H30 O7P 21 21 217.68291; 12.60214; 21.2697
90; 90; 90
2059.36Chen, Heng-Ye; Liu, Ting-Kai; Yang, Jian; Yang, Xiao-Long
Emerones A-C: three novel merosesquiterpenoids with unprecedented skeletons from Emericella sp. XL029.
Organic & biomolecular chemistry, 2019, 17, 8450-8455
7157068 CIFC30 H44 N O5 P SP 21 21 2110.584; 15.7917; 18.4493
90; 90; 90
3083.6Yuan, Minglei; Mbaezue, Ifenna I.; Zhou, Zhi; Topic, Filip; Tsantrizos, Youla S.
P-Chiral, N-phosphoryl sulfonamide Brønsted acids with an intramolecular hydrogen bond interaction that modulates organocatalysis.
Organic & biomolecular chemistry, 2019, 17, 8690-8694
7157069 CIFC10 H12 Br NP 21 21 2116.0321; 6.1532; 9.7828
90; 90; 90
965.06Yuan, Minglei; Mbaezue, Ifenna I.; Zhou, Zhi; Topic, Filip; Tsantrizos, Youla S.
P-Chiral, N-phosphoryl sulfonamide Brønsted acids with an intramolecular hydrogen bond interaction that modulates organocatalysis.
Organic & biomolecular chemistry, 2019, 17, 8690-8694
7157079 CIFC18 H13 Br O4P 21 21 218.8995; 12.8103; 13.9893
90; 90; 90
1594.85Shi, Taoda; Teng, Shenghan; Gopi Krishna Reddy, Alavala; Guo, Xin; Zhang, Yueteng; Moore, Kohlson T.; Buckley, Thomas; Mason, Damian J.; Wang, Wei; Chapman, Eli; Hu, Wenhao
Catalytic asymmetric synthesis of 2,5-dihydrofurans using synergistic bifunctional Ag catalysis.
Organic & biomolecular chemistry, 2019, 17, 8737-8744
7157081 CIFC21 H17 F N2 O2P 21 21 218.7924; 10.9272; 18.098
90; 90; 90
1738.79Xu, Yuanshuang; Zhang, Linghua; Liu, Mengyang; Zhang, Xiaopeng; Zhang, Xinying; Fan, Xuesen
Synthesis of benzoazepine derivatives via Rh(iii)-catalyzed inert C(sp<sup>2</sup>)-H functionalization and [4 + 3] annulation.
Organic & biomolecular chemistry, 2019, 17, 8706-8710
7157109 CIFC30 H36 Se2 Si2P 21 21 219.4081; 14.8474; 20.854
90; 90; 90
2913Hasegawa, Masashi; Kobayakawa, Kosuke; Nojima, Yuki; Mazaki, Yasuhiro
Synthesis and chiroptical properties of stereogenic cyclic dimers based on 2,2'-biselenophene and [2.2]paracyclophane.
Organic & biomolecular chemistry, 2019, 17, 8822-8826
7157123 CIFC28 H21 Cl N4 OP 21 21 217.5705; 11.9923; 27.772
90; 90; 90
2521.4Ji, Yan-Ling; Li, He-Ping; Ai, Yue-Yan; Li, Guo; He, Xiang-Hong; Huang, Wei; Huang, Rui-Zhen; Han, Bo
Enantio- and diastereoselective synthesis of spiropyrazolones via an organocatalytic [1 + 2 + 3] multicomponent reaction.
Organic & biomolecular chemistry, 2019, 17, 9217-9225
7157124 CIFC28 H21 Cl N4 OP 21 21 217.6734; 11.9044; 27.0141
90; 90; 90
2467.7Ji, Yan-Ling; Li, He-Ping; Ai, Yue-Yan; Li, Guo; He, Xiang-Hong; Huang, Wei; Huang, Rui-Zhen; Han, Bo
Enantio- and diastereoselective synthesis of spiropyrazolones via an organocatalytic [1 + 2 + 3] multicomponent reaction.
Organic & biomolecular chemistry, 2019, 17, 9217-9225
7157145 CIFC27 H24 N2 O5 SP 21 21 218.5917; 13.421; 21.279
90; 90; 90
2453.7Lu, Min; Li, Hong; Zou, Chuncheng; Li, Jianchang; Liu, Chengyu; Sun, Maolin; Ma, Yueyue; Cheng, Ruihua; Ye, Jinxing
Primary amine catalyzed diastereo- and enantioselective Michael reaction of thiazolones and α,β-unsaturated ketones.
Organic & biomolecular chemistry, 2019, 17, 9305-9312
7157147 CIFC25 H24 N2 O2 SP 21 21 219.0518; 12.1315; 18.9731
90; 90; 90
2083.47Luo, Shao-Xiong; Liu, Yanzhou; Lambrecht, Michael J.; Ortwine, Daniel F.; DiPasquale, Antonio G.; Liang, Jun; Wang, Xiaojing; Zbieg, Jason R.; Li, Jun
cis-Selective synthesis of 1,3-disubstituted tetrahydro-β-carbolines from N-sulfonyl N,S-acetals.
Organic & biomolecular chemistry, 2019, 17, 9510
7157148 CIFC23 H26 N2 O3 SP 21 21 219.2149; 11.3488; 19.7251
90; 90; 90
2062.81Luo, Shao-Xiong; Liu, Yanzhou; Lambrecht, Michael J.; Ortwine, Daniel F.; DiPasquale, Antonio G.; Liang, Jun; Wang, Xiaojing; Zbieg, Jason R.; Li, Jun
cis-Selective synthesis of 1,3-disubstituted tetrahydro-β-carbolines from N-sulfonyl N,S-acetals.
Organic & biomolecular chemistry, 2019, 17, 9510
7157162 CIFC24 H19 N O8P 21 21 2110.3112; 17.8036; 30.2278
90; 90; 90
5549.11Lv, Dan; Zhao, Min; Wang, Youming; Zhou, Zhenghong
3-Nitro-3,4-dihydrocoumarins: Valuable precursors for the synthesis of enantiomerically enriched masked quaternary α-amino acid derivatives with a 3,4-dihydrocoumarin scaffold
Organic & Biomolecular Chemistry, 2019
7157187 CIFC24 H24 Br2 O5P 21 21 2117.353; 24.435; 5.4165
90; 90; 90
2296.7Shit, Sudip; Devi, Namita; Devi, Ngangbam Renubala; Saikia, Anil K.
Stereoselective synthesis of hexahydrofuro[3,4-b]furan-4-ol and its dimer via tandem Prins and pinacol rearrangement.
Organic & biomolecular chemistry, 2019, 17, 7398-7407
7157189 CIFC32 H32 N2 O7P 21 21 2113; 13.405; 17.492
90; 90; 90
3048Sharma, Arun; Sharma, Vivek; Chimni, Swapandeep Singh
Organocatalytic enantioselective conjugate addition of pyrazolin-5-ones to arylomethylidene malonates.
Organic & biomolecular chemistry, 2019, 17, 9514
7157197 CIFC22 H22 O6P 21 21 216.8; 15.603; 17.7559
90; 90; 90
1883.91Liu, Zhaoming; Tan, Haibo; Chen, Kai; Chen, Yuchan; Zhang, Wenge; Chen, Shanchong; Liu, Hong-Xin; Zhang, Weimin
Rhizophols A and B, antioxidant and axially chiral benzophenones from the endophytic fungus Cytospora rhizophorae
Organic & Biomolecular Chemistry, 2019
7157204 CIFC24 H32 N4 O2P 21 21 218.83; 14.378; 17.669
90; 90; 90
2243.2Darapaneni, Chandra Mohan; Kaniraj, Prathap Jeya; Maayan, Galia
Water soluble hydrophobic peptoids via a minor backbone modification.
Organic & biomolecular chemistry, 2018, 16, 1480-1488
7157211 CIFC30 H48 O2P 21 21 216.44427; 25.748; 31.5946
90; 90; 90
5242.4Yu, Chun-Xue; Wang, Ru-Yue; Qi, Feng-Ming; Su, Pan-Jie; Yu, Yi-Fan; Li, Bing; Zhao, Ye; Zhi, De-Juan; Zhang, Zhan-Xin; Fei, Dong-Qing
Eupulcherol A, a triterpenoid with a new carbon skeleton from Euphorbia pulcherrima, and its anti-Alzheimer's disease bioactivity.
Organic & biomolecular chemistry, 2019, 18, 76-80
7157220 CIFC13 H9 F5 N2 O SP 21 21 216.07381; 10.7631; 19.448
90; 90; 90
1271.37Sansook, Supojjanee; Ocasio, Cory A.; Day, Iain J.; Tizzard, Graham J.; Coles, Simon J.; Fedorov, Oleg; Bennett, James M.; Elkins, Jonathan M.; Spencer, John
Synthesis of kinase inhibitors containing a pentafluorosulfanyl moiety.
Organic & biomolecular chemistry, 2017, 15, 8655-8660
7157235 CIFC44 H37 F N2 O4P 21 21 2111.3472; 20.551; 30.017
90; 90; 90
6999.9Zhan, Shao-Cong; Sun, Jing; Liu, Ru-Zhang; Yan, Chao-Guo
Diastereoselective construction of carbazole-based spirooxindoles via the Levy three-component reaction.
Organic & biomolecular chemistry, 2019, 18, 163-168
7157260 CIFC6 H13 K O9 SP 21 21 217.185; 10; 15.059
90; 90; 90
1082Zhang, Yunyang; Mui, Janice W.-Y.; Arumaperuma, Thimali; Lingford, James P.; Goddard-Borger, Ethan D; White, Jonathan M.; Williams, Spencer J.
Concise synthesis of sulfoquinovose and sulfoquinovosyl diacylglycerides, and development of a fluorogenic substrate for sulfoquinovosidases.
Organic & biomolecular chemistry, 2020, 18, 675-686
7157265 CIFC28 H36 O4P 21 21 217.7797; 13.9645; 21.3823
90; 90; 90
2322.96Mayorquín-Torres, Martha C; González-Orozco, Juan Carlos; Flores-Álamo, Marcos; Camacho-Arroyo, Ignacio; Iglesias-Arteaga, Martín A
Palladium catalyzed synthesis of benzannulated steroid spiroketals.
Organic & biomolecular chemistry, 2020, 18, 725-737
7157275 CIFC19 H17 N O2 SP 21 21 215.5128; 14.1945; 20.649
90; 90; 90
1615.8Zhou, Hui; Wang, Rui; Zhang, Hui; Chen, Wei; Lu, Xiao-Bing
Access to 1,3-oxazine-2,4-diones/1,3-thiazine-2,4-diones via organocatalytic CO<sub>2</sub>/COS incorporation into allenamides.
Organic & biomolecular chemistry, 2020, 18, 905-911
7157293 CIFC20 H26 O3 SP 21 21 217.14999; 12.6963; 20.1516
90; 90; 90
1829.33Hosokawa, Seijiro; Nakanishi, Keisuke; Udagawa, Yutaro; Maeda, Mitsutoshi; Sato, Seiya; Nakano, Keiji; Masuda, Toshiya; Ichikawa, Yoshiyasu
Total synthesis of exigurin: the Ugi reaction in a hypothetical biosynthesis of natural products.
Organic & biomolecular chemistry, 2020, 18, 687-693
7157305 CIFC14 H8 I2 N2P 21 21 217.7487; 8.3925; 21.639
90; 90; 90
1407.2Saha, Moumita; Das, Asish R.
Hypervalent iodine promoted ortho diversification: 2-aryl benzimidazole, quinazoline and imidazopyridine as directing templates.
Organic & biomolecular chemistry, 2020, 18, 941-955
7157307 CIFC35 H48 O7P 21 21 2111.3336; 16.1275; 18.2549
90; 90; 90
3336.68Hou, Ji-Qin; Yu, Jiang-Hong; Zhao, Heng; Dong, Ying-Ying; Peng, Qiu-Shi; Zhang, Bao-Bao; Wang, Hao
Biomimetic total syntheses of baefrutones A-D, baeckenon B, and frutescones A, D-F.
Organic & biomolecular chemistry, 2020, 18, 1135-1139
7157334 CIFC16 H16 Cl F3 O4P 21 21 215.6493; 14.4444; 21.6781
90; 90; 90
1768.95Yang, Hongzhou; Wang, Qingqing; Luo, Yuan; Ye, Ling; Li, Xinying; Chen, Feng; Zhao, Zhigang; Li, Xuefeng
Enantioselective synthesis of trifluoromethyl substituted cyclohexanones via an organocatalytic cascade Michael/aldol reaction.
Organic & biomolecular chemistry, 2020, 18, 1607-1611
7157351 CIFC25 H31 Br O4P 21 21 216.7572; 14.284; 23.8212
90; 90; 90
2299.2Miao, Jianzhuang; Zheng, Yi-Xuan; Wang, Linna; Lu, Shi-Chao; Zhang, Shi-Peng; Gong, Ya-Ling; Xu, Shu
Toward the total synthesis of grayanane diterpene mollanol A by a Prins [3 + 2] strategy.
Organic & biomolecular chemistry, 2020, 18, 1877-1880
7157370 CIFC24 H31 N OP 21 21 215.9119; 15.078; 23.745
90; 90; 90
2116.6Cao, An-Zhu; Xiao, Yu-Ting; Wu, Yan-Chen; Song, Ren-Jie; Xie, Ye-Xiang; Li, Jin-Heng
Copper-catalyzed C-H [3 + 2] annulation of N-substituted anilines with α-carbonyl alkyl bromides via C(sp<sup>3</sup>)-Br/C(sp<sup>2</sup>)-H functionalization.
Organic & biomolecular chemistry, 2020, 18, 2170-2174
7157382 CIFC20 H28 O3P 21 21 217.6786; 10.5655; 40.1904
90; 90; 90
3260.6Chen, He-Ping; Li, Jing; Zhao, Zhen-Zhu; Li, Xinyang; Liu, Shui-Lin; Wang, Qing-Yuan; Liu, Ji-Kai
Diterpenes with bicyclo[2.2.2]octane moieties from the fungicolous fungus Xylaria longipes HFG1018.
Organic & biomolecular chemistry, 2020, 18, 2410-2415
7157387 CIFC13 H14 N4 S2P 21 21 219.035; 11.727; 13.103
90; 90; 90
1388.3Teng, Qiaoqiao; Singh, Chandan; Han, Yuan; Huynh, Han Vinh
Fused azole-thiazolines via one-pot cyclization of functionalized N-heterocyclic carbene precursors.
Organic & biomolecular chemistry, 2020, 18, 2487-2491
7157408 CIFC10 H13 Br Cl O4 PP 21 21 218.7884; 9.1062; 34.664
90; 90; 90
2774.12Wang, Zexu; Zeng, Yiping; Wu, Xiaofan; Li, Zihan; Tao, Yuan; Yu, Xiaomin; Huang, Zedu; Chen, Fener
Access to chiral α-substituted-β-hydroxy arylphosphonates enabled by biocatalytic dynamic reductive kinetic resolution.
Organic & biomolecular chemistry, 2020, 18, 2672-2677
7157409 CIFC18 H21 N O6P 21 21 215.7158; 16.615; 19.036
90; 90; 90
1807.8Popik, Oskar; Grzeszczyk, Barbara; Staszewska-Krajewska, Olga; Furman, Bartłomiej; Chmielewski, Marek
Synthesis of β-lactams via diastereoselective, intramolecular Kinugasa reactions.
Organic & biomolecular chemistry, 2020, 18, 2852-2860
7157412 CIFC16 H20 B F O2P 21 21 218.532; 11.8108; 14.1961
90; 90; 90
1430.54Martínez-Aguirre, Mayte A; Flores-Alamo, Marcos; Medrano, Felipe; Yatsimirsky, Anatoly K.
Examination of pinanediol-boronic acid ester formation in aqueous media: relevance to the relative stability of trigonal and tetrahedral boronate esters.
Organic & biomolecular chemistry, 2020, 18, 2716-2726
7157413 CIFC18 H25 B O3P 21 21 216.2351; 12.5482; 20.861
90; 90; 90
1632.1Martínez-Aguirre, Mayte A; Flores-Alamo, Marcos; Medrano, Felipe; Yatsimirsky, Anatoly K.
Examination of pinanediol-boronic acid ester formation in aqueous media: relevance to the relative stability of trigonal and tetrahedral boronate esters.
Organic & biomolecular chemistry, 2020, 18, 2716-2726
7157415 CIFC31 H34 Cl N O3P 21 21 2110.3478; 14.7058; 18.6178
90; 90; 90
2833.1Qi, Suo-Suo; Jiang, Zhen-Hui; Chu, Ming-Ming; Wang, Yi-Feng; Chen, Xue-Yang; Ju, Wan-Zhen; Xu, Dan-Qian
Regioselective catalytic asymmetric N-alkylation of isoxazol-5-ones with para-quinone methides.
Organic & biomolecular chemistry, 2020, 18, 2398-2404
7157418 CIFC15 H12 O2 SP 21 21 217.5756; 8.7063; 19.34
90; 90; 90
1275.6Gharui, Chandan; Prakash, Satya; Chopra, Deepak; Pan, Subhas Chandra
Organocatalytic asymmetric addition of thioglycolates to o-quinone methides: a route to 5-substituted-5H-benzoxathiepine-2(3H)-ones.
Organic & biomolecular chemistry, 2020, 18, 2828-2833
7157420 CIFC37 H40 O2 P2P 21 21 2112.9764; 14.3781; 17.5765
90; 90; 90
3279.4Qiu, Mao-Ran; Zheng, Hong-Xing; Ye, Jing-Jing; Yan, Bing-Xia; Zhao, Chang-Qiu; Li, Qiang
Stereoselective preparation of P,axial-stereogenic allenyl bisphosphine oxides via chirality-transfer.
Organic & biomolecular chemistry, 2020, 18, 3017-3021
7157421 CIFC38 H42 O2 P2P 21 21 2113.2801; 14.3298; 17.9616
90; 90; 90
3418.1Qiu, Mao-Ran; Zheng, Hong-Xing; Ye, Jing-Jing; Yan, Bing-Xia; Zhao, Chang-Qiu; Li, Qiang
Stereoselective preparation of P,axial-stereogenic allenyl bisphosphine oxides via chirality-transfer.
Organic & biomolecular chemistry, 2020, 18, 3017-3021
7157422 CIFC26 H33 O3 PP 21 21 218.8154; 11.3911; 24.121
90; 90; 90
2422.2Qiu, Mao-Ran; Zheng, Hong-Xing; Ye, Jing-Jing; Yan, Bing-Xia; Zhao, Chang-Qiu; Li, Qiang
Stereoselective preparation of P,axial-stereogenic allenyl bisphosphine oxides via chirality-transfer.
Organic & biomolecular chemistry, 2020, 18, 3017-3021
7157427 CIFC28 H28 O2 SP 21 21 216.0742; 8.6056; 43.665
90; 90; 90
2282.5Chen, Jian-Ping; Xu, Ming-Hua
Chiral diene-promoted room temperature conjugate arylation: highly enantioselective synthesis of substituted chiral phenylalanine derivatives and α,α-di(arylmethyl)acetates.
Organic & biomolecular chemistry, 2020, 18, 4569-4574
7157433 CIFC19 H26 N2 O2P 21 21 216.0543; 8.5333; 34.582
90; 90; 90
1786.6Pan, Changduo; Huang, Gao; Shan, Yujia; Li, Yiting; Yu, Jin-Tao
Rh(iii)-Catalyzed regioselective C4 alkylation of indoles with allylic alcohols: direct access to β-indolyl ketones.
Organic & biomolecular chemistry, 2020, 18, 3038-3042
7157443 CIFC24 H18 N2 O2 SP 21 21 216.576; 16.9049; 17.5937
90; 90; 90
1955.83Arcadi, Antonio; Aschi, Massimiliano; Chiarini, Marco; Marinelli, Fabio; Marsicano, Vincenzo; Portalone, Gustavo
Experimental results and computational insight into sequential reactions of β-(2-aminophenyl)-α,β-ynones with aryl isocyanates/benzoyl isothiocyanate.
Organic & biomolecular chemistry, 2020, 18, 3177-3189
7157485 CIFC30 H52 O4P 21 21 216.61847; 9.54; 44.1844
90; 90; 90
2789.81Xiao, Long-Gao; Zhang, Yu; Zhang, Hong-Li; Li, Ding; Gu, Qiong; Tang, Gui-Hua; Yu, Qian; An, Lin-Kun
Spiroconyone A, a new phytosterol with a spiro [5,6] ring system from Conyza japonica.
Organic & biomolecular chemistry, 2020, 18, 5130-5136
7157497 CIFC17 H11 N O3 S2P 21 21 216.4978; 14.5164; 16.2262
90; 90; 90
1530.5Mondal, Santa; Mahato, Karuna; Arora, Neha; Kankane, Dheerendra; Singh, Umed Pratap; Ali, Saghir; Khan, Aftab Hossain; Ghosh, Siddhartha S.; Khan, Abu T.
Newly synthesized 3-sulfenylindole derivatives from 4-hydroxydithiocoumarin using an oxidative cross dehydrogenative coupling reaction (OCDCR): potential lead molecules for antiproliferative activity.
Organic & biomolecular chemistry, 2020, 18, 4104-4113
7157500 CIFC57 H77 N O6P 21 21 2112.008; 13.0066; 34.139
90; 90; 90
5331.9Peng, Xiaogang; Duan, Fangfang; He, Yangzhou; Gao, Ying; Chen, Juan; Chang, Jinling; Ruan, Hanli
Ergocytochalasin A, a polycyclic merocytochalasan from an endophytic fungus Phoma multirostrata XJ-2-1.
Organic & biomolecular chemistry, 2020, 18, 4056-4062
7157535 CIFC44 H46 Cl N3 O14P 21 21 218.1104; 19.5548; 27.2321
90; 90; 90
4318.9Sheppard, Daniel J.; Cameron, Scott A.; Tyler, Peter C.; Schwörer, Ralf
Comparison of disaccharide donors for heparan sulfate synthesis: uronic acids vs. their pyranose equivalents.
Organic & biomolecular chemistry, 2020, 18, 4728-4733
7157536 CIFC43 H45 N3 O14P 21 21 218.0833; 18.7876; 26.8116
90; 90; 90
4071.8Sheppard, Daniel J.; Cameron, Scott A.; Tyler, Peter C.; Schwörer, Ralf
Comparison of disaccharide donors for heparan sulfate synthesis: uronic acids vs. their pyranose equivalents.
Organic & biomolecular chemistry, 2020, 18, 4728-4733
7157550 CIFC16 H17 NP 21 21 217.2231; 14.5123; 22.3944
90; 90; 90
2347.47Zonker, Benjamin; Duman, Ediz; Hausmann, Heike; Becker, Jonathan; Hrdina, Radim
[1,2]-Rearrangement of iminium salts provides access to heterocycles with adamantane scaffold.
Organic & biomolecular chemistry, 2020, 18, 4941-4945
7157555 CIFC38 H40 Br N O2P 21 21 2110.382; 15.766; 20.036
90; 90; 90
3279.5Wu, Shu-Fang; Tu, Man-Su; Hang, Qing-Qing; Zhang, Shu; Ding, Haixia; Zhang, Yu-Chen; Shi, Feng
Construction of chiral chroman scaffolds via catalytic asymmetric (4 + 2) cyclizations of para-quinone methide derivatives with 3-vinylindoles.
Organic & biomolecular chemistry, 2020, 18, 5388-5399
7157564 CIFC46 H45 N6 O7 S2P 21 21 2110.295; 11.374; 36.37
90; 90; 90
4259Salunke, Rahul Vilas; Mishra, Pawan Kumar; Sanghvi, Yogesh S.; Ramesh, Namakkal G.
Synthesis of novel homoazanucleosides and their peptidyl analogs.
Organic & biomolecular chemistry, 2020, 18, 5639-5651
7157565 CIFC11 H20 Cl2 N4 O4P 21 21 215.4636; 15.231; 18.032
90; 90; 90
1500.6Salunke, Rahul Vilas; Mishra, Pawan Kumar; Sanghvi, Yogesh S.; Ramesh, Namakkal G.
Synthesis of novel homoazanucleosides and their peptidyl analogs.
Organic & biomolecular chemistry, 2020, 18, 5639-5651
7157566 CIFC44 H46 Cl Fe2 N2 O2 P Pd2P 21 21 2112.1801; 12.77485; 25.8213
90; 90; 90
4017.77Arthurs, Ross A.; Hughes, David L.; Richards, Christopher J.
Planar chiral palladacycle precatalysts for asymmetric synthesis.
Organic & biomolecular chemistry, 2020, 18, 5466-5472
7157590 CIFC16 H22 O4P 21 21 218.3946; 11.481; 15.2872
90; 90; 90
1473.36Ren, Panlong; Miao, Xinyu; Tang, Ting; Wu, Yueting; Wang, Jing; Zeng, Ying; Li, Yun; Gao, Kun; Yang, Yan-Long
Construction of a meroterpenoid-like compound collection by precursor-assisted biosynthesis.
Organic & biomolecular chemistry, 2020, 18, 5850-5856
7157620 CIFC20 H27 N7 O12P 21 21 219.29096; 14.5006; 20.3184
90; 90; 90
2737.39He, Huan; Cao, Ruiyuan; Cao, Ruidi; Liu, Xiao-Yu; Li, Wei; Yu, Di; Li, Yuexiang; Liu, Miaomiao; Wu, Yanmei; Wu, Pingzhou; Yang, Jin-Song; Yan, Yunzheng; Yang, Jingjing; Zheng, Zhi-Bing; Zhong, Wu; Qin, Yong
A light- and heat-driven glycal diazidation approach to nitrogenous carbohydrate derivatives with antiviral activity.
Organic & biomolecular chemistry, 2020, 18, 6155-6161
7157622 CIFC14 H16 Cl3 N6 O8P 21 21 218.6304; 10.8741; 22.9325
90; 90; 90
2152.2He, Huan; Cao, Ruiyuan; Cao, Ruidi; Liu, Xiao-Yu; Li, Wei; Yu, Di; Li, Yuexiang; Liu, Miaomiao; Wu, Yanmei; Wu, Pingzhou; Yang, Jin-Song; Yan, Yunzheng; Yang, Jingjing; Zheng, Zhi-Bing; Zhong, Wu; Qin, Yong
A light- and heat-driven glycal diazidation approach to nitrogenous carbohydrate derivatives with antiviral activity.
Organic & biomolecular chemistry, 2020, 18, 6155-6161
7157623 CIFC18 H24 N10 O10P 21 21 218.6075; 10.7485; 33.736
90; 90; 90
3121.2He, Huan; Cao, Ruiyuan; Cao, Ruidi; Liu, Xiao-Yu; Li, Wei; Yu, Di; Li, Yuexiang; Liu, Miaomiao; Wu, Yanmei; Wu, Pingzhou; Yang, Jin-Song; Yan, Yunzheng; Yang, Jingjing; Zheng, Zhi-Bing; Zhong, Wu; Qin, Yong
A light- and heat-driven glycal diazidation approach to nitrogenous carbohydrate derivatives with antiviral activity.
Organic & biomolecular chemistry, 2020, 18, 6155-6161
7157624 CIFC13 H16 N6 O8P 21 21 217.2784; 9.2019; 26.166
90; 90; 90
1752.5He, Huan; Cao, Ruiyuan; Cao, Ruidi; Liu, Xiao-Yu; Li, Wei; Yu, Di; Li, Yuexiang; Liu, Miaomiao; Wu, Yanmei; Wu, Pingzhou; Yang, Jin-Song; Yan, Yunzheng; Yang, Jingjing; Zheng, Zhi-Bing; Zhong, Wu; Qin, Yong
A light- and heat-driven glycal diazidation approach to nitrogenous carbohydrate derivatives with antiviral activity.
Organic & biomolecular chemistry, 2020, 18, 6155-6161
7157629 CIFC11 H11 N O2P 21 21 217.5291; 7.4902; 17.0281
90; 90; 90
960.29Braire, Julien; Dorcet, Vincent; Vidal, Joëlle; Lalli, Claudia; Carreaux, François
BINOL derivatives-catalysed enantioselective allylboration of isatins: application to the synthesis of (R)-chimonamidine.
Organic & biomolecular chemistry, 2020, 18, 6042-6046
7157630 CIFC12 H13 N O2P 21 21 217.3607; 8.0406; 17.598
90; 90; 90
1041.5Braire, Julien; Dorcet, Vincent; Vidal, Joëlle; Lalli, Claudia; Carreaux, François
BINOL derivatives-catalysed enantioselective allylboration of isatins: application to the synthesis of (R)-chimonamidine.
Organic & biomolecular chemistry, 2020, 18, 6042-6046
7157638 CIFC28 H30 N2 O3 S4P 21 21 219.4421; 14.8451; 19.2118
90; 90; 90
2692.9García de la Concepción, Juan; Ávalos, Martín; Jiménez, José L; Cintas, Pedro; Light, Mark E.
A fully diastereoselective oxidation of a mesoionic dipole with triplet molecular oxygen.
Organic & biomolecular chemistry, 2020, 18, 6328-6339
7157640 CIFC34 H26 N2 O3 S4P 21 21 2112.482; 12.8583; 19.5132
90; 90; 90
3131.82García de la Concepción, Juan; Ávalos, Martín; Jiménez, José L; Cintas, Pedro; Light, Mark E.
A fully diastereoselective oxidation of a mesoionic dipole with triplet molecular oxygen.
Organic & biomolecular chemistry, 2020, 18, 6328-6339
7157651 CIFC20 H23 Cl5 D N3 O4 S2P 21 21 2110.5857; 14.0014; 17.5197
90; 90; 90
2596.68Kletskov, Alexey V.; Zatykina, Anastasya D.; Grudova, Mariya V.; Sinelshchikova, Anna A.; Grigoriev, Mikhail S.; Zaytsev, Vladimir P.; Gil, Diego M.; Novikov, Roman A.; Zubkov, Fedor I.; Frontera, Antonio
Raise the anchor! Synthesis, X-ray and NMR characterization of 1,3,5-triazinanes with an axial tert-butyl group.
Organic & biomolecular chemistry, 2020, 18, 8386-8394
7157654 CIFC20 H23 Cl3 D F2 N3 O4 S2P 21 21 2110.4481; 14.3121; 16.4591
90; 90; 90
2461.2Kletskov, Alexey V.; Zatykina, Anastasya D.; Grudova, Mariya V.; Sinelshchikova, Anna A.; Grigoriev, Mikhail S.; Zaytsev, Vladimir P.; Gil, Diego M.; Novikov, Roman A.; Zubkov, Fedor I.; Frontera, Antonio
Raise the anchor! Synthesis, X-ray and NMR characterization of 1,3,5-triazinanes with an axial tert-butyl group.
Organic & biomolecular chemistry, 2020, 18, 8386-8394
7157667 CIFC15 H30 O S2P 21 21 215.0392; 8.4897; 38.3953
90; 90; 90
1642.6Scheutz, Georg M.; Rowell, Jonathan L.; Wang, Fu-Sheng; Abboud, Khalil A.; Peng, Chi-How; Sumerlin, Brent S.
Synthesis of functional 1,2-dithiolanes from 1,3-bis-<i>tert</i>-butyl thioethers.
Organic & biomolecular chemistry, 2020, 18, 6509-6513
7157675 CIFC34 H25 N O4P 21 21 217.2273; 12.6042; 29.1348
90; 90; 90
2654.02Mu, Yuanyang; Yuan, Yang; Wang, Ye; Xu, Murong; Feng, Ye; Zhao, Yulei; Li, Yanzhong
Synthesis of indoline-fused eight-membered azaheterocycles through Zn-catalyzed dearomatization of indoles and subsequent base-promoted C-C activation.
Organic & biomolecular chemistry, 2020, 18, 6916-6926
7157711 CIFC18 H24 O3P 21 21 217.0307; 8.666; 25.171
90; 90; 90
1533.6Chang, Fang-Rong; Wang, Shih-Wei; Chen, Shu-Rong; Lee, Ching-Ying; Sheu, Jyh-Horng; Cheng, Yuan-Bin
Aleuritin, a novel dinor-diterpenoid from the twigs of <i>Aleurites moluccanus</i> with an anti-lymphangiogenic effect.
Organic & biomolecular chemistry, 2020, 18, 7892-7898
7157712 CIFC20 H28 O2P 21 21 217.526; 13.1519; 17.4059
90; 90; 90
1722.9Chang, Fang-Rong; Wang, Shih-Wei; Chen, Shu-Rong; Lee, Ching-Ying; Sheu, Jyh-Horng; Cheng, Yuan-Bin
Aleuritin, a novel dinor-diterpenoid from the twigs of <i>Aleurites moluccanus</i> with an anti-lymphangiogenic effect.
Organic & biomolecular chemistry, 2020, 18, 7892-7898
7157731 CIFC16 H20 O5P 21 21 217.2801; 9.9611; 18.9298
90; 90; 90
1372.75Yan, Hai-Wei; Zhang, Xu; Yang, Ya-Nan; Feng, Zi-Ming; Jiang, Jian-Shuang; Zhang, Pei-Cheng
Archromones A-F, unusual polycyclic dearomatic geranylquinol derivatives from the roots of <i>Arnebia euchroma</i>.
Organic & biomolecular chemistry, 2020, 18, 8424-8432
7157733 CIFC16 H18 O3P 21 21 217.1617; 9.7401; 18.6984
90; 90; 90
1304.32Yan, Hai-Wei; Zhang, Xu; Yang, Ya-Nan; Feng, Zi-Ming; Jiang, Jian-Shuang; Zhang, Pei-Cheng
Archromones A-F, unusual polycyclic dearomatic geranylquinol derivatives from the roots of <i>Arnebia euchroma</i>.
Organic & biomolecular chemistry, 2020, 18, 8424-8432
7157740 CIFC26 H24 F N3P 21 21 215.6056; 17.422; 22.161
90; 90; 90
2164.3Tiwari, Vibha; Bingham, Jacob T.; Vyas, Shubham; Singh, Anand
Intermolecular fluoroamination of allenes towards substituted vinyl fluorides
Organic & Biomolecular Chemistry, 2020, 18, 9044-9049
7157745 CIFC36 H32 N2 O2P 21 21 219.3208; 15.9714; 19.0521
90; 90; 90
2836.21Yao, Chao; Wu, Piao; Huang, Yue; Chen, Yaoqi; Li, Lin; Li, Yue-Ming
Binaphthyl-based chiral ligands: design, synthesis and evaluation of their performance in enantioselective addition of diethylzinc to aromatic aldehydes.
Organic & biomolecular chemistry, 2020, 18, 9712-9725
7157758 CIFC31 H31 Cl Ir N OP 21 21 217.7357; 14.3256; 22.7397
90; 90; 90
2520Smith, Jennifer; Kacmaz, Aysecik; Wang, Chao; Villa-Marcos, Barbara; Xiao, Jianliang
Chiral cyclometalated iridium complexes for asymmetric reduction reactions.
Organic & biomolecular chemistry, 2021, 19, 279-284
7157774 CIFC17 H20 Cl N O2P 21 21 2110.4037; 10.6504; 13.4206
90; 90; 90
1487.05Thaima, Thanphat; Yazici, Arife; Auranwiwat, Chiramet; Willis, Anthony C.; Wille, Uta; Limtharakul, Thunwadee; Pyne, Stephen G.
Synthesis of spirocyclic heterocycles from α,β-unsaturated <i>N</i>-acyliminium ions.
Organic & biomolecular chemistry, 2021, 19, 259-272
7157791 CIFC28 H30 N2P 21 21 216.859; 17.0662; 19.6709
90; 90; 90
2302.6Gadigennavar, Savita; Ranganathan, Madhav; Sankararaman, Sethuraman
Which isomer is it, 1,2,5,6- or 1,4,5,8-tetrasubstituted cycloocta-1,3,5,7-tetraene? Synthesis of symmetrically tetrasubstituted cycloocta-1,3,5,7-tetraene derivatives
Organic & Biomolecular Chemistry, 2020, 18, 9284-9291
7157794 CIFC26 H32 O7P 21 21 218.0223; 13.6842; 21.6959
90; 90; 90
2381.75Kikuchi, Takashi; Akita, Keiko; Koike, Hiroki; In, Yasuko; Yamada, Takeshi; Tanaka, Reiko
Carapanins A–C: new limonoids from andiroba (Carapa guianensis) fruit oil
Organic & Biomolecular Chemistry, 2020, 18, 9268-9274
7157804 CIFC17 H16 O5P 21 21 219.5125; 10.2643; 14.9575
90; 90; 90
1460.4Gao, Yu-Qi; Hou, Yi; Chen, Junhan; Zhen, Yanxia; Xu, Dongyang; Zhang, Hongli; Wei, Hongbo; Xie, Weiqing
Asymmetric synthesis of 9-alkyl tetrahydroxanthenones <i>via</i> tandem asymmetric Michael/cyclization promoted by chiral phosphoric acid.
Organic & biomolecular chemistry, 2021, 19, 348-354
7157830 CIFC18 H17 N O3P 21 21 218.9919; 12.2777; 14.0831
90; 90; 90
1554.77Chang, Zhiqian; Zhu, Huilong; Wu, Changhui; Xing, Junhao; Dou, Xiaowei
A rhodium-catalysed conjugate addition/cyclization cascade for the asymmetric synthesis of 2-amino-4H-chromenes.
Organic & biomolecular chemistry, 2021, 19, 785-788
7157837 CIFC24 H25 Br N2 O5P 21 21 214.9355; 9.9998; 44.492
90; 90; 90
2195.9Marshall, James W.; de Mattos-Shipley, Kate M J; Ghannam, Iman A. Y.; Munawar, Asifa; Killen, Jonathan C.; Lazarus, Colin M.; Cox, Russell J.; Willis, Christine L.; Simpson, Thomas J.
Fusarochromene, a novel tryptophan-derived metabolite from <i>Fusarium sacchari</i>.
Organic & biomolecular chemistry, 2021, 19, 182-187
7157838 CIFC22 H18 Br F3 N2 O2P 21 21 216.2936; 14.1248; 23.296
90; 90; 90
2070.92Gao, Yang; Song, Xue; Yan, Ru-Jie; Du, Wei; Chen, Ying-Chun
Asymmetric β,γ'-regioselective [4 + 3] and [4 + 2] annulations of α-vinylenals <i>via</i> cascade iminium ion-dienamine catalysis.
Organic & biomolecular chemistry, 2021, 19, 151-155
7157851 CIFC25 H21 Br O4P 21 21 2110.0294; 10.8154; 19.2909
90; 90; 90
2092.52Xu, Yan-Li; Qin, Zhou-Zhou; Wang, Yu-Xia; Zhao, Peng-Fei; Li, Hong-Feng; Du, Zhi-Hong; Da, Chao-Shan
Highly enantioselective one-pot sequential synthesis of valerolactones and pyrazolones bearing all-carbon quaternary stereocentres.
Organic & biomolecular chemistry, 2021, 19, 1610-1615
7157852 CIFC25 H23 Cl N2 O3P 21 21 217.0441; 16.2447; 18.72
90; 90; 90
2142.12Xu, Yan-Li; Qin, Zhou-Zhou; Wang, Yu-Xia; Zhao, Peng-Fei; Li, Hong-Feng; Du, Zhi-Hong; Da, Chao-Shan
Highly enantioselective one-pot sequential synthesis of valerolactones and pyrazolones bearing all-carbon quaternary stereocentres.
Organic & biomolecular chemistry, 2021, 19, 1610-1615
7157855 CIFC26 H23 Cl N2 O3P 21 21 2110.234; 14.235; 30.529
90; 90; 90
4447Guo, Xing; Chen, Xuling; Cheng, Yuyu; Chang, Xiaoyong; Li, Xuechen; Li, Pengfei
Organocatalytic enantioselective [2 + 4]-annulation of γ-substituted allenoates with <i>N</i>-acyldiazenes for the synthesis of optically active 1,3,4-oxadiazines.
Organic & biomolecular chemistry, 2021, 19, 1727-1731
7157865 CIFC27 H36 N2 O3P 21 21 218.2965; 8.9484; 34.1519
90; 90; 90
2535.45Kimura, Yuto; Uraguchi, Daisuke; Ooi, Takashi
Catalytic asymmetric synthesis of 5-membered alicyclic α-quaternary β-amino acids <i>via</i> [3 + 2]-photocycloaddition of α-substituted acrylates.
Organic & biomolecular chemistry, 2021, 19, 1744-1747
7157880 CIFC19 H23 N O S2P 21 21 218.626; 9.2018; 22.6467
90; 90; 90
1797.58Welsh, Erin N.; Robertson, Katherine N.; Speed, Alexander W. H.
Short syntheses of 1-substituted dibenzothiophene derivatives.
Organic & biomolecular chemistry, 2021, 19, 2000-2007
7157901 CIFC13 H14 F N O5P 21 21 217.40072; 9.1371; 18.7024
90; 90; 90
1264.68Sperga, Arturs; Kazia, Armands; Veliks, Janis
Monofluorinated 5-membered rings via fluoromethylene transfer: synthesis of monofluorinated isoxazoline N-oxides.
Organic & biomolecular chemistry, 2021, 19, 2688-2691
7157918 CIFC10 H15 N3 O2P 21 21 216.577; 10.7154; 15.0191
90; 90; 90
1058.47Ptiček, Lucija; Hok, Lucija; Grbčić, Petra; Topić, Filip; Cetina, Mario; Rissanen, Kari; Pavelić, Sandra Kraljević; Vianello, Robert; Racané, Livio
Amidino substituted 2-aminophenols: biologically important building blocks for the amidino-functionalization of 2-substituted benzoxazoles.
Organic & biomolecular chemistry, 2021, 19, 2784-2793
7157923 CIFC16 H17 N O4P 21 21 215.2488; 7.5956; 33.4224
90; 90; 90
1332.48Liang, Leilei; Li, Ji; Shen, Baochun; Zhang, Yili; Liu, Jianping; Chen, Jingbo; Liu, Dandan
The effect of carbonyl on the isomerization of a galanthan ring system and total synthesis of (±)-β-lycorane.
Organic & biomolecular chemistry, 2021, 19, 2767-2772
7157931 CIFC15 H9 B Cl2 N2 OP 21 21 219.266; 11.4559; 12.8747
90; 90; 90
1366.65Iqbal, S. A.; Yuan, K.; Cid, J.; Pahl, J.; Ingleson, M. J.
Controlling selectivity in N-heterocycle directed borylation of indoles.
Organic & biomolecular chemistry, 2021, 19, 2949-2958
7157963 CIFC26 H21 N O SP 21 21 216.149; 16.882; 19.24
90; 90; 90
1997.3Li, Zhen; Vijaykumar, Gonela; Li, Xiangdong; Golz, Christopher; Alcarazo, Manuel
5-(Diarylimino)- and 5-(sulfoximido)dibenzothiophenium triflates: syntheses and applications as electrophilic aminating reagents.
Organic & biomolecular chemistry, 2021, 19, 2941-2948
7157984 CIFC38 H37 Cl F6 N2 P2 RuP 21 21 2110.4412; 11.3932; 29.2341
90; 90; 90
3477.65Huang, Ming; Li, Yinwu; Lan, Xiao-Bing; Liu, Jiahao; Zhao, Cunyuan; Liu, Yan; Ke, Zhuofeng
Ruthenium(II) complexes with N-heterocyclic carbene-phosphine ligands for the <i>N</i>-alkylation of amines with alcohols.
Organic & biomolecular chemistry, 2021, 19, 3451-3461
7157989 CIFC25 H19 Br N2 O4 SP 21 21 216.7354; 18.2897; 19.0257
90; 90; 90
2343.75Chang, Li; Zhu, Guang-Yu; Yang, Ting; Zhao, Xiao-Li; Shi, Min; Zhao, Mei-Xin
Organocatalytic asymmetric formal [3 + 2] cycloaddition reaction of isocyanoacetates with saccharin-derived 1-azadienes.
Organic & biomolecular chemistry, 2021, 19, 3687-3697
7157999 CIFC25 H35 N O7P 21 21 2110.8932; 17.0966; 39.2989
90; 90; 90
7318.9Kong, Xiang-Kai; Xiong, Zhi-Min; Zhi, Xiang; Meng, Xue-Ling; Zhao, Jing-Feng; Chen, Wen; Zhang, Hongbin
Lewis acid mediated cyclization: synthesis of 2 spirocyclohexylindolines.
Organic & biomolecular chemistry, 2021, 19, 4043-4047
7158001 CIFC25 H35 N O7P 21 21 2110.8971; 17.1101; 39.2778
90; 90; 90
7323.4Kong, Xiang-Kai; Xiong, Zhi-Min; Zhi, Xiang; Meng, Xue-Ling; Zhao, Jing-Feng; Chen, Wen; Zhang, Hongbin
Lewis acid mediated cyclization: synthesis of 2 spirocyclohexylindolines.
Organic & biomolecular chemistry, 2021, 19, 4043-4047

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